95 research outputs found
Chikungunya virus (CHIKV) inhibitors from natural sources: a medicinal chemistry perspective
- Author
- AA Rashad
- AK Sachdeva
- D Parashar
- DA Case
- E Guantai
- FE Koehn
- G Molinari
- G Molinari
- GA Belov
- H Malet
- IH Chowdhury
- IP Singh
- J Mann
- JE Voss
- JW Li
- JWH Li
- K Hirneisen
- L Pohjala
- L-F Nothias-Scaglia
- M Bourjot
- M Bourjot
- M Bourjot
- M Lucas-Hourani
- Mahmoud E. S. Soliman
- MP Williamson
- N Corlay
- P Kaur
- P-M Allard
- PTV Nguyen
- RR Teixeira
- S Bhakat
- S Kothandan
- S Lee
- S Mondal
- Soumendranath Bhakat
- T Wells
- X Lamballerie de
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Phenylalanine-Rich Peptides Potently Bind ESAT6, a Virulence Determinant of Mycobacterium tuberculosis, and Concurrently Affect the Pathogen's Growth
- Author
- A Bhatt
- A Jain
- A Ojha
- A Rao
- A Rao
- Anamika Ghosh
- Anand Ranganathan
- AS Pym
- Azeet Narayan
- BJ Wards
- C Abou-Zeid
- C Cheadle
- C Dye
- CE Barry 3rd
- CM Sassetti
- CM Sassetti
- Deepti Gupta
- E Dubnau
- F Berthet
- G Schumann
- Geeta Ram
- GR Khatri
- IH Lee
- J Volmink
- Jameel Ahmad Khan
- JH Miller
- JR Schwebach
- JWS Backlock
- K Weldingh
- Krishan Kumar
- Krishnamurthy Natarajan
- Kuhulika Bhalla
- L Majlessi
- M Harboe
- Megha Tharad
- MG Sonnenberg
- MI de Jonge
- Niyaz Ahmed
- P Andersen
- P Brodin
- P Peake
- PS Renshaw
- PS Renshaw
- R Mondal
- R Provvedi
- R Qamra
- Rana Pratap
- S Aravinda
- S Nagai
- SA Stanley
- Sachin Kumar Samuchiwal
- SC Derrick
- Sushil Kumar
- Swetha Ganapathy
- T Hsu
- TD Schmittgen
- WW Yew
- Y Yuan
- Yogendra Singh
- Publication venue
- Public Library of Science
- Publication date
- 01/11/2009
- Field of study
BACKGROUND:The secretory proteins of Mycobacterium tuberculosis (M. tuberculosis) have been known to be involved in the virulence, pathogenesis as well as proliferation of the pathogen. Among this set, many proteins have been hypothesized to play a critical role at the genesis of the onset of infection, the primary site of which is invariably the human lung. METHODOLOGY/PRINCIPAL FINDINGS:During our efforts to isolate potential binding partners of key secretory proteins of M. tuberculosis from a human lung protein library, we isolated peptides that strongly bound the virulence determinant protein Esat6. All peptides were less than fifty amino acids in length and the binding was confirmed by in vivo as well as in vitro studies. Curiously, we found all three binders to be unusually rich in phenylalanine, with one of the three peptides a short fragment of the human cytochrome c oxidase-3 (Cox-3). The most accessible of the three binders, named Hcl1, was shown also to bind to the Mycobacterium smegmatis (M. smegmatis) Esat6 homologue. Expression of hcl1 in M. tuberculosis H37Rv led to considerable reduction in growth. Microarray analysis showed that Hcl1 affects a host of key cellular pathways in M. tuberculosis. In a macrophage infection model, the sets expressing hcl1 were shown to clear off M. tuberculosis in much greater numbers than those infected macrophages wherein the M. tuberculosis was not expressing the peptide. Transmission electron microscopy studies of hcl1 expressing M. tuberculosis showed prominent expulsion of cellular material into the matrix, hinting at cell wall damage. CONCLUSIONS/SIGNIFICANCE:While the debilitating effects of Hcl1 on M. tuberculosis are unrelated and not because of the peptide's binding to Esat6-as the latter is not an essential protein of M. tuberculosis-nonetheless, further studies with this peptide, as well as a closer inspection of the microarray data may shed important light on the suitability of such small phenylalanine-rich peptides as potential drug-like molecules against this pathogen
Search for Higgs Boson Pair Production in the Four b Quark Final State in Proton-Proton Collisions at root s=13 TeV
- Author
- Aarrestad T
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdullah WW
- Abdullin S
- Abercrombie D
- Abreu A
- Acharya H
- Acosta D
- Adam W
- Adamidis K
- Adams E
- Adams M
- Adams T
- Addesa F
- Adloff C
- Adzic P
- AdĂĄn DP
- Afanasiev S
- Agapitos A
- Agarwal G
- Aggleton R
- Agram J
- Aguilar-Benitez M
- Ahmad A
- Ahmad M
- Ahmad WH
- Ahmed A
- Ahuja S
- Aime` C
- Akchurin N
- Akgun B
- Akpinar A
- Albergo S
- Albert A
- Albrecht S
- Albrow M
- Aleksandrov A
- Alexander J
- Alhusseini M
- Alimena J
- Alison J
- Almond J
- Alonso AG
- Alpana K
- Alvarez JR
- Alverson G
- Alves G
- Aly R
- Alyari M
- Amapane N
- Amaral SSD
- Amarilo KM
- Ambrozas M
- Amendola C
- Amin N
- Amram O
- Amsler C
- An S
- An Y
- Anagnostou G
- Anampa KH
- Andrea J
- Andreassi G
- Andreev V
- Andreev Y
- Andrejkovic J
- Andrews M
- Androsov K
- Angioni GP
- Anguiano J
- Antchev G
- Antequera JB
- Anthony D
- Antunovic Z
- Anuar AB
- Apollinari G
- Apparu D
- Appelt E
- Apresyan A
- Apyan A
- Araujo M
- Arcaro D
- Arcidiacono R
- Arenton M
- Argiro S
- Arneodo M
- Aruta C
- Asavapibhop B
- Asawatangtrakuldee C
- Asenov P
- Asghar M
- Asilar E
- Askew A
- Asmuss P
- Atakisi I
- Attikis A
- Auffray E
- Aushev T
- Auzinger G
- Avati V
- Avery P
- Avila C
- Awais A
- Awan M
- Ayala E
- Ayala G
- Azarkin M
- Azhgirey I
- Aziz T
- Azzi P
- Azzurri P
- Baarmand M
- Babaev A
- Bacchetta N
- Bachiller I
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- Baechler J
- Bagliesi G
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- Baillon P
- Bainbridge R
- Bakas G
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- Bakshi A
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- Band R
- Bandyopadhyay H
- Banerjee S
- Banos LE
- Bansal S
- Barbagli G
- Barberis E
- Bargassa P
- Baringer P
- Barnes V
- Barney D
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- Barrera CB
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- Yu G
- Yu I
- Yu P
- Yu S
- Yuan L
- Yuan S
- Yuldashev B
- Yumiceva F
- Yusli M
- Yzquierdo AP
- Zabi A
- Zacharopoulou A
- Zahid S
- Zaleski S
- Zalewski P
- Zanetti M
- Zarubin A
- Zarucki M
- Zecchinelli A
- Zeinali M
- Zeuner W
- Zghiche A
- Zhang F
- Zhang H
- Zhang J
- Zhang L
- Zhang W
- Zhang Y
- Zhang Z
- Zhao J
- Zhizhin I
- Zhokin A
- Zhu D
- Zhu R
- Ziemons T
- Zoi I
- Zolkapli Z
- Zorbakir I
- Zorbilmez C
- Zotto P
- Zotz A
- Zou D
- Zou R
- Zucchetta A
- Zumerle G
- Zuo X
- Zuolo D
- Zygala L
- Ălvarez CR
- Ăzçelik Ă
- Publication venue
- Publication date
- 01/01/2022
- Field of study
Search for dark matter produced in association with a Higgs boson decaying to a pair of bottom quarks in proton-proton collisions at root s=13TeV
- Author
- Aarrestad TK
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdullah WATW
- Abdullin S
- Abercrombie D
- Acharya H
- Acosta D
- Acosta JG
- Adam W
- Adams E
- Adams MR
- Adams T
- Adloff C
- Adzic P
- AdĂĄn DP
- Afanasiev S
- Agapitos A
- Agarwal G
- Aggleton R
- Agram J-L
- Aguilar-Benitez M
- Ahmad A
- Ahmad M
- Ahmad WH
- Ahmed A
- Ahuja S
- Aime' C
- Akchurin N
- Akgun B
- Akpinar A
- Albajar C
- Albergo S
- Albert A
- Albrow M
- Aleksandrov A
- Alexander J
- Alhusseini M
- Alimena J
- Alison J
- Allen B
- Almond J
- Alonso AG
- Alvarez JDR
- Alverson G
- Alves GA
- Aly R
- Alyari M
- Amapane N
- Amaral SMSD
- Amendola C
- Amin N
- Amram O
- Amsler C
- Anagnostou G
- Anampa KH
- Anderson D
- Andrea J
- Andreev V
- Andreev Y
- Andrews MB
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- Angioni GLP
- Antchev G
- Antunovic Z
- Anuar AAB
- Apanasevich L
- Apollinari G
- Appelt E
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- Araujo M
- Arbelaez NV
- Arbol PMRD
- Arcaro D
- Arcidiacono R
- Arenton MW
- Argiro S
- Arneodo M
- Aruta C
- Asavapibhop B
- Asawatangtrakuldee C
- Asenov P
- Asghar MI
- Asilar E
- Askew A
- Asmuss P
- Atakisi IO
- Atanasov I
- Ather MW
- Attikis A
- Auffray E
- Aushev T
- Auzinger G
- Avati V
- Avery P
- Avila C
- Awan MIM
- Ayala E
- Ayala G
- Azarkin M
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- Dimitrov A
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- Dupont N
- Durgut S
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- Dutta D
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- Ecklund KM
- Eckstein D
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- Elmetenawee W
- Elvira VD
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- Ăzçelik Ă
- Publication venue
- Publication date
- 01/01/2018
- Field of study
A search for dark matter produced in association with a Higgs boson decaying to a pair of bottom quarks is performed in proton-proton collisions at a center-of-mass energy of 13 TeV collected with the CMS detector at the LHC. The analyzed data sample corresponds to an integrated luminosity of 35.9 fb(-1). The signal is characterized by a large missing transverse momentum recoiling against a bottom quark-antiquark system that has a large Lorentz boost. The number of events observed in the data is consistent with the standard model background prediction. Results are interpreted in terms of limits both on parameters of the type-2 two-Higgs doublet model extended by an additional light pseudoscalar boson a (2HDM+a) and on parameters of a baryonic Z simplified model. The 2HDM+a model is tested experimentally for the first time. For the baryonic Z model, the presented results constitute the most stringent constraints to date.Peer reviewe
A Deep Neural Network for Simultaneous Estimation of b Jet Energy and Resolution
- Author
- Aarrestad TK
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdalla H
- Abdullah WATW
- Abdullin S
- Abercrombie D
- Acharya H
- Acosta D
- Acosta JG
- Adam W
- Adams MR
- Adams T
- Adzic P
- AdĂĄn DP
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- Ăzçelik Ă
- Publication venue
- Publication date
- 01/01/2020
- Field of study
We describe a method to obtain point and dispersion estimates for the energies of jets arising from b quarks produced in proton-proton collisions at an energy of s = 13 TeV at the CERN LHC. The algorithm is trained on a large sample of simulated b jets and validated on data recorded by the CMS detector in 2017 corresponding to an integrated luminosity of 41 fb - 1 . A multivariate regression algorithm based on a deep feed-forward neural network employs jet composition and shape information, and the properties of reconstructed secondary vertices associated with the jet. The results of the algorithm are used to improve the sensitivity of analyses that make use of b jets in the final state, such as the observation of Higgs boson decay to b b ÂŻ
Search for invisible decays of the Higgs boson produced via vector boson fusion in proton-proton collisions at root s=13 TeV
- Author
- Aarrestad T
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdelalim A
- Abdullin S
- Abercrombie D
- Abreu A
- Acharya H
- Acosta D
- Acosta HE
- Adam W
- Adamidis K
- Adams E
- Adams M
- Adams T
- Addesa F
- Adloff C
- Adzic P
- AdĂĄn DP
- Afanasiev S
- Agapitos A
- Agarwal G
- Aggleton R
- Agram J
- Aguilar-Benitez M
- Ahmad A
- Ahmad M
- Ahmad WH
- Ahmed A
- Ahuja S
- AimĂš C
- Akchurin N
- Akgun B
- Akpinar A
- Albergo S
- Albert A
- Albrecht S
- Albrow M
- Aleksandrov A
- Alexander J
- Alhusseini M
- Alimena J
- Alison J
- Almond J
- Alonso AG
- Alpana A
- Alvarez JR
- Alverson G
- Alves BFS
- Alves G
- Aly R
- Alyari M
- Amapane N
- Amaral SSD
- Amarilo KM
- Ambrozas M
- Amendola C
- Amin N
- Amram O
- Amsler C
- An S
- An Y
- Anagnostou G
- Anampa KH
- Andrea J
- Andreassi G
- Andreev V
- Andreev Y
- Andrejkovic J
- Andrews M
- Androsov K
- Anguiano J
- Antchev G
- Antequera JB
- Anthony D
- Antunovic Z
- Anuar AB
- Apollinari G
- Apparu D
- Appelt E
- Apresyan A
- Apyan A
- Araujo M
- Arcaro D
- Arcidiacono R
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- Auzinger G
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- Baarmand M
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- Bachiller I
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- Bagliesi G
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- Bandyopadhyay H
- Banerjee S
- Banos LE
- Bansal S
- Barbagli G
- Barberis E
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- Ălvarez CR
- Ăzçelik Ă
- Publication venue
- Publication date
- 01/01/2022
- Field of study
Serological Surveillance Development for Tropical Infectious Diseases Using Simultaneous Microsphere-Based Multiplex Assays and Finite Mixture Models
- Author
- A Clavijo
- A Kulshrestha
- AK Ngugi
- AL Baughman
- Anne Wanjiru Mwangi
- AW Solomon
- B Yang
- BS Everitt
- Chihiro Tanigawa
- DA Vignali
- Dinesh Mondal
- DM Moss
- DS Watson
- DW Njomo
- E Kimura
- F Nakamura-Uchiyama
- F Qadri
- H Otsubo
- H Tachibana
- H Takagi
- HD Romero
- Hiroshi Tachibana
- Ibrahim Kiche
- IH Khan
- James Kimotho
- JW Gnann Jr
- JW Pickering
- K Ishii
- Kazunari Ishii
- Ken-ichi Kamo
- Kenji Hirayama
- KL Kotloff
- KV Rao
- Lay Myint Yoshida
- M Sakikawa
- M Yazdanbakhsh
- Makoto Itoh
- Mamiko Niki
- Manabu Inoue
- Masashi Miura
- Matilu Mwau
- Mayuko Osada-Oka
- MC Rota
- MM Levine
- Mohamed Karama
- MV Marlet
- Mwatasa Changoma
- Patrick J. Lammie
- PJ Hotez
- PJ Hotez
- PJ Lammie
- Rashidul Haque
- S Dissanayake
- S Kaneko
- Sammy M. Njenga
- Samson Muuo Nzou
- Satoshi Kaneko
- Shinjiro Hamano
- SM Griffin
- SM Njenga
- Sohkichi Matsumoto
- T Waterboer
- Takafumi Tsuboi
- Tomonori Hoshi
- WJ Youden
- Yoshio Ichinose
- Yoshito Fujii
- YY Go
- Z Bentwich
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- 31/07/2014
- Field of study
Background:A strategy to combat infectious diseases, including neglected tropical diseases (NTDs), will depend on the development of reliable epidemiological surveillance methods. To establish a simple and practical seroprevalence detection system, we developed a microsphere-based multiplex immunoassay system and evaluated utility using samples obtained in Kenya.Methods:We developed a microsphere-based immuno-assay system to simultaneously measure the individual levels of plasma antibody (IgG) against 8 antigens derived from 6 pathogens: Entamoeba histolytica (C-IgL), Leishmania donovani (KRP42), Toxoplasma gondii (SAG1), Wuchereria bancrofti (SXP1), HIV (gag, gp120 and gp41), and Vibrio cholerae (cholera toxin). The assay system was validated using appropriate control samples. The assay system was applied for 3411 blood samples collected from the general population randomly selected from two health and demographic surveillance system (HDSS) cohorts in the coastal and western regions of Kenya. The immunoassay values distribution for each antigen was mathematically defined by a finite mixture model, and cut-off values were optimized.Findings:Sensitivities and specificities for each antigen ranged between 71 and 100%. Seroprevalences for each pathogen from the Kwale and Mbita HDSS sites (respectively) were as follows: HIV, 3.0% and 20.1%; L. donovani, 12.6% and 17.3%; E. histolytica, 12.8% and 16.6%; and T. gondii, 30.9% and 28.2%. Seroprevalences of W. bancrofti and V. cholerae showed relatively high figures, especially among children. The results might be affected by immunological cross reactions between W. bancrofti-SXP1 and other parasitic infections; and cholera toxin and the enterotoxigenic E. coli (ETEC), respectively.Interpretation:A microsphere-based multi-serological assay system can provide an opportunity to comprehensively grasp epidemiological features for NTDs. By adding pathogens and antigens of interest, optimized made-to-order high-quality programs can be established to utilize limited resources to effectively control NTDs in Africa
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Measurement of the differential ttÂŻ production cross section as a function of the jet mass and extraction of the top quark mass in hadronic decays of boosted top quarks
- Author
- Aarrestad TK
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdalla H
- Abdullin S
- Abercrombie D
- Abreu A
- Acharya H
- Acosta D
- Acosta HAE
- Adam W
- Adamidis K
- Adams E
- Adams MR
- Adams T
- Addesa FM
- Adloff C
- Adzic P
- AdĂĄn DP
- Afanasiev S
- Agapitos A
- Agarwal G
- Agram J-L
- Aguilar-Benitez M
- Agyel D
- Ahmad A
- Ahmad M
- Ahmad WH
- Ahmed A
- AimĂš C
- Akchurin N
- Akgun B
- Akpinar A
- Albert A
- Albrecht A
- Albrecht S
- Albrow M
- Alcerro LFA
- Aleksandrov A
- Alexander J
- Alhusseini M
- Alimena J
- Alison J
- Allmond B
- Almond J
- Alonso AG
- Alpana A
- Alvarez JDR
- Alverson G
- Alves BAFS
- Alves GA
- Aly R
- Alyari M
- Amapane N
- Amaral SMSD
- Amarilo KM
- Ambrozas M
- Amendola C
- Amin N
- Amram O
- Amsler C
- An S
- An Y
- Anagnostou G
- Anampa KH
- Andrea J
- Andreev V
- Andreev Y
- Andrejkovic JW
- Andrews MB
- Androsov K
- Anguiano J
- Antchev G
- Anthony D
- Antonello M
- Antunovic Z
- Anuar AAB
- Apollinari G
- Apparu D
- Appelt E
- Apresyan A
- Araujo M
- Arbol PMRD
- Arcaro D
- Arcidiacono R
- Argiro S
- Arneodo M
- Aruta C
- Asawatangtrakuldee C
- Asenov P
- Asghar MI
- Asilar E
- Askew A
- Asmuss P
- Assiouras P
- Assran Y
- Atakisi IO
- Attikis A
- Auffray E
- Aushev T
- Auzinger G
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- Avila C
- Awais A
- Awan MIM
- Ayala E
- Ayala G
- Aydilek O
- Azarkin M
- Aziz T
- Azzi P
- Azzurri P
- Baarmand MM
- Babaev A
- Babbar J
- Bacchetta N
- Bachtis M
- Backhaus M
- Baden A
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- Yumiceva F
- Yusuff I
- Yzquierdo AP-C
- Zabi A
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- Zaleski S
- Zalewski P
- Zanetti M
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- Zecchinelli AG
- Zeid SA
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- Zoi I
- Zolkapli Z
- Zorbakir IS
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- Zumerle G
- Zuo X
- Zuolo D
- Zygala L
- Ălvarez CR
- Publication venue
- Springer Nature
- Publication date
- 03/07/2023
- Field of study
Data Availability:
This manuscript has no associated data or the data will not be deposited. [Authorsâ comment: Release and preservation of data used by the CMS Collaboration as the basis for publications is guided by the CMS policy as stated in https://cms-docdb.cern.ch/cgibin/PublicDocDB/RetrieveFile?docid=6032 &filename=CMSDataPolicyV1.2.pdf &version=2.]A measurement of the jet mass distribution in hadronic decays of Lorentz-boosted top quarks is presented. The measurement is performed in the lepton + jets channel of top quark pair production (ttÂŻ
) events, where the lepton is an electron or muon. The products of the hadronic top quark decay are reconstructed using a single large-radius jet with transverse momentum greater than 400GeV
. The data were collected with the CMS detector at the LHC in proton-proton collisions and correspond to an integrated luminosity of 138fbâ1
. The differential ttÂŻ
production cross section as a function of the jet mass is unfolded to the particle level and is used to extract the top quark mass. The jet mass scale is calibrated using the hadronic W boson decay within the large-radius jet. The uncertainties in the modelling of the final state radiation are reduced by studying angular correlations in the jet substructure. These developments lead to a significant increase in precision, and a top quark mass of 173.06±0.84GeV.SCOAP
Recommended from our members
Precision measurement of the W boson decay branching fractions in proton-proton collisions at âs=13 TeV
- Author
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- Yumiceva F
- Yusli MN
- Yzquierdo AP-C
- Zabi A
- Zacharopoulou A
- Zahid S
- Zaleski S
- Zalewski P
- Zanetti M
- Zarubin A
- Zarucki M
- Zecchinelli AG
- Zeinali M
- Zeuner WD
- Zghiche A
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- Zhizhin I
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- Zoi I
- Zolkapli Z
- Zorbakir IS
- Zorbilmez C
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- Zou D
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- Zumerle G
- Zuo X
- Zuolo D
- Zygala L
- Ălvarez CR
- Ăzçelik Ă
- Publication venue
- 'American Physical Society (APS)'
- Publication date
- 26/04/2022
- Field of study
The leptonic and inclusive hadronic decay branching fractions of the W boson are measured using
proton-proton collision data collected at ffiffi s p Œ 13 TeV by the CMS experiment at the CERN LHC,
corresponding to an integrated luminosity of 35.9 fbâ1. Events characterized by the production of one or
two W bosons are selected and categorized based on the multiplicity and flavor of reconstructed leptons, the
number of jets, and the number of jets identified as originating from the hadronization of b quarks. A
binned maximum likelihood estimate of the W boson branching fractions is performed simultaneously in
each event category. The measured branching fractions of the W boson decaying into electron, muon, and
tau lepton final states are Ă°10.83 0.10Ă%, Ă°10.94 0.08Ă%, and Ă°10.77 0.21Ă%, respectively,
consistent with lepton flavor universality for the weak interaction. The average leptonic and inclusive
hadronic decay branching fractions are estimated to be Ă°10.89 0.08Ă% and Ă°67.32 0.23Ă%, respec tively. Based on the hadronic branching fraction, three standard model quantities are subsequently derived: the sum of squared elements in the first two rows of the CabibboâKobayashiâMaskawa (CKM) matrix
P ij jVijj 2 Œ 1.984 0.021, the CKM element jVcsj Œ 0.967 0.011, and the strong coupling constant at
the W boson mass scale, αSĂ°m2 WĂ ÂŒ 0.095 0.033
- âŠ