7 research outputs found
P2Y₂ Nucleotide Receptors Expressed Heterologously in Sympathetic Neurons Inhibit Both N-Type Ca²⁺ and M-Type K⁺ Currents
- Publication venue
- Publication date
- 15/07/1998
- Field of study
The P2Y₂ receptor is a uridine/adenosine triphosphate (UTP/ATP)-sensitive G-protein-linked nucleotide receptor that previously has been reported to stimulate the phosphoinositide signaling pathway. Messenger RNA for this receptor has been detected in brain tissue. We have investigated the coupling of the molecularly defined rat P2Y₂ receptor to neuronal N-type Ca²⁺ channels and to M-type K⁺ channels by heterologous expression in rat superior cervical sympathetic (SCG) neurons. After the injection of P2Y₂cRNA, UTP inhibited the currents carried by both types of ion channel. As previously reported [Filippov AK, Webb TE, Barnard EA, Brown DA (1997) Inhibition by heterologously expressed P2Y₂nucleotide receptors of N-type calcium currents in rat sympathetic neurones. Br J Pharmacol 121:849–851], UTP inhibited the Ca²⁺ current (I_{Ca(N)} by up to 64%, with an IC₅₀ of ∼0.5 μm. We now find that UTP also inhibited the K⁺_{M} current (I_{K(M)} by up to 61%, with an IC₅₀ of ∼1.5 μm. UTP had no effect on either current in neurons not injected with P2Y₂ cRNA. Structure–activity relations for the inhibition of I_{Ca(N)} and I_{K(M)} in P2Y₂ cRNA-injected neurons were similar, with UTP ≥ ATP > ITP ≫ GTP,UDP. However, coupling to these two channels involved different G-proteins: pretreatment withPertussis toxin (PTX) did not affect UTP-induced inhibition of I_{K(M)} but reduced inhibition of I_{Ca(N)} by ∼60% and abolished the voltage-dependent component of this inhibition. In unclamped neurons, UTP greatly facilitated depolarization-induced action potential discharges. Thus, the single P2Y₂ receptor can couple to at least two G-proteins to inhibit both Ca²⁺_{N} and K⁺_{M} channels with near-equal facility. This implies that the P2Y₂ receptor may induce a broad range of effector responses in the nervous system
Therapeutic applications of ATP-(P2)-receptors agonists and antagonists
- Author
- ABBRACCHIO MP
- ABBRACCHIO MP
- ABBRACHIO MP
- AKBER GKM DASARI VR, WEBB TE
- BARNARD EA
- BARNARD EA
- BENNETT WD
- BHAGWAT SS
- Bilha Fischer
- BOARDER MR HOURANI SMO
- BOGDANOV Y
- BOX ZHANG Y
- BOYER JL O&
- BRAKE AJ
- BURNSTOCK G
- BURNSTOCK G
- BURNSTOCK G
- CAMAIONI E
- CHAN CM
- CHEN CC
- COLLO G
- COMMUNI D
- COMMUNI D
- CUSACK NJ
- DAMER S
- DHULIPALA PDK WANG Y-X, KOTLIKOFF
- ECKSTEIN F
- ERB L
- FISCHER B
- FREDHOLM BB BURNSTOCK G, HARDEN TK, SPEDDING M
- GRACIA-GUZMAN B
- GRACIA-GUZMAN M
- HARDEN TK
- HILLAIRE-BUYS D
- HOURANI SMO WELFORD LA, CUSACK NJ
- INOUE K
- JACOBSON KA KIM Y-C
- JARLEBARK L
- JASSENS R
- JIANG Q
- KING BF
- LEON C
- LEON C
- LONGHURST PA
- LOUBATIERES-MARIAMI MM
- MORO S
- NORENBERG W
- PARR CE
- PEHK T
- PETIT P
- PODRASKY E
- RASSENDREN F
- RIBES G
- SALTER MW
- SIDDIQI SM
- SOUTHEY MC
- SPEDDING M
- URI A
- VALERA S
- VAN RHEE MA
- VIRGINIO C
- WEBB TE
- WEBB TE
- ZIMMERMAN H
- Publication venue
- 'Informa Healthcare'
- Publication date
- Field of study
Characteristics of ecto-ATPase of Xenopus oocytes and the inhibitory actions of suramin on ATP breakdown
- Author
- A Agarwal
- AK Nagy
- AL Bartlett
- AU Ziganshin
- BS Tuana
- CH Fiske
- CHV Hoyle
- E Honoré
- E Sigel
- EA Barnard
- EJ Grondal
- G Burnstock
- G Burnstock
- GB Segel
- GC Majumder
- GR Dubyak
- HF Zoellner
- JB Gurdon
- JD Pearson
- JE Smolen
- JF Manery
- KD Lustig
- KE Dombrowski
- KN Fedde
- L Erb
- LA Welford
- LC Nuttle
- LJ Greenfield Jr
- M Spedding
- MC Berman
- MD Rosenberg
- MP Abbracchio
- MW Beukers
- N Dascal
- NS Dhalla
- PM Murphy
- R Miledi
- RK Banerjee
- SE Hickman
- SH Lin
- SMO Hourani
- SN Russell
- T Kazic
- TE Webb
- TP Snutch
- X Xu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Regulation of Extracellular UTP-Activated Cl− Current by P2Y-PLC-PKC Signaling and ATP Hydrolysis in Mouse Ventricular Myocytes
- Author
- Balogh J Wihlborg AK, Isackson H, Joshi BV, Jacobson KA, Arner A, Erlinge D.
- Banfi C Ferrario S, De Vincenti O, Ceruti S, Fumagalli M, Mazzola A, N DA, Volonte C, Fratto P, Vitali E, Burnstock G, Beltrami E, Parolari A, Polvani G, Biglioli P, Tremoli E, Abbracchio MP.
- Bannister RA Melliti K, Adams BA.
- Erlinge D Harnek J, van Heusden C, Olivecrona G, Jern S, Lazarowski E.
- Gadsby DC Nairn AC.
- Hohl CM Wetzel S, Fertel RH, Wimsatt DK, Brierley GP, Altschuld RA.
- Hume JR Duan D, Collier ML, Yamazaki J, Horowitz B.
- KUNAPULI S P
- Lazarowski ER Boucher RC, Harden TK.
- Lin X Jo H, Sakakibara Y, Tambara K, Kim B, Komeda M, Matsuoka S.
- Matsuura H Ehara T.
- NAGEL G
- North RA.
- RALEVIC V
- Rossi A Olivares J, Aussedat J, Ray A.
- Scamps F Vassort G.
- Vassort G.
- Webb TE Barnard EA.
- Wihlborg AK Balogh J, Wang L, Borna C, Dou Y, Joshi BV, Lazarowski E, Jacobson KA, Arner A, Erlinge D.
- Yamamoto S Ehara T.
- Yamamoto-Mizuma S Wang GX, Hume JR.
- Yamamoto-Mizuma S Wang GX, Liu LL, Schegg K, Hatton WJ, Duan D, Horowitz TL, Lamb FS, Hume JR.
- ZAMBON A C
- Publication venue
- 'Physiological Society of Japan'
- Publication date
- 01/01/2007
- Field of study
Purinergic signalling in neuron–glia interactions
- Author
- A Araque
- A Colmar
- A Panatier
- A Pinto-Duarte
- A Townsend-Nicholson
- A Wieraszko
- AJ Brake
- AN Drury
- AR Light
- AS Kuperman
- B Grafstein
- B Innocent
- B Pearce
- B Stevens
- B Stevens
- B Stevens
- B Stevens
- B Zalc
- BB Fredholm
- BB Fredholm
- BM Altevogt
- BM Kucher
- BS Jahromi
- BS Khakh
- C Boucsein
- C Mayer
- CD Tweedle
- CE Jahr
- CG Schipke
- CH Kastritsis
- CM Wang
- D Davalos
- D Rochon
- D Van Calker
- DB Arthur
- DN Bowser
- DT Theodosis
- EA Barnard
- EA Newman
- EA Newman
- EA Newman
- EA Newman
- EA Newman
- EA Newman
- EC Toescu
- ER Lazarowski
- ER Stevens
- ES Vizi
- FA Edwards
- FA Holton
- FP Gendron
- FS Lee
- G Arcuino
- G Burnstock
- G Burnstock
- G Burnstock
- G Burnstock
- G Burnstock
- G Burnstock
- G Burnstock
- G Burnstock
- G Burnstock
- G Hollopeter
- G James
- GE Torres
- Geoffrey Burnstock
- GF Tian
- GR Dubyak
- GR Gordon
- H Zimmermann
- H Zimmermann
- H Zimmermann
- H Zimmermann
- HA Kolb
- I Hide
- J Kang
- J Saura
- J Sawynok
- J-Y Sul
- JA Markham
- JC Fowler
- JM Sanz
- JM Zhang
- JO Malva
- JT Neary
- JT Neary
- JT Neary
- JT Neary
- JT Neary
- JT Porter
- K Adrian
- K Inoue
- KA Jacobson
- KD Lustig
- KD McCarthy
- LK Parvathenani
- LV Lopes
- M Darby
- M Duner-Engstrom
- M Kukley
- M Nedergaard
- M Ryten
- M Ryten
- M Ryten
- M Simard
- M Tsuda
- M Zonta
- MH Teicher
- MJ Diogenes
- ML Cotrina
- MP Abbracchio
- MP Abbracchio
- MP Abbracchio
- MP Abbracchio
- MT Perez
- MT Tebano
- N Kaya
- N Rebola
- NE Reist
- O Pascual
- P Bodin
- P Illes
- P Illes
- PB Guthrie
- QS Liu
- QS Liu
- R Brambilla
- R Brambilla
- R Ciccarelli
- R Robitaille
- R Robitaille
- R. Douglas Fields
- RA Cunha
- RA Cunha
- RA Cunha
- RA Cunha
- RA Hauser
- RA North
- RC Choi
- RD Fields
- RD Fields
- RD Fields
- RD Fields
- RD Fields
- RJ Rodrigues
- RS Redman
- S Coco
- S Hindley
- S Kirischuk
- S Kriegler
- S Valera
- SA Lyons
- SA Masino
- SK Mishra
- SO Suadicani
- SO Suandicani
- T Almeida
- T Ishibashi
- T Yokomizo
- TA Fiacco
- TD Hassinger
- TE Webb
- V Lev-Ram
- V Maienschein
- V Parpura
- V Ralevic
- YD Bogdanov
- YJ Son
- Z Wang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Bareroot Seedling Culture
- Author
- A Webb
- AE Hassan
- AE Miller
- AE Romero
- AG Kais
- AG Kais
- AL MacKinney
- AR Gilmore
- AR Gilmore
- B Benzian
- BD Cleary
- BD McLendon
- BF Clark
- BF McLemore
- C Glerum
- C Hartley
- CG Bacon
- CJ Barden
- CL Tuttle
- CL Tuttle
- CM Stange
- CP Seymour
- CR Venator
- D Bowling
- D Raj
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DB South
- DG Simpson
- DGM Donald
- DGM Donald
- DGM Donald
- DH Marx
- DH Marx
- DH Marx
- DH Marx
- DH Marx
- DH Marx
- DH Marx
- DH Marx
- DH Marx
- DK Lauer
- DK Plank
- E Shoulders
- E Shoulders
- EA Sterling
- EC Stone
- EKS Nambiar
- EL Barnard
- EP Jones
- EV Hunt Jr.
- Forest Research Institute
- FT Ledig
- GA Fancher
- GA Kranzler
- GA Lang
- GA Ritchie
- GD Racy
- GE Hatchell
- GE Hatchell
- GE Hatchell
- GH Schubert
- GJ Bacon
- GK Slocum
- GK Xydias
- GL Switzer
- GL Switzer
- GL Switzer
- GL Switzer
- GL Switzer
- H Hellmers
- H Hellmers
- H Stanley
- HC Grigsby
- HJ Derr
- HL Williston
- HM Williams
- HM Williams
- HS Larsen
- HS Larsen
- HS Larsen
- I Arnold
- IAS Gibson
- JB White
- JC Brissette
- JC Brissette
- JC Brissette
- JC Brissette
- JC Brissette
- JD Johnson
- JD Johnson
- JD Walstad
- JG Mexal
- JG Mexal
- JG Mexal
- JG Mexal
- JG Mexal
- JG Mexal
- JG Mexal
- JG Mexal
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- JG Mexal
- JI Blake
- JJ Gill
- JJ Stransky
- JJ Stransky
- JL Ruehle
- JL Ruehle
- JM Balneaves
- JN Boyer
- JN Boyer
- JN Boyer
- JN Boyer
- JN Boyer
- JN Boyer
- JN Boyer
- JN Boyer
- JN Boyer
- JP Barnett
- JP Barnett
- JP Barnett
- JP Barnett
- JP Barnett
- JP Barnett
- JP Caulfield
- JR Dunlap
- JR Dunlap
- JR Seiler
- JR Toliver
- JS Boyce
- JT Auten
- JT Fisher
- JT May
- JT May
- JT May
- JT Paul
- KA Armson
- KA Baker
- KL McNabb
- LE Hinesley
- LH Reineke
- LL Autry
- LV Barton
- MB Bryan
- MGR Cannell
- ML Duryea
- MP Garber
- MW Bilan
- NM Scarbrough
- OG Langdon
- P Dougherty
- PC Wakeley
- PC Wakeley
- PC Wakeley
- PC Wakeley
- PC Wakeley
- PJ Hanson
- PP Feret
- PP Feret
- PP Feret
- PP Kormanik
- PR Larson
- R Blair
- R Driessche Van den
- R Driessche Van den
- R Driessche Van den
- R Taylor
- RD Shipman
- RD Shipman
- RF Sutton
- RG Wasser
- RJ Mitchell
- RJ Nebgen
- RL Bailey
- RM Burns
- RM Danielson
- RP Karrfalt
- RP Pharis
- SA Ardalan
- SA Ekwebelam
- SE McKeand
- SJ Colombo
- SJ Rowan
- SJ Rowan
- SJ Rowan
- SJ Rowan
- SJ Rowan
- SJ Rowan
- SW Hallgren
- T Hansbrough
- T Satoo
- TA Dierauf
- TA Dierauf
- TA Dierauf
- TA Dierauf
- TA Dierauf
- TA Dierauf
- TA Dierauf
- TE Maki
- TG Daniels
- TJ Hodgson
- U.S.D.A. Forest Service
- WA Retzlaff
- WA Retzlaff
- WC Carlson
- WC Carlson
- WC Carlson
- WC Carlson
- WD Kelley
- WD Kelley
- WF Beineke
- WG Morris
- WN Dixon
- WR Harms
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- WT Plass
- Y Tanaka
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/1991
- Field of study
Contributions of Quaternary botany to modern ecology and biogeography
- Author
- Aakala T
- Aalto M
- Aario R.
- Aartolahti T.
- Aartolahti T.
- Abel Schaad D
- Abel Schaad D
- Abraham V
- Abrams PA.
- Ackerly DD
- Ackerly DD.
- Ackerly DD.
- Adler PB
- Aitken SN
- Alba-Sánchez F
- Alba-Sánchez F
- Alberto FJ
- Alexander JM
- Alexander K
- Alexander K
- Allen K
- Allen MS
- Alley RB
- Allison TD
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- Alonso D
- Ammann B
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- Angeler DG
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- Armsworth PR
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- Tüxen R.
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- Urban MA
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- Valencia BG
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- van der Geer AAE
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- van der Knaap WO
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- van der Sande MT
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- Vellend M
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- Volkov I
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- Wingard GL
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- Publication venue
- 'Informa UK Limited'
- Publication date
- Field of study