11 research outputs found
A Steered Molecular Dynamics Study of Binding and Translocation Processes in the GABA Transporter
- Author
- A Bendahan
- A Rosenberg
- A Schousboe
- A Yamashita
- AK Meinild
- BI Kanner
- BI Kanner
- BK Mai
- C Braestrup
- C Jarzynski
- C Jarzynski
- CL Piscitelli
- DP Claxton
- E Zomot
- ER Bennett
- F Cherubino
- Flemming Steen JĂžrgensen
- G Forlani
- GI Keshet
- GZ Genchev
- H Grubmuller
- Heinrich Sticht
- J Andersen
- J Shan
- JR Dodd
- KJ Bowers
- KK Madsen
- KK Madsen
- L Celik
- L Celik
- L Shi
- Laurent David
- LK Henry
- LLC Schrodinger
- LLC Schrödinger
- LR Forrest
- M Quick
- M Sotomayor
- MO Jensen
- N Hansra
- N Kleinberger-Doron
- N MacAulay
- N Melamed
- N Yu
- Olivier Taboureau
- RE Amaro
- Research D. E. Shaw
- RP Clausen
- RP Clausen
- S Mager
- S Pantanowitz
- S Skovstrup
- S Tamura
- SK Singh
- SK Singh
- SL Deken
- SĂžren Skovstrup
- U Gether
- W Humphrey
- Y Bismuth
- Y Zhao
- Y Zhou
- Z Zhou
- Z Zhou
- Publication venue
- Public Library of Science
- Publication date
- 01/01/2012
- Field of study
The entire substrate translocation pathway in the human GABA transporter (GAT-1) was explored for the endogenous substrate GABA and the anti-convulsive drug tiagabine. Following a steered molecular dynamics (SMD) approach, in which a harmonic restraining potential is applied to the ligand, dissociation and re-association of ligands were simulated revealing events leading to substrate (GABA) translocation and inhibitor (tiagabine) mechanism of action. We succeeded in turning the transporter from the outward facing occluded to the open-to-out conformation, and also to reorient the transporter to the open-to-in conformation. The simulations are validated by literature data and provide a substrate pathway fingerprint in terms of which, how, and in which sequence specific residues are interacted with. They reveal the essential functional roles of specific residues, e.g. the role of charged residues in the extracellular vestibule including two lysines (K76 (TM1) and K448 (TM10)) and a TM6-triad (D281, E283, and D287) in attracting and relocating substrates towards the secondary/interim substrate-binding site (S2). Likewise, E101 is highlighted as essential for the relocation of the substrate from the primary substrate-binding site (S1) towards the cytoplasm
Erratum to: Comparison of the Z/Îł* + jets to Îł + jets cross sections in pp collisions at âs = 8
- Author
- Aarrestad TK
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdullah WATW
- Abdullin S
- Abdulsalam A
- Abu Zeid S
- Ackert A
- Acosta D
- Acosta JG
- Acosta MV
- Adair A
- Adam W
- Adams JR
- Adams MR
- Adams T
- Adiguzel A
- Adzic P
- Afanasiev S
- Agapitos A
- Aggleton R
- Agram J-L
- Ahmad A
- Ahmad M
- Ahmad M
- Ahmad WH
- Ahuja S
- Akbiyik M
- Akchurin N
- Akgun B
- Akin IV
- Albajar C
- Albayrak EA
- Albrow M
- Alcaraz Maestre J
- Alderweireldt S
- Aleksandrov A
- Alexander J
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- Alimena J
- Alvarez JDR
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- Alves GA
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- Aly S
- Alyari M
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- Anagnostou G
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- Zagozdzinska A
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- Publication venue
- 'Springer Fachmedien Wiesbaden GmbH'
- Publication date
- 01/04/2016
- Field of study
Erratum to: JHEP10(2015)128. ArXiv ePrint: 1505.06520. The online version of the original article can be found at http://dx.doi.org/10.1007/JHEP10(2015)128
Inclusive and differential measurements of the t(t)over-bar charge asymmetry in pp collisions at root s=8 TeV
- Author
- -Fernandez RL
- -Hernandez AS
- Aarrestad TK
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdelalim AA
- Abdullah WATW
- Abdullin S
- Abdulsalam A
- Abu Zeid S
- Ackert A
- Acosta D
- Acosta JG
- Acosta MV
- Adair A
- Adam W
- Adams JR
- Adams MR
- Adams T
- Adiguzel A
- Adzic P
- Afanasiev S
- Agapitos A
- Aggleton R
- Agram J-L
- Ahmad A
- Ahmad M
- Ahmad M
- Ahmed I
- Ahuja S
- Akbiyik M
- Akchurin N
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- Vorobyev A
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- Walczak M
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- Wallny R
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- Wang Z
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- Wasserbaech S
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- Wittmer B
- Woehrmann C
- Wohri HK
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- Wolfe E
- Womersley WJ
- Won S
- Wood D
- Wood J
- Wood JS
- Woodard A
- Woods N
- Worm SD
- Wright D
- Wu Z
- Wulsin HW
- Wulz C-E
- Wurthwein F
- Wyslouch B
- Xia F
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- Xiao M
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- Xu Z
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- Yazgan E
- Yelton J
- Yetkin T
- Yi K
- Yilmaz Y
- Yin H
- Yohay R
- Yonamine R
- Yoo HD
- Yoo J
- York A
- You C
- Yu I
- Yu SS
- Yumiceva F
- Yusli MN
- Zabel J
- Zabi A
- Zablocki J
- Zaganidis N
- Zagozdzinska A
- Zakaria M
- Zalewski P
- Zanetti A
- Zanetti M
- Zarubin A
- Zeinali M
- Zenoni F
- Zenz SC
- Zeuner WD
- Zeyrek M
- Zghiche A
- Zhang F
- Zhang H
- Zhang J
- Zhokin A
- Zhu RY
- Zhukov V
- Zhukova V
- Zorbilmez C
- Zotto P
- Zou D
- Zou W
- Zsigmond AJ
- Zucchetta A
- Zumerle G
- Zuranski A
- Publication venue
- ELSEVIER SCIENCE BV
- Publication date
- 10/06/2016
- Field of study
The charge asymmetry is measured in protonâproton collisions at a centre-of-mass energy of . The data, collected with the CMS experiment at the LHC, correspond to an integrated luminosity of 19.7 fbâ1. Selected events contain an electron or a muon and four or more jets, where at least one jet is identified as originating from b-quark hadronization. The inclusive charge asymmetry is found to be . In addition, differential charge asymmetries as a function of rapidity, transverse momentum, and invariant mass of the system are studied. For the first time at the LHC, the measurements are also performed in a reduced fiducial phase space of top quark pair production, with an integrated result of . All measurements are consistent within two standard deviations with zero asymmetry as well as with the predictions of the standard model
Multi-omics facilitated variable selection in Cox-regression model for cancer prognosis prediction
- Publication venue
- Publication date
- 01/07/2017
- Field of study
Motivation New developments in high-throughput genomic technologies have enabled the measurement of diverse types of omics biomarkers in a cost-efficient and clinically-feasible manner. Developing computational methods and tools for analysis and translation of such genomic data into clinically-relevant information is an ongoing and active area of investigation. For example, several studies have utilized an unsupervised learning framework to cluster patients by integrating omics data. Despite such recent advances, predicting cancer prognosis using integrated omics biomarkers remains a challenge. There is also a shortage of computational tools for predicting cancer prognosis by using supervised learning methods. The current standard approach is to fit a Cox regression model by concatenating the different types of omics data in a linear manner, while penalty could be added for feature selection. A more powerful approach, however, would be to incorporate data by considering relationships among omics datatypes. Methods Here we developed two methods: a SKI-Cox method and a wLASSO-Cox method to incorporate the association among different types of omics data. Both methods fit the Cox proportional hazards model and predict a risk score based on mRNA expression profiles. SKI-Cox borrows the information generated by these additional types of omics data to guide variable selection, while wLASSO-Cox incorporates this information as a penalty factor during model fitting. Results We show that SKI-Cox and wLASSO-Cox models select more true variables than a LASSO-Cox model in simulation studies. We assess the performance of SKI-Cox and wLASSO-Cox using TCGA glioblastoma multiforme and lung adenocarcinoma data. In each case, mRNA expression, methylation, and copy number variation data are integrated to predict the overall survival time of cancer patients. Our methods achieve better performance in predicting patientsâ survival in glioblastoma and lung adenocarcinoma. © 201
Molecular dynamics provides new insights into the mechanism of calcium signal transduction and interdomain interactions in cardiac troponin
- Author
- Aprahamian ML
- Baryshnikova OK
- Bernstein FC
- Bowman JD
- Brown JH
- Coldren WH
- Craig R
- Digel J
- Dong WJ
- Dvornikov AV
- Evenas J
- Evenas J
- Gagne SM
- Gagne SM
- Genchev GZ
- Genchev GZ
- Gillis TE
- Houdusse A
- Humphrey W
- Jaquet K
- Jayasundar JJ
- Jorgensen WL
- Kobayashi C
- Kobayashi T
- Kobayashi T
- Kobayashi T
- Kowlessur D
- Li MX
- Li MX
- Lin YH
- Lindert S
- Lindert S
- Lindert S
- Lu H
- Luo Y
- MacKerell AD
- Manning EP
- Marston S
- Mirny LA
- Nagy L
- Pearlstone JR
- Phillips JC
- PinedaâSanabria SE
- Robertson IM
- Sia SK
- Slupsky CM
- Stevens CM
- Strynadka NC
- Szatkowski L
- Takeda S
- Tardiff JC
- Varughese JF
- Vinogradova MV
- Yamada Y
- Publication venue
- 'Wiley'
- Publication date
- Field of study
Accelerated Molecular Dynamics and Protein Conformational Change: A Theoretical and Practical Guide Using a Membrane Embedded Model Neurotransmitter Transporter
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Evaluations of physicochemical and anti-oxidant properties of powdered leaves from lotus, shepherdâs purse and goldenrod in restructured duck/pork patties
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Molecular Dynamics Simulations of the Cardiac Troponin Complex Performed with FRET Distances as Restraints
- Author
- A Babu
- A Fiser
- A Fiser
- A Pirani
- A Schmidtmann
- AC Wallace
- AJ Franklin
- AM Gordon
- C Sheldahl
- CA Parker
- CG dos Remedios
- CS Farah
- D Kowlessur
- D Ritchie
- DA Parry
- E Lindahl
- E Potterton
- EP Manning
- G Vriend
- GZ Genchev
- HE Huxley
- Herbert C. Cheung
- HJC Berendsen
- J Xing
- Jayant James Jayasundar
- JC Haselgrove
- JD Potter
- JF Varughese
- Jie Zheng
- JM Robinson
- John M. Robinson
- JP Jin
- Jun Xing
- JW Howarth
- L Potterton
- L Spyracopoulos
- LB Smillie
- M Chandra
- MB Abbott
- MJ Calvert
- MV Vinogradova
- MX Li
- NM Cordina
- NM Cordina
- RA Sayle
- S Ebashi
- S Ramakrishnan
- S Takeda
- SP Robertson
- T Kobayashi
- V Gaponenko
- W-J Dong
- Wen-Ji Dong
- WJ Dong
- WJ Dong
- WJ Dong
- WJ Dong
- WJ Dong
- WJ Dong
- Z Dobrowolski
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- Field of study
Study of protein structural deformations under external mechanical perturbations by a coarse-grained simulation method
- Author
- A Wlodawer
- AR Atilgan
- AW Orr
- B Isralewitz
- B Liu
- B Liu
- BB Lim
- BR Care
- C Clementi
- C Hardin
- C Hyeon
- C Hyeon
- C Zhang
- CC DuFort
- CW Cairo
- DE Ingber
- DK Klimov
- DR Critchley
- DR Fooksman
- EH Lee
- EM Balzer
- F Cailliez
- F Cailliez
- F Rico
- GA Jeffrey
- GH Li
- GZ Genchev
- H Lu
- H Zhou
- HS Martin
- I Kostetskii
- J Chen
- J Hsin
- J Karanicolas
- J Karanicolas
- J Ma
- J Ma
- Jiawen Chen
- JS Patel
- K Burridge
- K Manibog
- K Svoboda
- KC Marshall
- KM Ravikumar
- M Cieplak
- M Cieplak
- M Gao
- M Karplus
- M Knott
- M Rief
- M Sotomayor
- M Sotomayor
- M Sotomayor
- M Sotomayor
- M Yao
- MA Schwartz
- MA Schwartz
- MM Martino
- N Koga
- NC Hartman
- OH Willemsen
- PA Janmey
- R Merkel
- RD Hills Jr
- S Improta
- S Kalyaanamoorthy
- S Wu
- S Yang
- T Ha
- TJ Boggon
- V Barsegov
- V Labrador
- VP Hytonen
- W Kabsch
- W Zheng
- W Zheng
- YH Wu
- Yinghao Wu
- YV Pereverzev
- Zhong-Ru Xie
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Introduction
- Author
- Aarrestad TK
- Abbaneo D
- Abbiendi G
- Abbrescia M
- Abdullah WATW
- Abdullin S
- Abdulsalam A
- Abu Zeid S
- Ackert A
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- Acosta JG
- Acosta MV
- Adair A
- Adam W
- Adams JR
- Adams MR
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- Adiguzel A
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- Agapitos A
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- Ahmad A
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- Alderweireldt S
- Aleksandrov A
- Alexander J
- Ali A
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- Alverson G
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- Anderson D
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- Publication venue
- Publication date
- 01/01/2013
- Field of study
In the original paper, the wrong plot was used in figure 6. The correct figure is given below. (figure presented.)