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36 research outputs found
An alternative approach to the synthesis of [1,2,4]triazolo[1,5â a
Author
Abudusaimi M.
Dyckman A.
+8Â more
Emmitte K.
Flohr K.
He Z.
Kawakaki K.
Mulwad V.
Parr R.
Trottmann G.
Wu L.
Publication venue
'Wiley'
Publication date
Field of study
No full text
Crossref
Development and kilogram-scale synthesis of mGlu5 negative allosteric modulator VU0424238 (auglurant)
Author
Anna L. Blobaum
Arlindo L. Castelhano
+40Â more
Berry-Kravis
Bezard
Busse
Carrie K. Jones
Conn
Cosford
Craig W. Lindsley
Devendrareddy Pallalu
Emmitte
Felts
Felts
Gasparini
Golubeva
Guerini
Jaeschke
Jaso
Kyle A. Emmitte
Lindsley
Lindsley
Litim
M. Rajendraswami
Michael J. Kates
Mihov
Nayak K. Prashanth
Niswender
P. Jeffrey Conn
Palanisamy
Pop
Porter
Quiroz
Rascol
Ribeiro
Rocher
Rutrick
Silverman
Thomas K. David
Tison
Vranesic
Wenthur
Zhang
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Evaluating the Disposition of a Mixed Aldehyde Oxidase/Cytochrome P450 Substrate in Rats with Attenuated P450 Activity
Author
Al-Salmy
Beedham
+14Â more
Beedham
C. W. Lindsley
F. W. Byers
Garattini
J. S. Daniels
K. A. Emmitte
Kitamura
Obach
Pryde
R. D. Crouch
R. D. Morrison
Sahi
Smeland
Zhang
Publication venue
'American Society for Pharmacology & Experimental Therapeutics (ASPET)'
Publication date
Field of study
No full text
Crossref
Discovery of ( R
Author
Andrew S. Felts
Campo B.
+24Â more
Caraci F.
Cody J. Wenthur
Conn P. J.
Conn P. J.
Conn P. J.
Craig W. Lindsley
Emmitte K. A.
Frank W. Byers
Harrision P. J.
J. Scott Daniels
Julie L. Engers
Katrina A. Smith
Kyle A. Emmitte
Melancon B. J.
Monn J. A.
Nelson S. D.
P. Jeffrey Conn
Robichaud A. J.
Ryan Morrison
Sheffler D. J.
Sheffler D. J.
Stauffer S. R.
Suzuki G.
Wood M. R.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
VU0477573: Partial Negative Allosteric Modulator of the Subtype 5 Metabotropic Glutamate Receptor with In Vivo Efficacy
Author
A. Thompson
B. S. Bates
+16Â more
C. K. Jones
C. M. Niswender
C. W. Lindsley
H. H. Nickols
J. P. Yuh
J. S. Daniels
K. A. Emmitte
K. J. Gregory
M. Bubser
M. T. Nedelcovych
P. J. Conn
R. D. Morrison
S. R. Stauffer
W. Peng
X. Lv
Z. Xiang
Publication venue
'American Society for Pharmacology & Experimental Therapeutics (ASPET)'
Publication date
Field of study
No full text
Crossref
Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate Receptors
Author
Bond A.
Colleen M. Niswender
+16Â more
Corey R. Hopkins
Craig W. Lindsley
Fraser C. M.
Gregory K. J.
Hall D. A.
Helton D. R.
Kalinichev M.
Karen J. Gregory
Kyle A. Emmitte
Litschig S.
Lovinger D. M.
Mezler M.
Nho K.
P. Jeffrey Conn
Thomas M. Bridges
Yacoubi M. E.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
Discovery of VU0409106: A negative allosteric modulator of mGlu5 with activity in a mouse model of anxiety
Author
Adams
Alice L. Rodriguez
+82Â more
Amato
Andrew S. Felts
Anna L. Blobaum
Berg
Berry-Kravis
Besheer
Bridges
Brittney S. Bates
Broekkamp
Busse
BĂ€ckstrom
Carrie K. Jones
Colleen M. Niswender
Conn
Conn
Cosford
Cosford
Craig W. Lindsley
Daryl F. Venable
de Vrij
Emmitte
Emmitte
Felts
Felts
FlĂŒck
Frank W. Byers
Frisby
Gasparini
Gasparini
Gass
Gass
Hughes
J. Scott Daniels
Jacquemont
Jason T. Manka
Jensen
Kalvass
Kenny
Kew
Keywood
Klodzinska
Kotlinska
Kumaresan
Kuresh
Kyle A. Emmitte
Lamb
Lee
Lindemann
Lindsley
Lindsley
Lominac
Martin-Fardon
Melancon
Michalon
Morin
Morrison
Mueller
Nicolas
Njungâe
Noetzel
P. Jeffrey Conn
Pajouhesh
Pietraszek
Platt
Ritzén
Rocher
Rodriguez
Rohof
Ryan D. Morrison
Schoepp
Schroeder
Sharma
Silverman
Silverman
Spooren
Tessari
Tison
Tronci
Yan
Zhou
Zhu
Zientek
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Identification of Specific LigandâReceptor Interactions That Govern Binding and Cooperativity of Diverse Modulators to a Common Metabotropic Glutamate Receptor 5 Allosteric Site
Author
Alagille D.
Alagille D.
+61Â more
Brittney S. Bates
Chen Y.
Chrysa Malosh
Cosford N. D.
Craig W. Lindsley
Davis I. W.
de Paulis T.
Deupi X.
Elizabeth D. Nguyen
Emma F. Squire
Emmitte K. A.
Eric M. Turner
Felts A. S.
Felts A. S.
Gasparini F.
Gregory K. J.
Gregory K. J.
Gregory K. J.
Gregory K. J.
Hammond A. S.
Jeffrey L. Mendenhall
Jens Meiler
Jerri M. Rook
Jessica Z. Zic
Kaae B. H.
Karen J. Gregory
Kinney G. G.
Kulkarni S. S.
Kyle A. Emmitte
Labute P.
Lamb J. P.
Lemmon G.
Malherbe P.
Malherbe P.
Meiler J.
Meredith J. Noetzel
Molck C.
Mueller R.
Muhlemann A.
Nguyen E. D.
Niswender C. M.
Noetzel M. J.
Ortiz A. R.
P. Jeffrey Conn
Pagano A.
Rodriguez A. L.
Rodriguez A. L.
Roppe J.
Sharma S.
Shaun R. Stauffer
Sheffler D. J.
Spear N.
Stauffer S. R.
Tautermann C. S.
Turlington M.
Varney M. A.
Wood M. R.
Xiong H.
Zhao Z.
Zhou Y.
Zou M. F.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
N-Alkylpyrido[1âČ,2âČ:1,5]pyrazolo-[4,3-d]pyrimidin-4-amines: A new series of negative allosteric modulators of mGlu1/5 with CNS exposure in rodents
Author
Achat-Mendes
Adams
+81Â more
Addex Pharmaceuticals Press Release
Alice L. Rodriguez
Amato
Andrew S. Felts
Anna L. Blobaum
Berg
Besheer
Bridges
Bridges
Busse
BĂ€ckstrom
Carrie K. Jones
Cho
Colleen M. Niswender
Conn
Conn
Craig W. Lindsley
Daryl F. Venable
Di
Emmitte
Emmitte
Engers
Felts
Frank W. Byers
Fukuda
Gasparini
Gass
Gass
Ito
J. Scott Daniels
Kalvass
Kenny
Kew
Klodzinska
Kohara
Kotlinska
Kumaresan
Kyle A. Emmitte
Lee
Lesage
Lindemann
Lindsley
Liu
Lominac
Lovering
Mantell
Martin-Fardon
Melancon
Mohamed
Mueller
Newell
Nicolas
Niswender
Niswender
Noetzel
Obach
Owen
P. Jeffrey Conn
Pietraszek
Platt
Quiroz
Ravez
Ritzén
Rocher
Rodriguez
Ryan D. Morrison
Schoepp
Schroeder
Shannon
Spooren
Steckler
Stocchi
Tessari
Tian
Tronci
Tsuritani
Xie
Zheng
Zhu
Zhu
Zientek
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Discovery of VU0431316: A negative allosteric modulator of mGlu5 with activity in a mouse model of anxiety
Author
Adams
Alice L. Rodriguez
+81Â more
Amato
Andrew S. Felts
Anna L. Blobaum
Berg
Berry-Kravis
Besheer
Bhagwanth
Bridges
Brittney S. Bates
Broekkamp
Busse
BĂ€ckstrom
Carrie K. Jones
Colleen M. Niswender
Conn
Conn
Cosford
Cosford
Craig W. Lindsley
Daryl F. Venable
de Vrij
Emmitte
Emmitte
Felts
Felts
Felts
Frank W. Byers
Frisby
Gasparini
Gasparini
Gass
Gass
J. Scott Daniels
Jacquemont
Jensen
Kalvass
Kenny
Kera P. Lawson
Kew
Keywood
Klodzinska
Kotlinska
Kumaresan
Kuresh
Kyle A. Emmitte
Lamb
Lee
Lindsley
Lindsley
Lominac
Martin-Fardon
Melancon
Morin
Morrison
Mueller
Nicolas
Njungâe
Noetzel
P. Jeffrey Conn
Pietraszek
Platt
Ritzén
Rocher
Rodriguez
Rohof
Ryan D. Morrison
Schoepp
Schroeder
Silverman
Spooren
Tessari
Thomas
Tison
Tronci
Wang
Yan
Yin
Zhang
Zhou
Zhu
Zientek
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
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