8 research outputs found
Intracolonic administration of zileuton, a selective 5-lipoxygenase inhibitor, accelerates healing in a rat model of chronic colitis
- Author
- Allgayer H.
- Allgayer H.
- Beno D.W.A.
- Betz M.
- Donowitz M.
- E Castella
- F Fernandez-Banares
- Gibson G.R.
- Goto T.
- Gould SR
- Gould SR, Brash
- Gryglewski R.J.
- Hawkey C.
- I Ojanguren
- J Mane
- Kauffmann H.J.
- Kunkel S.L.
- Lauritsen K.
- Lauritsen K.
- Laursen L.S.
- LeDuc L.E.
- M A Gassull
- M Esteve
- Morris G.P.
- Peppercorn M.
- Peskar B.M.
- Powell W.S.
- R Bartoli
- Rachmilewitz R.
- Ramis I.
- Rampton D.S.
- Sharon P.
- Sharon P.
- Sharon P.
- Stenson W.F.
- Surawicz C.M.
- Vilaseca J.
- Vilaseca J.
- Wallace J.L.
- Wallace J.L.
- Wallace J.L.
- Wallace J.L.
- X Bertran
- Yamada T.
- Zahner G.
- Zijlstra F.J.
- Zipser R.D.
- Publication venue
- 'BMJ'
- Publication date
- 01/01/1996
- Field of study
BACKGROUND: 5-Lipoxygenase products play a part in inflammatory response. AIMS: The effect of intracolonic administration of zileuton (a 5-lipoxygenase inhibitor) on colonic damage and eicosanoid local release was assessed in a rat model of colitis. METHODS: Ninety rats with trinitrobenzenesulphonic acid induced colitis were randomised to receive placebo, 5-aminosalicylic acid (50 mg/kg), or zileuton (50 mg/kg) intracolonically for four weeks. Local eicosanoid release was monitored by intracolonic dialysis throughout the study. The colon was removed for macroscopic and histological assessment at weeks 1, 2, and 4 after colitis induction in 10 rats of each group. RESULTS: Zileuton significantly reduced macroscopic damage score after four weeks of treatment in comparison with the other two groups (p = 0.034). In addition, zileuton administration significantly increased the intracolonic release of both thromboxane B2 at week 1 (p = 0.05) and prostaglandin E2 at weeks 2 and 4 (p < 0.05). Zileuton and 5-aminosalicylic acid decreased leukotriene B4 release by 90% at day 3. CONCLUSIONS: Intracolonic zileuton, compared with 5-aminosalicylic acid and placebo, seems to improve the course of the disease in a model of chronic colitis. This effect may be related to an increased and maintained production of prostaglandin E2 together with inhibition of leukotriene B4 synthesis
Studies on Biologically Relevant Iron (II) and Lead (II) Macrocyclic Complexes : Designed, Synthesis, Spectroscopic Characterization and Applied Potential
- Author
- Arora D.L.
- Baker A.T.
- Bhakuni D.S.
- Caddick S.
- Collins T.J.
- Dhawan B.N.
- Dixit S.K.
- Fahmi N.
- Fahmi N.
- Horsfall J.H.
- Howlader B.H.
- Ibrahim Y.A.
- Jain M.
- Kamal R.
- Kidwai M.
- Kimura E.
- Liakad A.
- Malik W.U.
- Mane P.S.
- Mckee V.
- Mishra A.P.
- Muller J.G.
- Parker D.
- Prasad R.N.
- Saxena C.
- Sharma K.
- Singh A.
- Singh R.V.
- Singh U.P.
- Srivastava R.S.
- Tandon S.
- Thimmaiah K.N.
- Publication venue
- 'Walter de Gruyter GmbH'
- Publication date
- Field of study
Brain Tumor Segmentation of T1w MRI Images Based on Clustering Using Dimensionality Reduction Random Projection Technique
- Author
- Adhikari S.K.
- Aslam H.A.
- Attique Khan M.
- Bingham E.
- Cheng Z.
- Guo L.
- Harchaoui NE.
- Jolliffe IT
- Kapoor L.
- Karuna Y.
- Kaya IE.
- Khan M.A.
- Khan M.A.
- Kumar D.
- Liu J.
- Madhukumar S.
- Majid A.
- Majumder S.
- Mane D.S.
- Masood S.
- Menze BJ.
- Nazir M.
- Ng S.C.
- Parsi A.
- Rehman A.
- Rodríguez-Méndez IA
- Sanghamitra T.
- Saunders C.
- Sharif M.
- Sharif M.I.
- Stewart G.W.
- Subhani S.K.
- Viswanath SE.
- Yousefi S.
- Zeng G.
- Publication venue
- 'Bentham Science Publishers Ltd.'
- Publication date
- Field of study
Prediction of optimum adsorption isotherm: comparison of chi-square and Log-likelihood statistics
- Author
- Afshin Maleki
- Agresti A.
- Allen S.
- Belhachemi M.
- Chernoff H.
- Choy K.K.H.
- Do Duong D.
- Dubinin M.M.
- Freundlich H.Z.
- Fritz W.
- Gordon McKay
- Hadi M.
- Hadi M.
- Halsey G.
- Harkins W.D.
- Ho Y.S.
- Ho Y.S.
- Ho Y.S.
- Honig J.M.
- Jossens L.
- Jovanovic D.S.
- Khan A.R.
- Koble R.A.
- Kumar K.V.
- Langmuir I.
- Liang J.
- Mahdi Hadi
- Malek A.
- Mane V.S.
- Matheswaran M.
- McDonald J.H.
- McKay G.
- Mehri Solaimany Aminabad
- Mohammad Reza Samarghandi
- Ncibi M.C.
- Ng J.C.Y.
- Radke C.J.
- Ratkowsky D.A.
- Redlich O.
- Ringot D.
- Samarghandi M.R.
- Seidel A.
- Seidel-Morgenstern A.
- Shih M.C.
- Sips R.
- Tóth J.
- Vieth W.R.
- Zhang L.
- Zhu H.
- Publication venue
- 'Informa UK Limited'
- Publication date
- Field of study
Analytical Techniques in the Analysis of Darunavir and Ritonavir: A Review
- Author
- Ahmad Z.
- AlOthman Z.A.
- Babu G.R.
- Bommella M.
- Cerezo G.E.
- Chaudhary P.G.
- Chemburkar S.R.
- Chiranjeevi K.
- Correa J.C.R.
- Curran A.
- Damle M.
- Dickinson L.
- Fan B.
- Fanales-Belasio E.
- Fathima N.
- Gadhvi M.
- Ghante M.
- Golucci A.P.
- Gorja A.
- Goswami Kashish
- Hiremath S.N.
- Jain H.K.
- Kadikar Hiren
- Kaduk J.A.
- Kanta V.
- Karthik A.
- Kiranmaie S.G.
- Kogawa A.C.
- Kogawa A.C.
- Kogawa A.C.
- Kumar K.V.
- Kumar P.J.
- Maddinapudi R.
- Mane M.B.
- Mohammad A.S.
- Mohammad H.A.
- Mohammad H.A.
- Mohana P.V.
- Nagano D.
- Nagendrakumar A.
- Nagulwar V.P.
- Parikh Nisha
- Patel A.
- Patel B.N.
- Patel B.N.
- Pawar D.S.
- Pereira E.A.
- Rahman N.
- Rao V.B.
- Rao V.B.
- Reddy B.V.R.
- Reddy J.S.K.
- Reddy Mp.
- Rizwan S.H.
- Salunke J.M.
- Sangshetti J.N.
- Shankpal P.D.
- Siddiqui M.R.
- Sindu P.D.
- Suneeth A.
- Sunitha N.
- Vasavi N.
- Publication venue
- 'Bentham Science Publishers Ltd.'
- Publication date
- Field of study
Dynamical Chaos
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- A. Akopov
- A. Amengual
- A. Arneodo
- A. Babloyantz
- A. Babloyantz
- A. Brandstater
- A. Garfinkel
- A. Libchaber
- A. Lichtenberg
- A. Morelli
- A. Neiman
- A. Neiman
- A. Pikovsky
- A. Pikovsky
- A. Pikovsky
- A. Pikovsky
- A. Shabunin
- A. Sherman
- A. Wolf
- A. Wolf
- A.A. Akopov
- A.A. Dvornikov
- A.A. Maltsev
- A.A. Samarskii
- A.B. Neiman
- A.G. Mayer
- A.I. Fomin
- A.L. Fradkov
- A.L. Shilnikov
- A.M. Fraser
- A.N. Kolmogorov
- A.N. Malakhov
- A.N. Pavlov
- A.N. Sharkovsky
- A.P. Kuznetsov
- A.P. Kuznetsov
- A.R. Volkovskii
- A.S. Dmitriev
- A.S. Gurtovnik
- A.S. Pikovsky
- A.S. Pikovsky
- A.S. Pikovsky
- A.S. Pikovsky
- A.S. Pikovsky
- A.T. Winfree
- A.T. Winfree
- A.V. Gaponov-Grekhov
- A.V. Gaponov-Grekhov
- A.V. Gaponov-Grekhov
- A.V. Ustinov
- A.W. Hübler
- B. Hu
- B. Hu
- B. Hu
- B. Malreison
- B.A. Huberman
- B.I. Shraiman
- B.I. Shraiman
- C. Baesens
- C. Elphik
- C. Giberti
- C. Grebogi
- C. Grebogi
- C. Grebogi
- C. Liverani
- C. Schäfer
- C. Schäfer
- C. Schäfer
- C.G. Schroer
- C.K. Duan
- C.S. Hsu
- C.S.M. Lainscsek
- C.W. Gardiner
- C.W. Wu
- D. Alonso
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- D. Ruelle
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- D.A. Gribkov
- D.A. Linkens
- D.E. Postnov
- D.F. Russell
- D.G. Aranson
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- D.I. Biswas
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- E. Baake
- E. Baretto
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- E. Ott
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- E. Rosa
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- Task Force of the European Society of Cardiology and the North American Society of Racing and Electrophysiology
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- V.S. Anishchenko
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- V.S. Anishchenko
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- V.S. Anishchenko
- V.S. Anishchenko
- V.S. Anishchenko
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- V.V. Astakhov
- W. Freeman
- W. Horsthemke
- W. Liebert
- W.L. Ditto
- Y. Aizawa
- Y. Braiman
- Y. Braiman
- Y. Jiang
- Y. Kuramoto
- Y. Kuramoto
- Y. Kuramoto
- Y. Pomeau
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- Yu.A. Kuznetsov
- Yu.M. Romanovsky
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- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/2006
- Field of study
Recent Developments in Medicinal Chemistry of Allosteric Activators of Human Glucokinase for Type 2 Diabetes Mellitus Therapeutics
- Author
- Ahmed A.M.
- Aicher T.D.
- Aicher T.D.
- Aicher TD
- Aicher TD
- Aicher TD
- Aicher TD
- Ajmer S. Grewal
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- Bizzarro FT
- Bonadonna R.C.
- Bonn P.
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Assessing the Reliability of Commercially Available Point of Care in Various Clinical Fields
- Author
- Abbai-Shaik N.S.
- Abdelazim I.A.
- Abdelazim I.A.
- Adams S.
- Agarwal A.
- Akinbami F.
- Alam M.S.
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- Alawad A.O.
- Alessandro Di Cerbo
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- Andersen G.N.
- Antonio Scarano
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- Apple F.S.
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- Asimos A.W.
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- Bornemann P.
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- Bénéteau-Burnat B.
- Carlotta Marini
- Ceplecha V.
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- Publication venue
- 'Bentham Science Publishers Ltd.'
- Publication date
- Field of study