16 research outputs found
Synthesis and Pharmacology of the Baclofen Homologues. 5-Amino-4-(4-chlorophenyl)pentanoic Acid and the R- and S-Enantiomers of 5-Amino-3-(4-chlorophenyl)pentanoic Acid
No full textConvergent synthesis and pharmacology of substituted tetrazolyl-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid analogues
No full textHeteroaryl analogues of AMPA. 2. Synthesis, absolute stereochemistry, photochemistry, and structure-activity relationships
No full textPharmacological characterization and binding modes of novel racemic and optically active phenylalanine-based antagonists of AMPA receptors
No full textA new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure:Synthesis, resolution, pharmacology, and crystal structure
No full textA stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors
No full textAryl and cycloalkyl analogues of AMPA: synthetic, pharmacological and stereochemical aspects
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