9 research outputs found
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- Publication venue
- 'Pharmaceutical Society of Japan'
- Publication date
- Field of study
Physico-chemiacl approach for prediction of the skin concentration of topically applied drugs
- Publication venue
- Wolters Kluwer Medknow Publications
- Publication date
- Field of study
Mathematical Model to Predict Skin Concentration after Topical Application of Drugs
- Publication venue
- 'MDPI AG'
- Publication date
- 01/12/2013
- Field of study
Skin permeation experiments have been broadly done since 1970s to 1980s as an evaluation method for transdermal drug delivery systems. In topically applied drug and cosmetic formulations, skin concentration of chemical compounds is more important than their skin permeations, because primary target site of the chemical compounds is skin surface or skin tissues. Furthermore, the direct pharmacological reaction of a metabolically stable drug that binds with specific receptors of known expression levels in an organ can be determined by Hillâs equation. Nevertheless, little investigation was carried out on the test method of skin concentration after topically application of chemical compounds. Recently we investigated an estimating method of skin concentration of the chemical compounds from their skin permeation profiles. In the study, we took care of â3Rsâ issues for animal experiments. We have proposed an equation which was capable to estimate animal skin concentration from permeation profile through the artificial membrane (silicone membrane) and animal skin. This new approach may allow the skin concentration of a drug to be predicted using Fickâs second law of diffusion. The silicone membrane was found to be useful as an alternative membrane to animal skin for predicting skin concentration of chemical compounds, because an extremely excellent extrapolation to animal skin concentration was attained by calculation using the silicone membrane permeation data. In this chapter, we aimed to establish an accurate and convenient method for predicting the concentration profiles of drugs in the skin based on the skin permeation parameters of topically active drugs derived from steady-state skin permeation experiments
Mathematical Model to Predict Skin Concentration after Topical Application of Drugs
- Author
- Publication venue
- 'MDPI AG'
- Publication date
- Field of study
A useful technique using imaging mass spectrometry for detecting the skin distribution of topically applied lidocaine
- Author
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Macromolecular Delivery into Skin Using a Hollow Microneedle
- Author
- Al-Qallaf B. Das D. B., Mori D., C
- Cormier M. Johnson B., Ameri M., N
- Hiroaki Todo
- Kenji Sugibayashi
- Nanthida Wonglertnirant
- Peppas N.A.
- Praneet Opanasopit
- Sugibayashi K. Todo H., Oshizaka T
- Tanasait Ngawhirunpat
- Verbaan F. J. Bal S. M., van den B
- Wang P. M. Cornwell M., Hill J., P
- Wu X. M. Todo H., Sugibayashi K.
- Publication venue
- 'Pharmaceutical Society of Japan'
- Publication date
- 01/01/2010
- Field of study
Lidocaine patches for postcesarean pain control in obese women: a pilot randomized controlled trial
- Author
- Abbott
- Adesope
- Altenau
- Alvarez
- Bai
- Bamigboye
- Bateman
- Bauchat
- Blake
- Bonnesen
- Catalano
- Champaneria
- Comer
- Dryden
- Elhafz
- Feeley
- Frieden
- Fyfe
- Gammaitoni
- Gammaitoni
- Gilhooly
- Gross
- Habib
- Hagle
- Hartge
- Horlocker
- Kessler
- Kessous
- Kleiman
- Klein
- Kwon
- Lam
- Lau
- Lebedevs
- Lee
- Lee
- Lloret-Linares
- Mace
- Magriples
- Mamun
- Martin
- Mason
- Mhyre
- Nightingale
- Oderda
- Ortega
- Oshizaka
- Overdyk
- OâDwyer
- Pallasmaa
- Patel
- Peahl
- Robinson
- Rosenberg
- Saber
- Sadigursky
- Schug
- Schwinghammer
- Sekhavat
- Sharawi
- Soens
- Stamilio
- Sutton
- Tan
- Upton
- Upton
- Weiss
- Zeisler
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Early Clinical Predictors of Hepatic Veno-Occlusive Disease/Sinusoidal Obstruction Syndrome after Myeloablative Stem Cell Transplantation
- Author
- Antin
- Armand
- Bearman
- Brett Glotzbecker
- Carreras
- Carreras
- Cheuk
- Coppell
- Corbacioglu
- Corbacioglu
- Corbacioglu
- Corey Cutler
- Cutler
- Cutler
- Dalle
- de Witte
- DeLeve
- Edwin P. Alyea
- Essell
- Gordon
- Haesook T. Kim
- Ho
- John Koreth
- Jones
- Joseph H. Antin
- Kantarjian
- Lindsey E. Roeker
- Liu
- Mahalati
- McDonald
- McDonald
- McDonald
- Mori
- Oshizaka
- Park
- Paul G. Richardson
- Philippe Armand
- Prashant Nageshwar
- Ricart
- Richardson
- Richardson
- Richardson
- Rio
- Robert J. Soiffer
- Ruutu
- Sarah Nikiforow
- Shin
- Strouse C
- Tanikawa
- Tay
- Toh
- Tsirigotis
- Vincent T. Ho
- Wadleigh
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
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- Lerner
- Lerner
- Lerner
- Lerner
- Lerner
- Leskowitz
- Leskowitz
- Lesley
- Lesley
- Levey
- Levine
- Levine
- Levine
- Levine
- Levine
- Lewis
- Lewis
- Liacopoulos
- Liang
- Lichtenberg
- Lieberman
- Liew
- Liew
- Lightbody
- Lilliehöök
- Lilly
- Lilly
- Lilly
- Lindahl
- Lindenmann
- Lindstrom
- Lipsky
- Lipsky
- Lischner
- Lischner
- Liskowska-Bernstein
- Litwin
- Litwin
- Lobo
- Loewi
- Lohmann-Matthes
- Lohrmann
- Lonai
- Lonai
- Lonai
- Lonai
- Lonai
- Lonai
- Lonai
- Loor
- Loor
- Loor
- LotzovĂĄ
- Louis
- Lozner
- Lundstedt
- Lynch
- MacDermott
- MacDonald
- MacDonald
- Mackaness
- MacLean
- MacLennan
- Mage
- Mage
- Mage
- Maguire
- Maguire
- Makinodan
- Makinodan
- Malchow
- Mandel
- Mandi
- Mann
- Mann
- Manning
- Manning
- Manson
- Many
- Marbrook
- Marchalonis
- Marchalonis
- Marchalonis
- Marchalonis
- Marchalonis
- Marchalonis
- Marchalonis
- Marker
- Marrack
- Marsh
- Martin
- Mason
- Matter
- McArthur
- McBride
- McBride
- McCalmon
- McCullagh
- McCullagh
- McDevitt
- McDevitt
- McDevitt
- McDevitt
- McDevitt
- McDevitt
- McDevitt
- McKearn
- McKearn
- McKearn
- McKenzie
- McKenzie
- McKenzie
- McKenzie
- McMaster
- McMichael
- McWilliams
- Medawar
- Melcher
- Melchers
- Melchers
- Melchers
- Meo
- Meo
- Meo
- Meo
- Meo
- Meo
- Merchant
- Merler
- Metcalf
- Metzgar
- Michael
- Micheel
- Michlmayr
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Miller
- Mills
- Miranda
- Mishell
- Mitchell
- Mitchell
- Mitchell
- Mitchell
- Mitchell
- Mitchell
- Mitchell
- Mitchell
- Mitchison
- Mitchison
- Mitchison
- Mitchison
- Mitchison
- Modabber
- Mond
- Mond
- Moore
- Moore
- Moore
- Moore
- Moorhead
- Moorhead
- Moroz
- Moroz
- Moroz
- Mosier
- Mosier
- Mosier
- Mosier
- Mosier
- Mosier
- Mosier
- Mosier
- Mosier
- Mota
- Mozes
- Mozes
- Mozes
- Mozes
- Mozes
- Mudd
- Munro
- Munro
- Munro
- Muramatsu
- Murphy
- Murphy
- Murphy
- Murphy
- Murphy
- MÀkelÀ
- MÀkelÀ
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Möller
- Nabholz
- Nabholz
- Nabholz
- Nagy
- Namba
- Naor
- Naor
- Nathenson
- Natvig
- Nauciel
- Neauport-Sautes
- Neauport-Sautes
- Nelson
- Neveu
- Newburger
- Niederhuber
- Niederhuber
- Niederhuber
- Niederhuber
- Nielsen
- Nordin
- Nordin
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nossal
- Nussenzweig
- Nussenzweig
- Nussenzweig
- Obata
- Ochiai
- Ogilvie
- Ogilvie
- Oka
- Okudaira
- Okudaira
- Okudaira
- Okumura
- Okumura
- Okumura
- Okumura
- Okumura
- Old
- Old
- Old
- Old
- Ollsson
- Opitz
- Opitz
- Oppenheim
- Ordal
- Ornellas
- Orr
- Osborne
- Osborne
- Osborne
- Osborne
- Osborne
- Osborne
- Oshizaka
- Osmond
- Osoba
- Osoba
- Ostberg
- Oudin
- Ovary
- Owen
- Owen
- Owen
- Owen
- Owen
- Ozato
- Paley
- Pang
- Pantelouris
- Papageorgious
- Papamichael
- Papamichael
- Paraskevas
- Paraskevas
- Paraskevas
- Paraskevas
- Parathenais
- Parish
- Parish
- Parish
- Parish
- Parish
- Parish
- Parish
- Parish
- Parish
- Parish
- Parish
- Parker
- Parkhouse
- Paul
- Paul
- Paul
- Paul
- Pauling
- Pawlak
- Pawlak
- Peavy
- Peavy
- Peavy
- Peavy
- Peck
- Pegrum
- Penn
- Pepys
- Pepys
- Perey
- Perini
- Perkins
- Perlmann
- Perlmann
- Perlmann
- Perlmann
- Pernis
- Pernis
- Pernis
- Pernis
- Pernis
- Pernis
- Pernis
- Pernis
- Perren
- Peter
- Pfizenmaier
- Pfizenmaier
- Phanuphak
- Phillips
- Phillips-Quagliata
- Pick
- Pickard
- Pierce
- Pierce
- Pierce
- Pierce
- Pierce
- Pierce
- Pierce
- Pierce
- Pierce
- Pierce
- Piessens
- Piguet
- Piguet
- Piguet
- Pincus
- Pincus
- Plate
- Plate
- Plate
- Plate
- Plate
- Playfair
- Playfair
- Playfair
- Playfair
- Playfair
- Poe
- Poe
- Poe
- Polak
- Poljak
- Potter
- Poulik
- Poulter
- Press
- Press
- Press
- Press
- Press
- Preud'homme
- Preud'homme
- Preud'homme
- Preud'homme
- Princler
- Pritchard
- Pryjma
- Pryjma
- Rabellino
- Rabellino
- Rabinowitz
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Raff
- Rajapakse
- Rajewsky
- Rajewsky
- Rajewsky
- Rajewsky
- Rajewsky
- Rajewsky
- Ramasamy
- Ramasamy
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Ramseier
- Rask
- Rask
- Rask
- Rehn
- Reif
- Reif
- Reif
- Reif
- Reif
- Reisfeld
- Revillard
- Revoltella
- Rich
- Rich
- Rich
- Rich
- Rich
- Rieke
- RiethmĂŒller
- Rittenberg
- Rocklin
- Roelants
- Roelants
- Roelants
- Roelants
- Roelants
- Romano
- Romano
- Roseman
- Rosenberg
- Rosenstreich
- Rosenthal
- Rosenthal
- Rosenthal
- Rosenthal
- Ross
- Ross
- Rotter
- Rotter
- Rotter
- Rotter
- Rouse
- Rowe
- Rowe
- Rowe
- Rowe
- Rowe
- Rowe
- Rowlands
- Rowley
- Rowley
- Rowley
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Rubin
- Ruddy
- Ruhl
- Rutishauser
- Rutishauser
- Ryan
- RychlĂkovĂĄ
- Ryder
- Ryser
- Röllinghoff
- Röllinghoff
- RĂŒde
- RĂŒde
- Sabbadini
- Sachs
- Sachs
- Sachs
- Sachs
- Sado
- Salvin
- Salvin
- Salvin
- Santer
- Sarkar
- Sarvas
- Sato
- Sauser
- Schaffner
- Scheid
- Scheid
- Scheid
- Scheid
- Schendel
- Schendel
- Scher
- Scher
- Scher
- Scher
- Scher
- Schierman
- Schimpl
- Schimpl
- Schimpl
- Schimpl
- Schimpl
- Schimpl
- Schirrmacher
- Schirrmacher
- Schirrmacher
- Schirrmacher
- Schirrmacher
- Schirrmacher
- Schlegel
- Schlegel
- Schlegel
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlesinger
- Schlossman
- Schmitt-Verhulst
- Schmitt-Verhulst
- Schrader
- Schrader
- Schrader
- Schrader
- Schrader
- Schrader
- Schrader
- Schrader
- Schrader
- Schreiner
- Schwartz
- Schwartz
- Schwartz
- Schwartz
- Schwartz
- Schwartz
- Schwartz
- Scibienski
- Scott
- Segal
- Segal
- Seger
- Sela
- Seligmann
- Sell
- Sell
- Sell
- Senyk
- Seon
- Shand
- Sharon
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Shearer
- Sheehy
- Shek
- Sher
- Sherwin
- Shevach
- Shevach
- Shevach
- Shevach
- Shevach
- Shevach
- Shevach
- Shevach
- Shigeno
- Shiku
- Shinohara
- Shortman
- Shortman
- Shortman
- Shreffler
- Shreffler
- Shreffler
- Shreffler
- Shreffler
- Shreffler
- Shreffler
- Sidman
- Sidman
- Sidman
- Siegal
- Silver
- Silver
- Silver
- Silver
- Silver
- Silver
- Silverman
- Silverstein
- Silverstein
- Silverstein
- Simonsen
- Simonsen
- Simonsen
- Simonsen
- Simpson
- Simpson
- Simpson
- Sinclair
- Singer
- Singh
- Siskind
- Sjöberg
- Sjöberg
- Sjöberg
- Sjöberg
- Sjöberg
- Sjöberg
- Sjögren
- Skidmore
- Skidmore
- Skidmore
- Skidmore
- Sledge
- Small
- Small
- Smith
- Smith
- Smith
- Smith
- Snary
- Snell
- Snell
- Snell
- Snell
- Snippe
- Solheim
- Solliday
- Solliday-Rich
- Solliday-Rich
- Solliday-Rich
- Sollinger
- Sollinger
- Sondel
- Sondel
- Sondel
- Spear
- Spear
- Spiegelberg
- Spiegelberg
- Sprent
- Sprent
- Sprent
- Sprent
- Sprent
- Stackpole
- Staines
- Staines
- Stavitsky
- Stecher
- Stern
- Sternberg
- Stimpfling
- Stimpfling
- Stobo
- Stobo
- Stobo
- Stobo
- Stobo
- Stobo
- Stobo
- Stocker
- Stocker
- Stockert
- Stockert
- Stockert
- Stockert
- Stockman
- Stollar
- Storrie
- Stout
- Stout
- Stout
- Stout
- Strand
- StrannegÄrd
- Strausbauch
- Strayer
- Strayer
- Strejan
- Strober
- Strober
- Strober
- Strober
- Strober
- Strober
- Strominger
- Strominger
- Ströbel
- Stulting
- Stutman
- Stutman
- Stutman
- Stutman
- Stutman
- Stutman
- Stutman
- StĂŒck
- Sulica
- Sultzer
- Szenberg
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Tada
- Takahashi
- Takahashi
- Takahashi
- Takahashi
- Takatsu
- Takatsu
- Takatsu
- Takemori
- Takemori
- Taliaferro
- Taliaferro
- Taliaferro
- Talmage
- Talmage
- Tamura
- Tanigaki
- Taniguchi
- Taniguchi
- Taniguchi
- Taniguchi
- Taniguchi
- Taniguchi
- Taussig
- Taussig
- Taussig
- Taussig
- Taussig
- Taussig
- Taylor
- Taylor
- Taylor
- Taylor
- Taylor
- Taylor
- Teodorczyk
- Terhorst
- Theodor
- Theofilopoulos
- Thomas
- Thompson
- Thompson
- Thorbecke
- Thorbecke
- Thorsby
- Thrasher
- Tigelaar
- Tigelaar
- Tigelaar
- Till
- Tittor
- Tittor
- Toivanen
- Toivanen
- Toivanen
- Toivanen
- Torrigiani
- Trainin
- Trenkner
- Trenkner
- Treves
- Trinchieri
- Triplett
- Trowbridge
- Trowbridge
- Truffa-Bachi
- Tung
- Tung
- Turk
- Turk
- Turk
- Turpen
- Tyan
- Tyan
- Tyan
- Uhr
- Uhr
- Uhr
- Uhr
- Umiel
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Unanue
- Vadas
- van Boxel
- van Boxel
- van Boxel
- van Boxel
- Van DenEngh
- Van Furth
- Van Rood
- Vann
- Vann
- Vann
- Vann
- Vaz
- Vaz
- Veit
- Verma
- Vischer
- Vischer
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vitetta
- Vogel
- Volpe
- von Boehmer
- von Boehmer
- von Boehmer
- von Boehmer
- von Boehmer
- von Boehmer
- von Boehmer
- von Boehmer
- von Boehmer
- Vossen
- Wagner
- Wagner
- Wagner
- Wagner
- Wagner
- Wagner
- Wagner
- Wagner
- Wagner
- Wagner
- Waksman
- Waksman
- Waksman
- Waldman
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waldmann
- Waltenbaugh
- Walters
- Walters
- Wang
- Wang
- Wang
- Warnatz
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warner
- Warr
- Watanabe
- Watanabe
- Watanabe
- Watanabe
- Watson
- Watson
- Watson
- Watson
- Watson
- Webb
- Weber
- Weber
- Weber
- Weigle
- Weigle
- Weigle
- Weinbaum
- Weissman
- Weissman
- Wekerle
- Welsh
- Werblin
- Wernet
- Wernet
- Weston
- White
- White
- Widmer
- Wigzell
- Wigzell
- Wigzell
- Wigzell
- Wigzell
- Willcox
- Willcox
- Williams
- Williamson
- Wilson
- Wilson
- Wilson
- Wilson
- Wilson
- Wilson
- Wilson
- Wilson
- Wilson
- Winchester
- Winkelstein
- Winn
- Winn
- Wittingham
- Wofsy
- Wolf
- Wolf
- Wood
- Wood
- Wood
- Wood
- Woodruff
- Wortis
- Wright
- Wunderlich
- Wybran
- Yagi
- Yamashita
- Yamashita
- Yoshida
- Yoshida
- Yu
- Yu
- Yu
- Yung
- Yung
- Yunis
- Yutoku
- Yutoku
- Yutoku
- Zaleski
- Zaleski
- Zembala
- Zembala
- Zembala
- Zier
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zinkernagel
- Zoschke
- Zvaifler
- Publication venue
- 'Elsevier BV'
- Publication date
- 01/01/1977
- Field of study