11 research outputs found
A PI3K-and GTPase-independent Rac1-mTOR mechanism mediates MET-driven anchorage-independent cell growth but not migration
- Publication venue
- 'American Association for the Advancement of Science (AAAS)'
- Publication date
- 23/06/2020
- Field of study
Receptor tyrosine kinases (RTKs) are often overexpressed or mutated in cancers and drive tumor growth and metastasis. In the current model of RTK signaling, including that of MET, downstream phosphatidylinositol 3-kinase (PI3K) mediates both cell proliferation and cell migration, whereas the small guanosine triphosphatase (GTPase) Rac1 mediates cell migration. However, in cultured NIH3T3 and glioblastoma cells, we found that class I PI3K mediated oncogenic MET-induced cell migration but not anchorage-independent growth. In contrast, Rac1 regulated both processes in distinct ways. Downstream of PI3K, Rac1 mediated cell migration through its GTPase activity, whereas independently of PI3K, Rac1 mediated anchorage-independent growth in a GTPase-independent manner through an adaptor function. Through its RKR motif, Rac1 formed a complex with the kinase mTOR to promote its translocation to the plasma membrane, where its activity promoted anchorage-independent growth of the cell cultures. Inhibiting mTOR with rapamycin suppressed the growth of subcutaneous MET-mutant cell grafts in mice, including that of MET inhibitor-resistant cells. These findings reveal a GTPase-independent role for Rac1 in mediating a PI3K-independent MET-to-mTOR pathway and suggest alternative or combined strategies that might overcome resistance to RTK inhibitors in patients with cancer
The Functions of Auxilin and Rab11 in Drosophila Suggest That the Fundamental Role of Ligand Endocytosis in Notch Signaling Cells Is Not Recycling
- Author
- A Chitnis
- A Rajan
- A Tomlinson
- A Tomlinson
- AK Satoh
- AL Parks
- ALM Cadavid
- Amit Singh
- B Pishavee
- Bomsoo Cho
- C Pitsouli
- CA Horvath
- David Bilder
- DP Alone
- E Eisenberg
- E Overstreet
- E Pavlopoulos
- E Yeh
- EC Lai
- EC Lai
- EJ Hagedorn
- G Emery
- G Scita
- GA Deblandre
- H Chen
- H Chen
- H Chen
- H Stenmark
- J Jafar-Nejad
- J-Y Roignant
- JA Fischer-Vize
- Janice A. Fischer
- Ji-Hoon Lee
- JT Nichols
- JT Nichols
- M Fanto
- M Furthauer
- M Itoh
- M Matsuda
- ME Fortini
- MTD Cooper
- N Benhra
- N Bogard
- NE Baker
- R Le Borgne
- R Le Borgne
- R Le Borgne
- RW Carthew
- S Robinow
- S Sigismund
- Sarah L. Windler
- SF Heuss
- SH Eun
- SH Eun
- SJ Bray
- SL Windler
- Suk Ho Eun
- Susan M. L. Banks
- T Bai
- T Vaccari
- T Wolff
- V Kandachar
- W Wang
- W Wang
- WE Gall
- WR Gordon
- X Sun
- X Tian
- Xuanhua Xie
- Y Huang
- Publication venue
- Public Library of Science
- Publication date
- 01/03/2011
- Field of study
Notch signaling requires ligand internalization by the signal sending cells. Two endocytic proteins, epsin and auxilin, are essential for ligand internalization and signaling. Epsin promotes clathrin-coated vesicle formation, and auxilin uncoats clathrin from newly internalized vesicles. Two hypotheses have been advanced to explain the requirement for ligand endocytosis. One idea is that after ligand/receptor binding, ligand endocytosis leads to receptor activation by pulling on the receptor, which either exposes a cleavage site on the extracellular domain, or dissociates two receptor subunits. Alternatively, ligand internalization prior to receptor binding, followed by trafficking through an endosomal pathway and recycling to the plasma membrane may enable ligand activation. Activation could mean ligand modification or ligand transcytosis to a membrane environment conducive to signaling. A key piece of evidence supporting the recycling model is the requirement in signaling cells for Rab11, which encodes a GTPase critical for endosomal recycling. Here, we use Drosophila Rab11 and auxilin mutants to test the ligand recycling hypothesis. First, we find that Rab11 is dispensable for several Notch signaling events in the eye disc. Second, we find that Drosophila female germline cells, the one cell type known to signal without clathrin, also do not require auxilin to signal. Third, we find that much of the requirement for auxilin in Notch signaling was bypassed by overexpression of both clathrin heavy chain and epsin. Thus, the main role of auxilin in Notch signaling is not to produce uncoated ligand-containing vesicles, but to maintain the pool of free clathrin. Taken together, these results argue strongly that at least in some cell types, the primary function of Notch ligand endocytosis is not for ligand recycling
c-Met signalling and endocytosis in clear cell ovarian cancer
- Publication venue
- Publication date
- 01/10/2018
- Field of study
Tracking Trafficking of Notch and Its Ligands in Mammalian Cells
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Deciphering the Glycolipid Code of Alzheimer's and Parkinson's Amyloid Proteins Allowed the Creation of a Universal Ganglioside-Binding Peptide
- Author
- A Kakio
- A Radhakrishnan
- BR Brooks
- D Hammache
- D Hammache
- D Hammache
- D Lingwood
- E Aubert-Jousset
- G Wu
- H Asou
- H Jang
- HA Hannson
- J Fantini
- J Fantini
- J Fantini
- J Fantini
- J Fantini
- J Fantini
- J Fantini
- J Fantini
- J Fantini
- Jacques Fantini
- JC DĂaz
- K Chakrabandhu
- K Matsuzaki
- K Yanagisawa
- L Svennerholm
- M Levy
- N Arispe
- N Guex
- N Izquierdo-Useros
- N Oikawa
- N Taieb
- N Yahi
- N Yamamoto
- Nouara Yahi
- P Hug
- R Kayed
- R Mahfoud
- R Mahfoud
- R Thomsen
- S Hamel
- S Hong
- S Rasool
- SF Heuss
- T Matsubara
- T Matsubara
- T Matsubara
- TJ Nelson
- V Mattei
- Vladimir N. Uversky
- WB Puryear
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- Field of study
Functional Analysis of the NHR2 Domain Indicates that Oligomerization of Neuralized Regulates Ubiquitination and Endocytosis of Delta during Notch Signaling
- Author
- Barsi JC
- Benhra N
- Boulianne GL
- Brand AH
- Bray SJ
- Chanet S
- Commisso C
- Corbin V
- Daskalaki A
- Deblandre GA
- Emery G
- Gho M
- Glittenberg M
- Gordon WR
- Hartenstein AY
- He F
- Heuss SF
- Hu Y
- Itoh M
- Justice NJ
- Klueg KM
- Koo BK
- Koutelou E
- Lai EC
- Lai EC
- Lai EC
- Lai EC
- Lamothe B
- Le Borgne R
- Le Borgne R
- Le Borgne R
- Lehmann R
- Li J
- Linares LK
- Lindsell CE
- Nastasi T
- Nichols JT
- Parks AL
- Pavlopoulos E
- Pitsouli C
- Portin P
- Rajan A
- Rorth P
- Skwarek LC
- Snow PM
- Tiyanont K
- Wang W
- Wang WD
- Weinmaster G
- Ye H
- Yeh E
- Yeh E
- Publication venue
- 'American Society for Microbiology'
- Publication date
- Field of study
Faster embryonic segmentation through elevated Delta-Notch signalling
- Author
- A Aulehla
- A Chitnis
- A Geling
- A Inoue
- A Mara
- A Meyer
- A Sawada
- AC Oates
- AJ Krol
- C Haddon
- C Schroter
- C Schroter
- C Schröter
- C Soza-Ried
- C Takke
- C Thisse
- C Zhang
- CB Kimmel
- D Henrique
- D Julich
- D Pan
- D Soroldoni
- D Soroldoni
- D Sprinzak
- DJ Jörg
- EA Delaune
- EM Ozbudak
- FJ van Eeden
- GJ Wright
- H Ogino
- H Ogino
- I Palmeirim
- IH Riedel-Kruse
- J Dubrulle
- J Fu
- J Schindelin
- JR Collier
- JS Taylor
- K Horikawa
- K Ishimatsu
- L Bajard
- L Herrgen
- L Herrgen
- LG Morelli
- M Inuzuka
- M Itoh
- M Matsuda
- M Sarov
- PJ Murray
- RK Ejsmont
- S Ares
- S Hans
- SA Holley
- SF Heuss
- V Thermes
- W Kim
- WC Jen
- Y Harima
- YJ Jiang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Transduction of group I mGluR-mediated synaptic plasticity by β-arrestin2 signalling
- Author
- A Contractor
- A Contractor
- AA Marusiak
- AC Emery
- AC Emery
- AS Nateri
- AY Hsia
- B Luan
- BP Clark
- C Heuss
- C Luscher
- CE Gee
- CE Gee
- CL Schmid
- CM Niswender
- DL Hunt
- DW Ali
- E Gomez
- ED Nosyreva
- EM Snyder
- G Dolen
- G Dolen
- GC Faas
- H Daniel
- H Kubota
- H Wei
- HA Hathaway
- HB Kwon
- J Bain
- JM Rook
- JT Brown
- K Xiao
- KH Ahn
- KM Huber
- KM Huber
- L Fagni
- L Iacovelli
- L Iacovelli
- LB Dale
- LM Luttrell
- LM Luttrell
- M Hirose
- M Pi
- MF Bear
- MJ Palmer
- MW Waung
- N Harata
- N Kemp
- N Rebola
- N Rebola
- ND Cosford
- P Benquet
- PH McDonald
- S Chiechio
- S Notartomaso
- S Piccinin
- S Sato
- SF Frausto
- SH Oliet
- SJ Mundell
- SK Shenoy
- SM Gallagher
- T Bouschet
- T Gelb
- V Chevaleyre
- XM Li
- Y Kawamura
- Y Sudo
- Z Gu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Organolead Compounds
- Author
- A Andeli
- A Astiglioni
- A Bellomo
- A Berezniak
- A Betta
- A Blumenthal
- A Boulard de
- A Burg
- A Cahours
- A Cahours
- A Cahours
- A Cahours
- A Demidowicz
- A D’Ulivo
- A Egerton
- A Egerton
- A Egerton
- A Egerton
- A Egerton
- A Egerton
- A Egerton
- A Egerton
- A Egerton
- A Febo
- A Febo
- A Ferro
- A Fookson
- A Ghira
- A Ghira
- A Girelli
- A Goldberg
- A GrĂĽnwald
- A GrĂĽnwald
- A Hager
- A Hager
- A Hager
- A Hager
- A Hamilton
- A Imhausen
- A Imhausen
- A Ivanov
- A Jennen
- A Kaufman
- A Klein
- A Klein
- A Klein
- A Klein
- A Laveskog
- A Laveskog
- A Malatesta
- A Marroni
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morelli
- A Morgan
- A Morgan
- A Richard
- A Richard
- A Richard
- A Rieche
- A Rizzoli
- A Rizzoli
- A Ross
- A Salemi
- A Sokolik
- A Terenin
- A Terenin
- A Terenin
- A Terenin
- A Terenin
- A Vardanis
- A Vardanis
- A Zanker
- A Zscharn
- A.L. Gol’dshtein
- AA Dobrinskaja
- AA Dobrinskaja
- AA Gureev
- AA Gureev
- AA Gureev
- AA Gureev
- AA Gureev
- AA Gureev
- AA Pashchenko
- AB Callear
- AB Callear
- AB Garrett
- AB Yaroshevskii
- AB Yaroshevskii
- ABF Duncan
- ABF Duncan
- ABF Duncan
- AC Chamberlain
- AC Chamberlain
- AC Egerton
- AC Egerton
- AC Egerton
- AC Egerton
- AC Egerton
- AC Egerton
- AC Egerton
- AC Egerton
- AD Walsh
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorin
- AD Zorjn
- AE Borisov
- AE BĂĽhler
- AE Chester
- AE Goddard
- AE Jukes
- AE Lutskii
- AE Lutskii
- AE Stearn
- AE Thiemann
- AF Zhigach
- AF Zhigach
- AG Allen
- AG Allen
- AG Baker
- AG Baker
- AG Panetsos
- AI Lavrinenko
- AI Slobodchikova
- AI Vogel
- AJ Barker
- AJ Fleming
- AJ Jakubowitsch
- AJ Jakubowitsch
- AJ Owen
- AJ Pahnke
- AJ Pahnke
- AK Monkevich
- AK Palmby
- AL Linch
- AL Linch
- AL Linch
- AL Linen
- AL Linen
- AL Linen
- AL McClellan
- AL Rheingold
- AL Rheingold
- AM Beccaria
- AM Beccaria
- AM Bond
- AM Bond
- AM Bond
- AM Bond
- AN Nesmejanow
- AN Nesmeyanov
- AN Nesmeyanov
- AN Pudovic
- AN Pudovic
- AN Pudovik
- Anonymous
- Anonymous
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- AO Melby
- AO Walker
- AP Batalov
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- AP Giraittis
- AP Kravchenko
- AP Thompson
- AP Tomilov
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- AR Belous
- AS Arkhipov
- AS Ghosh
- AS Karamayan
- AS Karamyan
- AS Ryabova
- Associated Octel Co. Ltd.
- Associated Octel Co. Ltd. (Belg. 610 109
- AT Gil’mutdinov
- AW Harman
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- AWP Jarvie
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- AY Pogosyan
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- B Barrett
- B Carli
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- B Hetnarski
- B Holle
- B Ivovic
- B Iwanicka
- B Kolb
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- B Lees
- B Mustafa
- B Radziuk
- B Radziuk
- B Radziuk
- B Radziuk
- B Skalicka
- B Smaller
- B Smaller
- B Steiger
- B Ventura
- B Ventura
- B Ventura
- B Wrackmeyer
- BA Thrush
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- BC Pant
- BD Quimby
- BE Buell
- BE Gordon
- BF Murashov
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- BG Maddock
- BI Tarunin
- BK Choudhuri
- BL Gulson
- BM Sturgis
- BR Blakley
- BraI.ThwaI.Te D.G.
- BS Kwak
- BS Strel’chjk
- BV Emel’yanov
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- BV Emel’yanov
- BV Smirnov
- BW Swanson
- C Alingaert
- C Alingaert
- C Alingaert
- C Allendar
- C Ampbell
- C Ampbell
- C Andeli
- C Apek
- C Arden
- C Arey
- C Armignani
- C Arr
- C Attaneo
- C Avallazzi
- C Beermann
- C Beermann
- C Bianchi
- C Bianchi
- C Botre
- C Campo
- C Cis
- C Colella
- C Giavarini
- C Klippel
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- C Löwig
- C Löwig
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- C Löwig
- C Löwig
- C Löwig
- C Löwig
- C Löwig
- C Marchetti
- C Nerin
- C Nicora
- C Nicora
- C Norris
- C Padovani
- C Sac
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- C Wronkowski
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- C.Alifornia Research Corp
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- California Research Corp.
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- CJ Feldhake
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- CS Marvel
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- CT Chu
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- CW Sortman
- D Amin
- D Bodiot
- D Britz
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- D Chakraborti
- D Chakraborti
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- D Chakraborti
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- D Danly
- D Downs
- D Downs
- D Downs
- D Downs
- D Downs
- D Eastman
- D Ferreira Da Silva
- D Ferreira Da Silva
- D Ferreira da Silva
- D Henneberg
- D Henneberg
- D Hunter
- D Husain
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- D Loroue
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- D Pletcher
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- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Aleksandrov
- YA Alexandrov
- YA Alexandrov
- YD Semchikov
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YK Chau
- YM Zinov’ev
- YM Zinov’ev
- YS Drugov
- YV Zhigailo
- Z Aneva
- Z Drabent
- Z Drabent
- Z Drabent
- Z Florjanczyk
- Z Forycki
- Z Karny
- Z Kowalski
- Z Kozarzewska
- Z Turlakiewicz
- Z Turlakiewicz
- Z Turlakiewicz
- Z Turlakiewicz
- Z Turlakiewicz
- ZK Lynkina
- ZM Manulkin
- ZM Manulkin
- ZM Manulkin
- ZM Manulkin
- ZV Veksler
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/1989
- Field of study
Glutamate as a Neurotoxin
- Author
- A Frandsen
- A Frandsen
- A Herb
- A Herb
- A Novelli
- A Ogawa
- A Riccio
- A Schrammel
- A Shuaib
- A Vliet van der
- A Zuddas
- AB Young
- AC Ludolph
- AE Kingston
- AH Schapira
- AH Schapira
- AI Faden
- AJ Baker
- AM Brown
- AM Buchan
- B Janetzky
- B McLaughlin
- B Reisberg
- B Zadow
- B Zingarelli
- BC Bowen
- BJ Snider
- BM Polster
- BT Faddis
- C Arias
- C Heuss
- C Ikonomidou
- C Ikonomidou
- C Ikonomidou
- C Ikonomidou
- C Ikonomidou
- C Ikonomidou
- C Ikonomidou
- C Malgouris
- C Portera-Cailliau
- C Zhang
- CA Boast
- CH Adler
- CJ Frederickson
- CT Sheline
- CV Borlongan
- D Blum
- D Giulian
- D Monte Di
- D Nakagawa
- D Pohl
- D Schmitz
- DB Calne
- DD Schoepp
- DJ Brooks
- DJ Cook
- DJ Laurie
- DJ Selkoe
- DJ Taylor
- DL Murman
- DM Rock
- DR Curtis
- DR Lucas
- DW Choi
- DW Choi
- DW Choi
- DW Cleveland
- E Bonfoco
- E Brouillet
- E Brouillet
- E Ozyurt
- E Urbanska
- F Block
- F Fonnum
- F Terro
- F Wahl
- F Wahl
- F Yamakura
- F Zipp
- F Zipp
- FJ Martinez-Guijarro
- G Bensimon
- G Cao
- G Lanzino
- G Lanzino
- GC Davis
- GD Zeevalk
- GE Hardingham
- GF Morris
- GJ Lees
- GJ Wang
- GK Steinberg
- GL Wenk
- GW Albers
- H Bernheimer
- H Braak
- H Ischiropoulos
- H Komuro
- H Monyer
- H Monyer
- H Monyer
- H Wachtel
- HA Krebs
- HS Sun
- I Nagano
- IJ Reynolds
- J Chen
- J Fearnley
- J Hugon
- J Zhang
- JA Dykens
- JB Schulz
- JD Rothstein
- JD Rothstein
- JE Chatterton
- JG Greene
- JG Greene
- JL Goodwin
- JL Montastruc
- JM Rabey
- JP Pin
- JR Brorson
- JR Brorson
- JR Geiger
- JS Fink
- JS Stamler
- JW Johnson
- JW Langston
- JW McDonald
- JW Olney
- JW Olney
- JW Olney
- JW Olney
- JY Koh
- K Inoue
- K Kieburtz
- K Matsuda
- K Tanaka
- K Tanaka
- K Williams
- KM Noh
- KR Lees
- KR Lees
- KW Lange
- KW Muir
- KW Muir
- L Guerrini
- L Hillered
- L Lacomblez
- L Molina y Vedia
- L Tenneti
- L Tenneti
- L Turski
- LF Marshall
- LL Dugan
- M Aarts
- M Benveniste
- M Enari
- M Frerking
- M Gaudette
- M Gonzalez-Zulueta
- M Gossel
- M Hollmann
- M Hollmann
- M Lafon-Cazal
- M Santiago
- M Takahashi
- M Tymianski
- M Tymianski
- M Vignes
- M Yokoyama
- MB Jorgensen
- MC Guyot
- ME Harris
- MF Beal
- MF Beal
- MF Beal
- MF Beal
- MF Beal
- MF Beal
- MJ Leach
- MJ Sheardown
- ML Mayer
- ML Mayer
- MP Mattson
- MR Hara
- MR Luquin
- MR Walton
- MY Globus
- MY Globus
- N Burnashev
- N Burnashev
- N Hattori
- N Sen
- N Tonder
- NM Seif el
- O Hansson
- OG McMaster
- P Chan
- P Chavis
- P Couratier
- P Couratier
- P Nicholls
- P Nilsson
- PE Castillo
- PJ Shaw
- PL McGeer
- PM Andersen
- PM Andersen
- PS Spencer
- PS Spencer
- PS Spencer
- PT Francis
- R Henshaw
- R Radi
- R Radi
- R Radi
- R Sattler
- R Sattler
- R Schwarcz
- R Schwarcz
- R Srivastava
- RC Crumrine
- RD Randall
- RD Terry
- RE Huie
- RH Singleton
- RR Hicks
- RS Schwab
- S Das
- S DiDonato
- S Du
- S Nakanishi
- S Ozawa
- S Rothman
- SA Jones-Humble
- SA Thayer
- SF Traynelis
- SL Sensi
- SL Sensi
- SM Davis
- SM Papa
- SM Rothman
- SP Palfi
- SR Bradley
- SS Koura
- SW Suh
- T Abe
- T Furukawa
- T Hayashi
- T Hayashi
- T Klockgether
- T Schewe
- T Yamaguchi
- TK McIntosh
- TL Perry
- TL Williams
- U WĂĽllner
- V Bruno
- V Bruno
- VL Dawson
- VL Dawson
- VM Mann
- WK Cullen
- X Tao
- Y Du
- Y Nakagawa-Hattori
- Y Tanabe
- Y Wang
- Y Zhang
- YG Jang
- YI Chen
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study