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10 research outputs found
An expedient strategy for the diversity-oriented synthesis of macrocyclic compounds with natural product-like characteristics
Author
Aeluri
Aeluri
+45Â more
Beckmann
Bock
Cornelius J. O'Connor
David R. Spring
Driggers
Galloway
Grossmann
Guduru
Hannah F. Sore
Hill
Horne
Isidro-Llobet
Isidro-Llobet
Jamie E. Stokes
Jefferson
Jimmidi
Joe J. Ciardiello
Kantevari
Kopp
Madsen
Marcaurelle
Marsault
Marsault
Maurya
Mullard
Muller
Newman
Nielsen
O'Connell
O'Connell
Russell
Sauer
Sauer
Schreiber
Socha
Ta
Thomas
Trabocchi
Warren R.J.D. Galloway
Wessjohann
Wessjohann
Wyatt
Wyatt
Yu
Yuteng Wu
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
The Dimroth rearrangement as a probable cause for structural misassignments in imidazo[1,2-a]pyrimidines: A N-labelling study and an easy method for the determination of regiochemistry
Author
Abignente
Aeluri
+26Â more
Anaflous
Angela J. Russell
Ashry
Borisov
Carballares
Chavignon
Chen
Francis X. Wilson
Ganesamoorthy
Goel
Graham M. Wynne
Guerret
Jacquier
Jensen
Li
Liu
Majumder
Maria Chatzopoulou
Mosquera
Nicky J. Willis
R. Fernando MartĂnez
Rasapalli
Rathke
Solberg
Stephen G. Davies
Timothy D.W. Claridge
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Design, Synthesis and Evaluation of 2,5-Diketopiperazines as Inhibitors of the MDM2-p53 Interaction
Author
A El-Faham
A Feki
+53Â more
A Ganesan
AD Borthwick
BP Orner
C Dalvit
D Reed
D Rognan
D Sun
DA Freedman
DC Fry
DG Myszka
ER Burkhardt
F Gonzalez-Lopez de Turiso
F Jam
F Mutulis
F Toledo
FP Gasparro
G Papalia
H Yin
J Momand
Jaeki Min
JC Brown
JD Park
JH Lee
JM Nigro
JP Plante
K Michelsen
KH Vousden
Kristina Luthman
LF Fieser
LG Milroy
LT Vassilev
Luigi Iconaru
M Aeluri
M Aeluri
M Tullberg
M Tullberg
M Wade
M. Brett Waddell
M. Tullberg
Maria Quant
Mariell Pettersson
Morten Grøtli
N Bharatham
PH Kussie
R Nishizawa
R. Kiplin Guy
Richard W. Kriwacki
S Shangary
SM Biros
T Stiewe
V Azzarito
Y Rew
Y Zhao
Publication venue
'Public Library of Science (PLoS)'
Publication date
Field of study
No full text
Crossref
Tetrahydroquinoline-Derived Macrocyclic Toolbox: The Discovery of Antiangiogenesis Agents in Zebrafish Assay
Author
Aeluri M.
Ajay A.
+33Â more
Arkin M. R.
Arya P.
Arya P.
Arya P.
Boger D. L.
Couve-Bonnaire S.
Dandapani S.
Dasari B.
Dockendorff C.
Driggers E. M.
Grubbs R. H.
Grubbs R. H.
Grubbs R. H.
Kimmel C. B.
Kitambi S. S.
Kitambi S. S.
Kitambi S. S.
Marcaurelle L. A.
Moretti J. D.
Newman D. J.
Pawson T.
Peng L. F.
Peterson R. T.
Prakesch M.
Prakesch M.
Reayi A.
Schreiber S. L.
Scott J. D.
Serbedzija G. N.
Sharma U.
Stanton B. Z.
Vogt A.
Wells J. A.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
8-Triazolylpurines: Towards Fluorescent Inhibitors of the MDM2/p53 Interaction
Author
A Dierckx
A Ganesan
+49Â more
AL Jochim
B Vogelstein
BP Orner
C Dalvit
C Dyrager
D Bliman
D Sun
DA Horton
David Bliman
DO Cicero
DS Pedersen
E Danelius
F Gonzalez-Lopez de Turiso
H Rosemeyer
H Yin
Jaeki Min
Jesper R. Nilsson
JH Lee
Jimmy Jacobsson
JJ Koivisto
Joakim Andréasson
JR Johansson
K Michelsen
KH Vousden
L Zhang
L Čechová
LT Vassilev
Luigi Iconaru
M Aeluri
M Fridén-Saxin
M Meldal
Mariell Pettersson
Morten Grøtli
MR Davis
N Bharatham
O Keskin
PH Kussie
R. Kiplin Guy
Richard W. Kriwacki
S Fletcher
S Fletcher
S Jones
SW Kwok
V Azzarito
WE Stites
WS Horne
Y Rew
Y Zhao
Y-T Chang
Publication venue
'Public Library of Science (PLoS)'
Publication date
Field of study
No full text
Crossref
A peptide mimicking the binding sites of VEGF-A and VEGF-B inhibits VEGFR-1/-2 driven angiogenesis, tumor growth and metastasis
Author
A Basile
A Pettersson
+42Â more
A Sadremomtaz
A Ĺ ali
B Gautier
B-Z Qian
C Dunk
CL Roland
D Hanahan
D-G Bae
DB Cines
ER Camp
H Matsuzaki
H Zeng
J Folkman
J Gille
JC Weddell
K Suto
L Rosa De
L Wang
L Wang
M Aeluri
M Prewett
M Shibuya
MJ Miller
MS O’Reilly
N Ferrara
N Ferrara
N Rahimi
P Chames
P-E Neagoe
PI Imoukhuede
PN Bernatchez
R Heidenreich
S Crespo
S Iyer
T Mesti
V Goncalves
Y Mebratu
Y Sakurai
Y Tu
YA Muller
YA Muller
Z Zhou
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Solvent-free silica-promoted multicomponent condensation: synthesis of highly functionalized piperidines
Author
A Corma
A Dömling
+64Â more
A Schotte
AB Beeler
AD Elbein
Adinath Majee
AK Banerjee
Alakananda Hajra
AT Khan
AT Khan
Avik Kumar Bagdi
BC Ranu
BC Ranu
BC Ranu
BC Ranu
BC Ranu
BC Ranu
BM Trost
C Mukhopadhyay
D O’Hagan
DJ RamĂłn
F Shi
FA Davis
G Brahmachari
G Spagnol
H Bin
H-J Wang
I Ugi
JA Dekus
JC Jaen
JH Clark
JH Clark
JP Yevich
JS Ghomi
JW Daly
K Kamei
K Takasu
M Baumann
M Lashkari
M Misra
M Rahman
M Sales
MJ Climent
MSR Murty
PA Clarke
PA Wender
PT Anastas
R Aeluri
R Ramachandran
RM Carballo
RS Verma
S Fustero
S Mishra
S Petit
S Targum
S Verma
SL Gwaltney II
Sougata Santra
SS Sajadikhah
Sudarshan Das
TP Lebold
V Nair
X Li
Y Matsushita
Y Yamanishi
Y Zhou
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
An Intriguing Correlation Based on the Superimposition of Residue Pairs with Inhibitors that Target Protein-Protein Interfaces
Author
A Whitty
AA Bogan
+53Â more
AE Robin
AJ Soures
AM Petro
AP Higeruelo
B Ma
BO Kuenemann
C Fang
CD Thanos
CM Labbé
CR Munteanu
D Marcotte
D Rajamani
DC Fry
DC Fry
DC Fry
DEV Pires
DL Buckley
G Zinzalla
GM KeserĂĽ
HC Fuller
I Van Molle
IS Moreira
J Porter
JA Wells
JM Davis
JM Zimmerman
KA Sharp
LMC Meireles
LMC Meireles
M Aeluri
M Asano
M Congreve
M Rickert
MR Arkin
MR Arkin
O Keskin
O Sperandio
PA Karplus
PJ Hajduk
R Bougeas
RM Brady
T Kortemme
T Ohta
T Oltersdorf
TL Nero
TS Peat
VM Gongçalves-Almeida
X Li
X Morell
Y Che
Y Cheng
Z Shiokawa
Z Zhang
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Resveratrol serves as a protein-substrate interaction stabilizer in human SIRT1 activation
Author
A Satoh
A Satoh
+58Â more
AS Banks
AW Gotz
BH Liu
BP Hubbard
BP Hubbard
CHS Aylett
CI Bayly
D Chen
D Chen
D Herranz
D Rooklin
DA Sinclair
DF Cao
EF Pettersen
EJ Kim
F Giordanetto
GT Diaz-Gerevini
GV Papamokos
H Dai
H Dai
HC Hsu
HJ Yang
HY Cohen
J Liang
JA Baur
JA Baur
JA IBaur
JA Maier
JC Milne
JG IWood
JH Chung
JL Avalos
JT Rodgers
JW Choi
KT Howitz
L Bordone
L Guarente
L Guarente
L Guarente
LG Milroy
M Aeluri
M Kaeberlein
M Lakshminarasimhan
M Pacholec
MB Peters
MS Cosgrove
MT Borra
NL Price
P Cieplak
P Gut
R Salomon-Ferrer
RI Tennen
S Imai
S Kume
S Schenk
TJ Dolinsky
U Ryde
YW Shi
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Spiro-oxindoles as a Promising Class of Small Molecule Inhibitors of p53–MDM2 Interaction Useful in Targeted Cancer Therapy
Author
A Aguilar
A Bertamino
+96Â more
A Czarna
A Kamal
A Khan
A Mullard
A Vazquez
AG Herman
AS Azmi
AS Azmi
AS Azmi
AZ Gonzalez
B Hu
B Vogelstein
B Yu
BA Chabner
BT Vassilev Vu
BT Vu
C Avendano
C Riedinger
C Tovar
CJ Ribeiro
D Sun
DE Gerber
DP Lane
G Jones
GA Masters
GM Popowicz
H Yin
HP Beck
I Collins
I Gomez-Monterrey
I Ray-Coquard
IR Hardcastle
J Canon
J Momand
JA Kritzer
JC Carry
JE Tanner
JG Allen
JJ Marugan
JJ Qin
JJ Qin
K Ding
K Ding
K Ding
K Zak
KH Khoo
KH Vousden
KL Bill
L Weber
LA Torre
M Aeluri
M Lacroix
M Millard
M Vanneman
M Wade
M Wade
M Wade
MJ Lind
ML Verdonk
MP Dickens
MR Stratton
N Chessum
NR Ball-Jones
P Chene
P Hainaut
P Raboisson
PH Kussie
Q Ding
Q Zhang
R Zhang
RM Mohammad
S Aggarwal
S Hoelder
S Kummar
S Shangary
S Shangary
S Shangary
S Wang
S Wang
S Yu
SH Sun
SL Schreiber
SM Picksley
SR Rheingold
T Fu
T Terzian
T Zheng
UM Moll
V Bottger
W Huang
Y Ma
Y Rew
Y Zhao
Y Zhao
Y Zhao
YH Bae
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref