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9 research outputs found
Simulations of Shikimate Dehydrogenase from Mycobacterium tuberculosis in Complex with 3-Dehydroshikimate and NADPH Suggest Strategies for MtbSDH Inhibition
Author
Hannongbua Supa
Kamsri Pharit
+4 more
Mulholland Adrian
Pungpo Pornpan
Punkvang Auradee
Spencer James
Publication venue
'American Chemical Society (ACS)'
Publication date
22/04/2019
Field of study
Get PDF
Explore Bristol Research
Insight into the Key Structural Features of Potent Enoyl Acyl Carrier Protein Reductase Inhibitors Based on Computer Aided Molecular Design
Author
Auradee Punkvang
Kodchakon Kun-asa
+5 more
Patchreenart Saparpakorn
Peter Wolschann
Pharit Kamsri
Pornpan Pungpo
Supa Hannongbua
Publication venue
'IntechOpen'
Publication date
07/12/2011
Field of study
Get PDF
IntechOpen
Discovery of novel and potent InhA inhibitors by an in silico screening and pharmacokinetic prediction
Author
Hannongbua Supa
Hanwarinroj Chayanin
+11 more
Kamsri Bundit
Kamsri Pharit
Ketrat Sombat
Kittakoop Prasat
Mulholland Adrian J
Phusi Nareudon
Pungpo Pornpan
Punkvang Auradee
Saparpakorn Patchreenart
Spencer James
Suttisintong Khomson
Publication venue
'Future Science Ltd'
Publication date
01/05/2022
Field of study
Get PDF
Explore Bristol Research
Discovery of New and Potent InhA Inhibitors as Anti-tuberculosis Agents:Structure Based Virtual Screening Validated by Biological Assays and X-ray Crystallography
Author
Blood Rosemary A
Chayajarus Kampanart
+25 more
Chen Zhaoqiang
Choowongkomon Kiattawee
Hannongbua Supa
Hanwarinroj Chayanin
Hinchliffe Philip
Hongmanee Poonpilas
Kamsri Pharit
Kittakoop Prasat
Mulholland Adrian J
Phusi Naruedon
Pornprom Thimpika
Pungpo Pornpan
Punkvang Auradee
Rattanabunyong Siriluk
Santanirand Pitak
Saparpakorn Patchreenart
Seetaha Supaporn
Songsiriritthigul Chomphunuch
Spencer James
Srimanote Potjanee
Sureram Sanya
Suttipanta Nitima
Suttisintong Khomson
Takebayashi Yuiko
Zhu Weiliang
Publication venue
'American Chemical Society (ACS)'
Publication date
27/01/2020
Field of study
Get PDF
Explore Bristol Research
Inhibition of Mycobacterium tuberculosis InhA by 3-nitropropanoic acid
Author
Hanwarinroj Chayanin
Kamsri Pharit
+10 more
Kittakoop Prasat
Pakamwong Bongkochawan
Pungpo Pornpan
Punkvang Auradee
Songsiriritthigul Chomphunuch
Spencer James
Srimanote Potjanee
Sureram Sanya
Suttipanta Nitima
Suttisintong Khomson
Publication venue
'Wiley'
Publication date
22/10/2022
Field of study
No full text
Explore Bristol Research
In silico design of novel quinazoline-based compounds as potential Mycobacterium tuberculosis PknB inhibitors through 2D and 3D-QSAR, molecular dynamics simulations combined with pharmacokinetic predictions
Author
Hannongbua Supa
Hanwarinroj Chayanin
+12 more
Kamsri Pharit
Ketrat Sombat Ketrat
Kittakoop Prasat
Mulholland Adrian J
Pungpo Pornpan
Punkvang Auradee
Saparpakorn Patchreenart
Spencer James
Sukchit Darunee
Suttisintong Khomson
Taveepanich Somjintana
Thongdee Paptawan
Publication venue
'Elsevier BV'
Publication date
28/05/2023
Field of study
No full text
Explore Bristol Research
Bioisosteric Design Identifies Inhibitors of Mycobacterium tuberculosis DNA Gyrase ATPase Activity
Author
Goudar Kirsty E
Hannongbua Supa
+18 more
Hongmanee Poonpilas
Kamsri Bundit
Kamsri Pharit
Ketrat Sombat
Kittakoop Prasat
Leanpolchareanchai Jiraporn
Mulholland Adrian J
Pakamwong Bongkochawan
Phusi Naruedon
Pungpo Pornpan
Punkvang Auradee
Sangswan Jidapa
Santanirand Pitak
Saparpakorn Patchreenart
Spencer James
Sureram Sanya
Suttisintong Khomson
Thongdee Paptawan
Publication venue
Publication date
19/04/2023
Field of study
No full text
Explore Bristol Research
Virtual Screening Identifies Novel and Potent Inhibitors of Mycobacterium tuberculosis PknB with Antibacterial Activity
Author
Ariyachaokun Kanchiyaphat
Blood Rosemary A
+19 more
Hannongbua Supa
Hanwarinroj Chayanin
Hongmanee Poonpilas
Kamsri Pharit
Ketrat Sombat
Kittakoop Prasat
Leanpolchareanchai Jiraporn
Mukamolova Galina V
Mulholland Adrian J
Pakamwong Bongkochawan
Pungpo Pornpan
Punkvang Auradee
Santanirand Pitak
Saparpakorn Patchreenart
Spencer James
Sureram Sanya
Suttisintong Khomson
Takebayashi Yuiko
Thongdee Paptawan
Publication venue
'American Chemical Society (ACS)'
Publication date
22/08/2023
Field of study
No full text
Explore Bristol Research
Curcumin protects mice from Staphylococcus aureus pneumonia by interfering with the self-assembly process of α-hemolysin
Author
A Punkvang
A Shehzad
+38 more
AF Sonnen
AM Rivera
B Hess
B Walker
BE Ragle
BE Ragle
BJ Berube
BT Kurien
C Schaffner-Barbero
CP Montgomery
CP Montgomery
D Sinha
DA Rasko
DM Elston
E Rubinstein
F Vandenesch
F Xu
G Kapakos
G Scatchard
HM Nguyen
J Bubeck Wardenburg
J Bubeck Wardenburg
J Dong
J Qiu
J Qiu
L Song
M Li
MR Eftink
MR Hanson
MT Holden
P Auradee
PA Subramani
RA Awad
T Esatbeyoglu
V Khodaverdian
VT Nguyen
W Gao
Y Ye
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
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