9 research outputs found
Prediction the probability of retrombosis in patients with acute coronary syndrome and ST-segment elevation during medical reperfusion therapy and percutaneous intervention
- Author
- Publication venue
- БНТУ
- Publication date
- 28/02/2020
- Field of study
Prediction the probability of retrombosis in patients with acute coronary syndrome and ST-segment elevation during medical reperfusion therapy and percutaneous intervention
- Author
- Publication venue
- БНТУ
- Publication date
- 01/01/2014
- Field of study
An X-ray diffraction investigation of the reaction between molybdenum powder and manganese additions during sintering
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Variability of oral bioavailability for low dose methotrexate in rats
- Author
- B. K. Reuter
- C. H. Lifschitz
- C. Lebbe
- D. D. Shen
- D. K. Smith
- D. Oguey
- G. D. Weinstein
- G. G. Altman
- G. G. Popovici
- H. Tanaka
- I. Cobden
- I. D. Capel
- J. G. Gispen
- J. Jolivet
- J. L. Dhondt
- J. M. Kremer
- J. M. Kremer
- J. W. L. Robinson
- K. Kobayashi
- L. Cuzzolin
- L. E. Jolly
- M. Ahern
- M. E. Weinblatt
- M. Masuda
- M. Nakamaru
- N. M. Davices
- P. Statkevich
- R. Kakuno
- S. H. Wan
- T. Kuroda
- V. M. K. Venho
- W. A. Bleyer
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Management of Elevated Low-Density Lipoprotein Cholesterol
- Author
- Anitschkow N
- Anum EA
- Ballantyne C
- Bauer KS
- Bays H
- Bittner V
- Canner PL
- Capuzzi DM
- Carlson LA
- Catapano AL
- Chambless LE
- Courtney RD
- Davidson MH
- Davidson MH
- Davidson MH
- Davis HR
- Dyer A
- Eklund G
- Enos W
- Faxon DP
- Genest J
- Goldstein JL
- Goldstein JL
- Gray DR
- Guyton JR
- Herrmann J
- Higgins M
- Hoeg JM
- Howard BV
- Hunt KJ
- Jackson S
- Jin FY
- Kennedy M
- Keung AC
- Keys A
- Keys A
- Knopp RH
- Knopp RH
- Kosoglou T
- Kosoglou T
- Kreisberg RA
- Krishna G
- LaBarthe D
- Law MR
- Leary T
- Liao Y
- Lloyd-Jones DM
- McMichael J
- Melani L
- Morgan JM
- Packard CJ
- Paulose-Ram R
- Pekkanen J
- Punwani N
- Reddy KS
- Reyderman L
- Reyderman L
- Rothstein WG
- Schaefer EJ
- Schneider WJ
- Stamler J
- Stamler J
- Statkevich P
- Stein EA
- Stemmermann G
- Steyn K
- Tunstall-Pedoe H
- van Heek M
- Windhaus A
- Wong N
- Worth R
- Zhu Y
- Zhu Y
- Publication venue
- 'Informa UK Limited'
- Publication date
- Field of study
A new role of AMP-activated protein kinase in regulating proliferation of mesenchymal stem cells
- Author
- A. A. B. Van Veen
- A. A. Lammertsma
- A. Akhmedov
- A. Angelini
- A. Angelini
- A. Bairamov
- A. Baldini
- A. Bayes-Genis
- A. Berezin
- A. Berezin
- A. Bye
- A. C. Meli
- A. Caporali
- A. Caporali
- A. Caporali
- A. Cardinali
- A. Carpi
- A. Chernova
- A. Chester
- A. Coulter
- A. Cross
- A. Czikora
- A. D. Kokkinos
- A. Daniels
- A. Darago
- A. De Pauw
- A. Dembinska-Kiec
- A. Didangelos
- A. E. Messer
- A. E. Messer
- A. E. Messer
- A. F. Leite-Moreira
- A. F. Leite-Moreira
- A. F. Leite-Moreira
- A. Farkas
- A. Frazier
- A. Friart
- A. G. Grdinic
- A. Garcia Escudero
- A. Gastaldelli
- A. Gonzalez-Tendero
- A. Gonzalez-Tendero
- A. Gorlach
- A. Graffeuil
- A. Grahl
- A. Grdinic
- A. H. Maass
- A. H. Ottesen
- A. H. Wagner
- A. Heidari
- A. Herman
- A. Hultgardh-Nilsson
- A. Hussain
- A. I. Suceveanu
- A. J. A. Raaijmakers
- A. J. Tijsen
- A. Jaiswal
- A. K. Dinda
- A. K. Najmi
- A. K. Sharma
- A. Kapoor
- A. Kelly
- A. Kiss
- A. Koller
- A. Kostareva
- A. Kristof
- A. L. Harris
- A. L. Pires
- A. Lacampagne
- A. Leite-Moreira
- A. Leuner
- A. Llacer
- A. Llucia-Valldeperas
- A. Lymperopoulos
- A. M. Lompre
- A. M. Marks
- A. M. Miller
- A. M. Murphy
- A. M. Soldatova
- A. M. Soldatova
- A. Mogielnicki
- A. N. Price
- A. Oikawa
- A. Oikawa
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- V. Y. Hoymans
- W. Buczko
- W. E. Louch
- W. G. Daniel
- W. H. Van Gilst
- W. Husada
- W. J. Koch
- W. J. Koch
- W. J. Paulus
- W. J. Van Der Laarse
- W. J. Wijnen
- W. Kuzyniak
- W. Linke
- W. M. Blankesteijn
- W. R. Giles
- W. S. Speidl
- W. Schgoer
- W.-T. Wu
- X. Yin
- X. Yin
- Y. Ajiro
- Y. M. Pinto
- Y. Rudy
- Y. U. A. Yuricheva
- Y. Y. Wong
- Y. Yao
- Z. Gaciong
- Z. H. N. Kot
- Z. Husti
- Z. Papp
- Z. Pesevski
- Z. S. Kohajda
- Z. V. Varga
- Z. Vamos
- Z. Vucinic
- Z. Yassin
- Z. Yassin
- Publication venue
- 'Oxford University Press (OUP)'
- Publication date
- 01/01/2012
- Field of study
Purpose: Natriuretic peptides (NPs) administered during early reperfusion are protective in models of myocardial infarction. A previous study examining the endogenous components of B-type natriuretic peptide (BNP) protection of reperfused myocardium, implicated both sarcolemmal (s) KATP and mitochondrial (m) KATP channels. The indirect evidence characterising the relationship between BNP signalling and KATP was obtained using sulphonylurea receptor inhibitors in a rat isolated heart model of ischaemia-reperfusion injury. Here we seek to further examine the relationship between NPs and sKATP openings using single channel electrophysiology. Given our previous findings and the overarching consensus that cardioprotective autacoids open KATP channels, it was hypothesised that NPs elicit sKATP opening.
Methods: Cardiomyocyte isolation. Left ventricular cardiomyocytes were isolated from male Sprague-Dawley rat hearts subjected to enzymatic digestion with Liberase Blendzyme DL. Cardiomyocytes were cultured overnight in Medium 199, prior to patch clamp. Single channel patch clamp. Single channel recordings at room temperature (22°C) were made from cell attached patches bathed in Na+ Locke, pH 7.2. The recording pipette contained high KCl (140 mM), pH 7.2. Recordings (45 sec) were made over a range of patch potentials (0, -30, -60, -90, -120 mV), in the absence (control) and in the presence of bath applied BNP (10, 100 nM and 1 µM), pinacidil (200 µM) or pinacidil vehicle (DMSO, 0.25%). Recordings were also made with BNP and pinacidil applied concomitantly. Data are mean ± S.E.M.
Results: The current voltage relationship of sKATP under control conditions was linear at –ve patch potentials, the mean conductance being 52.9 ± 1.8 pS (n = 18 hearts, n = 35 cells). Pinacidil caused a four fold increase in sKATP open probability compared to control. Mean channel conductance in the presence of pinacidil was 59.9 ± 1.9 pS (n = 16 hearts, n = 44 cells). Interestingly BNP at all concentrations had negligible effects on sKATP open probability and unitary conductance. However, BNP at all concentrations and patch potentials inhibited pinacidil induced sKATP openings, restoring channel open probability to baseline.
Conclusion: These data illustrate the inhibitory effect of NP signalling on sKATP function in the cardiomyocyte under normoxia. They are concordant with the inhibitory effect of atrial NP on KATP in the pancreatic beta cell, but are in apparent conflict with the current cardioprotection paradigm. However, differential effects on sKATP and mKATP and the effects of hypoxia-reoxygenation require further exploration
Renal Drug Transporters and Drug Interactions.
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- A Allen
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- T Watanabe
- T Yamazaki
- T Yasujima
- T Yokooji
- T Zoto
- TB Stage
- TB Tjandra-Maga
- TB Tjandramaga
- TF Solbach
- Thierry Buclin
- TJ Urban
- TN Kakuda
- TN Winter
- TS Bekaii-Saab
- TS Tracy
- U Jaehde
- U Roy
- U Schmitt
- V Gorboulev
- V Juhasz
- V Lecureur
- V Lecureur
- V Martin
- V Sikri
- V Vallon
- V Vallon
- VA Eagling
- VC Oliveira Almeida De
- VJ Wacher
- VL Damaraju
- VR Challa
- W Kim
- W Liu
- W Mueck
- W Siegmund
- W Wang
- W Yamashiro
- W Zhang
- W-Q Chen
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- WM Suhre
- X Bossuyt
- X Chu
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- X Li
- X Ming
- X Ming
- X Ming
- X Wang
- X Wu
- X Wu
- X Wu
- X Wu
- X Wu
- X Zhang
- X Zheng
- XJ He
- XY Chu
- Y Adachi
- Y Cheng
- Y Feng
- Y Fujita
- Y Fukuda
- Y Hagos
- Y Hagos
- Y Hagos
- Y Hagos
- Y Hashiguchi
- Y Honda
- Y Imamura
- Y Imamura
- Y Kato
- Y Kido
- Y Kido
- Y Kobayashi
- Y Kurata
- Y Matsuo
- Y Matsuo
- Y Moriyama
- Y Nagasaka
- Y Nozaki
- Y Nozaki
- Y Nozaki
- Y Pan
- Y Shibayama
- Y Shibayama
- Y Shima
- Y Shirasaka
- Y Shirasaka
- Y Shitara
- Y Shitara
- Y Shu
- Y Su
- Y Sugimoto
- Y Tanaka
- Y Tanigawara
- Y Tanihara
- Y Tanihara
- Y Tomita
- Y Tschuppert
- Y Uchida
- Y Urakami
- Y Urakami
- Y Urakami
- Y Urakami
- Y Urakami
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Uwai
- Y Yamakawa
- Y Yamasaki
- Y Zhang
- Y Zhang
- Y Zhou
- Y Zhu
- Y-F Cheng
- Y-H Han
- Y-H Zhang
- Y-J Piao
- YA Chen
- YH Oh
- YH Peng
- YR Ma
- Z Cheng
- Z Gai
- Z Li
- Z Shen
- Z Tong
- Z Yang
- Z-J Wang
- ZS Chen
- ZS Chen
- ZS Chen
- ZS Chen
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/08/2017
- Field of study
Transporters in proximal renal tubules contribute to the disposition of numerous drugs. Furthermore, the molecular mechanisms of tubular secretion have been progressively elucidated during the past decades. Organic anions tend to be secreted by the transport proteins OAT1, OAT3 and OATP4C1 on the basolateral side of tubular cells, and multidrug resistance protein (MRP) 2, MRP4, OATP1A2 and breast cancer resistance protein (BCRP) on the apical side. Organic cations are secreted by organic cation transporter (OCT) 2 on the basolateral side, and multidrug and toxic compound extrusion (MATE) proteins MATE1, MATE2/2-K, P-glycoprotein, organic cation and carnitine transporter (OCTN) 1 and OCTN2 on the apical side. Significant drug-drug interactions (DDIs) may affect any of these transporters, altering the clearance and, consequently, the efficacy and/or toxicity of substrate drugs. Interactions at the level of basolateral transporters typically decrease the clearance of the victim drug, causing higher systemic exposure. Interactions at the apical level can also lower drug clearance, but may be associated with higher renal toxicity, due to intracellular accumulation. Whereas the importance of glomerular filtration in drug disposition is largely appreciated among clinicians, DDIs involving renal transporters are less well recognized. This review summarizes current knowledge on the roles, quantitative importance and clinical relevance of these transporters in drug therapy. It proposes an approach based on substrate-inhibitor associations for predicting potential tubular-based DDIs and preventing their adverse consequences. We provide a comprehensive list of known drug interactions with renally-expressed transporters. While many of these interactions have limited clinical consequences, some involving high-risk drugs (e.g. methotrexate) definitely deserve the attention of prescribers
Renal Drug Transporters and Drug Interactions
- Author
- A Allen
- A Amphoux
- A Aslamkhan
- A Azzariti
- A Brandoni
- A Collett
- A Courtois
- A Crowe
- A Dahan
- A Dahan
- A Dahan
- A Dahlin
- A D’Emanuele
- A Enomoto
- A Enomoto
- A Futatsugi
- A Gaowa
- A Geick
- A Gupta
- A Hamada
- A Horie
- A Kamizono
- A Kawase
- A Koenen
- A Komatsuda
- A Kunze
- A Lazar
- A Lespine
- A Maeda
- A Maeda
- A McCormick
- A Milane
- A Mulgaonkar
- A Nakayama
- A Nies
- A Oka
- A Ose
- A Owen
- A Pawarode
- A Poirier
- A Rizwan
- A Servais
- A Soldner
- A Somogyi
- A Somogyi
- A Somogyi
- A Somogyi
- A Vildhede
- A Yamada
- A Yamada
- A Yonezawa
- A Yonezawa
- AA El-Sheikh
- AA Ela El
- AA Somogyi
- AA Somogyi
- AAK El-Sheikh
- AAK El-Sheikh
- AAK El-Sheikh
- AAK El-Sheikh
- AB Shapiro
- AE Busch
- AE Herwaarden van
- AE Kim
- AG Hotchkiss
- AH Schinkel
- AH Schinkel
- AH Schinkel
- AJ Dudley
- AJ Dudley
- AJ Scheen
- AL Dzierlenga
- AL VanWert
- AL VanWert
- AL Walker
- AM Al-Mohizea
- AM Bergman
- AM Hecken van
- AN Shaik
- Anton Ivanyuk
- AR Asif
- AS Mulato
- AS Ray
- AS Windass
- AS Windass
- AT Nies
- AT Wolman
- B Astorga
- B Feng
- B Feng
- B Fleisher
- B Greiner
- B Grover
- B Grover
- B Haenisch
- B Poller
- B Wenge
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- BC Burckhardt
- BC Ferslew
- BG Hardy
- BG Hardy
- BH Long
- BJ Gurley
- BL Lum
- BL Mason
- BM Schmitt
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- BR Green
- C Chen
- C Chen
- C Chu
- C Fahrmayr
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- YH Oh
- YH Peng
- YR Ma
- Z Cheng
- Z Gai
- Z Li
- Z Shen
- Z Tong
- Z Yang
- Z-J Wang
- ZS Chen
- ZS Chen
- ZS Chen
- ZS Chen
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
The state of the art of biospeleology in Russia and other countries of the former Soviet Union: A review of the cave (endogean) invertebrate fauna. 3. References
- Author
- A. Casale
- A. Evsyukov
- A. Jaworowski
- A. Riedel
- A. Schellenberg
- A. Sendra
- A. Vandel
- A. Winkler
- A. Winkler
- A.A. Nadolny
- A.A. Nadolny
- A.A. Nadolny
- A.A. Sadovsky
- A.A. Shileiko
- A.A. Shileiko
- A.B. Babenko
- A.B. Babenko
- A.B. Babenko
- A.D. Petrova-Nikitina
- A.G. Koval
- A.G. Koval
- A.G. Koval
- A.G. Koval
- A.G. Koval
- A.I. Andreev
- A.I. Camacho
- A.I. Yankovskaya
- A.I. Yankovskaya
- A.I. Yankovskaya
- A.I. Yankovskaya
- A.L. Behning
- A.L. Behning
- A.L. Behning
- A.L. Brodsky
- A.L. Brodsky
- A.L. Smirnov
- A.M. Shugurov
- A.M. Shugurov
- A.M. Sokolova
- A.N. Chemeris
- A.N. Derzhavin
- A.N. Derzhavin
- A.N. Derzhavin
- A.N. Derzhavin
- A.N. Derzhavin
- A.N. Derzhavin
- A.N. Korchagin
- A.N. Shumeev
- A.N. Tchemeris
- A.O. Kovtun
- A.P. Mylnikov
- A.P. Mylnikov
- A.P. Semenov
- A.P. Semenov-Tyan-Shansky
- A.P. Stadnichenko
- A.S. Reboleira
- A.S. Skorikow
- A.S. Skorikow
- A.S. Zamotajlov
- A.S. Zamotajlov
- A.V. Ereskovsky
- A.V. Martynov
- A.V. Martynov
- A.V. Martynov
- A.V. Martynov
- A.V. Martynov
- A.V. Mukhanov
- A.V. Puchkov
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- A.W. Skalski
- A.Ya. Bazikalova
- A.Ya. Bazikalova
- B. Matyushkin
- B. Szczęsny
- B. Wolf
- B.I. Ioffe
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- D.N. Kobakhidze
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- E.V. Komarov
- E.V. Mikhaljova
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- G.A. Prokopov
- G.A. Prokopov
- G.A. Prokopov
- G.E. Davidian
- G.J. Bey-Bienko
- G.M. Abdurakhmanov
- G.S. Karaman
- G.S. Karaman
- G.S. Poli
- G.Ya. Bey-Bienko
- G.Ya. Bey-Bienko
- H. Enghoff
- H. Lohmander
- H. Read
- H. Schmalfuss
- I. Balashov
- I. Balashov
- I. Belousov
- I. Belousov
- I. Eliava
- I. Marin
- I. S. Turbanov
- I. Turbanov
- I. Zagorodnyuk
- I.A. Belousov
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- I.I. Dedyu
- I.I. Dedyu
- I.I. Dedyu
- I.I. Dedyu
- I.I. Lapshov
- I.I. Malevich
- I.J. Kaprus
- I.J. Kaprus
- I.M. Karaman
- I.M. Likharev
- I.N. Marin
- I.S. Turbanov
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- I.S. Zharkova
- I.V. Dovgal
- I.V. Dovgal
- I.V. Dovgal
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- I.V. Dovgal
- I.V. Dovgal
- I.V. Zagorodnyuk
- J. Breit
- J. Carl
- J. Carl
- J. Christophoryová
- J. Martens
- J. Martens
- J.-P. Henry
- J.A. Birstein
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- K. Evtushenko
- K. Verhoeff
- K. Verhoeff
- K.A. Satunin
- K.B. Gongalsky
- K.V. Evtushenko
- K.V. Makarov
- K.V. Makarov
- K.W. Verhoeff
- L. Deharveng
- L.D. Arutyunova
- L.V. Kulkina
- L.V. Samchishina
- L.V. Vorobieva
- M. Krumpal
- M. Krumpal
- M. Murvanidze
- M. Potapov
- M. Straškraba
- M.-J. Turquin
- M.B. Potapov
- M.B. Potapov
- M.B. Potapov
- M.D. Moroz
- M.I. Shapovalov
- M.M. Kovblyuk
- M.M. Novikov
- M.S. Gilyarov
- M.S. Gilyarov
- M.S. Harvey
- M.S. Harvey
- M.V. Chertoprud
- M.V. Stolyarov
- M.V. Vinarski
- N. Gourbault
- N. Grese
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- N.A. Akatova
- N.A. Gvozdetski
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- N.D. Lebedev
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- O.A. Kovtun
- O.A. Kovtun
- O.A. Kovtun
- O.A. Kovtun
- O.G. Reznichenko
- O.I. Chibisova
- O.I. Schmalhauzen
- O.L. Kryzhanovskij
- O.L. Makarova
- O.V. Chekanovskaya
- O.V. Golovachev
- O.Yu. Derevenskaya
- P. Beauchamp de
- P. Hlaváč
- P. Hlaváč
- P.F.M.A. Dejean
- P.M. Giachino
- P.V. Kiyashko
- P.V. Kiyashko
- P.V. Kiyashko
- P.V. Kiyashko
- P.V. Kiyashko
- R. Djanashvili
- R. Djanashvili
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- R.V. Egorov
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- S. Barjadze
- S. Barjadze
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- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.I. Ljovuschkin
- S.K. Stebaeva
- S.L. Esyunin
- S.L. Karaman
- S.M. Iablokoff-Khnzorian
- S.M. Iablokoff-Khnzorian
- S.M. Iablokoff-Khnzorian
- S.M. Jusbaschjan
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- S.M. Khnzorian
- S.T. Lepneva
- S.V. Statkevich
- S.V. Statkevich
- S.Yu. Kleimenov
- S.Yu. Storozhenko
- Sh. Barjadze
- Sh. Barjadze
- Sh. Barjadze
- Sh. Barjadze
- Sh.R. Abdullin
- Sh.R. Abdullin
- Sh.R. Abdullin
- T. Timm
- T.N. Amelichev
- T.N. Komarova
- T.N. Vereshchagina
- T.N. Vereshchagina
- V. Golemansky
- V. Kniss
- V. Mahnert
- V. Mahnert
- V. Redikorzev
- V. Zakšek
- V.A. Isaev
- V.A. Isaev
- V.A. Kniss
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- V.A. Kniss
- V.A. Kniss
- V.A. Kniss
- V.A. Kniss
- V.A. Kniss
- V.B. Rizun
- V.E. Pichka
- V.F. Boldyrev
- V.F. Nikolyuk
- V.G. Pliginsky
- V.G. Pliginsky
- V.G. Pliginsky
- V.G. Shilenkov
- V.I. Gusarov
- V.I. Mikhalevich
- V.I. Monchenko
- V.I. Monchenko
- V.I. Monchenko
- V.I. Monchenko
- V.I. Monchenko
- V.I. Monchenko
- V.I. Monchenko
- V.I. Monchenko
- V.I. Shadin
- V.I. Shchurov
- V.I. Zhadin
- V.K. Chernyavsky
- V.M. Rylov
- V.N. Kurnakov
- V.N. Luchnik
- V.N. Vishnyakova
- V.O. Kozminykh
- V.P. Semernoi
- V.S. Labay
- V.V. Anistratenko
- V.V. Petryashev
- V.V. Polishchuk
- V.V. Takhteev
- V.V. Takhteev
- V.Yu. Dolzhanskij
- V.Yu. Dolzhanskij
- V.Yu. Dolzhanskij
- W. Michaelsen
- W. Michaelsen
- W. Schawaller
- W. Schawaller
- W. Szymczakowski
- Y.I. Kantor
- Ya.I. Starobogatov
- Ya.I. Starobogatov
- Ya.I. Starobogatov
- Ya.N. Lebedinsky
- Ya.N. Lebedinsky
- Ya.N. Lebedinsky
- Ya.P. Vlasov
- Yu. Mazei
- Yu.A. Mazei
- Yu.A. Rudyakov
- Yu.E. Gladkova
- Yu.E. Gladkova
- Yu.E. Gladkova
- Yu.G. Giginyak
- Yu.M. Marusik
- Yu.P. Malkov
- Yu.S. Volkova
- Z.I. Izzatullaev
- Z.I. Izzatullaev
- Z.S. Bronstein
- Publication venue
- 'Pleiades Publishing Ltd'
- Publication date
- 16/12/2020
- Field of study