26 research outputs found
Heterodimerization of Glycosylated Insulin-Like Growth Factor-1 Receptors and Insulin Receptors in Cancer Cells Sensitive to Anti-IGF1R Antibody
- Author
- A Belfiore
- A Belfiore
- A Belfiore
- A Gualberto
- A Keller
- A Ouban
- A Ullrich
- AI Nesvizhskii
- AL Frattali
- BD Cohen
- CP Moxham
- D Burtrum
- D Olmos
- DD Karp
- Do Youn Oh
- EC Yi
- Eugene C. Yi
- F Frasca
- F Frasca
- Frank T. Kolligs
- G Heller
- G Pandini
- G Pandini
- G Pandini
- Gyeong Hoon Kang
- H Yu
- Hwang-Phill Kim
- J Jassem
- J Rodon
- J Rosenfeld
- J Zha
- Jinah Park
- JK Eng
- JL Ku
- Jong-Wan Park
- Jun Gyu Kim
- Keon Wook Kang
- KR Kalli
- L Cao
- L Sciacca
- MA Soos
- MA Soos
- Min Jueng Kang
- P De Meyts
- P Haluska
- R Baserga
- R Nahta
- S Avnet
- Sae-Won Han
- Sang-Hyun Song
- Seock-Ah Im
- Tae-You Kim
- TS Olson
- V Papa
- V Papa
- V Vella
- V Vella
- V Vella
- Y Gong
- Young-Kwang Yoon
- Yung-Jue Bang
- Publication venue
- Public Library of Science
- Publication date
- 01/03/2012
- Field of study
Identification of predictive biomarkers is essential for the successful development of targeted therapy. Insulin-like growth factor 1 receptor (IGF1R) has been examined as a potential therapeutic target for various cancers. However, recent clinical trials showed that anti-IGF1R antibody and chemotherapy are not effective for treating lung cancer.In order to define biomarkers for predicting successful IGF1R targeted therapy, we evaluated the anti-proliferation effect of figitumumab (CP-751,871), a humanized anti-IGF1R antibody, against nine gastric and eight hepatocellular cancer cell lines. Out of 17 cancer cell lines, figitumumab effectively inhibited the growth of three cell lines (SNU719, HepG2, and SNU368), decreased p-AKT and p-STAT3 levels, and induced G 1 arrest in a dose-dependent manner. Interestingly, these cells showed co-overexpression and altered mobility of the IGF1R and insulin receptor (IR). Immunoprecipitaion (IP) assays and ELISA confirmed the presence of IGF1R/IR heterodimeric receptors in figitumumab-sensitive cells. Treatment with figitumumab led to the dissociation of IGF1-dependent heterodimeric receptors and inhibited tumor growth with decreased levels of heterodimeric receptors in a mouse xenograft model. We next found that both IGF1R and IR were N-linked glyosylated in figitumumab-sensitive cells. In particular, mass spectrometry showed that IGF1R had N-linked glycans at N913 in three figitumumab-sensitive cell lines. We observed that an absence of N-linked glycosylation at N913 led to a lack of membranous localization of IGF1R and figitumumab insensitivity.The data suggest that the level of N-linked glycosylated IGF1R/IR heterodimeric receptor is highly associated with sensitivity to anti-IGF1R antibody in cancer cells
A922 Sequential measurement of 1 hour creatinine clearance (1-CRCL) in critically ill patients at risk of acute kidney injury (AKI)
- Author
- Abbott TE
- Abdallah RI
- Abdel-Aal IR
- Abdelmonem SA
- Abdo WF
- Abellan AN
- Abellán AN
- Abellán AN
- Abellán AN
- Abrams ST
- Ackerley C
- Acuña M
- Adda M
- Adhikari NK
- Adriano G
- Adrie C
- Affatato R
- Affatato R
- Afonso-Rivero D
- Agarossi A
- Agarwal LK
- Ageeva T
- Agrawal R
- Aguayo-DeHoyos E
- Aguilar AL
- Aguilar-Alonso E
- Aguilar-Alonso E
- Aguilar-Alonso E
- Aguirregabyria M
- Ahmadnia E
- Ahn C
- Ahn JY
- Ahn JY
- Ahn MY
- Ahn MY
- Aitken LM
- Akalaev R
- Akbarzadeh A
- Akcan-Arikan A
- Akhlagh SH
- Akhtar N
- AKI Research Group
- Akiduki N
- Akin S
- Akizuki N
- Akkoc T
- Ala-Kokko T
- Alanio A
- Albaiceta GM
- Albaladejo P
- Alberto F
- Albuisson E
- Alcala MA
- Alcázar L
- Aldabo-Pallas T
- Aldana NN
- Aldecoa C
- Alegría L
- Alejandro R
- Alejo GC
- Alejos RM
- Alexandrova E
- Algarte R
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- Algieri I
- Algora-Weber A
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- Aliaga FA
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- Altıntas ND
- Alvarez J
- Alves SC
- Alzola LM
- Amargianitakis V
- Amaro R
- Amato MB
- Ambler M
- Amerongen MP
- Amininejad T
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- Amorim V
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- Araujo NJ
- Araujo VF
- ARIAM registry of adult cardiac surgery
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- Chhor V
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- Izdes S
- Jaber S
- Jacky A
- Jacobs FM
- Jacques T
- Jaffal K
- Jamali S
- Jang BH
- Janotka M
- Janotka M
- Janotka M
- Jansen D
- Jansen N
- Japan Septic Disseminated Intravascular Coagulation (JSEPTIC DIC) study group
- Jardim JJ
- Jardim M
- Jareño A
- Javadpour S
- Jayasinghe S
- Jean-Baptiste S
- Jean-Baptiste S
- Jensen AE
- Jensen JU
- Jeon YD
- Jeon YD
- Jeong IY
- Jeong IY
- Jeong WY
- Jeong WY
- Jian Z
- Jiao LR
- Jibaja M
- Jimenez-Herrera MF
- Jiménez GJ
- Jo YH
- Joachim J
- Jochmans S
- John G
- Jonas M
- Jonas M
- Jonas M
- Jones C
- Joshi R
- Joshi V
- Jovaisa T
- JSEPTIC (Japanese Society of Education for Physicians and Trainees in Intensive Care) Clinical Trial Group
- Juan WC
- Juanas CA
- Judickas S
- Juez A
- Juliarena A
- Jun IG
- Jun IG
- Jung K
- Jung KW
- Junior JM
- Kaczirek K
- Kaese S
- Kalani N
- Kalenka A
- Kalfon P
- Kamali E
- Kaminsky GE
- Kaneko M
- Kang M
- Kang M
- Kang PL
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- Kang Y
- Kao KC
- Kappler F
- Kara A
- Karachi F
- Karanjia N
- Karbing DS
- Karsten E
- Kasdan H
- Kashiya S
- Kashyap R
- Katabami K
- Katabami K
- Katabami K
- Katabami K
- Katira BH
- Kavanagh BP
- Kawamura N
- Kawano S
- Kay FU
- Kayaaslan B
- Kayambu G
- Kazutoshi F
- Ke MW
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- Keep J
- Keep J
- Keller E
- Kellner F
- Kelly JM
- Kenardy J
- Keough E
- Kerhuel L
- Kerr C
- Kezyte G
- Khadjibaev A
- Khaliq W
- Khine H
- Kim DJ
- Kim HJ
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- Kim KS
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- Kim MH
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- Kim W
- Kimmoun A
- King HS
- Kinnear J
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- Kirakli C
- Kirca H
- Kirman M
- Kirwan CJ
- Kittnar O
- Klapsing P
- Klaus DA
- Kleinpell R
- Kluge S
- Knafelj R
- Knight LD
- Ko JI
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- Kobayashi A
- Koco E
- Kodate A
- Kodate A
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- Kokkini S
- Kolnikova I
- Komuro T
- Kondili E
- Kongpolprom N
- Kooner G
- Kostalas M
- Kosuk ME
- Kotsopoulos A
- Kou PS
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- Kovacikova L
- Kox M
- Kraegpoeth A
- Krenn CG
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- Kristof J
- Kruger A
- Kruger A
- Krüger A
- Ku NS
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- Kubik M
- Kubota K
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- Kulaga EV
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- Kumari BK
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- Kunze-Szikszay N
- Kurmukov IA
- Kurth T
- Kurtz P
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- Kwon HM
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- Kye YC
- Kyle UG
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- Labaune MA
- Labra C
- Lacerda P
- Laerkner E
- Lafaurie M
- Lafuente E
- Lagonidis D
- Lagos R
- Lahmer T
- Lai CC
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- Latini R
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- Latorre J
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- Lebherz-Eichinger D
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- Letizia T
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- Liao X
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- Lipcsey M
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- Lissonde F
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- Litchfield K
- Liu CP
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- Liu D
- Llaurado-Serra M
- Llorente B
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- Lopes JA
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- Lortat-Jacob B
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- Ly H
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- Macfarlane B
- MacKay A
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- Maekawa K
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- Magnanimi E
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- Mezidi M
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- Mimoz O
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- Stretti F
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- Sun XM
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- Suwanpasu S
- Suzuki S
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- Sylla P
- Sáez VC
- Sánchez B
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- Sánchez MJ
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- Tabatabaei HR
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- Timsit JF
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- Tokyo Womens Medical University
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- WIND study group
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- Yamaguchi Y
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- Yan WW
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- Yasuda H
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- Yoshitake E
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- Zabini D
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- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/2016
- Field of study
Meeting abstrac
Development, effectiveness and cost-effectiveness of a new out-patient Breathlessness Support Service: study protocol of a phase III fast-track randomised controlled trial
- Author
- A Gift
- A Williams
- AJS Coats
- American Thoracic Society
- American Thoracic Society
- AP Abernethy
- AP Abernethy
- AS Zigmond
- BR Celli
- C Bausewein
- C Bausewein
- Caroline Jolley
- Caroline Murphy
- Caty Panell
- Charles Reilly
- Chiara De Biase
- Claudia Bausewein
- CP Escalante
- DB Reuben
- DG Altman
- Elmien Brink
- G Kasymjanova
- GH Guyatt
- H Katsura
- H Seow
- Helene Bellas
- HJ Schunemann
- I Higginson
- IJ Higginson
- Irene J Higginson
- J Austin
- J Corner
- J Hearn
- J Lynn
- J Yorke
- Jane Kelly
- John Moxham
- K Hill
- L Jennings Anne
- L Sewell
- M Bredin
- M Bédard
- M Campbell
- M Farquhar
- M Farquhar
- M Gysels
- M Gysels
- MA Puhan
- Medical Research Council
- MH Gysels
- MH Gysels
- MW Rabow
- National Institute for Clinical Excellence (NICE)
- P Edmonds
- Paul McCrone
- Paula Lobo
- Preety Madan
- R Garrod
- S Booth
- S Booth
- S Moore
- S Rennard
- W D-C Man
- Wei Gao
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
What is the role of trees and remnant vegetation in attracting people to urban parks?
- Author
- A Chiesura
- A Forsyth
- A Kazmierczak
- A Troy
- Australian Bureau of Statistics
- B. B. Lin
- BB Lin
- Brisbane City Council
- C Moxham
- CC Branas
- CH Ho
- CP Catterall
- CW Thompson
- CY Jim
- D Zanon
- D. F. Shanahan
- DC Dearborn
- DF Shanahan
- DF Shanahan
- DF Shanahan
- DQ Zhou
- E Pleson
- EK Nisbet
- GD Daniels
- GR McCormack
- GS Lovasi
- H Bai
- HEW Wende
- J Bigirimana
- J Garden
- J Maas
- JD Armston
- JG Wu
- JG Wu
- JWR Baur
- K Beil
- K Han
- K Hauru
- K Stagoll
- K. J. Gaston
- KC Matteson
- KJ Shinew
- KK Peschardt
- KN Irvine
- KP Burnham
- LE Jackson
- LE Keniger
- LW Clarke
- M Bodin
- M Ferre´
- M Strohbach
- MJ Brady
- MP White
- MW Strohbach
- N Heynen
- Natural England
- NM Wells
- P Bolund
- P Sikorski
- PS Sattler
- R Core Team
- R Home
- R Kaplan
- R Mitchell
- R Parsons
- R. A. Fuller
- R. Bush
- RA Fuller
- RD Bixler
- RJ Standish
- RS Ulrich
- SA Bekessy
- SD Piper
- SM Landry
- SME Dillen van
- T Bjerke
- T Hartig
- T Sugiyama
- T-T-H Pham
- Y Heezik van
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Anti-Peptide Monoclonal Antibodies to the β-Adrenergic Receptor: Use in Purification of β Receptor 1,2
- Publication venue
- 'Mary Ann Liebert Inc'
- Publication date
- Field of study
The type 1 insulin-like growth factor receptor signalling system and targeted tyrosine kinase inhibition in cancer
- Publication venue
- 'SAGE Publications'
- Publication date
- Field of study
Lack of specificity of antibodies against human beta-adrenergic receptors.
- Author
- Publication venue
- Publication date
- 01/01/2009
- Field of study
Insulin and GH secretion in adolescent girls with irregular cycles: Polycystic vs multifollicular ovaries
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Call for Consistency: the Need to Establish Gross Anatomy Learning Objectives for the Entry-Level Physical Therapist
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
The metabolic and mitogenic properties of basal insulin analogues
- Author
- Publication venue
- 'Informa UK Limited'
- Publication date
- Field of study