6 research outputs found
Non-peptide ligands for bradykinin receptors 1995 – 2004
- Author
- ALTAMURA M
- ARAMORI I
- ARAMORI I
- ARTIS DR
- ASANO M
- ASANO M
- ASANO M
- AUSTIN CE
- BELLUCCI F
- BHOOLA KD
- BOCK MG
- BOELS K
- BORKOWSKI JA
- BURKE JE
- CALIXTO JB
- CARRETERO OA
- CASSIM B
- DANKWARDT SM
- DZIADULEWICZ EK
- DZIADULEWICZ EK
- DZIADULEWICZ EK
- Edward K Dziadulewicz
- EVANS BE
- GOBEIL F JR MONTAGNE M, INAMURA N, REGOLI D
- GOODFELLOW VS
- GOUGAT J
- HEITSCH H
- HEITSCH H
- HEITSCH H
- HESS JF
- HOCK FJ
- HORLICK RA
- HOWL J
- HOYER D AWAD MMA
- HUANG HM
- KOZIK A. MOORE RB
- KUDUK SD
- LAM YK
- LEE J
- LEEB-LUNDBERG LMF
- LEEB-LUNDBERG LMF MARCEAU
- LIU C
- MACNEIL T
- MARCEAU F
- MARCEAU F
- MARCEAU F
- MARCEAU F
- MARCEAU F
- MEINI S
- MENKE JG
- MORISSETTE G
- PESQUERO JB
- PRUNEAU D
- RANSOM RW
- REGOLI D
- RITCHIE TJ
- SALVINO JM
- SALVINO JM
- SAMUEL CS
- SAWUTZ DG
- STEWART JM
- STEWART JM
- STEWART JM
- SU D-S MARKOWITZ MK, DIPARDO RM et al.
- SU D-S MARKOWITZ MK, MURPHY KL et al.
- WIRTH K
- WITHERUP KM
- WOTHERSPOON G
- YOUNGMAN MA
- Publication venue
- 'Informa Healthcare'
- Publication date
- Field of study
New insights into the stereochemical requirements of the bradykinin B2 receptor antagonists binding
- Author
- A Cordomi
- A Faussner
- A Sali
- B Wu
- C Gibson
- C Thurieau
- Cecylia S. Lupala
- D Pruneau
- D Pruneau
- D Regoli
- D Spoel Van Der
- DG Sawutz
- DJ Kyle
- DJ Kyle
- DJ Kyle
- ED Dziadulewicz
- EK Dziadulewicz
- EK Dziadulewicz
- ES Monteagudo
- F Bellucci
- F Marceau
- FJ Hock
- GM Burgess
- H Heitsch
- J Marie
- JJ Lopez
- JJ Perez
- JM Salvino
- JM Stewart
- Juan J. Perez
- K Bork
- LF Pineda
- LMF Leeb-Lundberg
- LR Steranka
- M Asano
- M Filizola
- N Blaes
- P Cucchi
- Patricia Gomez-Gutierrez
- RA Boissonnas
- RA Friesner
- RJ Vavrek
- S Krishna
- S Meini
- S Meini
- S Meini
- S Meini
- V Katritch
- Y Sawada
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Bradykinin receptors as a therapeutic target
- Author
- AHLUWALIA A
- ALFIE ME
- ARAMORI I
- ASANO M
- BARNES PJ
- BARTUS RT
- BELICHARD P
- BHOOLA KD
- BHOOLA R
- CHAN D
- CHAN D
- CHAVAKIS T
- CHERONIS JC
- CHERONIS JC
- COUTURE R
- CRUWYS SC
- DAFFIX I
- DE WITT BJ
- DOUILLET CD
- DRAY A
- DUNCAN A-M KLADIS A, JENNINGS GL, DART AM, ESLER M, CAMPBELL
- DUNCAN AM
- EGGERICKZ D
- EMANUELI C
- EMERICH DF
- FATHY DB
- FATHY DB
- GROVES E KURZ S JUST H
- HECQUET C
- HESS JF
- HOWL J
- HOWL J
- KOZIK A
- KUGA T
- LEEB-LUNDBERG LMF KANG DS
- MAD DEDU P
- MAJIMA M
- MARCEAU F
- MARGOLIUS HS
- MARIE J
- MCLEAN PG
- MENKE JG
- MURPHEY LJ
- NEUGEBAUER W
- NI A
- PESQUERO JB
- PHAGOO SB
- POLOSA R
- PRAT A
- PRAT A
- PROUD D
- RAIDOO DM
- REGOLI D
- RICCIARDOLO FLM GEPPETTI P
- RIZZI A
- ROISMAN GL
- SAHA JK
- SARDI SP
- SARDI SP
- SCHANSTRA JP
- SCHREMMER-DANNINGER E
- SCHREY MP
- SHIGEMATSU S
- SQUIRE IB
- STEWART JM
- STEWART JM
- STEWART JM
- STEWART JM
- STEWART JM
- THOMAS HD
- WARREN KE
- WIRTH KJ
- WOHLFART E DEDIO J WIRTH K, SCHOLKENS BA
- Publication venue
- 'Informa Healthcare'
- Publication date
- 01/01/2003
- Field of study
Biologically-active kinins, including bradykinin (BK) and Lys(0)-BK (kallidin), are short-lived peptide mediators predominantly generated by the enzymatic action of kallikreins on kininogen precursors. A diverse spectrum of physiological and pathological actions attributed to local kinin production is a consequence of the activation of G-protein-coupled receptors (GPCRs). Currently, two major subtypes of kinin receptor, designated B(1) and B(2), are recognised, although there is much evidence for pharmacological heterogeneity, particularly within the B(2) receptors. Considering these facts and the widespread distribution of kinin receptors in many human tissues, it is no surprise that the therapeutic potential of kinins and kinin receptor antagonists remains the focus of numerous investigations. Studies in animals and animal tissues, instrumental in elucidating the biological roles of kinins, are well-documented in numerous excellent reviews. Unfortunately, and despite the enormous potential illustrated by animal studies, attempts to develop kinin analogues as therapeutic agents to combat human disease have largely proven disappointing. Consequently, this review selectively focuses upon studies that are directly relevant to the targeting of human BK receptors as a therapeutic intervention. In addition to providing a succinct review of well-documented pathological conditions to which kinin receptors contribute, the authors have also included more recent data that illustrate new avenues for the therapeutic application of kinin analogues
Kinins in Glioblastoma Microenvironment
- Author
- A Bajetto
- A Del Fattore
- A Hossain
- A Nakamizo
- A Philips
- A Sottoriva
- A Torsvik
- A Zomer
- AH Klopp
- AP Patel
- AZ Rizvi
- B Gole
- B Yan
- Barbara Breznik
- BM Ogle
- BN Hannafon
- C Melzer
- C Schichor
- C Spinelli
- CA Trujillo
- CD Figueroa
- CO Rodini
- D Bastida-Ruiz
- D Yi
- D Zhang
- DA Aderetti
- DE Clapham
- DM Raidoo
- DN Louis
- DW Stuckey
- DY Lu
- E Kashuba
- E Milkina
- ED Gomes
- EG Thompson
- EG Van Meir
- ET Whalley
- F Appaix
- F Marceau
- F Papaccio
- F Ricklefs
- H Motaln
- H Motaln
- H Motaln
- Henning Ulrich
- HK Lee
- HS Phillips
- HY Lee
- I Bryukhovetskiy
- I Singec
- J Behnan
- J Behnan
- J Björkqvist
- J Côté
- J Felsberg
- J Figueroa
- J Mercapide
- J Skog
- J Teng
- JD Hood
- JD Lathia
- JM Stewart
- JS Rao
- K Ishihara
- K Kološa
- K Wolf
- KPL Bhat
- L Barki-Harrington
- L Barki-Harrington
- L Molina
- LF Pavon
- LMF Leeb-Lundberg
- M Ceccarelli
- M Diksin
- M Ifuku
- M Mohr
- M Overholtzer
- M Tavazoie
- M Uchida
- M Vittori
- M. Rocha e Silva
- MA Qazi
- MD Wood
- MD Wood
- ME Castro-Manrreza
- ME Hardee
- ME Hegi
- Micheli M. Pillat
- MM Pillat
- MN Oliveira
- Mona N. Oliveira
- N Levicar
- N Podergajs
- NF Nicoletti
- P Barcellos-de-Souza
- P Ehrenfeld
- P Friedl
- P Maiuri
- PD Negraes
- PLN da Costa
- PT Ronaldson
- Q Wang
- R Kozma
- R Kozma
- R Wang
- R WĂĽrth
- RGW Verhaak
- Ricardo L. Pereira
- RJ Molenaar
- RJ Molenaar
- S Bao
- S Seifert
- S Seifert
- S Shi
- SA van Lith
- SK Singh
- SR Baglio
- T Dittmar
- T Dittmar
- T Liu
- Tamara T Lah
- Tamara T. Lah
- TB Steinbichler
- TK Howcroft
- U Verbovšek
- V Montana
- V Montana
- VA Cuddapah
- VR Dasari
- VR Dasari
- VVV Hira
- VVV Hira
- WY Bao
- X Zhang
- X Zhang
- Y Iwadate
- Y Shi
- YD Teng
- YD Teng
- YM Kim
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Stroke: Pathophysiology and Therapy
- Author
- Aarts MM
- Abu Fanne R
- ADVANCE Collaborative Group Patel A, MacMahon S, Chalmers J, Neal B, Billot L, Woodward M, Marre M, Cooper M, Glasziou P, Grobbee D, Hamet P, Harrap S, Heller S, Liu L, Mancia G, Mogensen CE, Pan C, Poulter N, Rodgers A, Williams B, Bompoint S, de Galan BE, Joshi R, Travert F
- Albert-WeiĂźenberger C
- Altman J
- Amarenco P
- Amarenco P
- Amaro S
- Amaro S
- Andres RH
- Armstead WM
- Arvidsson A
- Arvin B
- Astrup J
- Austinat M
- Badaut J
- Baker RI
- Ballen KK
- Bath C
- Bath PMW
- Benowitz LI
- Beray-Berthat V
- Bernard SA
- Berrouschot J
- Besancon E
- Bjorklund LM
- Bochelen D
- Boncoraglio GB
- Brait VH
- Brecht S
- Brenneman M
- Brines M
- Broos K
- Brown CE
- Bruno V
- Burden 0.
- Burns DM
- Buss A
- Butenas S
- BĂĽhnemann C
- Caliezi C
- Camera M
- Cao C-X
- Caplan LR
- Carmeliet P
- Carmichael ST
- Carmichael ST
- Carmichael ST
- Carmichael ST
- Caso JR
- Chan PH
- Chan PH
- Chaudhry A
- Chen H
- Chen H
- Chen H
- Chen J
- Chen J
- Chen P
- Chen R-L
- Chimowitz MI
- Chobanian AV
- Chow DK
- Clifton GL
- Corbett D
- Courtine G
- Cozzo Picca C
- Cramer SC
- Crossley NA
- Czech B
- Daadi MM
- Dancause N
- Darsalia V
- Davis AE
- De Meyer SF
- De Simoni MG
- De Simoni MG
- Deb P
- Di Virgilio F
- Diederich K
- Diener H-C
- Ding-Zhou L
- Dirnagl U
- Dirnagl U
- Dirnagl U
- Doyle KP
- Durham JT
- Ehrenreich H
- Ehrenreich H
- Elvington A
- Empey PE
- Eriksson PS
- Fassbender K
- Feigin VL
- Ferro JM
- Fisher J W
- Fisher M
- Fouad K
- Furie B
- Furie KL
- Furlan A
- Furuichi Y
- Gaede P
- Gailani D
- Gelderblom M
- Gertz K
- Gesuete R
- Ginsberg MD
- Giraldi-GuimarĂŁes A
- Girolami A
- Go AS
- Go AS
- Goldstein LB
- Gould E
- Gralla J
- Grewer C
- Grimm RH
- Gröger M
- Guo R-B
- Hacke W
- Hacke W
- Hagedorn I
- Hakim AM
- Hallenbeck JM
- Hatton J
- Hemmen TM
- Hermann DM
- Heydenreich N
- Hillen T
- Hirt L
- Hovelsø N
- Hunt D
- Hurn PD
- Hypothermia after Cardiac Arrest Study Group
- Ikegame Y
- Izumi Y
- Jabaudon D
- Jackman KA
- Jackman KA
- Jin K
- Jones TA
- Jones TA
- Jung K-H
- Junger WG
- Kahles T
- Kaushansky K
- Kawada H
- Kawamata T
- Kernie SG
- Kettle AJ
- Kimelberg HK
- Kimelberg HK
- Kleinschnitz C
- Kleinschnitz C
- Kleinschnitz C
- Kleinschnitz C
- Kleinschnitz C
- Kleinschnitz C
- Koeffler HP
- Kolb B
- Kollmar R
- Kraft P
- Kunz A
- Kunz A
- Langhauser F
- Law MR
- Lawes CMM
- Lee HJ
- Lee J-K
- Lee S-T
- Lee S-T
- Leeb-Lundberg LMF
- Lees KR
- Lees KR
- Lehnardt S
- Lewington S
- Li L
- Li Q
- Li S
- Li Y
- Liesz A
- Liman TG
- Lin J-Y
- Liu B
- Liu D-Z
- Lozano R
- Lumenta DB
- Luo Y
- Madeddu P
- Makrilia N
- Manley GT
- Mao Q-Q
- Marceau F
- Martins SB
- Matsuda T
- Mazzeo AT
- Mazzeo AT
- McIntosh TK
- Ming G-L
- Minnerup J
- Minnerup J
- Minnerup J
- Minnerup J
- Minnerup J
- Minnerup J
- Mostany R
- MRI.
- Muir KW
- Murikinati S
- Nader-Kawachi J
- Nagata S
- Nakamura K
- Nakano-Doi A
- Nassar T
- Navarro-Sobrino M
- Nieswandt B
- Nogueira RG
- Noto T
- O'Collins VE
- O'Donnell ME
- Oki K
- Opitz N
- Osman MM
- Papadopoulos CM
- Park D-H
- Paton JA
- Pellegrini-Giampietro DE
- Pham M
- Pham M
- Phng L-K
- Pignataro G
- Pignataro G
- Planas AM
- Pollock JD
- Popa-Wagner A
- Psaty BM
- Quaegebeur A
- Radermacher KA
- Radermacher KA
- Rashid P
- Reeves MJ
- Ren X
- Ren X
- Ren X
- Reubinoff BE
- Ribeiro C
- Ringelstein EB
- Risau W
- Risher WC
- Roberts T
- Romanos E
- Rosell A
- Rossi DJ
- Rubattu S
- RĂos C
- Sacco RL
- Sachs L
- Sahota P
- Salomon O
- Saver JL
- Saver JL
- Savitz SI
- Savitz SI
- Schaechter JD
- Schmidt-Hieber C
- Schneider A
- Schneider A
- Schäbitz WR
- Sealy-Jefferson S
- Sharkey J
- Sharma S
- Shaw CM
- Shichita T
- Shichita T
- Shuaib A
- Siegerink B
- Silver J
- Simard JM
- Sirén AL
- Smith WS
- Stoll G
- Storini C
- Stroke Unit Trialists' Collaboration
- Strong K
- Su J
- Sugiyama Y
- Sun Y
- Sutherland BAB
- Tait MJ
- Takahashi K
- Tang S-C
- Tang XN
- Tashiro A
- The Lancet Neurology
- Tortiglione A
- Touzé E
- Turnbull F
- Unterberg AW
- Vahedi K
- Valable S
- Vantourout P
- Vendrame M
- Vermeer SE
- Wagner DD
- Wagner JE
- Wang L
- Ward NS
- Wardlaw JM
- Warner DS
- Wei Y
- Whelton PK
- Wright JM
- Yagita Y
- Yan J
- Yanamoto H
- Yenari MA
- Yilmaz G
- Zausinger S
- Zausinger S
- Zerangue N
- Zhang ZG
- Zhang ZG
- Zhao B-Q
- Zhao C
- Zhu YI
- Ziegler G
- Publication venue
- 'Morgan & Claypool Publishers LLC'
- Publication date
- Field of study
Anti-inflammatory Activity
- Author
- A Ahluwalia
- A Akeson
- A Alfieri
- A Blackham
- A Boris
- A Cabrero
- A Castrillo
- A Colorado
- A Crummey
- A Daniel
- A Ferrante
- A Golebiowski
- A GraneĂź
- A Hedberg
- A Lee
- A Mortellaro
- A Nagahisa
- A Naya
- A Nencioni
- A Pouleau
- A Robert
- A Rubino
- A Sabatino Di
- A Saria
- A Tanaka
- A Tomlinson
- A Tubaro
- A Zlotnik
- AA Miles
- AB Dietz
- AC Castro
- AC Issekutz
- AC Lennard
- AD Fryer
- AD Medhurst
- AE McEachern
- AEI Proudfoot
- AJ Bennett
- AJ Lewis
- AJ Miller
- AK Roshak
- AKW Tse
- AL Akeson
- AL Willis
- AM Wolf
- Anonymous
- AP Alexenko
- AP Alexenko
- AP Roszkowski
- AR Renzetti
- AS Kalgutkar
- AT Evans
- AW Ford-Hutchinson
- AW Yem
- B Beutler
- B Dubinsky
- B Goffe
- B Jarvis
- B Kaltschmidt
- B Moser
- B Rudas
- B Samuelsson
- B Sander
- B Sander
- BA Jakschik
- BA Whittle
- BB Aggarwal
- BB Aggarwal
- BD Gitter
- BL Daugherty
- C Blanquart
- C Bombardier
- C Brideau
- C Emond
- C Gloxhuber
- C Jiang
- C Kemal
- C Kunsch
- C Laudanna
- C Liebmann
- C Liebmann
- C Liu
- C Liu
- C Mendoza-Milla
- C Pfeifer
- C Shen
- C Takeguchi
- CA Dinarello
- CA Dinarello
- CA Dinarello
- CA Maggi
- CA Maggi
- CA Smith
- CA Winter
- CA Winter
- CC Chan
- CD Anderson
- CD Funk
- CH Hannum
- CH Pontzer
- CJ Dunn
- CJ Hawkey
- CJ Mussap
- CM Lee
- CM Yang
- CN Hensby
- CSJ Walpole
- CV Winder
- D Bishop-Bailey
- D Branceni
- D D’Ambrosio
- D Eggerickx
- D Faust
- D Ignar
- D Kollias
- D Kontoyiannis
- D Lorenz
- D Mastrangelo
- D O’Gradaigh
- D Pruneau
- D Riendeau
- D Riendeau
- D Rossi
- DA Flick
- DA Kalbhen
- DB Carter
- DB Colagiovanni
- DC Manning
- DE Furst
- DE Griswold
- DE Griswold
- DE Moller
- DF Woodward
- DJ Grainger
- DJ McCarty
- DJ McCarty
- DK Gemmel
- DL Saussy Jr
- DM Butler
- DM Crothers
- DM Knight
- DM Siegel
- DT Beattie
- E Arrigoni-Martelli
- E Bosio
- E Fujihira
- E Fujii
- E Moore
- E Sarrubi
- E Schött
- E Whitehorn
- E Wong
- EA Graham
- EA Higgs
- EE Opas
- EF Webb
- EG Weirich
- EH Karran
- EJ Fernandez
- EK Ainscow
- EM Eugui
- EM Kudlacz
- EM Lasché
- ES Alnemri
- ES Tai
- F D’Acquisto
- F Erdö
- F Gbahou
- F Gobeil
- F Herrmann
- F Lembeck
- F Marceau
- F Marceau
- F Nantel
- F Sallusto
- F Yan
- F Zhang
- FJ Legat
- FJT Staal
- FR Cochran
- G Buell
- G Camussi
- G Cirino
- G D’Amato
- G Hofrichter
- G Jancso
- G Tonelli
- G Wagner
- G Wiemer
- G Wilhelmi
- G Woerly
- GA FitzGerald
- GA Higgs
- GB Penn
- GC Sen
- GC Viscomi
- GD Anderson
- GJ Hankey
- GN Prado
- GP Lewis
- GP O’Neill
- GR Bobalik
- GR Drummond
- GT Le
- GV Lucca De
- GW Moe
- H Abt
- H Akiyama
- H Cambridge
- H Fahmi
- H Heitsch
- H Kojo
- H Safayhi
- H Salari
- H Schmidt
- H Selye
- H Shionoya
- H Shirota
- H Umehara
- HA Schreuder
- HD Lim
- HD Lim
- HG Alpermann
- HG Schaible
- HG Vogel
- HG Vogel
- HG Vogel
- HG Vogel
- HG Vogel
- HG Vogel
- I Nicoletti
- IE Bush
- IJ Esch De
- IL Bonta
- IM Adcock
- IM McLay
- IS Figari
- J Agnholt
- J Berg
- J Bouthillier
- J Braun
- J Carleson
- J Chang
- J Chin
- J Harvey
- J Keffer
- J Marek
- J Mizrahi
- J Norman
- J Rinder
- J Tian
- J Vane
- J Vane
- J Vane
- J Veenstra
- J Waugh
- JA Gracie
- JA Kim
- JA Mitchell
- JB Calixto
- JB Cheng
- JB Warren
- JC Beaujouan
- JC Souza Pinto
- JD Winkler
- JF Kachur
- JG Meingassner
- JG Menke
- JG Vallejo
- JH Lee
- JH Ruth
- JI Braga da Motta
- JI Shigeta
- JJ Chen
- JJ Haringman
- JJ Moreno
- JJ Young
- JK Gierse
- JKF Hess
- JL Bascands
- JL Field
- JL Field
- JL Henry
- JL Kang
- JL Kang
- JL Martal
- JM Young
- JM Young
- JM Young
- JP Fortin
- JP Galizzi
- JP Portanova
- JP Tarayre
- JR Bing
- JR Burke
- JR Vane
- JS Faires
- JS Warren
- JS Yuan
- JT Whicher
- JW Christman
- JW Christman
- JW Watson
- K Akassoglou
- K Bon
- K Heynink
- K Hirota
- K Iwasaki
- K Nagata
- K Natarajan
- K Paulini
- K Paulini
- K Pfizenmaier
- K Redlich
- K Ren
- K Seibert
- K Seibert
- K Sugio
- K Tanaka
- K Thiam
- K Tiku
- K Tsumuri
- K Vuoltteenaho
- K Watanabe
- K Watanabe
- K Wirth
- KA Schneck
- KB Gordon
- KC Appell
- KH Sensch
- KJ Wirth
- KM Mohler
- KP Meyers
- KR Aupperle
- KU Weithmann
- KU Weithmann
- L Acarin
- L Chen
- L Harvath
- L Quartara
- L Reber
- L Sancilio
- L Seguin
- L Seguin
- L Singh
- LA Davis
- LA Tomchek
- LA Urban
- LB Hough
- LF Sancilio
- LH Kligman
- LJ Crofford
- LL Iversen
- LM Blatt
- LM Young De
- LM Young De
- LMF Leeb-Lundberg
- LO Randall
- M Boucher
- M Bradford
- M Broccardo
- M Feldmann
- M Frimmer
- M Félétou
- M Hiramoto
- M Katin
- M Katsumata
- M Lassila
- M Liang
- M Liang
- M Matsubara
- M Murakawa
- M MĂĽhlbauer
- M Otsuka
- M Ouellet
- M Peterfalvi
- M Roch-Arveiller
- M Tramontana
- M Zhang
- MA Botrel
- MA Cascieri
- MA Hull
- MA Matuszek
- MB Lawrence
- MD Brand
- MD Brand
- ME Poynter
- ME Rosenthale
- ME Rosenthale
- MG Fried
- MG O’Sullivan
- MG Tovey
- MH Perrone
- MJ Uddin
- MK Pugsley
- ML Richards
- MM Campos
- MM Chang
- MM Chaturvedi
- MM Krause
- MM Teixeira
- MM Tropea
- MN Perkins
- MNJ Rupniak
- MR Shalaby
- MS Kramer
- MS Nanes
- MSS Palanki
- MSS Palanki
- N Ackerman
- N Fujioka
- N McClure
- N Minami
- N Mukaida
- N Rouissi
- N Scheinfeld
- N Selve
- NE Rhaleb
- NE Rhaleb
- NJ Brenner
- NMJ Rupniak
- NMJ Rupniak
- NV Chandrasekharan
- O RĂĄdmark
- OP Gupta
- P Borgeat
- P Clarke
- P Cole
- P Delerive
- P D’Orléans-Juste
- P Holm-Pedersen
- P Houshmand
- P Kuhl
- P Li
- P Phelps
- P Schiatti
- P Schönhöfer
- P Traxler
- PB Simpson
- PC Atkins
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