15 research outputs found
Structural Features Underlying Raloxifene’s Biophysical Interaction with Bone Matrix
- Author
- Publication venue
- 'Elsevier BV'
- Publication date
- 01/02/2016
- Field of study
Raloxifene, a selective estrogen receptor modulator (SERM), reduces fracture risk at least in part by improving the mechanical properties of bone in a cell- and estrogen receptor-independent manner. In this study, we determined that raloxifene directly interacts with the bone tissue. Through the use of multiple and complementary biophysical techniques including nuclear magnetic resonance (NMR) and Fourier transform infrared spectroscopy (FTIR), we show that raloxifene interacts specifically with the organic component or the organic/mineral composite, and not with hydroxyapatite. Structure–activity studies reveal that the basic side chain of raloxifene is an instrumental determinant in the interaction with bone. Thus, truncation of portions of the side chain reduces bone binding and also diminishes the increase in mechanical properties. Our results support a model wherein the piperidine interacts with bone matrix through electrostatic interactions with the piperidine nitrogen and through hydrophobic interactions (van der Waals) with the aliphatic groups in the side chain and the benzothiophene core. Furthermore, in silico prediction of the potential binding sites on the surface of collagen revealed the presence of a groove with sufficient space to accommodate raloxifene analogs. The hydroxyl groups on the benzothiophene nucleus, which are necessary for binding of SERMs to the estrogen receptor, are not required for binding to the bone surface, but mediate a more robust binding of the compound to the bone powder. In conclusion, we report herein a novel property of raloxifene analogs that allows them to interact with the bone tissue through potential contacts with the organic matrix and in particular collagen
Global patient outcomes after elective surgery: prospective cohort study in 27 low-, middle- and high-income countries.
- Author
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- Ab Rahman AS
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- Zsisku L
- Publication venue
- 'Oxford University Press (OUP)'
- Publication date
- 01/01/2016
- Field of study
BACKGROUND: As global initiatives increase patient access to surgical treatments, there remains a need to understand the adverse effects of surgery and define appropriate levels of perioperative care. METHODS: We designed a prospective international 7-day cohort study of outcomes following elective adult inpatient surgery in 27 countries. The primary outcome was in-hospital complications. Secondary outcomes were death following a complication (failure to rescue) and death in hospital. Process measures were admission to critical care immediately after surgery or to treat a complication and duration of hospital stay. A single definition of critical care was used for all countries. RESULTS: A total of 474 hospitals in 19 high-, 7 middle- and 1 low-income country were included in the primary analysis. Data included 44 814 patients with a median hospital stay of 4 (range 2-7) days. A total of 7508 patients (16.8%) developed one or more postoperative complication and 207 died (0.5%). The overall mortality among patients who developed complications was 2.8%. Mortality following complications ranged from 2.4% for pulmonary embolism to 43.9% for cardiac arrest. A total of 4360 (9.7%) patients were admitted to a critical care unit as routine immediately after surgery, of whom 2198 (50.4%) developed a complication, with 105 (2.4%) deaths. A total of 1233 patients (16.4%) were admitted to a critical care unit to treat complications, with 119 (9.7%) deaths. Despite lower baseline risk, outcomes were similar in low- and middle-income compared with high-income countries. CONCLUSIONS: Poor patient outcomes are common after inpatient surgery. Global initiatives to increase access to surgical treatments should also address the need for safe perioperative care. STUDY REGISTRATION: ISRCTN5181700
Conformational analysis of phosphine ligands, using molecular mechanics and cone angle calculations
- Author
- Publication venue
- Publication date
- 01/01/1988
- Field of study
An empirical approach to the study of phosphine compounds was completed using Molecular Mechanics 2 (MM2), and several computer programs written to descibe and analyze the final geometric orientations of the molecules. The calculations were performed on 64 conformers of 16 different phosphines. Results from these calculations were compared to those previously obtained for MNDO and MINDO/3 calculations, and to experimental data. Cone angles calculated from the MM2 optimized geometries, were compared to Tolman's original work, and to values obtained from semiempirical calculations, and to experimental results. In general, it was found that weighted average cone angles best represent the size of phosphine ligands.Thesis (M.S.)Department of Chemistr
Corrigendum to “Structural features underlying raloxifene’s biophysical interaction with bone matrix” [Bioorg. Med. Chem. 24 (2016) 759–767]
- Author
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Kuluttajabarometri maakunnittain 2000, 2. neljännes
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- Yuliana A
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- Zamudio D
- Zangrillo A
- Zapata DDM
- Zbitnew G
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- Zoerner F
- Zonneveldt H
- Zou X
- Zoulamoglou M
- Zsisku L
- Publication venue
- Tilastokeskus
- Publication date
- 11/07/2000
- Field of study
Suomen virallinen tilasto (SVT
Use of failure-to-rescue to identify international variation in postoperative care in low-, middle- and high-income countries: a 7-day cohort study of elective surgery
- Author
- Ab Majid MA
- Ab Rahman AS
- Ab Rahman R
- Abayasinghe C
- Abbott T
- Abdullah NH
- Abdur-Rahman L
- Abeloos J
- Abernethy C
- Abidin UN
- Abrunhosa A
- Absar M
- Adam S
- Adams D
- Adams G
- Adamson M
- Adekola O
- Adelaja Y
- Ademola A
- Adenekan A
- Adenike O
- Adeolu AA
- Adetoye A
- Adewale B
- Adigun T
- Adolfsson A
- Aflori L
- Africander C
- Afshari A
- Agarwal V
- Agodirin O
- Aguero Vera M
- Aguzzoli C
- Ahmad A
- Ahmad N
- Ahmad T
- Ahmad T
- Ahmad Y
- Ahmed A
- Ahmed J
- Ai Y
- Aignatoaie M
- Aimoniotou-Georgiou E
- Akanmu O
- Akerman N
- Akinwale M
- Akring I
- Al 'Amri K
- Al Anizi M
- Al hussaini S
- Al-Soudaine Y
- Aladin H
- Alagbe-Briggs O
- Alaman Laguarda G
- Albaj S
- Alcock D
- Alcock L
- Aldecoa C
- Aldecoa C
- Aleixo FB
- Alexander H
- Alexander M
- Alexander-Sefre F
- Alherz F
- Ali H
- Ali M
- Ali S
- Alias A
- Alias AH
- Alias RLR
- Alit MA
- Allen S
- Allen SJ
- Allison J
- Alloj C
- Allorto NL
- Allsop J
- Almeida W
- Alonso E
- Alphonsus C
- Alvares D
- Alves MJ
- Amador JCB
- Ameer Y
- Amendola CP
- Ami N
- Amstrup-Hansen L
- Anagnou A
- Andersen C
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- Anderson C
- Anderson F
- Anderson P
- Andreadaki E
- Andreou A
- Andreou P
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- Angermair S
- Angus K
- Anillo V
- Antal O
- Antill P
- Antoniadou E
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- Ardern D
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- Attwood C
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- Avila Sanchez FJ
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- Chicken D-W
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- Chin II
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- Chisbert Cuenca V
- Chlorou D
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- Chung CKE
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- Cirstea E
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- Codita A
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- Suen A
- Sukawi I
- Sulaiman HA
- Sule UM
- Sumner M
- Sun C
- Sun H
- Sun Y
- Sun Y
- Sundayi S
- Sung W
- Susanti A
- Swain A
- Swarbrick G
- Swift D
- Sylvan A
- Synekidou E
- Syrogianni P
- Szabo C
- Szafranski J
- Szakmany T
- Tabajara FB
- Taddeo D
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- Tai J
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- Tameem A
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- Tantri A
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- Tchekulaev A
- Tebar Soto MT
- Teixeira Jesus JS
- Templer P
- ten Bokkel-Andela J
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- Tessera G
- Testa V
- Theodorakopoulou M
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- Thomas R
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- Vanluchene A
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- Vasileiou M
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- Veerakumaran J
- Veevaete L
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- Vilela dos Santos AM
- Virdi P
- Visser L
- Visvalingam S
- Vivian M
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- Vohra A
- Vohra R
- Voldaeva O
- Voloudakis N
- Volta CA
- Von Heymann C
- von Rhaden R
- Voruz F
- Wadams B
- Waggett H
- Walder B
- Walkden G
- Walker A
- Walker E
- Walker R
- Walker R
- Walker T
- Wallace A
- Wallace K
- Wallet F
- Walsgrove J
- Walsh D
- Wan X
- Wang D
- Wang D
- Wang F
- Wang G
- Wang H
- Wang H
- Wang J
- Wang J
- Wang J
- Wang J
- Wang J
- Wang K
- Wang L
- Wang L
- Wang L
- Wang S
- Wang S
- Wang S
- Wang T
- Wang W
- Wang X-L
- Wang Y
- Wang Y
- Wang Z
- Wang Z
- Wang Z
- Wang Z
- Ward J
- Wasmund C
- Wassall R
- Watanabe Oliveira HR
- Watson A
- Watson N
- Watt P
- Waugh D
- Waweru P
- Waworuntu N
- Waymouth E
- Weatherall L
- Weatherill J
- Webb S
- Weber E
- Wei J
- Weimann J
- Weller D
- Welsh S
- Wen XH
- Wen Y
- Wen Z
- Wendling PR
- Wessels JD
- Wetzel P
- Weyland A
- White S
- White S
- whitehouse A
- Whitman Z
- Whittle N
- Whitworth H
- Whysall K
- Wibrandt I
- Wickboldt N
- Wickenhauser R
- Wid WM
- Widmark C
- Wiegand-Loehnert C
- Wighton E
- Wigmore G
- Wijeysundera D
- Wikner M
- Wild J
- Wildes T
- Wildi S
- Williams A
- Williams M
- Williams S
- Wilscott-Davids C
- Wilson A
- Wilson D
- Wilson L
- Wilson N
- Wima S
- Winch D
- Winstone U
- Winterton D
- Wir WM
- Wise R
- Wittmann M
- Wolfer A
- Wollaston J
- Wong C
- Wong CW
- Wong JY
- Wong K
- Wong KWK
- Wong SM
- Wong T
- Wong WL
- Woodgate A
- Woolsey A
- Woon YL
- Worreth M
- Wouters P
- Wrench I
- Wright S
- Wu C
- Wu C
- Wu J
- Wu J
- Wu Q
- Wu S
- Wyffels P
- Wylie K
- Xia J
- Xia Y
- Xia Z-Y
- Xiao W
- Xiao W
- Xie G
- Xie J
- Xie J
- Xie K
- Xifara A
- Xiong X
- Xiong Y
- Xouplidis K
- Xu G-J
- Xu L
- Xu L
- Xu Q
- Xu S
- Xue R
- Yagnik A
- Yan Y
- Yang J
- Yang L
- Yang Q
- Yang S
- Yang T
- Yang Y
- Yao S
- Yao Y
- Yap HL
- Yarwood J
- Yassaee A
- Ye H
- Ye H
- Yegnaram S
- Yeh E
- Yin N
- Yip CP
- Yong J
- Yu HC
- Yu S
- Yu T
- Yu Y
- Yuan D
- Yuan F
- Yuan J
- Yuan J
- Yuan Y
- Yuliana A
- Zaimi D
- Zakynthinos S
- Zamudio D
- Zangrillo A
- Zapata DDM
- Zbitnew G
- Zeidan L
- Zeng Q
- Zerman L
- Zettergren J
- Zhang B
- Zhang E
- Zhang H
- Zhang H
- Zhang H
- Zhang J
- Zhang K
- Zhang L
- Zhang M
- Zhang M
- Zhang Q
- Zhang R
- Zhang S
- Zhang W
- Zhang X
- Zhang X
- Zhang X
- Zhang X
- Zhang Y
- Zhang Y
- Zhang Y
- Zhang Y
- Zhao B
- Zhao B
- Zhao C
- Zhao J
- Zhao J
- Zhao L
- Zhao L
- Zhao S
- Zhao T
- Zhao W
- Zhao W
- Zhao X
- Zhen J
- Zheng K
- Zheng L
- Zheng T
- Zhong Y
- Zhou C
- Zhou D
- Zhou H
- Zhou H
- Zhou J
- Zhou J
- Zhou J
- Zhou X-J
- Zhu X
- Zhu X
- Zhu Y
- Zhu Z
- Zhuang X
- Zilis G
- Zin NHM
- Zingerle N
- Zingg U
- Zoerner F
- Zonneveldt H
- Zou X
- Zoulamoglou M
- Zsisku L
- Publication venue
- 'Oxford University Press (OUP)'
- Publication date
- 01/01/2017
- Field of study
This was an investigator-initiated study funded by Nestle Health Sciences through an unrestricted research grant and by a National Institute for Health Research (UK) Professorship held by R.P. The study was sponsored by Queen Mary University of London
Molecular mechanisms of viral oncogenesis in humans
- Author
- A Ciccia
- A Decorsiere
- A Eulalio
- A Fradet-Turcotte
- A Gessain
- A Honegger
- A Lavorgna
- A Lujambio
- A Morales-Sanchez
- A Sodhi
- AM Price
- AP South
- AR Marquitz
- B Gruhne
- BJ Poiesz
- BS Blumberg
- BS Bowser
- C Bagneris
- C McCormick
- C Porta
- C Vernin
- CA Moody
- CC Tomlinson
- CE Lilley
- CJ Sherr
- CK Yuen
- CL Curry
- CM Murphy
- CW Dawson
- D Chen
- D Olagnier
- DA Thorley-Lawson
- DC Cho
- DG Wright
- DM Harper
- E Gottwein
- E Gottwein
- E Noch
- EK Kim
- EW Hewitt
- F Cheng
- F Scholle
- G Ma
- G Matusali
- G Stallone
- G Zhang
- GA Sowd
- H Feng
- H Takeda
- H zur Hausen
- HC Jha
- HH Chang
- HL Kaufman
- J Doorbar
- J Gao
- J Guito
- J Li
- JA Morrison
- JA Morrison
- JA Wendzicki
- Jianxin You
- JJ Wu
- JK Mitchell
- JL Petersen
- JM Luna
- JM Meyers
- JM Taylor
- JP Wong
- K Lan
- K Machida
- K McFadden
- K Yasuma
- KA Gillespie
- KJ Mackenzie
- L Coscoy
- L Lau
- L Xia
- L Zhang
- LS Young
- LW Wang
- L A Yates
- M Chatterjee
- M Daud
- M Durst
- M Fujimuro
- M Fukuda
- M Karin
- M Levrero
- M Luftig
- M Matsuoka
- M Ringelhan
- M Rowe
- M Schiffman
- M Shuda
- M Shuda
- MA Epstein
- MD Weitzman
- MD Weitzman
- ME McLaughlin-Drubin
- MJ Tan
- N Brimer
- N Goossens
- N Menzel
- N Prooyen Van
- N Raab-Traub
- N Rosewick
- N Sakakibara
- NA Wallace
- Nathan A. Krump
- O Rozenblatt-Rosen
- OL Hatton
- P Banerjee
- P Chugh
- P Ranganathan
- PA Nikitin
- PM Howley
- PS Moore
- PT Nghiem
- Q Chen
- Q Zhang
- QL Choo
- R Gopalakrishnan
- R Liu
- R Nusse
- RE Means
- RG Caldwell
- RJ Dowling
- S Duensing
- S Ishido
- S Knoll
- S Nitta
- S Yu
- SE Hopcraft
- SH Tsang
- SM Gregory
- SR Jacobs
- T McQuaid
- T Minamitani
- T Taga
- T Xia
- TF Schulz
- V Emuss
- W Kulwichit
- W Liu
- W Liu
- X Wang
- Y Chang
- Y Liu
- Z Dou
- Z Ma
- Z Surviladze
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
GNU Radio
- Author
- a-andre
- Abele Jason
- aidan
- Aigner Philipp
- AlexandraTrifan
- Alok Aradhana
- Anastasopoulos Achilleas
- Anderson Douglas
- Antetokounpo
- Apitzsch André
- Arnold Julian
- AsciiWolf
- Ashton Brennan
- Atreides Paul
- Baier Gerald
- Bailey Josh
- Balister Philip
- Banti Stefano
- Barnhart William
- Bauer Mark
- Becker Johannes K
- Beeri Gilad
- Behar Doron
- beitler
- Bell Richard C.
- Berman Michael
- Berndt Luke
- beroset
- Bhowmick Abhishek
- Bigot Peter A.
- Bird Alistair
- Bisht Rohit
- Bloessl Bastian
- Blomberg Tobias
- Blossom Eric
- Blot Emmanuel
- Blum Josh
- Boone Jared
- Bottoms A. Maitland
- Boven Paul
- Braun Martin
- Bruce Nicholas
- Brucker Jonathan
- Bruns Stefan
- Byers Michael
- Callyan
- Cate
- Cercueil Paul
- Chavez Christopher
- Chiang Johann
- Clark Bill
- cmrincon
- Collins Travis F.
- Conn Tracie
- Corgan Johnathan
- Corgan Nicholas
- Cornelius Mike
- Cottrell Mark
- Cox Grant
- Csete Alexandru
- cswiger
- Cuervo Nicolas
- Cutler Justin R.
- danielnachun
- David Paul
- Davis Andrew
- Demel Johannes
- Dhruvadityamittal
- Diaconescu Bogdan
- Dickens Michael
- Dijke Martyn van
- Dobrodii Roman
- Donohue Chris
- Drake Jeremy
- Duffy Charles
- Duggan Barry
- Dulmage Jared
- Dumps Jeff
- Durst Julius
- DvH Martin
- eb
- Economos Ron
- efardin
- ejk
- elms
- Enochs Brandon P.
- Eslinger Gregory
- esrh
- Estévez Daniel
- Ettus Matt
- Federico
- Feng Zhe
- Fischer Moritz
- Flamewires
- Flynn Toby
- Foster Nick
- FranBoric
- Franzen Florian
- Freire Igor
- Garver Paul
- Gauthier Philippe
- gdt
- Geiger Douglas
- Gelman Andriy
- Gentile Kevin
- Gerhard Davide
- Gerlits Ferenc
- Ghani Armin
- Gilbert Jacob
- Glass Steve
- gmazilla
- Goavec-Merou Gwenhael
- Goergen Nate
- Gottula Brett
- Govostes Ryan
- gr-sp
- Grambihler Daniel
- Griffiths Matt
- Gupta Alekh
- Gupta Arpit
- Gupta Sugandha
- Habets Thomas
- haru-02
- hatsunearu
- Haynal Steve
- Head4che
- Heel Martin Dudok van
- Hein Jason
- Hennepe Harm te
- Hermann Uwe
- Hilburn Ben
- Hitefield Seth
- Horden Adam
- Horvath Peter
- Hostetter Matt
- Hsu Bolin
- Huggins Tim
- Hübner Martin
- Iannucci Bob
- ilovezfs
- Inci Christian
- Ipsit
- Jackson Barry
- Jameson Mike
- japm48
- JaredD
- jb41997
- jcoy
- Johnson Eric
- Joost Laur
- Kalør Anders
- Kamat Jay
- Kapoor Siddharth
- karel
- karel-
- Kat Kerem
- Kawamoto Darek
- kc1212
- Kerler Bjoern
- Kigwana Edward
- Koehler Christoph
- Koehn Thaddeus
- Komulainen Tommi
- Koslowski Sebastian
- Kozel Derek
- Kravchuk Oleksandr
- Krysik Piotr
- Krämer Jan
- Kuester Tim
- Kuethe Chris
- Kurtle250
- Kuzmiak Lukas
- Lajovic Andrej
- LANGE Ludovic
- Larew Stephen
- Ledbetter William
- Ledet-Pedersen Jeppe
- Leech Marcus
- lenhart
- Lennart
- Lessard Louis Philippe
- Lichtman Marc
- Lindfors Timo
- linwei
- Litzenberger Darsey
- Lobo Pedro
- Long Jeff
- Ludwig Stephan
- luzpaz
- Løfaldli André
- M Nick
- Madeira Joao
- Madeira João
- Maier Kristian
- mark
- Markgraf Steve
- Maroti Miklos
- masw
- matt
- May Terry
- Mayer Christoph
- Mayo Chris
- MBoerschig
- McCarthy Nicholas
- McCarthy Nick
- McCodeface Codey
- McDiarmid Campbell
- McGwier Bob
- McQuiggin Kevin
- Mendez Alba
- Meyerhoff Grant
- mi-a
- michael-roe
- Michel Adrien
- Mills Matt
- Mochalov Konstantin
- Moeller
- Molenkamp Ray
- Monahan-Mitchell Tim
- Morin Cyrille
- Morman Josh
- Munaut Sylvain
- Muzika Bill
- Muñoz Eduardo Sánchez
- Müller Marcus
- Müller Sebastian
- Naranjo Carlos Alberto Ruiz
- Negi Swapnil
- Newman Tim
- Nguyễn Chí-Thanh Christopher
- Nieboer Geof
- Niedermayer Philipp
- Niki
- Nil Michael De
- Nowlan Sean
- Nychis George
- NZSmartie
- O'Shea Tim
- Olivain Julien
- Oliver
- Olsen Sebastian
- Oltmanns Stefan
- Orlando John
- Orr Brian
- Ossmann Michael
- P Vladisslav
- Padalino Brian
- Patel Kartik
- Patulea Catalin
- Pavon
- Pendlum Jonathon
- Pentler Mark
- ph1t0
- phansel
- Pi David
- Pinkava Jiri
- Pinkava Jiří
- Pisarenko Artem
- Piscopo Mike
- Plett Mark
- Porges Donald
- Pyle Hugh
- Quaresma Jose
- R-ohit-B-isht
- Radulescu Bogdan
- rajb245
- Rajendran Sreeraj
- Rasmussen Mathias
- rear1019
- RedStone002
- Reid Kevin
- Rene Mathieu
- Reynwar Ben
- Ribero Marco
- Richardson Glenn
- Roberts Wayne
- Robertson Dan
- Rocca Federico La
- Rode Andrej
- Roe Michael
- Rondeau Tom
- Ross Spencer
- Rui Huang
- Saari James
- Sabaghi Behnam
- Sallay John
- samwhiting
- Savoye Rob
- Schmidt Fabian P.
- Schmitz Johannes
- Schneider Eric
- schneider42
- Schroer Volker
- Schueler Joshua
- Schutt Ryan
- Seeber Balint
- Seeker
- Seguinot Christophe
- Semich Karl
- Shane
- Sharan Ravi
- Sharma Rohan
- Shepard Tim
- shwhiti
- Siddiq Sahil
- Singh Adarsh
- Sloane Andy
- Smith Clayton
- soggysec
- Solano Camilo
- Sorber David
- Spanbauer Rick
- Spytz Zackery
- Srairi Imad-Eddine
- Stapleton Brent
- Statzer Eric
- Stef Mihai
- Stiefel Maximilian
- Stolnikov Dimitri
- Suciu Adrian
- Swiger Chuck
- Szymaniak Jon
- Tagunov Ilya
- Talbert Scott
- Tan Solomon
- TASAKA Mamoru
- Temple Nate
- Thakur Anshul
- theartful
- Thomas Aditya
- Thompson Roy
- Torborg Scott
- Trewhitt Ethan
- Trotter Brett L.
- Tsiligiannis Vasilis
- Tsou Thomas
- tttx
- Tuerkyilmaz Eral
- Tyers Bernard
- Uher Jason
- Undheim Ruben
- Unice Kyle
- Unknown
- Vanhoy Garrett
- Velichkov Vasil
- vermillionsands
- Vierinen Juha
- Volz Ryan
- Vutukuri Srinivas Naga
- Vågsether Håkon
- wakass
- Walls Andy
- Walters Mike
- Ward Don
- Warnes Gregory
- wcampbell
- Weber Douglas
- Wecksell Elof
- West Nathan
- Wicks Paul
- Wiedemann Bernhard M.
- Willecke Alexander
- Winter David
- Witkowski Peter
- Wollesen Victor
- Wunsch Felix
- Wunsch Stefan
- Wyk Hendrik van
- Xu Henry
- yang dae hyun,
- Z Liu, Andrew
- Zapodovnikov Valerii
- Zehl Stefan
- Zero_Chaos
- Zhao Alick
- Zheng Kevin
- Zhu Chuang
- Zy Jakub
- Østergaard Nick
- Šafář Jan
- Škarvada Jaroslav
- Publication venue
- Zenodo
- Publication date
- 13/12/2022
- Field of study
GNU Radio is a free & open-source software development toolkit that provides signal processing blocks to implement software radios. It can be used with readily-available, low-cost external RF hardware to create software-defined radios, or without hardware in a simulation-like environment. It is widely used in hobbyist, academic, and commercial environments to support both wireless communications research and real-world radio systems