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7 research outputs found
Design, Synthesis, and Biological Evaluation of a New Series of Biphenyl/Bibenzyl Derivatives Functioning as Dual Inhibitors of Acetylcholinesterase and Butyrylcholinesterase
Author
Ai-lin Liu
Bo Feng
+6Â more
Dong-mei Wang
Guan-hua Du
Hui Fu
Lin Wang
Schelterns
Song Wu
Publication venue
'MDPI AG'
Publication date
Field of study
No full text
Crossref
3′-R/S-Hydroxyvoacamine, a potent acetylcholinesterase inhibitor from Tabernaemontana divaricata
Author
Braga
Chattipakorn
+33Â more
Ellman
Farfara
Greig
Henriques
Howes
I.C.H. Guideline
Ingkaninan
Ingkaninan
Jan Schripsema
Johnson
Kam
Kam
Kam
Kornkanok Ingkaninan
Lefèvre
Mercier
Mukherjee
Nakdook
Neddermeyer
Perera
Pratchayasakul
Rhee
Schelterns
Selkoe
Siriporn Okonogi
Snyder
Van Beek
Van Beek
Van Beek
Wantida Chaiyana
Wentrup
Winblad
Zhao
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Synthesis and evaluation of 6-substituted 3-arylcoumarin derivatives as multifunctional acetylcholinesterase/monoamine oxidase B dual inhibitors for the treatment of Alzheimer’s disease
Author
Alonso
Asadipour
+53Â more
Axelsen
Binda
Bolea
Castro
Chen
Desideri
Di
Ellman
Ghosh
Goedert
Hardy
Jakob-Roetne
Jones
Jucker
Kumar
Lan
LeĂłn
Lu
Lu
LĂłpez
Matos
Miller
Mitoma
Naiki
Novaroli
Pan
Piazzi
Pisani
Polinsky
Ramsay
Rizzo
Rosini
Samadi
Schelterns
Scott
Son
Soto-Ortega
Stege
Sterling
Suzuki
Talesa
Tumiatti
Viña
Wang
Wang
Watkins
Weyler
Xie
Xie
Xu
Youdim
Zheng
Zhou
Publication venue
'Royal Society of Chemistry (RSC)'
Publication date
01/01/2015
Field of study
No full text
Crossref
Multitarget drug design strategy against Alzheimer’s disease: Homoisoflavonoid Mannich base derivatives serve as acetylcholinesterase and monoamine oxidase B dual inhibitors with multifunctional properties
Author
Agis-Torres
Carradori
+54Â more
Da Prada
Da Silva
Desideri
Di
Dávalos
Engelbrecht
Fang
Foroumadi
Fu Su
Gan
Ganyuan Xiao
He
Hou
Huang
Huang
Inestrosa
Kontogiorgis
Kurt
Legoabe
Li
Li
Li Luo
Liu
Lu
Matos
Maynard
Mostofi
Nepovimova
Novaroli
Park
Patil
Qiang
Roman
Roy
Sang
Sang
Schelterns
Shaikh
Sharma
Siddaiah
Strydom
Sun
Tanada
Wang
Wilhelm
Xia Yang
Xiaoming Qiang
Yan Li
Yang
Yong Deng
Yunxiaozhu Zheng
Zheng
Zhipei Sang
Zhongcheng Cao
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Comparative study of selective in vitro and in silico BACE1 inhibitory potential of glycyrrhizin together with its metabolites, 18α- and 18β-glycyrrhetinic acid, isolated from Hizikia fusiformis
Author
A Kurz
Aditi Wagle
+53Â more
Alzheimer’s Association
Bing Tian Zhao
BM Jung
C Fiore
CC Tan
D Langer
D Zou
GA Tolstikov
GL Ellman
GR Fenwick
GW Huh
H Lineweaver
H Sugimoto
HA Jung
Hyun Ah Jung
J Cinatl
J Folch
J Hardy
Jae Sue Choi
JG Koo
JH Kim
K Mizoguchi
K Zhao
KE Park
KI Kim
L Luo
M Damle
M Wu
MA Farag
Mi Hee Woo
MN Asl
MW Sung
MY Ali
P Link
P Schelterns
P Seeman
PT Francis
R Karawita
R Khan
S Sen
S Takeda
SJ Pang
SS Eteghad
Su Hui Seong
T Akao
T Akao
T Ishida
WJ Geldenhuys
Y Yamamura
YR Han
Z Ma
Z Wang
ZQ Shao
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Computational exploration and experimental validation to identify a dual inhibitor of cholinesterase and amyloid-beta for the treatment of Alzheimer’s disease
Author
A Tripathi
AD MacKerell Jr
+54Â more
B Klimova
D Shivakumar
EK Perry
FH Darras
G Kryger
GL Ellman
GM Sastry
H Lineweaver
I Manoharan
IIIH Levine
J Cheung
J Hartmann
K Iqbal
L Peauger
L Santarpia
LS Goodman
LS Schneider
M Carmo Carreiras
M Dixon
M Kontoyianni
MA Silva
MA Smith
MF Eskander
MP Jacobson
MS Albert
N Kandiah
NC Inestrosa
NC Inestrosa
ND Heindel
NH Greig
P Mishra
P Schelterns
P Sharma
P Sharma
P Sharma
P Sharma
P Srivastava
P Srivastava
PN Tripathi
PN Tripathi
R Bullock
R Cacabelos
R Wang
RA Friesner
RM Lane
RN Kalaria
RS Wilson
S Agatonovic-Kustrin
SK Shrivastava
SN Dighe
SS More
W Luo
X-h Gao
Y Xu
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
In silico modeling for dual inhibition of acetylcholinesterase (AChE) and butyrylcholinesterase (BuChE) enzymes in Alzheimer’s disease
Author
Achintya Saha
Ahmad
+150Â more
Ahmad
Ahmed
Anand
Anand
Andreani
Awasthi
Bacalhau
Bagheri
Barreiro
Bolognesi
Bukhari
Buldurun
Camps
Cardoso
Carlier
Carlier
Ceschi
Cho
Conejo-GarcĂa
Contreras
Czarnecka
da Costa
Das
Das
De Souza
DeBernardis
Decker
Decker
dos Santos
Du
Ekins
Ercan
Erlanson
Fang
Fang
Feng
Feng
Fink
Ganeshpurkar
Girisha
Gray
Gregor
Hameed
Hameed
Han
Hasan
He
Hu
Hu
Huang
Huang
Högenauer
Ishihara
Jaén
Jia
Jiang
Kanhed
Kapples
Kavitha
Khan
Komersova
Krátký
Krátký
Kumar
Kumar
Kumar
Kunal Roy
Kurt
Leader
Leng
Leonard
Li
Li
Li
Li
Li
Lin
Liston
Liu
Luo
Mauri
McKenna
Minitab IN
Mohamed
Mohammadi
Morini
Mouchlis
Murzin
Najafi
Nekoei
Nordberg
Orhan
Pal
Pang
Pool
Pouramiri
RodrĂguez
RodrĂguez-Franco
Roy
Roy
Rydberg
Sadashiva
Saeed
Saeedi
Samadi
Samadi
Sang
Sang
Sang
Sarfraz
Schelterns
Shao
Shen
Sheng
Sheng
Sheng
Shi
Shi
Shi
Shinada
Shrivastava
Shutske
Simoni
Skrzypek
Sterling
Sugimoto
Sugimoto
Szymański
Tang
Taslimi
Tropsha
TĂĽrkan
Valenti
Veerasamy
Vidaluc
Vidaluc
Villalobos
Vinay Kumar
Wen
Wong
Yang
Yanovsky
Yap
YurttaĹź
Zakhari
ZelĂk
Zeng
Zhan
Zheng
Zhu
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref