1 research outputs found
Iodine-Catalyzed Oxidative Cross-Coupling of Indoles and Azoles: Regioselective Synthesis of <i>N</i>‑Linked 2‑(Azol-1-yl)indole Derivatives
A highly
efficient iodine-catalyzed regioselective oxidative cross-coupling
of an indole C–H bond and azole N–H bond is described.
This metal-free reaction can be easily carried out at room temperature
under mild and environmentally friendly conditions and provides a
series of <i>N</i>-linked 2-(azol-1-yl)Âindole derivatives
in moderate to excellence yields