14 research outputs found
Selective 5-HT7 receptor agonists LP 44 and LP 211 elicit an analgesic effect on formalin-induced orofacial pain in mice
- Author
- Ahmet DOĞRUL
- Albayrak A
- Bardin L
- Benyamin R
- Brenchat A
- Brenchat A
- Buğra ŞENEL
- Chen Y
- Dogrul A
- Dogrul A
- Enza LACİVİTA
- Godínez-Chaparro B
- Hargreaves K
- Kadriye DEMİRKAYA
- Luccarini P
- Marcello LEOPOLDO
- Mehlisch DR
- Melik SEYREK
- Miranda HF
- Nakajima K
- Okamoto K
- Rocha-González HI
- Russell R
- Tamaddonfard E
- Viguier F
- Yang EJ
- Yesilyurt O
- Zeynep ÖNCEL TORUN
- Özlem Martı AKGÜN
- Publication venue
- 'FapUNIFESP (SciELO)'
- Publication date
- Field of study
Targeting the Serotonin 5-HT7 Receptor in the Search for Treatments for CNS Disorders: Rationale and Progress to Date
- Author
- A Brenchat
- A Brenchat
- A Brenchat
- A Brenchat
- A Gasbarri
- A Gasbarri
- A Matthys
- A Meneses
- A Meneses
- A Meneses
- A Meneses
- A Nikiforuk
- A Nikiforuk
- A Nikiforuk
- A Ulugol
- A Wesolowska
- A Wesolowska
- A Wesolowska
- Agnieszka Nikiforuk
- AI Abbas
- AJ Roberts
- AJ Roberts
- B Dean
- B Filippis De
- B Pouzet
- BB Garcia-Iglesias
- BL Roth
- C Kikuchi
- CR Guthrie
- D Guseva
- D Leo
- D Pericic
- DE Heidmann
- DL Braff
- DR Thomas
- DR Thomas
- E Gellynck
- E Kvachnina
- E Kvachnina
- F Kobe
- F Viguier
- F Viguier
- G Beaudet
- G Liy-Salmeron
- G Sarkisyan
- G Sarkisyan
- GS Perez-Garcia
- J Shelton
- J Shelton
- J Sprouse
- JA Bard
- JA Terron
- JA Terron
- JC Ehlen
- JC Neill
- JJ Hagan
- JM Monti
- JM Monti
- JM Monti
- JM Witkin
- K Tokarski
- K Tokarski
- KA Krobert
- KA Krobert
- KA Waters
- L Ciranna
- L Costa
- L Westrich
- L Westrich
- LA Ruocco
- LN Cates
- M Cuesta
- M Gardani
- M Graf
- M Guscott
- M Horiguchi
- M Hołuj
- M Ikeda
- M Leopoldo
- M Leopoldo
- M Ruat
- M Teitler
- O Mnie-Filali
- P Atanes
- P Bonaventure
- P Bonaventure
- P Bonaventure
- P Pilato Di
- P Willner
- PB Hedlund
- PB Hedlund
- PJ Lovell
- R Canese
- R Galici
- S Semenova
- SJ Ballaz
- SJ Ballaz
- SL McLean
- SR Hauser
- SW Ying
- SZ East
- T Freret
- T Horisawa
- T Horisawa
- T Kenakin
- TM Eriksson
- TW Lovenberg
- U Renner
- W Adriani
- X Wang
- YC Li
- Z Yang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Esc‐1GN shows therapeutic potentials for acne vulgaris and inflammatory pain
- Publication venue
- 'Wiley'
- Publication date
- Field of study
HTR7 Mediates Serotonergic Acute and Chronic Itch
- Author
- Abbott
- Adham
- Ahn
- Akiyama
- Anjaneyulu
- Anne Sofie Braun Olsen
- Bardin
- Bautista
- Bautista
- Bayer
- Blardi
- Bonnet
- Brandt
- Brenchat
- Brenchat
- Browning
- Brueggemann
- Caterina
- Cederberg
- Cevikbas
- Cheryl L. Stucky
- Cho
- Cookson
- Diana M. Bautista
- Garibyan
- Gerhold
- Giaever
- Glass
- Green
- Hampton
- Han
- Hedlund
- Hedlund
- Hoon
- Huang
- Idzko
- Imamachi
- Julius
- Justin F. Wong
- Jørgensen
- Kalz
- Karai
- Kayser
- Kerr
- Kim
- Kuraishi
- Kuraishi
- Kwan
- Kyle Lyman
- Kyriakides
- LaMotte
- Li
- Lin
- Liu
- Liu
- Liu
- Lovenberg
- Lundeberg
- Lyn M. Batia
- Manteniotis
- Matterne
- Maurizio Pellegrino
- Metz
- Michael A. Kienzler
- Mishra
- Mollanazar
- Moser
- Nair
- Nascimento
- Nojima
- Nordlind
- Oh
- Rachel B. Brem
- Rausl
- Roberts
- Ross
- Sannicandro
- Santello
- Sarah R. Wilson
- Schadt
- Schmidt
- Schwörer
- Shannan P. McClain
- Soga
- Spergel
- Takeshi Morita
- Tang
- Taylor
- Tepper
- Van Steenwinckel
- Vanhoenacker
- Warnock
- Wilson
- Wilson
- Wilson
- Xie
- Yun
- Zeitz
- Zhao
- Zylicz
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Low-basicity 5-HT7 Receptor Agonists Synthesized Using the van Leusen Multicomponent Protocol
- Author
- A Agarwal
- A Brenchat
- A Dömling
- A Gasbarri
- A Gasbarri
- A Matthys
- A Meneses
- A Meneses
- A Sali
- A Wesolowska
- A Wesolowska
- AJ Bojarski
- AJ Roberts
- AK Tiwari
- AM Leusen Van
- AP Bento
- B Dean
- B Filippis De
- B Pouzet
- C Mahe
- D Hoyer
- DA Nugiel
- E Deau
- E Kvachnina
- E Lacivita
- ES Vermeulen
- FC Bernstein
- FJ Monsma
- G Sarkisyan
- HD Hansen
- HI Rocha-Gonzalez
- J Andries
- J Watson
- JA Bard
- JA Terron
- JJ Hagan
- L Costa
- L Zhang
- M Leopoldo
- M Leopoldo
- M Leopoldo
- M Ruat
- MH Paluchowska
- P Pilato Di
- P Zajdel
- PB Hedlund
- PB Hedlund
- PB Hedlund
- PN James
- R Canese
- RA Glennon
- RN Harris 3rd
- RS Obach
- S Semenova
- T Ladduwahetty
- TM Eriksson
- TT Wager
- TW Lovenberg
- UL Mullins
- V Isberg
- W Stoll
- Y Cheng
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Fisetin exerts antihyperalgesic effect in a mouse model of neuropathic pain: engagement of spinal serotonergic system
- Author
- A Brenchat
- B Gustorff
- B Hu
- C Vogel
- D Bridges
- E Eisenberg
- F Viguier
- GJ Bennett
- H Cheong
- I Yalcin
- I Yalcin
- JA Micó
- JA Ross
- JG Villarinho
- JH Liang
- JL Hylden
- K Hargreaves
- K Roeska
- L Zhen
- M Benbouzid
- M Tanabe
- MJ Millan
- MY Patel
- N Choucair-Jaafar
- N Ravichandran
- NB Finnerup
- RD Porsolt
- T Dowdall
- T Suzuki
- T Vo
- TJ Haley
- V Krishnan
- X Zhao
- X Zhao
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Serotonergic Modulation of Nociceptive Circuits in Spinal Cord Dorsal Horn
- Author
- Abe K.
- Ahn A.H.
- Al Ghamdi K.S.
- Alhaider A.A.
- Ali Z.
- Amaya-Castellanos E.
- Attal N.
- Bardin L.
- Bardoni R.
- Basbaum A.I.
- Betelli C.
- Bonnefont J.
- Brenchat A.
- Brenchat A.
- Brenchat A.
- Buhler A.V.
- Buritova J.
- Cai Y.Q.
- Cardenas C.G.
- Cardenas C.G.
- Cardenas L.M.
- Colpaert F.C.
- Conte D.
- Cui M.
- Daval G.
- Del Mar L.P.
- Dickie A.C.
- Doly S.
- Doly S.
- Eide P.K.
- el-Yassir N.
- el-Yassir N.
- Fields H.L.
- Fonseca M.I.
- Fukushima T.
- García-Ramírez D.L.
- Garraway S.M.
- Garraway S.M.
- Garraway S.M.
- Gautier A.
- Gjerstad J.
- Gjerstad J.
- Glaum S.R.
- Goadsby P.J.
- Hammond D.L.
- Hayashida K.I.
- Headley P.M.
- Hentall I.D.
- Hori Y.
- Horiuchi H.
- Huang J.
- Hylden J.L.
- Ito A.
- Jennings E.A.
- Jeong H.J.
- Jordan L.M.
- Kato G.
- Kayser V.
- Khasabov S.G.
- Kia H.K.
- Kidd E.J.
- Kim J.M.
- Kwiat G.C.
- Laporte A.M.
- Li H.
- Li P.
- Lin Q.
- Liu F.Y.
- Liu F.Y.
- Liu X.G.
- Liu X.G.
- Lopez-Garcia J.A.
- Lopez-Garcia J.A.
- Lopez-Garcia J.A.
- Lu Y.
- Lucas-Osma A.M.
- Maeshima T.
- Marlier L.
- Marlier L.
- Maxishima M.
- Meuser T.
- Millan M.J.
- Morales M.
- Murase K.
- Nadeson R.
- Nicholson R.
- Nitanda A.
- Oatway M.A.
- Obata H.
- Obata H.
- Okamoto K.
- Okazaki R.
- Paul D.
- Perrin F.E.
- Peters C.M.
- Pierce P.A.
- Pierce P.A.
- Pompeiano M.
- Pompeiano M.
- Potrebic S.
- Rahman W.
- Ren L.Q.
- Ridet J.L.
- Rita Bardoni
- Robertson B.
- Rocha-González H.I.
- Rudomin P.
- Sasaki M.
- Sasaki M.
- Schmauss C.
- Schwaller F.
- Scott J.A.
- Shay B.L.
- Smith K.M.
- Sorkin L.S.
- Svensson C.I.
- Tecott L.H.
- Thibault K.
- Thor K.B.
- Todd A.J.
- Todorovic S.
- Tomoyose O.
- Tsuchiya M.
- Van Steenwinckel J.
- Van Steenwinckel J.
- Viguier F.
- Viguier F.
- Wang J.K.
- Wang Y.Y.
- Wattiez A.S.
- Wei F.
- Worsley M.A.
- Xie D.J.
- Xu W.
- Yasaka T.
- Yoshimura M.
- You H.J.
- Zeitz K.P.
- Zemlan F.P.
- Zhang Y.Q.
- Zhang Z.
- Zhao Z.Q.
- Zhao Z.Q.
- Zhuo M.
- Zhuo M.
- Zuena A.R.
- Publication venue
- 'Bentham Science Publishers Ltd.'
- Publication date
- Field of study
5-HT 7
- Author
- Abbas AI
- Antle MC
- Belenky MA
- Bonaventure P
- Bonaventure P
- Brenchat A
- Diaz-Reval MI
- Dogrul A
- Doly S
- Duncan MJ
- Ehlen JC
- Enza Lacivita
- Francesco Berardi
- Gardani M
- Glass JD
- Guscott M
- Gustafson EL
- Harte SE
- Hedlund PB
- Hedlund PB
- Hedlund PB
- Hedlund PB
- Holmberg P
- Hoyer D
- Johnson KW
- Kim SH
- Leopoldo M
- Leopoldo M
- Leopoldo M
- Lovenberg TW
- Marcello Leopoldo
- Martínez-García E
- Mengod G
- Monsma FJ
- Neumaier JF
- Perez-García GS
- Pittalà V
- Raubo P
- Roberto Perrone
- Roberts AJ
- Ruat M
- Sarkisyan G
- Schoeffter P
- Sethy VH
- Shibata M
- Sprouse J
- Sprouse J
- Terrón JA
- Terrón JA
- Thomas DR
- Tjølsen A
- To ZP
- Vanhoenacker P
- Varnäs K
- Verheggen R
- Villalon CM
- Volk B
- Waeber C
- Wesolowska A
- Wesolowska A
- Witkin JM
- Ying SW
- Yu GD
- Publication venue
- 'Informa Healthcare'
- Publication date
- Field of study
Towards metabolically stable 5-HT7 receptor ligands: a study on 1-arylpiperazine derivatives and related isosters
- Author
- A Brenchat
- A Wesolowska
- AI Abbas
- AJ Bojarski
- Andrzej J. Bojarski
- B Volk
- Beata Duszynska
- C Kikuchi
- C Prakash
- CB Reese
- D Hoyer
- D Hoyer
- D Leo
- Daniela Patarnello
- E Kvachnina
- E Lacivita
- Enza Lacivita
- Francesco Berardi
- G Luo
- G Sarkisyan
- GE Martin
- Grzegorz Satala
- H Geneste
- IT Forbes
- K Natsui
- L Citrome
- L Costa
- L Jia
- L Speranza
- M Guscott
- M Leopoldo
- M Leopoldo
- M Leopoldo
- M Leopoldo
- M Leopoldo
- M Nakamura
- M Paillet-Loilier
- Marcello Leopoldo
- Mauro Niso
- MH Paluchowska
- Nicola A. Colabufo
- P Bonaventure
- P Raubo
- P Zajdel
- Paola De Giorgio
- PB Hedlund
- PB Hedlund
- R Mannhold
- RA Medina
- Roberto Perrone
- S Caccia
- SE Harte
- TR Elworthy
- V Pittala
- V Pittalà
- W Spooren
- W-N Wu
- Y Cheng
- Z Miao
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study