5 research outputs found
Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathway
- Author
- Akhlaq Mohammed
- Bloomfield Graham C
- Bruce Ian
- Budd Emma
- Cox Brian
- Cuenoud Bernard
- Finan Peter
- Gedeck Peter
- Hatto Julia
- Hayler Judy F
- Head Denise
- Keller Thomas
- Kirman Louise
- Le Grand Darren
- Leblanc Catherine
- McCarthy Clive
- O'Connor Desmond
- Owen Charles
- Oza Mrinalini S
- Pilgrim Gaynor
- Press Nicola E
- Sviridenko Lilya
- Whitehead Lewis
- Publication venue
- 'Elsevier BV'
- Publication date
- 01/09/2012
- Field of study
Using a parallel synthesis approach to target a non-conserved region of the PI3K catalytic domain a pan-PI3K inhibitor 1 was elaborated to provide alpha, delta and gamma isoform selective Class I PI3K inhibitors 21, 24, 26 and 27. The compounds had good cellular activity and were selective against protein kinases and other members of the PI3K superfamily including mTOR and DNA-PK
Synthesis and biological properties of novel glucocorticoid androstene C-17 furoate esters.
- Author
- Barker Lucy
- Beattie David
- Beer David
- Bentley David
- Bidlake Louise
- Butler Keith
- Craig Sarah
- Cuenoud Bernard
- Farr David Colin
- Ffoulkes-Jones Claire
- Fozard John R.
- Haberthuer Sandra
- Howes Colin
- Hynx Deborah
- Jeffers Sarah
- Keller Thomas
- Kirkham Paul
- Maas Janet
- Mazzoni Lazzaro
- Nicholls Andy
- Pilgrim Gaynor
- Sandham David
- Schaebulin Elisabeth
- Spooner Gillian M
- Stringer Rowan
- Tranter Pamela
- Turner Katharine
- Tweed Morris
- Walker Christoph
- Watson Simon
- Publication venue
- 'Elsevier BV'
- Publication date
- 01/01/2004
- Field of study
A series of novel corticosteroid derivatives featuring C-17 furoate ester functionality have been synthesised. Profiling in vitro and in vivo has resulted in the identification of a compound with a longer duration of action and a lower oral side effect profile in rodents compared to budesonide
Kinetics of the CH 2
- Author
- Astholz D. C.
- Atkinson R.
- Atkinson R.
- Barat R. B.
- Bernshtein V.
- Chao J.
- Chase M. W.
- Chen Y.
- Dobis O.
- Engels B.
- Frisch M. J.
- Gaynor B. J.
- Gilbert R. G.
- Gilbert R. G.
- Hoz T.
- Hoz T.
- Iyer S. R.
- Kaiser E. W.
- Kaiser E. W.
- Knyazev V. D.
- Knyazev V. D.
- Knyazev V. D.
- Lee F. S. C.
- Marcus R. A.
- Maricq M. M.
- Minton T. K.
- Pilgrim J. S.
- Rabinovitch B. S.
- Schlegel H. B.
- Schlegel H. B.
- Schlegel H. B.
- Seetula J. A.
- Sewell T. D.
- Sewell T. D.
- Slagle I. R.
- Slagle I. R.
- Stutz J.
- Tsang W.
- Tsang W.
- Wallington T. J.
- Wallington T. J.
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
Arson in Review: From Profit to Pathology
- Author
- Andreason
- Appelbaum
- Arlow
- Ashton
- Awad
- Bach-Y-Rita
- Baker
- Bartlett
- Blumberg
- Boling
- Bourget
- Bourget
- Bradford
- Bradford
- Brahams
- Bucknill
- Bumpass
- Bumpass
- Bumpass
- Byrne
- Carpenter
- Carroll
- Carstens
- Cohen
- Cole
- Cowen
- Dalton
- Dalton
- Day
- Day
- Denckla
- Denholtz
- Dunglison
- Eberle
- Eisler
- Eiwell
- Esquirol
- Everall
- Faulk
- Felthous
- Fineman
- Fleszar-Szumigajowa
- Foust
- Francis
- Freud
- Fry
- Fräs
- Gaynor
- Geller
- Geller
- Geller
- Geller
- Goodwin
- Greenberg
- Griesinger
- Gruber
- Gualtieri
- Gunderson
- Hall
- Hall
- Hall
- Hall
- Harmon
- Harris
- Hartshome
- Heath
- Heath
- Heilman
- Heller
- Herjanic
- Hill
- Hoffman
- Holland
- Hurley
- Inciardi
- Innes
- Jackson
- Jacobson
- Jacobson
- Jayaprakash
- Jeffrey L. Geller
- Jones
- Justice
- Kafry
- Kaler
- Kane
- Karter MJ
- Kazdin
- Koles
- Kolko
- Kolko
- Kolko
- Kolko
- Kolko
- Kolko
- Koson
- Kraepelin
- Kuhnley
- Köret
- Lande
- Levin
- Lewis
- Liberman
- Liberman
- Liberman
- Linnoila
- Linnoila
- Lowenstein
- Lowenstein
- Lukoff
- Macdonald
- Macdonald
- Madanes
- Marlatt
- Marshall
- Mavromatis
- McGrath
- McKerracher
- Meinhard
- Mercilliott
- Miller
- Minuchin
- Molnar
- Nielsen
- Nielsen
- Nielsen
- O’Connor
- O’Sullivan
- Pascoe
- Pilgrim
- Pisani
- Post
- Powers
- Prentky
- Prichard
- Prichard
- Prins
- Prins
- Prins
- Prins
- Quinsey
- Rabain
- Ray
- Rice
- Rice
- Rice
- Rider
- Ritvo
- Robbins
- Robbins
- Rodenhauser
- Roy
- Royer
- Schaefer
- Schaefer
- Scott
- Scott
- Showers
- Soothill
- Soothill
- Sorensen
- Stawar
- Steinbach
- Stekel
- Stewart
- Stoddard
- Strachan
- Taylor
- Taylor
- Tennent
- Tonkonogy
- Topp
- Trent
- Tuke
- Virkkunen
- Virkkunen
- Virkkunen
- Virkkunen
- Virkkunen
- Virkkunen
- Vogltance
- Vreeland
- Vreeland
- Waldrop
- Wax
- Webb
- Weiss
- Welsh
- Wiklund
- Wilson
- Wing
- Wooden
- Woolf
- Yassa
- Yesavage
- Zeegers
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Melanin: The organizing molecule
- Author
- Abbott
- Abraham
- Abramowitz
- Acher
- Acheson
- Adey
- Adey
- Adey
- Adey
- Adey
- Akil
- Albert
- Alder
- Alderson
- Altschule
- Altschule
- Amaral
- Andrew
- Andrew
- Andrews
- Aronin
- Autillo-Touati
- Babitch
- Bagnara
- Bagnara
- Bappy
- Barbeau
- Barker
- Bass
- Battersby
- Baweja
- Bazelon
- Becker
- Becker
- Becker
- Becker
- Beckwith
- Benkovic
- Bennett
- Bennett
- Berger
- Berger
- Berridge
- Berson
- Betterle
- Bettger
- Beynam
- Blackshaw
- Blank
- Bleehan
- Bloch
- Bloch
- Bloch
- Bloom
- Bogerts
- Bohm
- Bohm
- Borbely
- Borgens
- Bornens
- Botez
- Boudier
- Bower
- Bowers
- Braak
- Braak
- Bray
- Breathreach
- Brewer
- Brill
- Brooks
- Brown
- Brown
- Brown
- Brown
- Bruinvels
- Brunngraber
- Buck
- Bullock
- Bunney
- Bunney
- Burbach
- Burbach
- Burger
- Burnstock
- Bygrove
- Cahill
- Cameron
- Cammer
- Cardinali
- Cerrito
- Cheramy
- Chertow
- Cheung
- Chock
- Chretien
- Chvapil
- Cline
- Cohen
- Cooper
- Cooper
- Cope
- Cope
- Cope
- Cope
- Cope
- Cope
- Cornfield
- Cotman
- Coulombre
- Covey
- Crawford
- Crayton
- Creel
- Crippa
- Cross
- Crow
- Crutcher
- Cumming
- Cumming
- Curzon
- Czeisler
- D'Adamo
- D'Espagnant
- Dafny
- Daly
- Daniels
- Das
- Das
- Datta
- Davies
- Davies
- Davis
- Dawson
- De Brabander
- De Luca
- De Luca
- de Rotte
- De Wied
- De Wied
- De Wied
- De Wied
- DeBault
- Dedman
- Dennis
- Derby
- Dismukes
- Docherty
- Dolman
- Donaldson
- Drucker-Colin
- Dwyer
- Eccles
- Edelman
- Edelstein
- Eguchi
- Eipper
- Ekstrand
- Eppig
- Eranko
- Eskay
- Fauquet
- Fekete
- Felix
- Filatovs
- Filatovs
- Fillion
- Floyd
- Foley
- Folk
- Forno
- Forrest
- Fox
- Fujimori
- Fulton
- Gagnon
- Gagnon
- Gal
- Gallon
- Galzigna
- Gan
- Gan
- Garcia
- Gaynor
- Gerber
- German
- Gold
- Golde
- Golden
- Goldyne
- Goodal
- Goodman
- Gordon
- Gospodarowicz
- Goudie
- Gramsch
- Grant
- Gray
- Green
- Greene
- Greengard
- Greiner
- Greiner
- Griffiths
- Grossman
- Guille
- Gulza
- Guraya
- Gutnick
- Gutwein
- Gwynn
- Habener
- Hahn
- Haider
- Haken
- Hale
- Hamberger
- Hare
- Harsa-King
- Hasilek
- Hassell
- Hatotani
- Hawkins
- Hearing
- Hearing
- Hegedus
- Hegedus
- Heinz
- Heinz
- Helen
- Henkart
- Henkart
- Henn
- Henn
- Henn
- Heritage
- Hertz
- Hertz
- Hertzberg
- Hervonen
- Heym
- Higgens
- Hirata
- Hobson
- Hogino
- Holtzman
- Hooper
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Horrobin
- Huang
- Hui
- Hurley
- Hökfelt
- Hökfelt
- Iacovitti
- Ide
- Irwin
- Israel
- Jacobowitz
- Jacobs
- Jacobson
- Jaffee
- Jaffee
- Jaffee
- Jaffee
- Jantsch
- Jaques
- Jaques
- Jope
- Jouvet
- Kaliner
- Kanaseki
- Karson
- Kastin
- Kastin
- Kastin
- Katchalsky
- Kaufman
- Keller
- Kilbridge
- Kinnier
- Kirkpatrick
- Kirschner
- Kissel
- Klebanoff
- Kobayaski
- Korneeva
- Kosker
- Koszinowski
- Krebs
- Kress
- Kreutzberg
- Krieger
- Kripke
- Krynicki
- Krynicki
- Kuehl
- La Ferriere
- La Hoste
- Laborit
- Lackovie
- Lamey
- Landers
- Landis
- Lands
- Langer
- Larsson
- Larsson
- Lasek
- Lavie
- Le Douarin
- Le Douarin
- Le Roith
- Leconte
- LeDouarin
- LeDouarin
- Lee
- Lennarz
- Lerner
- Lerner
- Levitski
- Levitt
- Lewin
- Lewis
- Lidsky
- Liesi
- Lindquist
- Lindquist
- Lindquist
- Lodisk
- Loewenstein
- Lovenberg
- Lovenberg
- Luft
- Lund
- Lyttkens
- Maas
- Mackenzie
- MacVicar
- Maden
- Maden
- Mahadoo
- Maines
- Maker
- Manasek
- Mandel
- Mandell
- Mandell
- Mandell
- Mandell
- Manitto
- Mann
- Margolis
- Margullo
- Marks
- Marnett
- Maro
- Marsden
- Marsden
- Marsh
- Marx
- Marx
- Mason
- Massa
- Masters
- Matsuda
- Matthyse
- Maudsley
- McAuliffe
- McBurney
- McClain
- McCord
- McCormack
- McGaugh
- McGeer
- McGinness
- McGinness
- McGinness
- McGinness
- McGrath
- McGuire
- McNutt
- Means
- Meister
- Mendelson
- Menon
- Mertz
- Mescher
- Meyskens
- Michaelis
- Milby
- Mills
- Mittal
- Molokhia
- Moore
- Moore
- Morris
- Moskowitz
- Moyer
- Murad
- Mytilineou
- Nabel
- Naber
- Nagatsu
- Nagatsu
- Nasjletti
- Nathan
- Nelson
- Nenci
- Nes
- Neskovic
- Niall
- Nias
- Nichols
- Nicholson
- Nicholson
- Nicolis
- Nicolson
- Nockels
- Noden
- Nonhebel
- Norman
- Norris
- Nuccitelli
- Nuccitelli
- Nuccitelli
- O'Donahue
- O'Donahue
- O'Flaherty
- Oberley
- Oberley
- Obika
- Okun
- Okun
- Okun
- Okun
- Okun
- Okun
- Okun
- Olson
- Oomen
- Orci
- Ordonez
- Oski
- Oster
- Padawer
- Palmer
- Palombo
- Pannese
- Parker
- Parker
- Paston
- Patel
- Patterson
- Pavel
- Pawelek
- Pazo
- Pearse
- Pearse
- Pearse
- Pearse
- Pearse
- Pearse
- Pepplinkhuizen
- Peracchia
- Persad
- Persinger
- Peterson
- Peterson
- Pethig
- Pfeiffer
- Pfenniger
- Phillis
- Pierce
- Pietsch
- Pilgrim
- Pintar
- Pirozzolo
- Pober
- Pohjanpelto
- Popp
- Popper
- Por
- Porter
- Post
- Potts
- Potts
- Prasad
- Pribram
- Prigogine
- Proctor
- Proctor
- Prota
- Prusiner
- Pryor
- Psychoyos
- Quarterman
- Quastel
- Quesney-Huneeus
- Rabe
- Raese
- Rajan
- Raphan
- Rastogi
- Raynor
- Razin
- Regan
- Reid
- Reinherz
- Rennert
- Revel
- Ribeiro
- Rich
- Richardson
- Riedl
- Rifat
- Riley
- Riley
- Riordan
- Robinson
- Robinson
- Rodbard
- Rodbell
- Rodgers
- Roll
- Roney
- Rosenblum
- Rosenfeld
- Rosenthal
- Ross
- Roth
- Roth
- Roth
- Rothman
- Rotrosen
- Routtenberg
- Routtenberg
- Rowland
- Rusinov
- Sabesan
- Sadler
- Sagan
- Salazar
- Saper
- Sara
- Sarna
- Sarnat
- Sawchenko
- Schaeffer
- Scheibel
- Scheving
- Schlessinger
- Schliwa
- Schmitt
- Schmitt
- Schousboe
- Schubert
- Schultz
- Schulzberg
- Schwartz
- Schwartz
- Scott
- Sealy
- Segal
- Seije
- Seiler
- Seiler
- Seiler
- Seite
- Semm
- Seregi
- Shank
- Shank
- Shapavalov
- Shapiro
- Shapiro
- Shaw
- Shepherd
- Shimada
- Shimuzu
- Shindler
- Shine
- Shur
- Siegel
- Simon
- Sinet
- Singer
- Singhal
- Sissoeff
- Skolnick
- Skrabanek
- Skutsch
- Slavkin
- Sloper
- Smythies
- Smythies
- Snell
- Snyderman
- Sokol
- Solomon
- Solursk
- Somjen
- Somjen
- Somjen
- Somjen
- Spiegel
- Spirites
- Spirites
- Spoerri
- Spokes
- Spray
- Springer
- Stadtman
- Stein
- Steinfels
- Stengaard-Pederson
- Steriade
- Stern
- Stevens
- Stevens
- Stevens
- Stevens
- Stevens
- Stevens
- Stevens
- Stewart
- Stoclet
- Stocum
- Stoddart
- Stone
- Stone
- Stricker
- Subramanian
- Sunkara
- Suttie
- Swan
- Swanson
- Szent-Gyoergyi
- Taben
- Takahashi
- Tanford
- Tank
- Tapp
- Tartakoff
- Taugner
- Taylor
- Thathachari
- Thathachari
- Theoharides
- Thody
- Tizabi
- Tjalve
- Tolbert
- Tolbert
- Tomita
- Toran-Allerand
- Trams
- Trifaro
- Trulson
- Turin
- Turk
- Turner
- Turner
- Turner
- Turner
- Uemura
- Uemura
- Unanue
- Usdin
- Usdin
- Uvnas
- Uy
- Van Calker
- van Ree
- Van Ree
- Van Wimersma Greidanus
- Van Wimersma Greidanus
- van Woert
- Vander Wende
- Vander Wende
- Varela
- Varela
- Varon
- Verhoef
- Verhofstad
- Vernadakis
- Villars
- Villegas
- Vizi
- Volavka
- Volle
- von der Malsburg
- Waechter
- Walker
- Walters
- Walz
- Wang
- Warner
- Wasserman
- Wasserman
- Wasserman
- Watson
- Weatherbee
- Webster
- Webster
- Weiss
- Weitzman
- Wenk
- Werb
- Weston
- Whaley
- Wheeler
- Wheler
- Wiegant
- Williams
- Williams-Ashman
- Williams-Ashman
- Williford
- Winfree
- Winfree
- Witkop
- Witkop
- Witting
- Wojcik
- Wold
- Wolf
- Wolf
- Woods
- Yoshikawa
- Young
- Young
- Young
- Young
- Young
- Young
- Zametkin
- Zarcone
- Zatz
- Zeleny
- Zieglgansberger
- Zimmerman
- Zinn
- Zisapel
- Zwiller
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study