7 research outputs found
CD34-related coexpression of MDR1 and BCRP indicates a clinically resistant phenotype in patients with acute myeloid leukemia (AML) of older age
- Author
- A Suvannasankha
- A Zon van
- Alan K. Burnett
- B Holt van der
- B Holt van der
- B Lowenberg
- B Uggla
- BD Cheson
- BL Abbott
- BL Abbott
- Bob Löwenberg
- Bronno van der Holt
- C Baldus
- CL Willman
- CP Leith
- CP Leith
- CS Wilson
- D Damiani
- D Israeli
- D Steinbach
- DD Ross
- DD Ross
- DM Kolk van der
- DM Kolk van der
- DR Cox
- DW Hosmer
- E Kaplan
- Edo Vellenga
- Gert J. Ossenkoppele
- Gregor E. G. Verhoef
- LA Doyle
- M Filipits
- M Hunault
- MA Goodell
- MA Pol van der
- Marry M. van den Heuvel-Eibrink
- Martin F. Fey
- MH Mossink
- MH Raaijmakers
- MM Heuvel-Eibrink van den
- MM Heuvel-Eibrink van den
- N Mantel
- O Legrand
- Pieter Sonneveld
- S Zhou
- Wolfgang U. Knauf
- Z Benderra
- Publication venue
- Springer-Verlag
- Publication date
- 01/01/2007
- Field of study
Clinical resistance to chemotherapy in acute myeloid leukemia (AML) is associated with the expression of the multidrug resistance (MDR) proteins P-glycoprotein, encoded by the MDR1/ABCB1 gene, multidrug resistant-related protein (MRP/ABCC1), the lung resistance-related protein (LRP), or major vault protein (MVP), and the breast cancer resistance protein (BCRP/ABCG2). The clinical value of MDR1, MRP1, LRP/MVP, and BCRP messenger RNA (mRNA) expression was prospectively studied in 154 newly diagnosed AML patients ≥60 years who were treated in a multicenter, randomized phase 3 trial. Expression of MDR1 and BCRP showed a negative whereas MRP1 and LRP showed a positive correlation with high white blood cell count (respectively, p < 0.05, p < 0.001, p < 0.001 and p < 0.001). Higher BCRP mRNA was associated with secondary AML (p < 0.05). MDR1 and BCRP mRNA were highly significantly associated (p < 0.001), as were MRP1 and LRP mRNA (p < 0.001) expression. Univariate regression analyses revealed that CD34 expression, increasing MDR1 mRNA as well as MDR1/BCRP coexpression, were associated with a lower complete response (CR) rate and with worse event-free survival and overall survival. When adjusted for other prognostic actors, only CD34-related MDR1/BCRP coexpression remained significantly associated with a lower CR rate (p = 0.03), thereby identifying a clinically resistant subgroup of elderly AML patients
Bendamustine compared with chlorambucil in previously untreated patients with chronic lymphocytic leukaemia: updated results of a randomized phase III trial
- Author
- Publication venue
- 'Wiley'
- Publication date
- 01/01/2012
- Field of study
The efficacy of bendamustine versus chlorambucil in a phase III trial of previously untreated patients with Binet stage B/C chronic lymphocytic leukaemia (CLL) was re-evaluated after a median observation time of 54months in May 2010. Overall survival (OS) was analysed for the first time. At follow-up, investigator-assessed complete response (CR) rate (21.0% vs 10.8%), median progression-free survival (21.2 vs 8.8months; P65 years, responders and non-responders. However, patients with objective response or a CR experienced a significantly longer OS than non-responders or those without a CR. Significantly more patients on chlorambucil progressed to second/further lines of treatment compared with those on bendamustine (78.3% vs 63.6%; P=0.004). The benefits of bendamustine over chlorambucil were achieved without reducing quality of life. In conclusion, bendamustine is significantly more effective than chlorambucil in previously untreated CLL patients, with the achievement of a CR or objective response appearing to prolong OS. Bendamustine should be considered as a preferred first-line option over chlorambucil for CLL patients ineligible for fludarabine, cyclophosphamide and rituximab
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- Publication date
- 01/01/1999
- Field of study
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- Görg Manfred
- Görg Manfred
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- Herzog
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- Hill
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- Lohfink Norbert
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- Luker Lamontte M
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- Thompson Henry O
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- Toombs Lawrence E
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- Waldmann Helmut
- Waldmann Rademacher
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- Wallis Gerhard
- Wallis Gerhard
- Wallis Gerhard
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- Weippert Manfred
- Weippert Manfred
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- Weißbach Franz Heinrich
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- Welten Peter
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- Wenning Zenger
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- Westenholz Joan Goodnick
- Westenholz Joan Goodnick
- Westenholz Joan Goodnick
- Whitehouse Helen
- Wilhelm Gernot
- Willeitner Joachim
- Williams David Salter
- Wilson Kevin A
- Wimmer Stefan Jakob
- Wiseman Donald John
- Witte Markus
- Witte Markus
- Wolff Hans Walter
- Wolters Albert M
- Wood Bryant G
- Wood Bryant G
- Wood Bryant G
- Woolley
- Woolley Charles
- Woolley Charles Leonard
- Woolley Charles Leonard
- Worschech Udo
- Wright G. Ernest
- Wright George R.H.
- Wright George R.H.
- Wächter Ludwig
- Würthwein Ernst
- Wüst Manfried
- Wüst Manfried
- Yeivin Zeev
- Yisraeli Yael
- Younker Randall W
- Yule Paul
- Zadok Ran
- Zadok Ran
- Zakovitch Yair
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- Zertal Adam
- Zettler Richard L
- Ziemer Benjamin
- Ziemer Benjamin
- Zilberbod Irina
- Zimmerli Walther
- Zucconi Laura Marie
- Zwickel Wolfgang
- Zwickel Wolfgang
- Zwickel Wolfgang
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- Zwickel Wolfgang
- Zwickel Wolfgang
- Zwickel Wolfgang
- Publication venue
- 'Vandenhoeck & Ruprecht GmbH & Co, KG'
- Publication date
- Field of study
Targeting the CNS to treat type 2 diabetes
- Author
- A Benani
- A Cohen
- A Gyte
- A Nakagawa
- A Pocai
- A Pocai
- A Pocai
- AA Dunn-Meynell
- AC Konner
- AD Cherrington
- AF Chintoh
- AH Cincotta
- AS Garfield
- B Kreymann
- B Williams
- BE Levin
- BE Levin
- BP Bullock
- C Buettner
- C Cruciani-Guglielmacci
- C Garcia-Echeverria
- C Giussani
- C Knauf
- C Perrin
- CD Morrison
- CM Taniguchi
- D Aftab Guy
- D Cota
- D Cota
- D Cota
- D Dardevet
- D Greenberg
- D Matzinger
- D Williams-Herman
- DA Sandoval
- DA Sandoval
- Darleen A. Sandoval
- DF Bertelli
- DG Hardie
- DJ Clegg
- DJ Drucker
- DS Edgerton
- DW Biggers
- EL Air
- FG Banting
- G Thomas
- G Tulipano
- GJ Morton
- GK McConell
- GV Ronnett
- H Ono
- H-R Berthoud
- I Merchenthaler
- J Kreuter
- J Rosenstock
- J Schirra
- J von Mering
- JA Lieberman
- JC Donahey
- JE Ayala
- JE Lindsley
- JL Dunphy
- JW Hill
- K Lee
- K Nonogaki
- K Proulx
- KA Anderson
- KD Niswender
- KD Niswender
- KL Houseknecht
- L Kang
- L Khamzina
- L Liu
- L Ozcan
- L Plum
- L Sokoloff
- L Zhou
- LE Parton
- LJ Stein
- M Ader
- M Claret
- M Fukushima
- M Stumvoll
- MB Wheeler
- MD Wortman
- ME Brewster
- MG Wallis
- MJ Wolfgang
- ML Hakansson
- ML Villanueva-Penacarrillo
- MM Meguid
- MM Patel
- MR Davis
- MS Haque
- MW Schwartz
- MW Schwartz
- N Bodor
- N McIntyre
- PA Israel
- PA Tataranni
- PB Dennis
- PY Wang
- R Coppari
- R Goke
- R Gutierrez-Juarez
- R Wang
- Randy J. Seeley
- RH Unger
- RH Unger
- RJ McCrimmon
- RJ Seeley
- RJ Shaw
- RL Prigeon
- RV Considine
- S Inoue
- S Mirshamsi
- S Obici
- S Obici
- S Obici
- S Obici
- S Obici
- S Troy
- S Wullschleger
- SC Benoit
- SC Woods
- SC Woods
- SE Kahn
- SH Bates
- SH Um
- Silvana Obici
- SM Han
- SR Heller
- SS Gill
- SY Zhou
- T Alquier
- T Shimazu
- T Shimokawa
- T Woltman
- TK Lam
- TK Lam
- TK Lam
- TL Horvath
- TM Loftus
- TP Vahl
- U Andersson
- V Ionut
- VA Narkar
- W He
- WA Banks
- WA Banks
- WA Banks
- X Zhang
- Y Minokoshi
- Y Minokoshi
- Y Xu
- Z Hu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Literatur
- Author
- Aboud Jehad
- Achenbach Reinhard
- Achenbach Reinhard
- Ackroyd Peter R
- Adam Klaus-Peter
- Ahn Dietrich
- Aischylos Tragödien
- Aitken Dell
- Albani Matthias
- Albertz Rainer
- Albertz Rainer
- Albertz Rainer
- Albertz Rainer
- Albrecht Christian
- Albrektson Bertil
- Alt Albrecht
- Alt Albrecht
- Alt Albrecht
- Altmann Peter
- Anderson Charles A
- Angenendt Vorgrimler
- Appian
- Arneth Gerechtigkeit
- Arnim
- Assmann Jan
- Assmann Jan
- Atkinson Kenneth
- Augustinus Aurelius
- Augustinus Aurelius
- Augustinus Aurelius
- Aurelius Erik
- Aurelius Erik
- Avalos Hector
- Avemarie Lichtenberger
- Avigad Nahman
- Axelsson Lars Eric
- Bachmann Veronika
- Bak Dong Hyun
- Baldermann
- Balentine Samuel E
- Balentine Samuel E
- Baltzer Klaus
- Barr James
- Barr James
- Barr James
- Barrett William
- Barth Christoph
- Barth Karl
- Barthelmus Rüdiger
- BarthØlemy Rickenbacher
- Barton John
- Bauks Liess
- Baumann Gerlinde
- Beck Schorn
- Becker Eva-Marie
- Becker Joachim
- Becker Joachim
- Becker Joachim
- Becker Jürgen
- Becker Uwe
- Becker Uwe
- Bees Robert
- Begrich Joachim
- Ben Zvi Ehud
- Benz Ernst
- Benzinger Immanuel
- Berger Klaus
- Berges Klaus
- Berlejung Angelika
- Berlejung Schmid
- Betz Otto
- Beuken Willem A. M.
- Beuken Willem A. M.
- Beuken Willem A.M
- Beyerlin Walter
- Beyse Karl-Martin
- Biblia Hebraica Stuttgartensia
- Bickermann Elias
- Bickermann Elias
- Bietenhard Hans
- Black Mathew
- Black Mathew
- Blischke Mareike V
- Blum Erhard
- Bobzien Susanne
- Bobzin Hartmut
- Bobzin Hartmut
- Bonnet Hans Zum
- Borgen Peder
- Borger Rykle
- Borger Rykle
- Braulik Georg
- Braulik Georg
- Braulik Georg
- Braun Rainer
- Brekelmans C.H.W.
- Brenner Martin L
- Bringmann Klaus
- Bringmann Klaus
- Brown Peter
- Brown Peter
- Bultmann Rudolf
- Burkert Walter
- Burkert Walter
- Böcher Otto
- Casetti Pierre
- Chadwick Henry
- Chadwick Henry
- Charlesworth James H
- Cheon Samuel
- Chirichigno Gregory C
- Christ Karl
- Christ Karl
- Cicero M.
- Cicero M.
- Cicero M.
- Cicero M.
- Clements Ronald E
- Clements Ronald E
- Collins John J
- Collins John J
- Collins John J
- Conrad Diethelm
- Coppens Joseph
- Corley Jeremy
- Corley Jeremy
- Crenshaw James L
- Crüsemann Frank
- Dahlmann Gustaf H
- Dahm Ulrike
- Dahm Ulrike
- Day John
- Day John
- Day Peggy L
- Debus Jörg
- Delitzsch Franz
- Dell Katharine J
- Denis Albert-Marie
- Denis Albert-Marie
- Di Lella Alexander A
- Diesel Antje A
- Dietrich Loretz
- Dietrich Loretz
- Dietrich Loretz
- Dietrich Loretz
- Dietrich Loretz
- Dietrich Walter
- Diogenes Laertius
- Diogenes Laertius
- Dochhorn Jan
- Dohmen Christoph
- Doll Peter
- Donner Herbert
- Donner Herbert
- Donner Herbert
- Donner Herbert
- Durhaime Jean
- Ebert Theodor
- Eckstein Landmesser
- Edzard Dietz Otto
- Egger-Wenzel Renate
- Egger-Wenzel Renate
- Egger-Wenzel Renate
- Ehrenberg Victor
- Eißfeldt Otto
- Ellermeier Friedrich
- Elliger Karl
- Emerton J. A.
- Engel Helmut
- Erman Adolf
- Essler Holger
- Evangelisches Gesangbuch
- Ewald Heinrich
- Fahlgren K.H.
- Falkenstein
- Finsterbusch Karin
- Fischer Alexander A
- Fischer Alexander A
- Fischer Alexander A
- Fischer Herrmann
- Fischer Irmtraud
- Fischer Stefan
- Fischer Ulrich
- Fleischer Günther
- Fohrer Georg
- Fohrer Georg
- Forschner Maximilian
- Fox Michael V
- Fox Michael V
- Frevel Christian
- Frevel Christian
- Fritz Volkmar
- Fritz Volkmar
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- Gadamer Hans Georg
- Gadamer Hans Georg
- Galling Kurt
- Galling Kurt
- Galling Kurt
- Galling Kurt
- Galling Kurt
- Gammy John G
- Gammy John G
- Gelassenheit
- Gelassenheit
- Gelassenheit
- Gerstenberger Erhard S
- Gerstenberger Erhard S
- Gerstenberger Erhard S
- Gerstenberger Erhard S
- Gertz Jan
- Gertz Jan
- Gertz Jan Christian
- Gese Hartmut
- Gese Hartmut
- Gilbert Maurice
- Gilbert Maurice
- Gordon Robert P
- Gowan Donald E
- Grabbe Lester L
- Grabe Peter J
- Graf Fritz
- Granerød Gard
- Graupner Axel
- Gressmann Hugo
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- Gustav
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- Janowski Bernd
- Janowski Bernd
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- Mettinger Tryggve N.D.
- Mettinger Tryggve N.D.
- Mettinger Tryggve N.D.
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