6 research outputs found
Blockade of EGFR Activation Promotes TNF-Induced Lung Epithelial Cell Apoptosis and Pulmonary Injury
- Author
- Publication venue
- 'MDPI AG'
- Publication date
- 17/08/2019
- Field of study
Pneumonitis is the leading cause of death associated with the use of epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors (EGFR-TKIs) against non-small cell lung cancer (NSCLC). However, the risk factors and the mechanism underlying this toxicity have not been elucidated. Tumor necrosis factor (TNF) has been reported to transactivate EGFR in pulmonary epithelial cells. Hence, we aimed to test the hypothesis that EGFR tyrosine kinase activity regulates TNF-mediated bronchial epithelial cell survival, and that inhibition of EGFR activity increases TNF-induced lung epithelial cell apoptosis. We used surfactant protein C (SPC)-TNF transgenic (tg) mice which overexpress TNF in the lungs. In this model, gefitinib, an EGFR-TKI, enhanced lung epithelial cell apoptosis and lymphocytic inflammation, indicating that EGFR tyrosine kinase prevents TNF-induced lung injury. Furthermore, IL-17A was significantly upregulated by gefitinib in SPC-TNF tg mice and p38MAPK activation was observed, indicative of a pathway involved in lung epithelial cell apoptosis. Moreover, in lung epithelial cells, BEAS-2B, TNF stimulated EGFR transactivation via the TNF-α-converting enzyme in a manner that requires heparin binding (HB)-EGF and transforming growth factor (TGF)-α. These novel findings have significant implications in understanding the role of EGFR in maintaining human bronchial epithelial cell homeostasis and in NSCLC treatment
Blockade of EGFR Activation Promotes TNF-Induced Lung Epithelial Cell Apoptosis and Pulmonary Injury
- Author
- Publication venue
- 'MDPI AG'
- Publication date
- Field of study
GROUND-BASED Paα NARROW-BAND IMAGING OF LOCAL LUMINOUS INFRARED GALAXIES. I. STAR FORMATION RATES AND SURFACE DENSITIES
- Author
- Agüero
- Alonso-Herrero
- Alonso-Herrero
- Alonso-Herrero
- Alonso-Herrero
- Ann
- Asami Nakashima
- Barnes
- Calzetti
- Calzetti
- Caputi
- Colina
- Corbett
- Daddi
- Davies
- de Vaucouleurs
- Dopita
- Díaz-Santos
- Falcke
- Fernández
- Grimes
- Hidenori Takahashi
- Ho
- Hopkins
- Iono
- Kazushi Okada
- Ken Tateuchi
- Ken'ichi Tarusawa
- Kennicutt
- Kennicutt
- Kentaro Asano
- Kentaro Motohara
- Kewley
- Kim
- Kim
- Kimiaki Kawara
- Koji Toshikawa
- Komugi
- Konishi
- Koss
- Kotaro Kohno
- Lada
- Lai
- Lauberts
- Levenson
- Liu
- Liu
- Lord
- Lutz
- Malmquist
- Mamoru Doi
- Masahiro Konishi
- Masuo Tanaka
- Mauder
- Mizuho Uchiyama
- Morganti
- Motohara
- Murphy
- Naim
- Natsuko Mitani Kato
- Peterson
- Rieke
- Roche
- Rothberg
- Rujopakarn
- Rujopakarn
- Rujopakarn
- Ryou Ohsawa
- Saito
- Sanders
- Schweizer
- Scoville
- Scoville
- Sheen
- Shigeyuki Sako
- Shintaro Koshida
- Shinya Komugi
- Sho Manabe
- Skrutskie
- Soifer
- Soifer
- Soifer
- Soya Todo
- Spergel
- Stritzinger
- Takafumi Kamizuka
- Takashi Miyata
- Takeo Minezaki
- Takeo Soyano
- Tateuchi
- Tateuchi
- Tomohiko Nakamura
- Tomoki Morokuma
- Toshihiko Tanabé
- Toshihiro Handa
- Toshinobu Takagi
- Tran
- Tsutomu Aoki
- van den Broek
- Vorontsov-Vel'Yaminov
- West
- Yoichi Tamura
- Yoshifusa Ita
- Yuan
- Yuka K. Uchimoto
- Yutaro Kitagawa
- Yuzuru Yoshii
- Publication venue
- 'IOP Publishing'
- Publication date
- Field of study
Miscible Polymer Blends
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- Z Benabdelghani
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