9 research outputs found
Esters of quinoxaline-7-carboxylate-1,4-di-N-oxide as Trichomonas vaginalis triosephosphate isomerase inhibitors
- Author
- Publication venue
- 'Walter de Gruyter GmbH'
- Publication date
- 01/01/2021
- Field of study
Trichomoniasis is a public health problem worldwide. Trichomoniasis treatment consists of the use of nitroimidazole derivatives; however, therapeutic ineffectiveness occurs in 5 to 20 % of the cases. Therefore, it is essential to propose new pharmacological agents against this disease. In this work, esters of quinoxaline-7-carboxylate-1,4-di-N-oxide (EQX-NO) were evaluated in in vitro assays as novel trichomonicidal agents. Additionally, an in vitro enzyme assay and molecular docking analysis against triosephosphate isomerase of Trichomonas vaginalis to confirm their mechanism of action were performed. Ethyl (compound 12) and n-propyl (compound 37) esters of quinoxaline-7-carboxylate-1,4-di-N-oxide derivatives showed trichomonicidal activity comparable to nitazoxanide, whereas five methyl (compounds 5, 15, 19, 20 and 22), four isopropyl (compounds 28, 29, 30 and 34), three ethyl (compound (4, 13 and 23) and one n-propyl (compound 35) ester derivatives displayed activity comparable to albendazole. Compounds 6 and 20 decreased 100 % of the enzyme activity of recombinant protein triosephosphate isomerase
Multi-messenger observations of a binary neutron star merger
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- Zong Z
- Zorn J
- Zornoza JD
- Zou CL
- Zuccarello F
- Zucker ME
- Zuniga J
- Zweizig J
- Zywucka N
- Publication venue
- 'American Astronomical Society'
- Publication date
- 01/01/2017
- Field of study
On 2017 August 17 a binary neutron star coalescence candidate (later designated GW170817) with merger time 12:41:04 UTC was observed through gravitational waves by the Advanced LIGO and Advanced Virgo detectors. The Fermi Gamma-ray Burst Monitor independently detected a gamma-ray burst (GRB 170817A) with a time delay of ~1.7 s with respect to the merger time. From the gravitational-wave signal, the source was initially localized to a sky region of 31 deg2 at a luminosity distance of 40+8-8 Mpc and with component masses consistent with neutron stars. The component masses were later measured to be in the range 0.86 to 2.26 Mo. An extensive observing campaign was launched across the electromagnetic spectrum leading to the discovery of a bright optical transient (SSS17a, now with the IAU identification of AT 2017gfo) in NGC 4993 (at ~40 Mpc) less than 11 hours after the merger by the One- Meter, Two Hemisphere (1M2H) team using the 1 m Swope Telescope. The optical transient was independently detected by multiple teams within an hour. Subsequent observations targeted the object and its environment. Early ultraviolet observations revealed a blue transient that faded within 48 hours. Optical and infrared observations showed a redward evolution over ~10 days. Following early non-detections, X-ray and radio emission were discovered at the transient’s position ~9 and ~16 days, respectively, after the merger. Both the X-ray and radio emission likely arise from a physical process that is distinct from the one that generates the UV/optical/near-infrared emission. No ultra-high-energy gamma-rays and no neutrino candidates consistent with the source were found in follow-up searches. These observations support the hypothesis that GW170817 was produced by the merger of two neutron stars in NGC4993 followed by a short gamma-ray burst (GRB 170817A) and a kilonova/macronova powered by the radioactive decay of r-process nuclei synthesized in the ejecta
Outcomes from elective colorectal cancer surgery during the SARS-CoV-2 pandemic
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- Uzunoglu F. G. (University Medical Center Hamburg–Eppendorf). Greece: Antonakis P.
- Vaccarella G. (Azienda Ospedaliera Ospedali Riuniti Villa Sofia-Cervello)
- Valbuena Jabares V. (Marqués de Valdecilla University Hospital)
- Valdes- Hernandez J. (Hospital Universitario Virgen Macarena)
- Valero Soriano M. (Hospital General Reina Sofía)
- Valle Rubio A. (Getafe University Hospital)
- Valverde S. (Hospital Clinic Barcelona)
- Van den Eynde J.
- Van den Eynde R. (Uz Leuven). Bulgaria: Sokolov M. (University Hospital Alexandrovska). Canada: Boutros M.
- Varma M. (University of California
- Vasljević J.
- Vassiliu P. (Attikon University General Hospital)
- Vaz Pereira R.
- Vaz S. (Centro Hospitalar e Universitário de São João)
- Velchuru V.
- Velickovic D. (Clinic for Digestive Surgery
- Velidedeoglu M.
- Venn M. (Royal London Hospital)
- Venskutonis D. (Lithuanian University of Health Sciences Kaunas Clinical Hospital). Madagascar: Rasoaherinomenjanahary F.
- Vera Mansilla C. (Hospital Universitario Principe de Asturias)
- Verberne C. (John Radcliffe Hospital)
- Vergari R. (Ospedali Riuniti di Ancona)
- Vernon L. (Cork University Hospital)
- Vervoort D.
- Vescio G. (University ‘Magna Graecia’ of Catanzaro)
- Vezakis A. (Aretaieion Hospital)
- Videira J. F. (IPO Porto). Réunion: Kassir R.
- Vieira B. (Centro Hospitalar de Trás-Os-Montes e Alto Douro
- Vieira Caroço T. (IPO Coimbra)
- Vieira Paiva Lopes A. C. (Hospital de Torres Vedras – Centro Hospitalar do Oeste)
- Vignali A. (San Raffaele Scientific Institute
- Vigorita V. (Álvaro Cunqueiro Hospital)
- Vijayan D. (Queen Elizabeth Hospital Birmingham)
- Villalabeitia Ateca I. (Hospital Universitario Cruces)
- Vimalachandran D. (Countess of Chester Hospital)
- Viswanath Y. K. S. (James Cook University Hospital)
- Vitali A. (Ospedale San Giovanni di Dio)
- Vitone L. (Royal Blackburn Hospital)
- Vives R. V. (Bellvitge University Hospital)
- Vo U. G. (Fiona Stanley Hospital)
- Von Papen M.
- Vovola F. (Ospedali Riuniti Azienda Ospedaliera Universitaria Foggia)
- Vucic N.
- Vázquez Fernández A. (Hospital Clínico Universitario de Valladolid)
- Wadham B. (The University Hospital of South Manchester)
- Walkes K. (Queen Elizabeth Hospital). Belgium: Flamey N.
- Wani R. (Sher-I-Kashmir Institute of Medical Sciences)
- Waqar S. H. (Pakistan Institute of Medical Sciences). Poland: Major P. (Jagiellonian University Medical College). Portugal: Azevedo C.
- Warren O. (Chelsea and Westminster Hospital)
- Watson L. J. (Sunderland Royal Hospital)
- Watson N. (King’s Mill Hospital)
- Weitz J.
- Welsch T. (Carl-Gustav-Carus University Hospital
- Werner J. (LMU Klinikum Campus Innenstadt)
- Westwood E. (James Paget University NHS Foundation Trust Hospital)
- Whelan M. (Tallaght University Hospital)
- Whitmore H. (Torbay and South Devon NHS Trust)
- Wilkin R. J. W. (South Warwickshire NHS Foundation Trust)
- Wilkins A. (Hull University Teaching Hospitals NHS Trust)
- Williams G. (Royal Gwent Hospital)
- Williams K. (St George’s Hospital)
- Wilson M. (Forth Valley Royal Hospital)
- Wimmer A. (Paracelsus Medical University Salzburg). Barbados: Barker D.
- Wong M.
- Worku D. (Queens Medical Centre)
- Wullschleger M. (Gold Coast University Hospital)
- Xavier R. G.
- Xenaki S.
- Xynos E. (University Hospital of Heraklion Crete and Interclinic Hospital of Crete). Hong Kong: Futaba K.
- Yang W.
- Yassin N. (Royal Wolverhampton NHS Trust)
- Ye G.
- Yesantharao P.
- Yetkin S. G. (Sisli Hamidiye Etfal Training and Research Hospital)
- Yeşilyurt D. (University of Health Sciences Tepecik Training and Research Hospital)
- Yiallourou A. (Nicosia General Hospital). Czechia: Martinek L.
- Yıldırım A.
- Yildiz A. (Yildirim Beyazit University Yenimahalle Training and Research Hospital). Uganda: Lule H.
- Young R. (York Teaching Hospitals NHS Trust)
- Yousof E. A. (Assiut University Hospital)
- Youssef M. (Norfolk and Norwich University Hospital)
- Yurttas C. (University Hospital Tuebingen)
- Yánez C. (Royo Villanova)
- Yüksel E. (Kocaeli University Teaching Hospital)
- Zafar S. N. (University of Wisconsin)
- Zakaria A. D.
- Zakaria Z. (School of Medical Sciences and Hospital
- Zambon M. (Policlinico Umberto I Sapienza University of Rome)
- Zanus G. (Ca’ Foncello Treviso – DISCOG – Università di Padova)
- Zegarac M. (Institute for Oncology and Radiology of Serbia)
- Zelić M. (University Hospital Center Rijeka)
- Zengin A. K. (Istanbul Universty – Cerrahpaşa Medical Faculty)
- Zerbib P. (CHU Lille)
- Zervas K.
- Zese M. (Santa Maria degli Angeli Hospital ULSS 5 – Adria)
- Zhang H. (Concord Repatriation General Hospital)
- Zizzo M. (Azienda Unità Sanitaria Locale – IRCCS di Reggio Emilia)
- Zografos C. (Laiko University Hospital)
- Zorrilla Ortúzar J. (Hospital General Universitario Gregorio Marañón)
- Zourntou S. (General Hospital of Larissa ‘Koutlimpaneio and Triantafylleio’)
- Zubaidi A. M. (King Saud University). Serbia: Aleksić L.
- Ângelo M.
- Çelebi F.
- Çolak E.
- Öfner D. (Medical University of Innsbruck)
- Öhlberger L.
- Özçelık M. F.
- Öğücü H.
- Überrück L.
- Ćoza I.
- Publication venue
- 'Wiley'
- Publication date
- 01/01/2020
- Field of study
This study aimed to describe the change in surgical practice and the impact of SARS-CoV-2 on mortality after surgical resection of colorectal cancer during the initial phases of the SARS-CoV-2 pandemic
In silico evaluation of phenothiazine derivatives as trypanothione reductase inhibitors
- Author
- Publication venue
- ScholarWorks @ UTRGV
- Publication date
- 28/09/2023
- Field of study
Background: American trypanosomiasis is caused by parasite Trypanosoma cruzi, and it is considered a worldwide health problem. Current treatment consists of benznidazole and nifurtimox, which are not fully effective against both disease stages and have adverse effects. There is thus a need to find parasite-specific alternative treatments. Search of specific inhibitors of parasite-exclusive crucial enzymes is a known strategy. Trypanothione reductase (TR) enzyme is central in parasite’s redox system both for detoxification of reactive oxygen and nitrogen species as well as amino acid and nucleotide biosynthesis. Phenothiazine scaffold is known by pharmacologists as a very versatile structure and its derivatives have shown TR inhibition. A virtual screening of phenothiazine derivatives from PubChem database may permit finding potential TR inhibitors.
Methodology: TR crystal was obtained from the PDB database (1GXF). A total of 100 phenothiazine derivatives complying with Lipinski’s rules were docked in TR active site using AutoDock Vina 1.1.2. Binding energy and interaction profiles, determined with PLIP (Protein-Ligand Interaction Profiler) server, were used to discriminate among derivatives.
Results: Binding energy was found to be in the range of -10.9 to -6.1 kcal/mol compared to -8.8 kcal/mol of natural ligand trypanothione disulfide (TS2). Forty-two compounds showed a binding energy greater than or equal to natural ligand, top ten were determined interactions. Main interactions were found with residues important to TS2 binding: Phe396, Leu399, His461, Glu466 and Glu467.
Conclusion: Best ranked compounds both by binding energy and interactions may be proposed as TR inhibitors and assayed in vitro to test effectivity
Esters of quinoxaline-7-carboxylate-1,4-di-N-oxide as Trichomonas vaginalis triosephosphate isomerase inhibitors
- Author
- Publication venue
- 'Walter de Gruyter GmbH'
- Publication date
- 01/09/2021
- Field of study
Trichomoniasis is a public health problem worldwide. Trichomoniasis treatment consists of the use of nitroimidazole derivatives; however, therapeutic ineffectiveness occurs in 5 to 20 % of the cases. Therefore, it is essential to propose new pharmacological agents against this disease. In this work, esters of quinoxaline-7-carboxylate-1,4-di-N-oxide (EQX-NO) were evaluated in in vitro assays as novel trichomonicidal agents. Additionally, an in vitro enzyme assay and molecular docking analysis against triosephosphate isomerase of Trichomonas vaginalis to confirm their mechanism of action were performed. Ethyl (compound 12) and n-propyl (compound 37) esters of quinoxaline-7-carboxy-late-1,4-di-N-oxide derivatives showed trichomonicidal activity comparable to nitazoxanide, whereas five methyl (compounds 5, 15, 19, 20 and 22), four isopropyl (compounds 28, 29, 30 and 34), three ethyl (compounds 4, 13 and 23) and one npropyl (compound 35) ester derivatives displayed activity comparable to albendazole. Compounds 6 and 20 decreased 100 % of the enzyme activity of recombinant protein triosephosphate isomerase
Triose Phosphate Isomerase Structure-Based Virtual Screening and In Vitro Biological Activity of Natural Products as <i>Leishmania mexicana</i> Inhibitors
- Author
- Publication venue
- MDPI AG
- Publication date
- 01/07/2023
- Field of study
Cutaneous leishmaniasis (CL) is a public health problem affecting more than 98 countries worldwide. No vaccine is available to prevent the disease, and available medical treatments cause serious side effects. Additionally, treatment failure and parasite resistance have made the development of new drugs against CL necessary. In this work, a virtual screening of natural products from the BIOFACQUIM and Selleckchem databases was performed using the method of molecular docking at the triosephosphate isomerase (TIM) enzyme interface of Leishmania mexicana (L. mexicana). Finally, the in vitro leishmanicidal activity of selected compounds against two strains of L. mexicana, their cytotoxicity, and selectivity index were determined. The top ten compounds were obtained based on the docking results. Four were selected for further in silico analysis. The ADME-Tox analysis of the selected compounds predicted favorable physicochemical and toxicological properties. Among these four compounds, S-8 (IC50 = 55 µM) demonstrated a two-fold higher activity against the promastigote of both L. mexicana strains than the reference drug glucantime (IC50 = 133 µM). This finding encourages the screening of natural products as new anti-leishmania agents
Genomewide Clonal Analysis of Lethal Mutations in the Drosophila melanogaster Eye: Comparison of the X Chromosome and Autosomes
- Author
- Abrams Anna
- Abramson Amanda
- Allen Christopher M.
- Alli Latifat
- Amado Latiffe
- An Ju
- Anderson Jenny
- Anwar Abbas
- Arevalo Sonia
- Ayoub Danny
- Badal Shawn S.
- Baghdanian Armonde
- Baghdanian Arthur H.
- Banerjee Utpal
- Bashour Keenan
- Baumann Sara A.
- Becerra Vivian N.
- Beyer Elsa
- Bibikova Elena
- Bookatz Allen
- Brewer Sarah
- Bui Chris
- Buu Natalie
- Call Gerald B.
- Calvillo Stephanie
- Cao Joseph
- Cespedes Albert
- Chan Amy
- Chan Cheryl
- Chan Hei J.
- Chan Jenny
- Chan Stacy
- Chang Aileen
- Chang Aileen E.
- Chang Daniel
- Chang Yuli
- Cheema Amrita K.
- Chen Jiong
- Chen YiBing
- Cheng Xibin A.
- Chhabra Akanksha
- Chin Mabel
- Chitsazzadeh Vida
- Choi Joo
- Chong Fleurette
- Chou Jeyling
- Cokus Shawn
- Crisostomo Carlyn
- Dang Peter
- Datta Sanjit
- Datta Sumit
- Davarifar Ardy
- Delosreyes Angela
- Deravanesian Artemis
- Desai Poonam
- Diep Francie
- Do Minh-Tu
- Ekanayake Preethika
- Engeln Mark
- Evers Elizabeth
- Fabrikant Jordan
- Fang Q. Angela
- Farnad Shahbaz
- Farshidi Farzin
- Fischer Katrina
- Folick Andrew
- Formanes Arlene J.
- Fu Katherine
- Garcia Eddie
- Garrone Nick
- Gasparyan Srpouhi
- Gayda Phyllis
- Go Sherrylene
- Goffstein Chad
- Gong Jun
- Gonzalez Courtney
- Goodstein Gelsey L.
- Guirguis Mariam
- Gupta Riju
- Haas Blake E.
- Hahm Vicky
- Hassid Ryan
- Hermogeno Brenda
- Hong Aria
- Hong Julie
- Hovestreydt Lindsay
- Hsieh Michael
- Hu Charles
- Huang Cheng R.
- Huff Devon
- Hui James Z.
- Hung Tony
- Iao Mei L.
- Jamshidian Farid
- Jen James
- Jin Sophia D.
- Kahen Katrin
- Kao Linda
- Kelley Melissa
- Kho Thomas
- Kim Angela Y.
- Kim Eunha
- Kim Lydia S-H.
- Kim Sarah
- Kim William
- Kim Yein
- Kim Yulee
- King Megan
- Kirkpatrick Brian
- Knudsen-Robbins Chloe
- Kohan Emil
- Kohanchi David
- Kovshilovskaya Bogdana
- Ku Amy
- Kung Raymond W.
- Kuoy Edward
- Kwak Robert
- Landig Mark E. L.
- Langenbacher Adam
- Latterman Stephanie S.
- Lauw Stephanie S.
- Laxamana Santino
- Lee Chris
- Lee Daniel S.
- Lee Eric
- Lee Janet
- Lee JiEun
- Lee Joann S.
- Lee So-Youn
- Lee ToHang S.
- Lee Toni
- Lei Kai C.
- Lerner Renata
- Leung Lesley L.
- Lewis Gemma
- Lezcano Sheila
- Lim Bryon C.
- Lin Henry
- Lin Jian-ya
- Lin Kathleen
- Lin Peter
- Liu H-C. Angela
- Liu Tiffany Q.
- Lui Crystal P. Y.
- Luong Vincent
- Luu Julie
- Luu Thanh
- Makshanoff Jacob
- Marrs Will
- Marsh Erin
- Marshall Jamie
- Mei An-Chi
- Meza Miguel
- Mikhaeil Yara A.
- Min Sarah
- Minasian Tanya
- Minye Helena
- Misra Amit
- Moarefi Majid
- Morimoto Miles
- Moroz Tatiana
- Moshfegh Yasaman
- Murray Jessica
- Ngo Kathy T.
- Nguyen Cynthia
- Nguyen Kha
- Nguyen Long H.
- Nodado Ernesto
- O'Donahue Amanda
- Olson John M.
- Onugha Ndidi
- Orjiakor Nneka
- Padhiar Bhavin
- Pai Shekhar S.
- Pandya Manish
- Patananan Alexander N.
- Patel Aadit R.
- Paul Eric
- Pavel-Dinu Mara
- Pavlenko Alex
- Paz Edwin
- Pellegrini Matteo
- Phaklides Sarah
- Pham Lephong
- Picard Paul D.
- Poulose Preethi
- Powell Russell
- Prasad Tharani
- Prashad Sacha L.
- Pusic Aya
- Ramola Divi
- Rangel Alma
- Regalia Kirsten
- Ribbens Meghann
- Rifai Bassel
- Rosselli Desiree
- Saakyan Manyak
- Saarikoski Pamela
- Safaee Michael M.
- Salame Carol
- Sanchez Christian
- Sanchez Nina
- Segura Miriam
- Seifert Christina C.
- Shadpour Farnaz
- Shah Abhishek
- Shemmassian Aram
- Shilgevorkyan Oganes H.
- Sidhu Sohrab
- Singh Inderroop
- Singh Ramnik
- Singh Vivek
- Sitz Daniel
- Skinner Emily
- Solomin Daniel
- Soma Vanessa
- Soneji Kosha
- Song Junia J.
- Spivey Kristin
- Srivastava Neetika
- Sta.Ana Jennifer L.
- Stageberg Erika
- Stavchanskiy Marina
- Sun Christie
- Taber Chelsea E.
- Tan Diane
- Tan Jingwen
- Tekchandani Leena
- Teruya Alison S.
- Thai Leo
- Thiyanaratnam Jayantha
- Tikia Robyn
- Tong Maurine
- Toor Aneet
- Topp Kasey
- Tovar Steve
- Tran PhuongThao
- Tran Quynh-Minh
- Tran Trinh
- Trangsrud Kelly
- Travis Emily G.
- Trinh Jennifer D.
- Tsang Wah-Yung
- Uemura Marc
- Unkovic Mary
- Villarasa Nikki
- Vo Diane
- Vollmer Emily
- Walsh Thomas
- Weiss Emily
- Wells Maggie
- Wickland Jessica
- Wong Regan S.
- Wood Damien
- Wu Joy
- Wu Katherine
- Wu Sophia
- Wu Winston
- Wu Ya-Whey
- Xu Qing
- Yabroff Allison M.
- Yackle Kevin
- Yamauchi Yuki
- Yang Nkau X. V.
- Yarosh Will
- Yavari Amir
- Yee Laura
- Yen George
- Yeranosian Michael
- Yu James S.
- Zaretsky Jesse M.
- Zhou Jennifer J.
- Zhu Ran X.
- Publication venue
- Copyright © 2007 by the Genetics Society of America
- Publication date
- Field of study
Using a large consortium of undergraduate students in an organized program at the University of California, Los Angeles (UCLA), we have undertaken a functional genomic screen in the Drosophila eye. In addition to the educational value of discovery-based learning, this article presents the first comprehensive genomewide analysis of essential genes involved in eye development. The data reveal the surprising result that the X chromosome has almost twice the frequency of essential genes involved in eye development as that found on the autosomes
Correction to: Comparative effectiveness and safety of non-vitamin K antagonists for atrial fibrillation in clinical practice: GLORIA-AF Registry
- Author
- Abban Dzifa Wosornu
- Abdul Nasser
- Abud Atilio Marcelo
- Adams Fran
- Addala Srinivas
- Adragão Pedro
- Ageno Walter
- Aggarwal Rajesh
- Agosti Sergio
- Agostoni Piergiuseppe
- Aguilar Francisco
- Aguinaga Luis
- Ahmed Jameel
- Aiello Allessandro
- Ainsworth Paul
- Aiub Jorge Roberto
- Al-Dallow Raed
- Alderson Lisa
- Alexopoulos Dimitrios
- Aliyar Pareed
- Almeida Luísa Fonseca
- Alonso David
- Alvaro Feliz
- Amado José
- Amara Walid
- Amelot Mathieu
- Amjadi Nima
- Ammirati Fabrizio
- Andrade Marianna
- Andrawis Nabil
- Annoni Giorgio
- Ansalone Gerardo
- Ariani M. Kevin
- Arias Juan Carlos
- Armero Sébastien
- Arora Chander
- Asensi Joaquín Osca
- Aslam Muhammad Shakil
- Asselman M.
- Audouin Philippe
- Augenbraun Charles
- Ayala Carlos Antero Chavez
- Aydin S.
- Ayryanova Ivaneta
- Aziz Emad
- Backes Luciano Marcelo
- Badings E.
- Bagni Ermentina
- Baker Seth
- Bala Richard
- Baldi Antonio
- Bando Shigenobu
- Banerjee Subhash
- Bank Alan
- Barr Craig
- Bartlett Maria
- Basic Kes Vanja
- Baula Giovanni
- Behrens Steffen
- Bell Alan
- Benedetti Raffaella
- Benhalima Bouziane
- Berg J.
- Bergler-Klein Jutta
- Berneau Jean-Baptiste
- Bernstein Richard
- Berrospi Percy
- Berti Sergio
- Berz Andrea
- Best Elizabeth
- Bettencourt Paulo
- Betzu Robert
- Bhagwat Ravi
- Bhatta Luna
- Biscione Francesco
- Bisignani Giovanni
- Black Toby
- Bloch Michael
- Bloom Stephen
- Blumberg Edwin
- Bo Mario
- Bodes Rafael Salguero
- Bollmann Andreas
- Bongiorni Maria Grazia
- Boriani Giuseppe
- Boswijk D.
- Bott Jochen
- Bottacchi Edo
- Bradman Drew
- Brautigam Donald
- Breton Nicolas
- Briones Ignacio Rodriguez
- Brkljacic Diana Delic
- Brouwers P.
- Browne Kevin
- Bruni A.
- Brunschwig Claude
- Buathier Hervé
- Buenostro Gabriel Contreras
- Buhl Aurélie
- Bullinga John
- Bøhmer Ellen
- Cabrera Jose Walter
- Caccavo Alberto
- Cai Shanglang
- Caine Sarah
- Calvi Valeria
- Calò Leonardo
- Campos Rodrigo Noronha
- Candeias Rui
- Capuano Vincenzo
- Capucci Alessandro
- Caputo Ronald
- Cardona Francisco
- Carolei Antonio
- Carreño Susana
- Carvalho Paula
- Cary Susanna
- Casu Gavino
- Cavallini Claudio
- Cayla Guillaume
- Celentano Aldo
- Cha Kwang Soo
- Cha Tae-Joon
- Chae Jei Keon
- Chalamidas Kathrine
- Challappa Krishnan
- Chand Sunil Prakash
- Chandrashekar Harinath
- Chartier Ludovic
- Chatterjee Kausik
- Cheema Aamir
- Cheema Amjad
- Chen Jyh Hong
- Chen Lin
- Chen Shih-Ann
- Chiang Fu-Tien
- Chiarella Francesco
- Chih-Chan Lin
- Cho Yong Keun
- Choi Dong Ju
- Choi Jong-Il
- Chouinard Guy
- Chow Danny Hoi-Fan
- Chreih Rami Mihail
- Chrysos Dimitrios
- Chumakova Galina
- Cislowski David
- Clay Anthony
- Clifford Piers
- Cohen Andrew
- Cohen Michael
- Cohen Serge
- Colivicchi Furio
- Collins Ronan
- Colonna Paolo
- Compton Steve
- Connolly Derek
- Conti Alberto
- Coodley Gregg
- Cooper Martin
- Coronel Julian
- Corso Giovanni
- Cortada Jordi Bruguera
- Cottin Yves
- Covalesky John
- Cracan Aurel
- Crea Filippo
- Crean Peter
- Crenshaw James
- Cullen Tina
- da Costa Darrieux Francisco Carlos
- da Costa Fernando Augusto Alves
- Dahl Jürgen Vom
- Darius Harald
- Dary Patrick
- Dascotte Olivier
- Dauber Ira
- Davalos Vicente
- Davies Ruth
- Davis Gershan
- Davy Jean-Marc
- Dayer Mark
- de Biasio Marzia
- de Bonis Silvana
- de Caterina Raffaele
- de Franceschi Teresiano
- de Groot J.
- de Horta José
- de La Briolle Axel
- de La Pena Topete Gilberto
- de Los Rios Ibarra Manuel Odin
- de Paola Angelo Amato Vicenzo
- de Souza Olga Ferreira
- de Souza Weimar
- de Veer A.
- de Wolf Luc
- Decoulx Eric
- Deepak Sasalu
- Defaye Pascal
- del Río Jorge Eduardo Hernández
- Deumite N. Joseph
- Di Legge Silvia
- Diemberger Igor
- Diener Hans-Christoph
- Dietz Denise
- Dionísio Pedro
- Dong Qiang
- dos Santos Fabio Rossi
- Dotcheva Elena
- Doukky Rami
- Dubner Sergio
- Dubrey Simon
- Ducrocq Xavier
- Dupljakov Dmitry
- Duque Mauricio
- Dutta Dipankar
- Duvilla Nathalie
- Duygun A.
- Dziewas Rainer
- D’souza Anthony
- Eaton Charles
- Eaves William
- Ebels-Tuinbeek L.
- Ehrlich Clifford
- Eichinger-Hasenauer Sabine
- Eisenberg Steven
- Escudero Aldo Edwin Rodriguez
- Esperon Guillermo Llamas
- Esquivias Gonzalo Barón
- Evonich Rudolph
- Evseeva Oksana
- Ezhov Andrey
- Fahmy Raed
- Fang Quan
- Farsad Ramin
- Fauchier Laurent
- Favale Stefano
- Fayard Maxime
- Fedele Francesco
- Fedele Jose Luis
- Fedorishina Olga
- Fera Steven
- Fernández Marcelo Sanmartín
- Ferreira Jorge
- Ferreira Luis Gustavo Gomes
- Ferri Claudio
- Ferrier Anna
- Ferro Hugo
- Filho Adalberto Menezes Lorga
- Filho Dario Sobral
- Finsen Alexandra
- First Brian
- Fischer Stuart
- Fonseca Catarina
- Forman Steven
- Fragoso Juan Carlos Nunez
- Frandsen Brad
- French William
- Friedman Keith
- Friese Athena
- Fruntelata Ana Gabriela
- Fujii Shigeru
- Fumagalli Stefano
- Fundamenski Marta
- Furukawa Yutaka
- Gabelmann Matthias
- Gabra Nashwa
- Gadsbøll Niels
- Galinier Michel
- Gammelgaard Anders
- Ganeshkumar Priya
- Gans Christopher
- Garcéa Jose Polo
- Gartenlaub Olivier
- Gaspardone Achille
- Genz Conrad
- Georger Frédéric
- Georges Jean-Louis
- Georgeson Steven
- Giedrimas Evaldas
- Gierba Mariusz
- Gillespie Eve
- Giniger Alberto
- Giudici Michael
- Gkotsis Alexandros
- Glotzer Taya
- Gmehling Joachim
- Gniot Jacek
- Goethals Peter
- Goldbarg Seth
- Goldberg Ronald
- Goldmann Britta
- Golitsyn Sergey
- Gonzalez Vicente Bertomeu
- González Salvador León
- Gorka Hervé
- Gornick Charles
- Gorog Diana
- Gottipaty Venkat
- Goube Pascal
- Goudevenos Ioannis
- Grado Carlos Antonio Raffo
- Graham Brett
- Greer G. Stephen
- Gremmler Uwe
- Grena Paul
- Grond Martin
- Gronda Edoardo
- Grönefeld Gerian
- Gu Xiang
- Guardigli Gabriele
- Guevara Carolina
- Guignier Alexandre
- Gulizia Michele
- Gumbley Michael
- Gurusamy Venkatesh Kumar
- Gómez Silvia
- Günther Albrecht
- Ha Andrew
- Hahalis Georgios
- Hakas Joseph
- Hall Christian
- Halperin Jonathan
- Han Bing
- Han Seongwook
- Hargrove Joe
- Hargroves David
- Haruna Tetsuya
- Hayek Emil
- Healey Jeff
- Hearne Steven
- Heffernan Michael
- Heggelund Geir
- Heijmeriks J.
- Hemels Maarten
- Hendriks I.
- Henein Sam
- Her Sung-Ho
- Hermany Paul
- Hermosillo Jesus Antonio Gonzalez
- Hernandes Mauro Esteves
- Hernandez Norberto Matadamas
- Higashino Yorihiko
- Hill Michael
- Hisadome Tetsuo
- Hishida Eiji
- Hoffer Etienne
- Hoghton Matthew
- Hong Kui
- Hong Suk Keun
- Horbach Stevie
- Horiuchi Masataka
- Hou Yinglong
- Hsing Jeff
- Huang Chi-Hung
- Huckins David
- Hughes Kathy
- Huisman Menno
- Huizinga A.
- Hulsman E.
- Hung Kuo-Chun
- Hurtado Helard Andres Manrique
- Hwang Gyo-Seung
- Ikpoh Margaret
- Imberti Davide
- Ince Hüseyin
- Indolfi Ciro
- Inoue Shujiro
- Irles Didier
- Iseki Harukazu
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- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/05/2022
- Field of study
International audienceIn this article, the name of the GLORIA-AF investigator Anastasios Kollias was given incorrectly as Athanasios Kollias in the Acknowledgements. The original article has been corrected
Patterns of oral anticoagulant use and outcomes in Asian patients with atrial fibrillation: a post-hoc analysis from the GLORIA-AF Registry
- Author
- Abban Dzifa Wosornu
- Abdul Nasser
- Abud Atilio Marcelo
- Adams Fran
- Addala Srinivas
- Adragão Pedro
- Ageno Walter
- Aggarwal Rajesh
- Agosti Sergio
- Agostoni Piergiuseppe
- Aguilar Francisco
- Aguinaga Luis
- Ahmed Jameel
- Aiello Allessandro
- Ainsworth Paul
- Aiub Jorge Roberto
- Al-Dallow Raed
- Alderson Lisa
- Aldrete Velasco Jorge Antonio
- Alexopoulos Dimitrios
- Aliyar Pareed
- Almeida Luísa Fonseca
- Alonso David
- Alves da Costa Fernando Augusto
- Amado José
- Amara Walid
- Amelot Mathieu
- Amjadi Nima
- Ammirati Fabrizio
- Andrade Marianna
- Andrawis Nabil
- Angela Koh Su Mei
- Annoni Giorgio
- Ansalone Gerardo
- Ariani M Kevin
- Arias Juan Carlos
- Armero Sébastien
- Arora Chander
- Asensi Joaquín Osca
- Aslam Muhammad Shakil
- Asselman M
- Audouin Philippe
- Augenbraun Charles
- Aydin S
- Ayryanova Ivaneta
- Aziz Emad
- Backes Luciano Marcelo
- Badings E
- Bagni Ermentina
- Baker Seth H
- Bala Richard
- Baldi Antonio
- Bando Shigenobu
- Banerjee Subhash
- Bank Alan
- Barr Craig
- Bartlett Maria
- Baula Giovanni
- Behrens Steffen
- Bell Alan
- Benedetti Raffaella
- Benhalima Bouziane
- Berg JM ten
- Bergler-Klein Jutta
- Berneau Jean-Baptiste
- Bernstein Richard A
- Berrospi Percy
- Berti Sergio
- Berz Andrea
- Best Elizabeth
- Bettencourt Paulo
- Betzu Robert
- Bhagwat Ravi
- Bhatta Luna
- Biscione Francesco
- Bisignani Giovanni
- Bisson Arnaud
- Black Toby
- Bloch Michael J
- Bloom Stephen
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- Bo Mario
- Bodes Rafael Salguero
- Bollmann Andreas
- Bongiorni Maria Grazia
- Boriani Giuseppe
- Boriani Giuseppe
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- Jarmukli Nabil
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- Jenkins Ronald D
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- Jobe Robert
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- Keeling P
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- Kmetzo James J
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- Koschutnik Martin
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- Lorraine Richard S
- Luengas Carlos Alberto
- Luke Robert
- Luo Ming
- Lupovitch Steven
- Lyrer Philippe
- López Amador
- López-Sendón José Luís
- Ma Changsheng
- Ma Genshan
- Madariaga Irene
- Maeno Koji
- Magnin Dominique
- Maid Gustavo
- Mainigi Sumeet K
- Makaritsis Konstantinos
- Malhotra Rohit
- Manning Rickey
- Manolis Athanasios
- Manrique Hurtado Helard Andres
- Mantas Ioannis
- Manterola Fernando Alfonso
- Maqueda Vicky
- Marchionni Niccolo
- Martinez Jorge
- Maskova Petra
- Matsuda Katsuhiro
- Maurer Tillmann
- Mauro Ciro
- May Erik
- Mayer Nolan
- Mazuecos Juan Benezet
- McClure John
- McCormack Terry
- McGarity William
- McIntyre Hugh
- McLaurin Brent
- Medina Palomino Feliz Alvaro
- Mei Davide Antonio
- Melandri Francesco
- Meno Hiroshi
- Menzies Dhananjai
- Mercader Marco
- Mesa Juan Gomez
- Meyer Beat J
- Meyer Christian
- Miarka Jacek
- Mibach Frank
- Michalski Dominik
- Michel Patrik
- Miguel Ricardo Nicolás
- Mikdadi Ghiath
- Mikus Milan
- Milicic Davor
- Militaru Constantin
- Minaie Sedi
- Minescu Bogdan
- Mintale Iveta
- Mirault Tristan
- Mirro Michael J
- Mistry Dinesh
- Miu Nicoleta Violeta
- Miyamoto Naomasa
- Miño
- Moccetti Tiziano
- Mohammed Akber
- Mollerus Michael
- Molon Giulio
- Mondillo Sergio
- Moniz Patrícia
- Mont Lluis
- Montagud Vicente
- Montaña Oscar
- Monti Cristina
- Moretti Luciano
- Mori Kiyoo
- Moriarty Andrew
- Morka Jacek
- Moschini Luigi
- Moschos Nikitas
- Moura Jorge Jose Carlos
- Mulhearn Thomas J
- Muresan Carmen
- Muriago Michela
- Musial Wlodzimierz
- Musser Carl W
- Musumeci Francesco
- Mügge Andreas
- Nageh Thuraia
- Nakagawa Hidemitsu
- Nakamura Yuichiro
- Nakayama Toru
- Nam Gi-Byoung
- Nanna Michele
- Natarajan Indira
- Navarro Nassip Llerena
- Nayak Hemal M
- Naydenov Stefan
- Nazlić Jurica
- Nechvatal Libor
- Negron Sandra Adela
- Neiman James
- Neuenschwander Fernando Carvalho
- Neves David
- Neykova Anna
- Nica Nicoleta Cindea
- Nijmeh George
- Nizov Alexey
- Nor Azlisham Mohd
- Nossan Janko
- Novikova Tatiana
- Nowalany-Kozielska Ewa
- Nsah Emmanuel
- Nunez Fragoso Juan Carlos
- Nurgalieva Svetlana
- Nuyens Dieter
- Nyvad Ole
- O'Donnell Martin
- O'Donnell Philip
- O'Hara Gilles
- Odin de Los Rios Ibarra Manuel
- Oh Dongjin
- Oh Seil
- Oh Yong Seog
- Oi Yan Yannie Soo
- Oikonomou Kostas
- Olivares Claudia
- Oliver Richard
- Olshansky Brian
- Olympios Christoforos
- omaszuk-Kazberuk Anna
- Ortega Ignacio Gil
- Ortuno Francisco Marin
- Padilla Padilla Francisco Gerardo
- Pajes Giuseppe
- Pandey Shekhar
- Paparella Gaetano
- Paris F
- Park Hyung Wook
- Park Jong Sung
- Parthenakis Fragkiskos
- Pascual Carlos Rodríguez
- Passamonti Enrico
- Patel Jaydutt
- Patel Mehool
- Patel Rajesh J
- Patrick Janice
- Paz Analía
- Pengo Vittorio
- Pentz William
- Perlman Richard
- Persic Viktor
- Perticone Francesco
- Peters Terri K
- Petkar Sanjiv
- Pezo Luis Felipe
- Pflücke Christian
- Pham David N
- Phillips Roland T
- Phlaum Stephen
- Pieters Denis
- Pineau Julien
- Pinter Arnold
- Pinto Fausto
- Pisters R
- Pivac Nediljko
- Pocanic Darko
- Podoleanu Cristian
- Politano Alessandro
- Poljakovic Zdravka
- Pollock Stewart
- Poppert Holger
- Porcu Maurizio
- Prasad Neeraj
- Prelle Alessandro
- Prodafikas John
- Proietti Marco
- Protasov Konstantin
- Précoma Dalton Bertolim
- Pye Maurice
- Pérez Ríos Alma Minerva
- Pérez Beatriz
- Pérez-Cabezas Alejandro
- Qiu Zhaohui
- Quedillac Jean-Michel
- Quintana Antonio Garcia
- Raev Dimitar
- Raffo Grado Carlos Antonio
- Rahimi Sidiqullah
- Raisaro Arturo
- Rama Bhola
- Ramos Ricardo
- Ranieri Maria
- Raposo Nuno
- Rashba Eric
- Rauch-Kroehnert Ursula
- Reddy Ramakota
- Reino Antonio Pose
- Renda Giulia
- Reza Shabbir
- Ria Luigi
- Richter Dimitrios
- Rickli Hans
- Rieker Werner
- Rios Victoria Padilla
- Ritt Luiz Eduardo
- Rizo Tatiana Cárdenas
- Roberts Douglas
- Rodriguez Escudero Aldo Edwin
- Roman Mark
- Romeo Francesco
- Romiti Giulio Francesco
- Ronner E
- Rossi dos Santos Fabio
- Roux Jean-Francois
- Rozkova Nadezda
- Rubacek Miroslav
- Rubalcava Frank
- Ruiz Rafael Olvera
- Russo Andrea M
- Rutgers Matthieu Pierre
- Rybak Karin
- Said Samir
- Sakamoto Tamotsu
- Salacata Abraham
- Salem Adrien
- Sales Juan Cosín
- Saltzman Marco A
- Salvioni Alessandro
- Santana Antonio Martín
- Saporito Wladmir Faustino
- Sarikonda Kesari
- Sasaoka Taishi
- Sati Hamdi
- Savelieva Irina
- Scala Pierre-Jean
- Schellinger Peter
- Scherr Carlos
- Schmitz Bettina
- Schmitz Karl-Heinz
- Schmitz Lisa
- Schnabel Teresa
- Schnupp Steffen
- Schoeniger Peter
- Schwimmbeck Peter
- Schön Norbert
- Seamark Clare
- Searles Greg
- Seidl Karl-Heinz
- Seidman Barry
- Sek Jaroslaw
- Sekaran Lakshmanan
- Serrati Carlo
- Shah Anil
- Shah Neerav
- Shah Shujahat
- Shah Vinay
- Sharma Vijay Kumar
- Shaw Louise
- Sheikh Khalid H
- Shimizu Naruhito
- Shimomura Hideki
- Shin Dong-Gu
- Shin Eun-Seok
- Shite Junya
- Sibilio Gerolamo
- Silver Frank
- Sime Iveta
- Simmers Tim A
- Singh Takhar Amrit Pal
- Singh Narendra
- Siostrzonek Peter
- Smadja Didier
- Smith David W
- Snitman Marcelo
- Soda Hassan
- Sofley Carl
- Sokal Adam
- Sotolongo Rodolfo
- Sparby Jon Arne
- Spinar Jindrich
- Sprigings David
- Spyropoulos Alex C
- Stakos Dimitrios
- Steinwender Clemens
- Stergiou Georgios
- Stiell Ian
- Stoddard Marcus
- Stoikov Anastas
- Streb Witold
- Styliadis Ioannis
- Su Guohai
- Su Xi
- Sudnik Wanda
- Sukles Kai
- Sun Xiaofei
- Swart H
- Szavits-Nossan Janko
- Sánchez Carlos Jerjes
- Sánchez Mauricio Camarillo
- Taggeselle Jens
- Takagi Yuichiro
- Tamm Angelika
- Tanaka Katsumi
- Tanawuttiwat Tanyanan
- Tang Aylmer
- Tang Sherman
- Tarsi Giovanni
- Tassinari Tiziana
- Tayal Ashis
- Tayebjee Muzahir
- Tesloianu Dan
- The Salem HK
- Thomas Dierk
- Timsit Serge
- Tobaru Tetsuya
- Tomasik Andrzej R
- Topete Gilberto de la Pena
- Torosoff Mikhail
- Torres Torres Ivett Guadalupe
- Touze Emmanuel
- Trendafilova Elina
- Tsai W Kevin
- Tse Hung Fat
- Tsutsui Hiroshi
- Tu Tian Ming
- Tuininga Ype
- Turakhia Minang
- Turk Samir
- Turner Wayne
- Tveit Arnljot
- Tytus Richard
- Valadão C
- Valenzuela Chuquiure
- Vallejo Gregorio Sanchez
- van Bergen PFMM
- van de Borne Philippe
- van den Berg BJ
- van der Zwaan C
- Van Eck M
- Vanacker Peter
- Vasilev Dimo
- Vasilikos Vasileios
- Vasilyev Maxim
- Veerareddy Srikar
- Vera Tomas Ripolil
- Verdecchia Paolo
- Versaci Francesco
- Vester Ernst Günter
- Vial Hubert
- Vicenzo de Paola Angelo Amato
- Victory Jason
- Villamil Alejandro
- Vincent Marc
- Vlastaris Anthony
- Vora Kishor
- Vranian Robert B
- Wakefield Paul
- Wang Feng
- Wang Mingsheng
- Wang Ningfu
- Wang Tian
- Wang Xinhua
- Warner Alberta L
- Watanabe Kouki
- Wei Jeanne
- Weimar Christian
- Weiner Stanislav
- Weinrich Renate
- Wen Ming-Shien
- Wiemer Marcus
- Wiggers Preben
- Wilke Andreas
- Williams David
- Williams Marcus L
- Witzenbichler Bernhard
- Wong Brian
- Wozakowska-Kaplon Beata
- Wu Richard C
- Wu Shulin
- Wunderlich Silke
- Wyatt Nell
- Wylie John Jack
- Xu Xiangdong
- Xu Yong
- Yamanoue Hiroki
- Yamashita Takeshi
- Yang Tianlun
- Yao Jing
- Yeh Kuo-Ho
- Yin Wei Hsian
- Yotov Yoto
- Zahn Ralf
- Zanetti Fernando Lanas
- Zarich Stuart
- Zenin Sergei
- Zeuthen Elisabeth Louise
- Zhang Donghui
- Zhang Huanyi
- Zhang Jun
- Zhang Ping
- Zhang Xingwei
- Zhao Shui Ping
- Zhao Yujie
- Zhao Zhichen
- Zheng Yang
- Zhou Jing
- Zimmermann Sergio
- Zini Andrea
- Zizzo Steven
- Zong Wenxia
- Zukerman L Steven
- Publication venue
- Elsevier BV
- Publication date
- 01/01/2023
- Field of study
Background: Previous studies suggested potential ethnic differences in the management and outcomes of atrial fibrillation (AF). We aim to analyse oral anticoagulant (OAC) prescription, discontinuation, and risk of adverse outcomes in Asian patients with AF, using data from a global prospective cohort study. Methods: From the GLORIA-AF Registry Phase II-III (November 2011-December 2014 for Phase II, and January 2014-December 2016 for Phase III), we analysed patients according to their self-reported ethnicity (Asian vs. non-Asian), as well as according to Asian subgroups (Chinese, Japanese, Korean and other Asian). Logistic regression was used to analyse OAC prescription, while the risk of OAC discontinuation and adverse outcomes were analysed through Cox-regression model. Our primary outcome was the composite of all-cause death and major adverse cardiovascular events (MACE). The original studies were registered with ClinicalTrials.gov, NCT01468701, NCT01671007, and NCT01937377. Findings: 34,421 patients were included (70.0 ± 10.5 years, 45.1% females, 6900 (20.0%) Asian: 3829 (55.5%) Chinese, 814 (11.8%) Japanese, 1964 (28.5%) Korean and 293 (4.2%) other Asian). Most of the Asian patients were recruited in Asia (n = 6701, 97.1%), while non-Asian patients were mainly recruited in Europe (n = 15,449, 56.1%) and North America (n = 8378, 30.4%). Compared to non-Asian individuals, prescription of OAC and non-vitamin K antagonist oral anticoagulant (NOAC) was lower in Asian patients (Odds Ratio [OR] and 95% Confidence Intervals (CI): 0.23 [0.22-0.25] and 0.66 [0.61-0.71], respectively), but higher in the Japanese subgroup. Asian ethnicity was also associated with higher risk of OAC discontinuation (Hazard Ratio [HR] and [95% CI]: 1.79 [1.67-1.92]), and lower risk of the primary composite outcome (HR [95% CI]: 0.86 [0.76-0.96]). Among the exploratory secondary outcomes, Asian ethnicity was associated with higher risks of thromboembolism and intracranial haemorrhage, and lower risk of major bleeding. Interpretation: Our results showed that Asian patients with AF showed suboptimal thromboembolic risk management and a specific risk profile of adverse outcomes; these differences may also reflect differences in country-specific factors. Ensuring integrated and appropriate treatment of these patients is crucial to improve their prognosis. Funding: The GLORIA-AF Registry was funded by Boehringer Ingelheim GmbH