7 research outputs found
Organometallic Complex Strongly Impairs Chikungunya Virus Entry to the Host Cells
- Author
- Publication venue
- 'Frontiers Media SA'
- Publication date
- 15/12/2020
- Field of study
Chikungunya fever is a disease caused by the Chikungunya virus (CHIKV) that is transmitted by the bite of the female of Aedes sp. mosquito. The symptoms include fever, muscle aches, skin rash, and severe joint pains. The disease may develop into a chronic condition and joint pain for months or years. Currently, there is no effective antiviral treatment against CHIKV infection. Treatments based on natural compounds have been widely studied, as many drugs were produced by using natural molecules and their derivatives. Alpha-phellandrene (α-Phe) is a naturally occurring organic compound that is a ligand for ruthenium, forming the organometallic complex [Ru2Cl4(p-cymene)2] (RcP). Organometallic complexes have shown promising as candidate molecules to a new generation of compounds that presented relevant biological properties, however, there is a lack of knowledge concerning the anti-CHIKV activity of these complexes. The present work evaluated the effects of the RcP and its precursors, the hydrate ruthenium(III) chloride salt (RuCl3â
xH2O) (Ru) and α-Phe, on CHIKV infection in vitro. To this, BHK-21 cells were infected with CHIKV-nanoluciferase (CHIKV-nanoluc), a viral construct harboring the nanoluciferase reporter gene, at the presence or absence of the compounds for 16 h. Cytotoxicity and impact on infectivity were analyzed. The results demonstrated that RcP exhibited a strong therapeutic potential judged by the selective index > 40. Antiviral effects of RcP on different stages of the CHIKV replicative cycle were investigated; the results showed that it affected early stages of virus infection reducing virus replication by 77% at non-cytotoxic concentrations. Further assays demonstrated the virucidal activity of the compound that completely blocked virus infectivity. In silico molecular docking calculations suggested different binding interactions between aromatic rings of RcP and the loop of amino acids of the E2 envelope CHIKV glycoprotein mainly through hydrophobic interactions. Additionally, infrared spectroscopy spectral analysis indicated interactions of RcP with CHIKV glycoproteins. These data suggest that RcP may act on CHIKV particles, disrupting virus entry to the host cells. Therefore, RcP may represent a strong candidate for the development of anti-CHIKV drugs
ICAR: endoscopic skullâbase surgery
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- Publication date
- 01/07/2019
- Field of study
n/
Post-transcriptional inhibition of hepatitis C virus replication through small interference RNA
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- A Parfieniuk
- A Pause
- AD Kwong
- AM Anesti
- AP McCaffrey
- AR Zekri
- B Bartosch
- BD Lindenbach
- C Guha
- CC Mello
- CC Pacca
- G Meister
- J Zhang
- J Zhong
- JA Wilson
- JA Wilson
- JH Hoofnagle
- KE Reed
- M Lopez-Fraga
- MJ Alter
- MK el-Awady
- MP Manns
- MP Walker
- Muhammad Ansar
- Muhammad Tahir Sarwar
- MY Seo
- NSJK Raja
- PC Haasnoot
- QL Choo
- SB Kapadia
- Sheikh Riazuddin
- Sidra Rehman
- SM Hammond
- Tariq Javed
- Usman Ali Ashfaq
- V Bitko
- VJ Leveque
- Y Takigawa
- YP Liu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Type I interferons are essential while type II interferon is dispensable for protection against St. Louis encephalitis virus infection in the mouse brain
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- Abbas AK
- Bamming D
- Boussif O
- Burguillos MA
- Calisher CH
- Chang T-H
- Chazal M
- Clark DC
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- Tang H
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- Vedovello D
- Wang T
- Xavier-Neto J
- Zmurko J
- Publication venue
- 'Informa UK Limited'
- Publication date
- Field of study
Distribution and phylogenetic analysis of Culex flavivirus in mosquitoes in China
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- A Shuyi
- A Vazquez
- A Yamanaka
- AE Firth
- BG Bolling
- BJ Blitvich
- C Barreau
- CC Pacca
- Chunxia Jing
- DC Machado
- DY Kim
- EA Gould
- G Kuno
- Guang Yang
- Guifang Liu
- Guodong Liang
- H Cammisa-Parks
- Hongyue Jiang
- Huanyu Wang
- J Hobson-Peters
- JA Farfan-Ale
- K Hoshino
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- Lei Feng
- M Calzolari
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- MB Crabtree
- MB Crabtree
- ME Morales-Betoulle
- Min Wang
- P Burivong
- R Saiyasombat
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- RC Sang
- RJ Kent
- RS Nasci
- S Cook
- S Cook
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- S Cook
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- Shaobai Zhang
- Shihong Fu
- T Solomon
- V Stollar
- W Huanyu
- W Zuoshu
- Weijun Hu
- Weixin Chen
- Wenkai Liang
- Xiaojuan Lin
- Xiaoxia He
- Xiaoyan Gao
- Xiaoyan Tao
- Yan Liu
- Ying He
- Yuxi Cao
- YY Chen
- Z Lu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
The RNAi pathway plays a small part in Wolbachia-mediated blocking of dengue virus in mosquito cells
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- A Sabchareon
- A Takaoka
- A Untergasser
- AA Hoffmann
- AG Ferreira
- AM Fallon
- B Lemaitre
- C Chang
- C Dostert
- CB Ocampo
- CC Pacca
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- CJ McMeniman
- CL Campbell
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- DJ Gubler
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- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
ICAR: endoscopic skullâbase surgery
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- American Academy of Pediatrics Steering Committee on Quality Improvement and Management
- Amichetti M
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- Lee TJ
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- Likhacheva A
- Lin EM
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- Linsler S
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- Little AS
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- Liu CL
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- London SD
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- Lorenz RR
- Loy AH
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- Lund V
- Lund VJ
- Lund VJ
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- Luong A
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- McLaughlin EJ
- McLaughlin N
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- Mehta BS
- Mehta GU
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- Mendelson ZS
- Mendenhall WM
- Merchant TE
- Mesquita Filho PM
- Messerer M
- Meyers SP
- Michel G
- Midilli R
- Milanese L
- Miller NR
- Minamida Y
- Minniti G
- Minniti G
- Mitchell EH
- Miyajima Y
- Miyamoto RC
- Miyamura S
- Modesto A
- Mohammadi M
- MohammadiâAraghi H
- Mohsenifar Z
- Molitch ME
- Montava M
- Monteith SJ
- Montgomery WW
- Montiero E
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- Nicolai P
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- NORDIC Idiopathic Intracranial Hypertension Study Group Writing Committee
- Nuwer MR
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- O'Connell BP
- O'Reilly AG
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- Palani A
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- Park JH
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- Pasztor E
- Patel KS
- Patel MR
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- Patel SN
- Patel TD
- Patil VM
- Patrona A
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- Pereira EAC
- Peris Celda M
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- PinheiroâNeto CD
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- Pledger CL
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- Weiland DA
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- Wiseman SM
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- Yunoue S
- YuâWaiâMan P
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- Publication venue
- 'Wiley'
- Publication date
- Field of study