13 research outputs found
PARP14 promotes the warburg effect in hepatocellular carcinoma by inhibiting JNK1-dependent PKM2 phosphorylation and activation
- Author
- A Barbarulo
- AE Vaughn
- AJ Levine
- B Chaneton
- C Bubici
- CC Wong
- CV Dang
- D Anastasiou
- D Anastasiou
- D Beyoğlu
- D Beyoğlu
- DY Gui
- E Kakazu
- E Wurmbach
- GK Abou-Alfa
- H Ke
- H Mohammed
- H Shim
- HJ Huber
- HR Christofk
- HR Christofk
- JL Andersen
- JS Boehm
- K Bensaad
- K Herzer
- K Kitamura
- K Wang
- L Lv
- L Lv
- M Cortés-Cros
- M Hatziapostolou
- M Wiznerowicz
- MG Vander Heiden
- NM Grüning
- NN Danial
- P Chinnaiyan
- P Mehrotra
- Q Geissmann
- R Koschny
- R Ma
- R Yang
- RA Cairns
- RA Gatenby
- RG Jones
- S Papa
- SH Cho
- SH Cho
- SK McBrayer
- SM Jang
- SY Peng
- T Amann
- T Hitosugi
- T Hitosugi
- T Yamashita
- T Yanagawa
- TH Nguyen
- V Schreiber
- W Luo
- W Yang
- WJ Israelsen
- Y Hoshida
- Z Chen
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 23/06/2015
- Field of study
Most tumour cells use aerobic glycolysis (the Warburg effect) to support anabolic growth and evade apoptosis. Intriguingly, the molecular mechanisms that link the Warburg effect with the suppression of apoptosis are not well understood. In this study, using loss-of-function studies in vitro and in vivo, we show that the anti-apoptotic protein poly(ADP-ribose) polymerase (PARP)14 promotes aerobic glycolysis in human hepatocellular carcinoma (HCC) by maintaining low activity of the pyruvate kinase M2 isoform (PKM2), a key regulator of the Warburg effect. Notably, PARP14 is highly expressed in HCC primary tumours and associated with poor patient prognosis. Mechanistically, PARP14 inhibits the pro-apoptotic kinase JNK1, which results in the activation of PKM2 through phosphorylation of Thr365. Moreover, targeting PARP14 enhances the sensitization of HCC cells to anti-HCC agents. Our findings indicate that the PARP14-JNK1-PKM2 regulatory axis is an important determinant for the Warburg effect in tumour cells and provide a mechanistic link between apoptosis and metabolism
Molecular association of glucose-6- phosphate isomerase and pyruvate kinase M2 with glyceraldehyde-3-phosphate dehydrogenase in cancer cells
- Author
- A Sawa
- Alok Ghosh
- Arup K. Bag
- AT Cordeiro
- B Khatua
- B You
- C Tristan
- Chitra Mandal
- D Anastasiou
- D Kozakov
- D Kozakov
- D Schneidman-Duhovny
- D Wang
- DE Epner
- E Krissinel
- EJ Tisdale
- F Ferreira-da-Silva
- H Nakajima
- HM Berman
- HR Christofk
- JH Roe
- JJ Laschet
- JL Jenkins
- K Tokunaga
- M Cortés-Cros
- M Ray
- M Torchala
- Mahua R. Das
- Manju Ray
- N Schek
- O Warburg
- PA Saunders
- PE Glaser
- Provas Das
- Q Huang
- Q Zhang
- RA Gomes
- RE Ferguson
- S Bagui
- S Carujo
- S Mazurek
- S Patra
- S Ray
- S Saha
- S Saha
- Saikat Chakrabarti
- Shekhar Saha
- Siddhartha S. Jana
- Subhankar Ray
- Sumit K. Dey
- T Funasaka
- T Funasaka
- T Li
- T Noguchi
- V Ravichandran
- W Luo
- W Yang
- W Yang
- X Gao
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/2016
- Field of study
Background: For a long time cancer cells are known for increased uptake of glucose and its metabolization through
glycolysis. Glyceraldehyde-3-phosphate dehydrogenase (GAPDH) is a key regulatory enzyme of this pathway and can
produce ATP through oxidative level of phosphorylation. Previously, we reported that GAPDH purified from a variety of malignant tissues, but not from normal tissues, was strongly inactivated by a normal metabolite, methylglyoxal (MG).Molecular mechanism behind MG mediated GAPDH inhibition in cancer cells is not well understood.
Methods: GAPDH was purified from Ehrlich ascites carcinoma (EAC) cells based on its enzymatic activity. GAPDH
associated proteins in EAC cells and 3-methylcholanthrene (3MC) induced mouse tumor tissue were detected by mass spectrometry analysis and immunoprecipitation (IP) experiment, respectively. Interacting domains of GAPDH
and its associated proteins were assessed by in silico molecular docking analysis. Mechanism of MG mediated GAPDH
inactivation in cancer cells was evaluated by measuring enzyme activity, Circular dichroism (CD) spectroscopy, IP and mass spectrometry analyses.
Result: Here, we report that GAPDH is associated with glucose-6-phosphate isomerase (GPI) and pyruvate kinase M2
(PKM2) in Ehrlich ascites carcinoma (EAC) cells and also in 3-methylcholanthrene (3MC) induced mouse tumor tissue.
Molecular docking analyses suggest C-terminal domain preference for the interaction between GAPDH and GPI.
However, both C and N termini of PKM2 might be interacting with the C terminal domain of GAPDH. Expression of both PKM2 and GPI is increased in 3MC induced tumor compared with the normal tissue. In presence of 1 mM MG,association of GAPDH with PKM2 or GPI is not perturbed, but the enzymatic activity of GAPDH is reduced to 26.8 ± 5 % in 3MC induced tumor and 57.8 ± 2.3 % in EAC cells. Treatment of MG to purified GAPDH complex leads to glycation at R399 residue of PKM2 only, and changes the secondary structure of the protein complex.
Conclusion: PKM2 may regulate the enzymatic activity of GAPDH. Increased enzymatic activity of GAPDH in tumor cells may be attributed to its association with PKM2 and GPI. Association of GAPDH with PKM2 and GPI could be a signature for cancer cells. Glycation at R399 of PKM2 and changes in the secondary structure of GAPDH complex could be one of the mechanisms by which GAPDH activity is inhibited in tumor cells by MG
Phytoplankton across Tropical and Subtropical Regions of the Atlantic, Indian and Pacific Oceans
- Author
- A Amato
- A Herbland
- A Sournia
- Ana María Cabello
- AR Longhurst
- AT Haidar
- B Fernández-Castro
- B Li
- BJ Finlay
- C De Vargas
- C Duarte
- CR Tomas
- CR Tomas
- CS Rousseaux
- D Blasco
- D Blasco
- D Kamykowski
- Dolors Blasco
- E Balech
- E Balech
- EL Venrick
- EL Venrick
- EL Venrick
- Eugenio Fraile-Nuez
- F Gómez
- F Gómez
- F Gómez
- F Gómez
- F Gómez
- G Monterey
- GM Hallegraeff
- H Utermöhl
- Hans G. Dam
- I Kaczmarska
- I Percopo
- JBH Martiny
- JF Saldarriaga
- JJ Cullen
- JR Beers
- JR Young
- K Grasshoff
- KB Padmakumar
- L Bérard-Thérriault
- L Cros
- L Rampi
- LK Medlin
- M Delgado
- M Edwards
- M Estrada
- M Estrada
- M Estrada
- M Latasa
- M Levandowski
- Marta Estrada
- Maximino Delgado
- MD Guiry
- MD Iglesias-Rodríguez
- MD Mackey
- Mikel Latasa
- MJ Chrétiennot-Dinet
- Montserrat Vidal
- MY Cortés
- P Cermeño
- P Jolicoeur
- P Légendre
- Patricija Mozetič
- PC Fiedler
- PG Falkowski
- PG Falkowski
- R Margalef
- RA Andersen
- RW Gould
- S Alvain
- SW Jeffrey
- V Smetacek
- Verónica Benítez-Barrios
- WG Sunda
- WW Gregg
- Y Fukuyo
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- 01/01/2016
- Field of study
Postprint4,411
Outcomes from elective colorectal cancer surgery during the SARS-CoV-2 pandemic
- Author
- 14 | COVIDSurg COllabOratIVe Tzovaras G. (General University Hospital of Larissa)
- Aawsaj Y.
- Abad Gurumeta A.
- Abad-Motos A.
- Abate E.
- Abbott D.
- Abdalla M.
- Abdeldayem H.
- Abdelkader Salama I.
- Abdelkarim M.
- Abdur-Rahman L.
- Abel M. K.
- Aboelkassem Ibrahim A.
- Abou Chaar M. K.
- Abreu da Silva A.
- Abubakar A.
- Acebes García F.
- Achalandabaso Boira M. Sales Mallafré R. (Hospital Universitari de Tarragona Joan XXIII)
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- Adamina M.
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- Adiamah A.
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- Aguado H. (Hellín Hospital)
- Aguilar Gonzalez M. Talukder S. (West Suffolk Hospital)
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- Aiken T.
- Aimé A.
- Akalin M.
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- Akhtar M. A.
- Akhter Rahman M. M.
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- Al Awwad S.
- Al Habes H.
- Al Maadany F. S. (Al-Jalaa Hospital)
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- Al-Masri M.
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- Alam F.
- Alawneh F. (King Hussein Cancer Center). Libya: Alkadeeki G.
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- Alghamdi M.
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- Ali M.
- Ali S.
- Aliyeva Z.
- Aljiffry M.
- Alma Mater Studiorum University of Bologna)
- Almeida A. C.
- Almeida J. I.
- Almeida-Reis R.
- Alnumani T. (King Fahad 16 | COVIDSurg COllabOratIVe General Hospital)
- Alobeed O.
- Alonso de la Fuente N. Jimenez Toscano M. (Hospital del Mar)
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- Alselaim N. (King Saud Bin Abdulaziz University for Health Sciences
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- Argentina: Alurralde C.
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- Castellammare di Stabia)
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- Clinical Centre of Serbia)
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- COVIDSurg COllabOratIVe | 15 Violante T. (IRCCS Azienda Ospedaliero – Universitaria di Bologna
- Cozza V.
- Creavin B.
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- Day A. (East Surrey Hospital)
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- Department of Biomedical Sciences
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- Government Medical College). Ireland: Aremu M.
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- Smith L.
- Smith. J (St James’s Hospital)
- Soares A. P.
- Soh J. Y.
- Sohrabi C.
- Solari F.
- Soriero D. (IRCCS Ospedale Policlinico San Martino)
- Sorrentino L. (Fondazione IRCCS Istituto Nazionale dei Tumori
- Sorribas Grifell M.
- Soto Montesinos C. (Fundació Althaia – Xarxa Assistencial Universitària de Manresa)
- Souadka A. (Institut National d’Oncologie
- Soulikia K.
- Sousa Fernandes M. (Hospital Beatriz Angelo)
- Sousa R. (Centro Hospitalar Universitário Lisboa Central)
- Sousa S.
- Spagni G.
- Spampinato M. G. (Vito Fazzi
- Spartalis E.
- Spencer N.
- Spiezio G. (Colorectal Surgical Oncology Unit – Istituto Nazionale Tumori Fondazione
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- Sreedharan L.
- Sriram R. K.
- Srishankar S. (Teaching Hospital Anuradhapura). Sudan Ali Adil A. K. (Al-Rajhi). COVIDSurg COllabOratIVe | 17 Sweden: Älgå A.
- St John S.
- Stafford J. (George Eliot Hospital)
- Stavrinidou O.
- Steele C. (Sheffield Teaching Hospital NHS Foundation Trust)
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- Steinke J.
- Stevens K.
- Stevenson J. (The Ottawa Hospital). Croatia: Bačić G.
- Stevic D.
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- Stylianidis G. (Evaggelismos General Hospital)
- Subhi M. T. (Alkhadra Hospital)
- Subocius A.
- Subramaniam S. (Queen Elizabeth Hospital and Universiti Malaysia Sabah
- Sundaram Venkatesan G. (Glan Clwyd Hospital)
- Suszták N. (Szent Borbála Kórház). India: Bhat G. A.
- Sutherland A. (Coffs Harbour Health Campus)
- Swinson B. (Royal Brisbane and Women’s Hospital). Austria: Messner F.
- Syed W. A. S.
- Syllaios A.
- Szatmary P.
- Szubota I. (Hospital and Oncological Centre Novy Jicin). Denmark: Ebbehøj A. L.
- Sánchez del Pueblo C.
- Sánchez Fuentes N.
- Sánchez- Pernaute A.
- Sánchez- Rubio M.
- Sánchez-García S.
- Taddei A.
- Tadic B.
- Taibi A. (Chu Limoges)
- Talal El-Abur I.
- Talwar R. (Luton and Dunstable University Hospital)
- Tammaro P.
- Tan J. A.
- Tan X. S.
- Tanal M.
- Tang A. M.
- Tanzanu M.
- Tartaglia D. (Azienda Ospedaliero Universitaria Pisana)
- Tasis N. (Athens Naval and Veterans Hospital)
- Tatar O. C.
- Tavares F.
- Tayeh S. (Homerton University Hospital)
- Tebala G. D.
- Teixeira J. (Centro Hospitalar Universitário do Algarve – Unidade de Faro)
- Teixeira M. (Centro Hospitalar do Tamega e Sousa)
- Tejero- Pintor F. J. (Hospital Universitario Río Hortega)
- Testa V. (Santa Croce E. Carle Hospital
- Tewari N. (University Hospitals Coventry and Warwickshire NHS Trusts)
- Tezas S. (Furness General Hospital)
- Thaha M.
- Thanapal M. R. (Hospital Kuala Lumpur)
- Theodosopoulos T.
- Theophilidou E. (Royal Derby Hospital)
- Thian A.
- Thomas A. (Royal Liverpool University Hospital)
- Thompson D. (Morriston Hospital Swansea)
- Thornhill M. (Dell Seton Medical Center at the University of Texas)
- Thrumurthy S. (Epsom and St Helier University Hospitals NHS Trust)
- Thulasiraman S. V.
- Timbrell S.
- Tirloni L.
- Titu S. (Prof. Dr. Ion Chiricuta Institute of Oncology). Russia: Garmanova T.
- Tonini V. (S. Orsola-Malpighi Hospital)
- Torres A. (Hospital Clínico de Madrid)
- Torres Arcos C.
- Townson A.
- Trabulsi N. (King Abdulaziz University Hospital)
- Travaglio E. (Regina Montis Regalis Hospital
- Tribillon E. (Institut Mutualiste Montsouris)
- Troncoso Pereira P. (Hospital Mateu Orfila)
- Tropeano F. P. (Federico II University Hospital)
- Trujillo Díaz J.
- Tsai L.
- Tsarkov P.
- Tsiamalou I.
- Tsiaoussis I.
- TU Dresden)
- Tucci R. (Azienda Ospedaliera Universitaria Careggi)
- Tufo A. (Ospedale del Mare)
- Tugmen C.
- Tulina I. (Clinic of Coloproctology and Minimally Invasive Surgery
- Tuncer K.
- Turnbull A. (Victoria Hospital Kirkcaldy)
- Turrado-Rodriguez V.
- Turri G. (Azienda Ospedaliera Universitaria Integrata di Verona)
- Tweedle E. (Addenbrooke’s Hospital)
- Ugarte-Sierra B. (Hospital Universitario de Galdakao)
- Uludağ S. S.
- Umair M.
- Universiti Sains Malaysia)
- University of Amsterdam)
- Università di Ferrara)
- Université Mohammed V Rabat). Netherlands: Hompes R.
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- Urbani A. (Azienda Ospedaliero Universitaria San’anna)
- Urbieta A. (Hospital Universitario la Paz)
- Uslu G.
- Utkan N. Z.
- Uyanik M. S. (Samsun Training and Research Hospital)
- Uzunoglu F. G. (University Medical Center Hamburg–Eppendorf). Greece: Antonakis P.
- Vaccarella G. (Azienda Ospedaliera Ospedali Riuniti Villa Sofia-Cervello)
- Valbuena Jabares V. (Marqués de Valdecilla University Hospital)
- Valdes- Hernandez J. (Hospital Universitario Virgen Macarena)
- Valero Soriano M. (Hospital General Reina Sofía)
- Valle Rubio A. (Getafe University Hospital)
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- Van den Eynde J.
- Van den Eynde R. (Uz Leuven). Bulgaria: Sokolov M. (University Hospital Alexandrovska). Canada: Boutros M.
- Varma M. (University of California
- Vasljević J.
- Vassiliu P. (Attikon University General Hospital)
- Vaz Pereira R.
- Vaz S. (Centro Hospitalar e Universitário de São João)
- Velchuru V.
- Velickovic D. (Clinic for Digestive Surgery
- Velidedeoglu M.
- Venn M. (Royal London Hospital)
- Venskutonis D. (Lithuanian University of Health Sciences Kaunas Clinical Hospital). Madagascar: Rasoaherinomenjanahary F.
- Vera Mansilla C. (Hospital Universitario Principe de Asturias)
- Verberne C. (John Radcliffe Hospital)
- Vergari R. (Ospedali Riuniti di Ancona)
- Vernon L. (Cork University Hospital)
- Vervoort D.
- Vescio G. (University ‘Magna Graecia’ of Catanzaro)
- Vezakis A. (Aretaieion Hospital)
- Videira J. F. (IPO Porto). Réunion: Kassir R.
- Vieira B. (Centro Hospitalar de Trás-Os-Montes e Alto Douro
- Vieira Caroço T. (IPO Coimbra)
- Vieira Paiva Lopes A. C. (Hospital de Torres Vedras – Centro Hospitalar do Oeste)
- Vignali A. (San Raffaele Scientific Institute
- Vigorita V. (Álvaro Cunqueiro Hospital)
- Vijayan D. (Queen Elizabeth Hospital Birmingham)
- Villalabeitia Ateca I. (Hospital Universitario Cruces)
- Vimalachandran D. (Countess of Chester Hospital)
- Viswanath Y. K. S. (James Cook University Hospital)
- Vitali A. (Ospedale San Giovanni di Dio)
- Vitone L. (Royal Blackburn Hospital)
- Vives R. V. (Bellvitge University Hospital)
- Vo U. G. (Fiona Stanley Hospital)
- Von Papen M.
- Vovola F. (Ospedali Riuniti Azienda Ospedaliera Universitaria Foggia)
- Vucic N.
- Vázquez Fernández A. (Hospital Clínico Universitario de Valladolid)
- Wadham B. (The University Hospital of South Manchester)
- Walkes K. (Queen Elizabeth Hospital). Belgium: Flamey N.
- Wani R. (Sher-I-Kashmir Institute of Medical Sciences)
- Waqar S. H. (Pakistan Institute of Medical Sciences). Poland: Major P. (Jagiellonian University Medical College). Portugal: Azevedo C.
- Warren O. (Chelsea and Westminster Hospital)
- Watson L. J. (Sunderland Royal Hospital)
- Watson N. (King’s Mill Hospital)
- Weitz J.
- Welsch T. (Carl-Gustav-Carus University Hospital
- Werner J. (LMU Klinikum Campus Innenstadt)
- Westwood E. (James Paget University NHS Foundation Trust Hospital)
- Whelan M. (Tallaght University Hospital)
- Whitmore H. (Torbay and South Devon NHS Trust)
- Wilkin R. J. W. (South Warwickshire NHS Foundation Trust)
- Wilkins A. (Hull University Teaching Hospitals NHS Trust)
- Williams G. (Royal Gwent Hospital)
- Williams K. (St George’s Hospital)
- Wilson M. (Forth Valley Royal Hospital)
- Wimmer A. (Paracelsus Medical University Salzburg). Barbados: Barker D.
- Wong M.
- Worku D. (Queens Medical Centre)
- Wullschleger M. (Gold Coast University Hospital)
- Xavier R. G.
- Xenaki S.
- Xynos E. (University Hospital of Heraklion Crete and Interclinic Hospital of Crete). Hong Kong: Futaba K.
- Yang W.
- Yassin N. (Royal Wolverhampton NHS Trust)
- Ye G.
- Yesantharao P.
- Yetkin S. G. (Sisli Hamidiye Etfal Training and Research Hospital)
- Yeşilyurt D. (University of Health Sciences Tepecik Training and Research Hospital)
- Yiallourou A. (Nicosia General Hospital). Czechia: Martinek L.
- Yıldırım A.
- Yildiz A. (Yildirim Beyazit University Yenimahalle Training and Research Hospital). Uganda: Lule H.
- Young R. (York Teaching Hospitals NHS Trust)
- Yousof E. A. (Assiut University Hospital)
- Youssef M. (Norfolk and Norwich University Hospital)
- Yurttas C. (University Hospital Tuebingen)
- Yánez C. (Royo Villanova)
- Yüksel E. (Kocaeli University Teaching Hospital)
- Zafar S. N. (University of Wisconsin)
- Zakaria A. D.
- Zakaria Z. (School of Medical Sciences and Hospital
- Zambon M. (Policlinico Umberto I Sapienza University of Rome)
- Zanus G. (Ca’ Foncello Treviso – DISCOG – Università di Padova)
- Zegarac M. (Institute for Oncology and Radiology of Serbia)
- Zelić M. (University Hospital Center Rijeka)
- Zengin A. K. (Istanbul Universty – Cerrahpaşa Medical Faculty)
- Zerbib P. (CHU Lille)
- Zervas K.
- Zese M. (Santa Maria degli Angeli Hospital ULSS 5 – Adria)
- Zhang H. (Concord Repatriation General Hospital)
- Zizzo M. (Azienda Unità Sanitaria Locale – IRCCS di Reggio Emilia)
- Zografos C. (Laiko University Hospital)
- Zorrilla Ortúzar J. (Hospital General Universitario Gregorio Marañón)
- Zourntou S. (General Hospital of Larissa ‘Koutlimpaneio and Triantafylleio’)
- Zubaidi A. M. (King Saud University). Serbia: Aleksić L.
- Ângelo M.
- Çelebi F.
- Çolak E.
- Öfner D. (Medical University of Innsbruck)
- Öhlberger L.
- Özçelık M. F.
- Öğücü H.
- Überrück L.
- Ćoza I.
- Publication venue
- 'Wiley'
- Publication date
- 01/01/2020
- Field of study
This study aimed to describe the change in surgical practice and the impact of SARS-CoV-2 on mortality after surgical resection of colorectal cancer during the initial phases of the SARS-CoV-2 pandemic
The ERK and JNK pathways in the regulation of metabolic reprogramming.
- Author
- A Barbarulo
- A Barthel
- A Hall
- A Kosteli
- A Shapouri-Moghaddam
- AD Panopoulos
- AJ Levine
- AJ Marko
- AM Mingo-Sion
- AP West
- AR Grassian
- B Everts
- B Faubert
- B Ghesquière
- B Zheng
- C Bubici
- C Cantó
- C Cellurale
- C Taha
- CD Folmes
- CD Folmes
- CH Chang
- CH Chang
- CJ Caunt
- CJ David
- CJ Hedeskov
- CM Krawczyk
- CN Lumeng
- Concetta Bubici
- CV Dang
- CV Dang
- CV Dang
- D Anastasiou
- D Dixit
- D Senyilmaz
- DG Hardie
- DG Hardie
- ED Michelakis
- EK Wiese
- EM Palsson-McDermott
- ES Goetzman
- EV Dang
- F Li
- G Dontu
- G Kroemer
- G Solinas
- GM Tannahill
- GV Long
- H Deng
- H Ke
- H Kondoh
- H Semba
- H Shim
- H Ying
- H Zhang
- HL Fritz
- HL Wieman
- HR Christofk
- HR Christofk
- I Kawashima
- J Bossche Van den
- J Cui
- J Pouysségur
- J Yun
- JA Graves
- JJ Lum
- JR Hom
- JW Locasale
- K Birsoy
- K Gottlob
- K Tech
- KM Lee
- KN Hardeman
- L Galluzzi
- L Hui
- LA O’Neill
- LA O’Neill
- LB Sullivan
- LM Ferreira
- LR Edmunds
- LZ Shi
- M Agathocleous
- M Anbalagan
- M Cargnello
- M Cortés-Cros
- M Gururajan
- M Kishore
- M Raman
- MF Miniotis
- MG Heiden Vander
- MG Heiden Vander
- MG Heiden Vander
- MH Lee
- MS Goyal
- MV Liberti
- N Chen
- N Hay
- N Wu
- NN Pavlova
- NP Shanware
- O Warburg
- OJ Martin
- PC Ho
- PG Través
- PP Hsu
- PP Hsu
- PS Ward
- Pui Man Choy
- Q Zhou
- R Haq
- R Khamari
- R Wang
- R Yang
- RA Cairns
- RA Gatenby
- RD Michalek
- RE Board
- RG Jones
- RL Elstrom
- S Aras
- S Chung
- S John
- S Miyamoto
- S Nemoto
- S Papa
- S Papa
- S Varum
- S Vernia
- Salvatore Papa
- SH Lee
- SK Biswas
- SK Biswas
- SO Lim
- SY Lunt
- SY Lunt
- T Finkel
- T Hitosugi
- TJ Parmenter
- TL Dayton
- TL Dayton
- UE Martinez-Outschoorn
- V Iansante
- W Yang
- W Zhou
- WH Munyon
- WJ Israelsen
- WJ Israelsen
- X Li
- X Zheng
- Y Zhao
- YH Wang
- ZE Stine
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 23/10/2018
- Field of study
Most tumor cells reprogram their glucose metabolism as a result of mutations in oncogenes and tumor suppressors, leading to the constitutive activation of signaling pathways involved in cell growth. This metabolic reprogramming, known as aerobic glycolysis or the Warburg effect, allows tumor cells to sustain their fast proliferation and evade apoptosis. Interfering with oncogenic signaling pathways that regulate the Warburg effect in cancer cells has therefore become an attractive anticancer strategy. However, evidence for the occurrence of the Warburg effect in physiological processes has also been documented. As such, close consideration of which signaling pathways are beneficial targets and the effect of their inhibition on physiological processes are essential. The MAPK/ERK and MAPK/JNK pathways, crucial for normal cellular responses to extracellular stimuli, have recently emerged as key regulators of the Warburg effect during tumorigenesis and normal cellular functions. In this review, we summarize our current understanding of the roles of the ERK and JNK pathways in controlling the Warburg effect in cancer and discuss their implication in controlling this metabolic reprogramming in physiological processes and opportunities for targeting their downstream effectors for therapeutic purposes.Brunel Research Initiative & Enterprise Fund, Brunel University
of London (to CB), Kay Kendall Leukemia Fund (KKL443) (to CB),
250 Great Minds Fellowship, University of Leeds (to SP), AMMF
Cholangiocarcinoma Charity (to SP and PMC), and Bloodwise
(17014) (to SP and CB)
Lack of Evidence for PKM2 Protein Kinase Activity
- Author
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Small-Molecule Screens: A Gateway to Cancer Therapeutic Agents with Case Studies of Food and Drug Administration–Approved Drugs
- Author
- Anton Simeonov
- Banasik
- Buchdunger
- Cashin
- Cortés-Cros
- Drew
- Epstein
- Fleuren
- Fong
- G. Sitta Sittampalam
- Giuliani
- Green
- Hall
- Hsiang
- Johannes
- John C. Braisted
- Kast
- Lazo
- Mak
- Manley
- Martinez
- Martinez Molina
- Matthew D. Hall
- Mezencev
- Michael M. Gottesman
- Nathan P. Coussens
- Padmanabha
- Plückthun
- Stein
- Tyler Peryea
- Uitdehaag
- Wakeling
- Wall
- Wassermann
- Zhao
- Publication venue
- 'American Society for Pharmacology & Experimental Therapeutics (ASPET)'
- Publication date
- Field of study
Targeting cancer cell metabolism: evidences and perspectives
- Author
- A Schulze
- BA Teicher
- BK Mohanti
- BR Landau
- C Frezza
- C Sebastián
- C. Massard
- CV Dang
- D Braas
- D Daye
- D Hanahan
- D Singh
- DB Longley
- DR Wise
- EA Raetz
- ED Michelakis
- F Bost
- F Zhang
- G Hatzivassiliou
- G Sutendra
- HR Christofk
- I Ben Sahra
- IB Sahra
- J Cao
- J-A Losman
- J. Hadoux
- JA Menendez
- K Holen
- L Jerby
- L Liu
- LE Raez
- M Ayala-Ramirez
- M Cortés-Cros
- M Gallí
- M Laplante
- MG Vander Heiden
- MJ Seltzer
- NC Duarte
- O Folger
- O Warburg
- P Gao
- PW Stacpoole
- S Bonnet
- S Farber
- T Puig
- V Behar
- W Liu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
PKM2 Isoform-Specific Deletion Reveals a Differential Requirement for Pyruvate Kinase in Tumor Cells
- Author
- Aaron M. Hosios
- Allali-Hassani
- Anastasiou
- Anastasiou
- Ayala
- Bardeesy
- Baumhoer
- Brian P. Fiske
- Cairns
- Cerami
- Chaneton
- Chaneton
- Chen
- Christofk
- Christofk
- Clary B. Clish
- Clower
- Commisso
- Cortés-Cros
- David
- Dolores Di Vizio
- Dombrauckas
- Gao
- Gary Bellinger
- Gerburg M. Wulf
- Goldberg
- Gordon B. Mills
- Hitosugi
- Imamura
- Jain
- James W. Horner
- Jianxin Xie
- Jie Li
- Jurczak
- Keller
- Laura N. Burga
- Lewis C. Cantley
- Liang
- Luo
- Lv
- Maquat
- Matthew G. Vander Heiden
- Mazurek
- Michael J. Jurczak
- Mika Sasaki
- Noguchi
- Parnell
- Raymond
- Richard G. Kibbey
- Ronald A. DePinho
- Salk
- Schraml
- Shawn M. Davidson
- Sonveaux
- Talya L. Dayton
- Tyler Jacks
- Vander Heiden
- Vander Heiden
- Vander Heiden
- Varghese
- Vaupel
- Wang
- Wang
- William J. Israelsen
- Xu
- Yang
- Yang
- Yang
- Yimin Yu
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Delaying surgery for patients with a previous SARS-CoV-2 infection
- Author
- A A Ali Karar
- A A Kerawala
- A A Marra
- A Abad Gurumeta
- A Abad-Motos
- A Abdelmajeed
- A Abdelrahman
- A Abdelsamed
- A Abdulkareem
- A Aboelkassem Ibrahim
- A Abouassi
- A Abreu da Silva
- A Abubakar
- A Acher
- A Aderombi
- A Adeyeye
- A Adiamah
- A Aggarwal
- A Aghayeva
- A Agnes
- A Agrawal
- A Ahmeidat
- A Aimé
- A Ajlan
- A Al-Habib
- A Al-Mohammad
- A Al-Mukhtar
- A Aladeojebi
- A Alamri
- A Alanbuki
- A Alatar
- A Alburakan
- A Alfaro-Goldaracena
- A Alhamed
- A Alhefdhi
- A Almeciga
- A Almeida
- A Alomair
- A Alonso Poza
- A Alsaif
- A Anastasi
- A Antic
- A Anzak
- A Aprile
- A Arminio
- A Arulanantham
- A Askari
- A Asqalan
- A Athanasiou
- A Ayhan
- A Ayman
- A Ayubi
- A Azizi
- A B Martins
- A Bacon
- A Baker
- A Balakrishnan
- A Bandiera
- A Banerjee
- A Barrabe
- A Beamish
- A Bellacci
- A Belli
- A Belvedere
- A Benkabbou
- A Bhalla
- A Bhangu
- A Billè
- A Bin Nasser
- A Biondi
- A Blatt
- A Blazquez Martin
- A Boddy
- A Bokhari
- A Bondurri
- A Boulton
- A Boutall
- A Branquinho
- A Brunelli
- A Brunt
- A Bruscino
- A Budacan
- A Burahee
- A Böttcher
- A C Almeida
- A C Deus
- A C Roslani
- A C Soares
- A C Vieira Paiva Lopes
- A Caiado
- A Camillo
- A Canas-Martinez
- A Cano
- A Carabias
- A Chandock
- A Charalabopoulos
- A Che Jusoh
- A Chebaro
- A Chessa
- A Chiappini
- A Chitul
- A Choudhry
- A Chowdhury
- A Colquhoun
- A Conesa
- A Cordova
- A Costanzi
- A Cotoia
- A Cotter
- A Crichton
- A Cuadrado-García
- A Currie
- A Cvetkovic
- A D Bueno Cañones
- A D Rajgor
- A D Zakaria
- A D'Amore
- A D'Urso
- A Daly
- A Davies
- A Day
- A De Gea Rico
- A De Manzoni Garberini
- A De Pablo García-Cuenca
- A De Troia
- A De Virgilio
- A Dehal
- A Desai
- A Di Bartolomeo
- A Di Bella
- A Di Somma
- A Diamantis
- A Doyle
- A Durrani
- A E Arikan
- A E Sherif
- A Eastmond
- A El Ouahabi
- A Elawad
- A Eldaly
- A Elhamshary
- A Esposito
- A Esteban
- A Ezanno
- A Fadzli
- A Fagotti
- A Fancellu
- A Farsi
- A Faustino
- A Fazenda
- A Fernández-López
- A Ferrero
- A Ferrés
- A Fiorini
- A Fisher
- A Fletcher
- A Fowler
- A Fox
- A Frampton
- A Frankel
- A Frati
- A Freitas
- A Frena
- A Fuson
- A G Carta
- A G Zarabini
- A Gabre-Kidan
- A Gagliano
- A Gainza
- A Gatti
- A Gattolin
- A Gaunt
- A Geddes
- A Gegúndez Simón
- A Ghanbari
- A Ghannam
- A Giaglaras
- A Gianni
- A Giblin
- A Gillis
- A Gklavas
- A Glencer
- A Gomes da Costa
- A Gori
- A Goyal
- A Gronchi
- A Gueutier
- A Guglielmi
- A Guimarães
- A Gupta
- A Gutierrez Calvo
- A Gvaramadze
- A Gómez-Pedraza
- A H Hussain
- A H Khan
- A Habeeb
- A Hainsworth
- A Hamad
- A Hannah
- A Hanson
- A Harky
- A Hasenburg
- A Hawkins
- A Haynes
- A Haynes
- A Henry
- A Herman
- A Hernández Gutierrez
- A Heuer
- A Hmedat
- A Hogan
- A Hunt
- A I Gutiérrez Fernández
- A I Kilani
- A I Soriano
- A I Tercero-Uribe
- A Ibrahim
- A Ionescu
- A Jah
- A Jain
- A Jamal
- A Jibril
- A Jiménez
- A Joshi
- A Jotic
- A K Ali
- A K Andrade
- A K Lala
- A K Scafa
- A K Zengin
- A Kahn
- A Kamocka
- A Kanatas
- A Kappenberger
- A Karamarkovic
- A Karim
- A Kattakayam
- A Kaufmann
- A Kawai
- A Kent
- A Khajuria
- A Khan
- A Khoja
- A Kirk
- A Kisiel
- A Kler
- A Kocataş
- A Koh
- A Kolias
- A Kollàr
- A Kolusarı
- A Kourdouli
- A Kouyoumdjian
- A Kredan
- A Kumar
- A Königsrainer
- A L De Oliveira López
- A L Ebbehøj
- A L Picardo
- A Laforest
- A Lagares
- A Laios
- A Laird
- A Landaluce-Olavarria
- A Lanzon
- A Larentzakis
- A Lauretta
- A Lim
- A Loayza
- A Loehrer
- A Lopez Abad
- A Louvrier
- A Lovece
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- N Dawe
- N Depalma
- N Donlon
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- N Eardley
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- N Howes
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- N Kamal
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- N Laskar
- N Lavagen
- N Lott
- N Lynch
- N Löfgren
- N M Mariani
- N Machado
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- N Manu
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- N Michalopoulos
- N Moeckelmann
- N Morales Palacios
- N N Dudi-Venkata
- N Neal
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- N Osman
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- N Pigadas
- N Prat
- N Prijović
- N Q Fathi
- N Rajaretnam
- N Ratnavelu
- N Ravi
- N Ryan
- N S Pipitone Federico
- N Salgado-Nesme
- N Savković
- N Schlesinger
- N Sharma
- N Shugg
- N Silva
- N Slijepcevic
- N Spencer
- N Stylianides
- N Sureshkumar Shah
- N Suszták
- N Sánchez Fuentes
- N Tamini
- N Tasis
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- N Tewari
- N Trabulsi
- N Vucic
- N Watson
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- N Z Utkan
- N Zeller
- Naomi Wright
- Neil J Smart
- Neil Sharma
- Ng Ssm
- NIgra Ma
- O Alaamer
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- O Cullivan
- O Dwidar
- O Dülgeroğlu
- O E Posadas-Trujillo
- O Esteban Sinovas
- O Fuwa
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- R A Castillejos-Molina
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- R Kassir
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- R Mahmoud
- R Mannion
- R Marques
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- R Massoud
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- R Memba Ikuga
- R Mihai
- R Mithany
- R Mohsine
- R Morgan
- R Myatt
- R Nafees Ahmed
- R Nath
- R O'Neill
- R Oliva
- R Ooi
- R Palaia
- R Parreira
- R Patrone
- R Peevor
- R Pereira
- R Persiani
- R Picón Rodríguez
- R Piper
- R Potter
- R Pujol Pina
- R Rahman
- R Ramamoorthy
- R Reehal
- R Reis
- R Ribeiro
- R Rimonda
- R Robles
- R S Martins
- R S Prichard
- R Sales Mallafré
- R Salvia
- R Salvioni
- R Sanchez Jimenez
- R Sanchez-Santos
- R Santos
- R Sanz-Lopez
- R Sayyed
- R Scheri
- R Schiavina
- R Schiemer
- R Schneider
- R Schwab
- R Scott
- R Scurrah
- R Shaw
- R Silva
- R Singh
- R Skipworth
- R Smeets
- R Smillie
- R Smith
- R Sousa
- R Talwar
- R Thomas
- R Torné
- R Tucci
- R Tudisco
- R Turkington
- R V Iosifescu
- R V Vives
- R Valero
- R Van den Eynde
- R Vaz Pereira
- R Vergari
- R Vidya
- R Vinayagam
- R Wade
- R Wilkin
- R Young
- R Zakaria
- R Çapoğlu
- Rachel A Khaw
- Rachel Moore
- Raghavan Vidya
- Raghavan Vidya
- Raghavan Vidya
- Rahel Ghebre
- Ravi Barod
- Raza Sayyed
- Rene Pareja
- Richard Jw Wilkin
- Richard Pt Evans
- Richard Shaw
- Richard Shaw
- Richard Shaw
- Risk Obf
- Rob Bristow
- Rohan R Gujjuri
- Rory J Piper
- Ruth A Benson
- Ruth A Benson
- Ruth Blanco-Colino
- S A Güler
- S A Landeo Agüero
- S Abdel Al
- S Ahad
- S Al Awwad
- S Alaa
- S Alfieri
- S Ali
- S Alkarak
- S Alshammari
- S Alsobhi
- S Amonkar
- S Andrijasevic
- S Annamalai
- S Antic
- S Anwar
- S Aribi
- S Banting
- S Barnard
- S Bhasin
- S Bonnet
- S Boucher
- S Boussedra
- S Bowman
- S Bradulskis
- S Brown
- S Brown
- S Bulathsinhala
- S Burg
- S Cadwell-Sneath
- S Caird
- S Cavaleiro
- S Cenciarelli
- S Chen
- S Chidambaram
- S Chopra
- S Clatworthy
- S Coiro
- S Corbin
- S Correia
- S D'Ugo
- S Dakpé
- S Demirli Atıcı
- S Demyttenaere
- S Di Maria Grimaldi
- S Domingo
- S Duff
- S Dumitra
- S Dwerryhouse
- S E Xyda
- S Elwatidy
- S Ergün
- S Evans
- S F Fulginiti
- S F Hon
- S Ferrero
- S Folli
- S Ford
- S Fordington
- S Frade
- S Fraser
- S Fusetti
- S G Aoun
- S Gacic
- S Gahunia
- S Gananadha
- S Garrido
- S Gennari
- S Gentilli
- S Goodrum
- S Gore
- S Gortázar
- S Granieri
- S Green
- S Guadagni
- S H Waqar
- S Hamrang-Yousefi
- S Handa
- S Henriques
- S Higgs
- S Humphries
- S Ibrahim
- S Iwata
- S Jang
- S Jog
- S Jordan
- S Kadija
- S Kapoor
- S Karandikar
- S Kazzaz
- S Killeen
- S Klimopoulos
- S Kmezić
- S Krajnak
- S Kudchadkar
- S Lam
- S Latinčić
- S Lawday
- S Laws
- S Leeson
- S Lester
- S Liau
- S M Isolani
- S M Lucchini
- S Macina
- S Majrashi
- S Mancini
- S Manfredelli
- S Mastoridis
- S Math
- S Matić
- S Mccluney
- S Melghazaly
- S Meneghini
- S Millar
- S Mills
- S Mochet
- S Moug
- S Mukherjee
- S Munot
- S Murphy
- S N Zafar
- S N Zafar
- S Nazir
- S Nikolic
- S Nobile
- S Novello
- S O'Brien
- S O'Malley
- S Ojha
- S Oosterling
- S Paiella
- S Palagi
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- S Pantovic
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- S Parmar
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- S Patauner
- S Patil
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- S Politis
- S Ponce
- S Powell
- S Prabhu
- S Preston
- S Price
- S Pringle
- S Rakhshani-Moghadam
- S Ramcharan
- S Rapaport
- S Rathinam
- S Rattizzato
- S Ravindrakumar
- S Ravindran
- S Rayamajhi
- S Reijers
- S Ricci
- S Robertson
- S Rodimov
- S Rooney
- S Rossi
- S Roy Mahapatra
- S Rozwadowski
- S S Uludağ
- S Saeed
- S Salimoğlu
- S Salindera
- S Santarrufina Martinez
- S Saso
- S Saudí
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- S Scasso
- S Shah
- S Shaikh
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- S Shaw
- S Shehata
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- S Singh
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- S Sravanam
- S Srinathan
- S Srishankar
- S St John
- S Subramaniam
- S Sumrak
- S Sundar
- S Sánchez-García
- S Talukder
- S Tayeh
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- S Tezas
- S Thole
- S Thrumurthy
- S Timbrell
- S Tingle
- S Titu
- S Tormey
- S Tornese
- S Torretta
- S Truant
- S Tzedakis
- S V Thulasiraman
- S Valverde
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- S Xenaki
- S Yordanov
- S Zani
- S Zanotti
- S Zonta
- S Zourntou
- Salomone Di Saverio
- Sameh Emile
- Sampaio da Nóvoa Gomes Miguel 2nd
- Samuel Ford
- Samuel Ford
- Samuel Lawday
- Santos Pmdd
- Sattar Alshryda
- Schelto Kruijff
- Sean Dowdy
- Sebastian Shu
- Sef Jones
- Sezai Leventoglu
- Shebani Farik
- Shelley Hwang
- Shylasree Ts Rajkumar
- Sinziana Dumitra
- Siobhan C Mckay
- Siobhan McKay
- Sivesh K Kamarajah
- Sivesh K Kamarajah
- Sohei Satoi
- Sohei Satoi
- Sohini Chakrabortee
- Ssa Qadri
- Stephen J Price
- Stephen Tabiri
- Steve Bromage
- Stuart C Winter
- Sudha Sundar
- Sudha Sundar
- Susan Moug
- Susan Moug
- Syed Was
- Symeon Metallidis
- T A Lawal
- T Abbott
- T Aiken
- T Alnumani
- T Arif
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- T Avlund
- T Bin Traiki
- T Boyle
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- T Fullmer
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- T Hilton
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- T Janjic
- T Jones
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- T Karahasanoğlu
- T Kato
- T Kaya
- T Khan
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- T Liakakos
- T M Sorour
- T Maccabe
- T Marina Martin
- T Martin
- T Miguel
- T Nambirajan
- T Nelli
- T Newman
- T Nicolás-López
- T Nouh
- T Nugent
- T O Klatte
- T Perra
- T Pina-Vaz
- T Pissanou
- T Poli
- T Raymond
- T Reinhard
- T Revez
- T Richards
- T Routledge
- T Royle
- T Saafan
- T Sammour
- T Santarius
- T Schiergens
- T Sehgal
- T Shortland
- T Sian
- T Sidiropoulos
- T T Sholadoye
- T Tammaro
- T Theodosopoulos
- T Tsirlis
- T Uson-Bouthelier
- T Van Wyngaard
- T Vanounou
- T Vieira Caroço
- T Violante
- T Vollkommer
- T Walton
- T Wasim
- T Welsch
- T Williams
- Tabassum Khan
- Tatiana Garmanova
- Thomas D Pinkney
- Thomas Konney
- Thomas M Drake
- Tobias Klatte
- Tom Ef Abbott
- U Akgor
- U Andaleeb
- U Bork
- U Bumbasirevic
- U Butt
- U De Andres Olabarria
- U Fernandes
- U Fumagalli Romario
- U G Vo
- U Grossi
- U Jayarajah
- U M Jariod Ferrer
- U Ribeiro Junior
- U Ronellenfitsch
- U Selbong
- U Speth
- V Alexoudi
- V Annessi
- V Bascarevic
- V Capizzi
- V Chiarella
- V Cozza
- V D Mandato
- V De Simone
- V Devezas
- V Drubay
- V Duque-Mallén
- V Fernandes
- V Garcia Soria
- V García Pineda
- V Gata
- V Granata
- V H Baptista
- V Hudson
- V I Ribeiro
- V Irvine
- V J García Porcel
- V Javurkova
- V Jimenez
- V Jokic
- V Kakotkin
- V Kantola
- V Kasivisvanathan
- V Konstantinovic
- V Kubyshkin
- V Lago
- V Linz
- V Lizzi
- V Luoma
- V Mahendran
- V Markovic
- V Mastrofilippo
- V Mazzaferro
- V Milutinović
- V Miu
- V Muñoz-Atienza
- V Ng
- V Ng
- V Oktseloglou
- V Ozben
- V Papadopoulos
- V Picotti
- V Pinto
- V Pla-Marti
- V Pérez Simón
- V Quintodei
- V Rizzo
- V Rossi
- V S Ban
- V S Kolli
- V S Rodrigo
- V Testa
- V Tonini
- V Tsaousis
- V Turrado-Rodriguez
- V Valbuena Jabares
- V Valtzoglou
- V Velchuru
- V Vigorita
- V Vujanac
- V Yip
- V Zamvar
- V Šćepanović
- Veeru Kasivisvanathan
- W Butt
- W Campbell
- W Cymes
- W Garrett
- W H Khan
- W J Wong
- W Knight
- W Lee
- W Marx
- W McCormick
- W McGahan
- W Mugla
- W Oosterlinck
- W Raby-Smith
- W Smolka
- W Van Houdt
- W Yang
- Willemijn van der Plas
- Wong Mpk
- X De Sousa
- X Morales
- X S Tan
- Y Aawsaj
- Y Al-Tamimi
- Y Arkha
- Y Ayasra
- Y Bashir
- Y El Bouazizi
- Y Fayed
- Y H Lam
- Y Kanemitsu
- Y Kara
- Y Kirmizi
- Y Levy-Zauberman
- Y Litvina
- Y Perez
- Y T Liew
- Y Tanase
- Y Viswanath
- Y Ying
- Z Al-Ishaq
- Z Aldayri
- Z Aliyeva
- Z Bayhan
- Z Chia
- Z Dzamic
- Z H Belkhadir
- Z Inic
- Z Jawad
- Z Jezdic
- Z Katusic
- Z Krivokapic
- Z Lakkis
- Z Li
- Z M Barrett-Brown
- Z Mahasin
- Z Seymour
- Z Vilendecic
- Z Zakaria
- Á De la Hoz Rodríguez
- Á Fernández Camuñas
- É Ryan
- Ž Grubač
- А Камалов
- Publication venue
- 'Wiley'
- Publication date
- 01/01/2020
- Field of study
Not availabl