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7 research outputs found
Identification of a Promising Drug Candidate for the Treatment of Type 2 Diabetes Based on a P2Y 1
Author
Adeghate E.
Belli S. I.
+55 more
Bilha Fischer
Boarder M. R.
Brandenberger H.
Burgess K.
Cattaneo M.
Cattaneo M.
Chapal J.
Chapal J.
Chung W. K.
David Varon
Ela Shai
Eliahu S.
Eliahu S. E.
Farret A.
Fernandez-Alvarez J.
Fischer B.
Fujii A.
Garrad R. C.
Gary A. Weisman
Gendaszewska-Darmach E.
Green J. B.
Griffin B. E.
Haim M. Barr
Halbfinger E.
Harada M.
Hegarty B. D.
Hillaire-Buys D.
Hoyle C. H. V.
Ishida H.
Jakubowski J. A.
Jean Camden
Jin J.
Kikugawa K.
Krishnan P.
Lenzen S.
Leon C.
Li P.
Li P.
Li P.
Loubatieres-Mariani M. M.
Macfarlane D. E.
Major D. T.
Moss D. W.
Nahum V.
Nahum V.
Parr C. E.
Schachter J. B.
Scheen A. J.
Selvin E.
Shaver S. R.
Shir Yelovitch
Srivastava P. C.
U.K. Prospective Diabetes Study (UKPDS) Group
Yelovitch S.
Zatorski A.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
Preparation of Synthetically Challenging Nucleotides Using Cyanoethyl P-Imidazolides and Microwaves
Author
Ahmadibeni Y.
Ahmadibeni Y.
+37 more
Amir A.
Batra V. K.
Boyle N. A.
Caton-Williams J.
Chamberlain B. T.
Connolly B. A.
Eckstein F.
Gille A.
Hirao I.
Jacek Jemielity
Joanna Kowalska
Kadokura M.
Kowalska J.
Kresse J.
Li P.
Li P.
Lin L.
Ludwig J.
Ludwig J.
Ludwig J.
Ma Q. F.
Malwina Strenkowska
Marcin Ziemniak
Mikkola S.
Milligan J. F.
Misiura K.
Mohamady S.
Mohamady S.
Nahum V.
Przemyslaw Wanat
Rydzik A. M.
Sheu K. R.
Spelta V.
Wu Y.
Xia S.
Yelovitch S.
Zlatev I.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
The enzymatic activity of the VEGFR2 receptor for the biosynthesis of dinucleoside polyphosphates
Author
A Wiedon
Anna Schulz
+42 more
Axel Kretschmer
Consortium TU
DJ Ma
DN Perkins
Doreen Janke
E Rapaport
Falko Boehringer
G Yegutkin
H Flodgaard
H Sase
H Schlüter
Harald Mischak
J Gobom
J Jankowski
J Lüthje
JE Girling
Joachim Jankowski
K Holmqvist
K Lehmann
K Spiekermann
K Tanaka
L Liu
MA Larkin
Markus van der Giet
Mirjam Schuchardt
PP Roux
Ralf Herwig
S Yelovitch
S Zhang
S Zhu
SP Dineen
T Matsumoto
T Matsumoto
V Jankowski
V Jankowski
V Jankowski
V Jankowski
V Jankowski
Vera Jankowski
Walter Zidek
Y Gui
Z Zhou
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Boranophosphate Isoster Controls P2Y-Receptor Subtype Selectivity and Metabolic Stability of Dinucleoside Polyphosphate Analogues
Author
Abbracchio M. P.
Bilha Fischer
+35 more
Delicado Esmerilda G.
Flores N. A.
Flores N. A.
Garrad R. C.
Gary A. Weisman
Han Q.
Hoard D. E.
Hoyle C. H. V.
Jacobson K. A.
Jacobson K. A.
Jankowski V.
Jankowski V.
Jean Camden
Kikugawa K.
Kikuta Y.
Li P.
Ludwig J.
Major D. T.
Maminishkis A.
McLennan A. G.
Mundasad M. V.
Nahum V.
Nahum V.
Pendergast W.
Pintor J.
Pintor J.
Randerath K.
Schlueter H.
Shaver S. R.
Shir Yelovitch
van der Giet M.
Vollmayer P.
Yegutkin G. G.
Yerxa B. R.
Zamecnik P. C.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
2,4-Dichloro-5-[(N-aryl/alkyl)sulfamoyl]benzoic Acid Derivatives: In Vitro Antidiabetic Activity, Molecular Modeling and In silico ADMET Screening
Author
Ahmadi A.
Altug C.
+55 more
Balam S.K.
Berendsen H.J.C.
Bhuva N.H.
Bian X.
Biasini M.
Cardoso M.F.
Chohan Z.H.
Dassault Systèmes B.I.O.V.I.A.
Dauter Z.
de Oliveira K.N.
Di Cesare Mannelli L.
Dudutiene V.
El‐Gohary N.S.
Gawin R.
Ghorab M.M.
Hsieh J.F.
Husain A.
Jhong C.H.
Jorgensen W.L.
Kam A.
Kim D.K.
Kim K.Y.
Li J.J.
Lipinski C.A.
Meltzer-Mats E.
Mishra C.B.
Murugavel S.
Navarrete-Vázquez G.
Nguyen T.H.
Patel H.S.
Poreba K.
Puranik N.V.
Rahim F.
Rani N.
Renzi G.
Riaz S.
Samridhi Thakral
Seo W.D.
Silva F.S.
Singh R.
Sun H.
Taha M.
Trott O.
Ugwu D.I.
Van Der Spoel D.
Veber D.F.
Vikramjeet Singh
Wang G.
Wang G.
Wang G.
Xu G.
Yamamoto K.
Yaseen S.
Yelovitch S.
Zani F.
Publication venue
'Bentham Science Publishers Ltd.'
Publication date
Field of study
No full text
Crossref
Synthesis and preclinical validation of novel P2Y1 receptor ligands as a potent anti-prostate cancer agent
Author
A Barzegar
A Delekate
+59 more
A. B. Parrish
AA Khalil
B Hechler
C Ferroni
CH Yao
D Zhang
DA Rudzka
DB Kitchen
DB Zorov
DB Zorov
EL Piatnitski Chekler
G Burnstock
G Roman
GM Sastry
HTT Le
HX Wan
HX Zhou
I Bellezza
I Masgras
J Shen
JA Pfefferkorn
JV Tapia-Vieyra
JW Putney
K Boland
K Liu
KA Jacobson
L Ouyang
LK Mamedova
M Kontoyianni
M Lamkanfi
M Shabbir
M Van Hemelrijck
M Wang
MT van Jaarsveld
NR Latorraca
P Doan
PC Wong
PS Bilbao
Q Wei
R Corriden
R Janssens
R Janssens
R Kaur
R Lappano
RA Friesner
RA Friesner
RC Calvert
RE Kumon
S Fulda
S McKenzie
S Yelovitch
SJ Guzman
SM Man
T Fiaschi
WH Li
X Wang
Y Ogawa
Y Yadav
Z Li
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Structure-Based Approaches to Ligands for G-Protein-Coupled Adenosine and P2Y Receptors, from Small Molecules to Nanoconjugates
Author
Abagyan R. A.
Abbracchio M. P.
+123 more
Abbracchio M. P.
Algaier I.
Andrews S. P.
Avila M. Y.
Balasubramanian R.
Ballesteros J. A.
Baraldi P. G.
Bennett K. A.
Borea P. A.
Canny S. A.
Carlsson J.
Carlsson J.
Chen D.
Chen J. F.
Chen Z.
Cheong S. L.
Chorna N. E.
Cohen R.
Conklin B. R.
Costanzi S.
Costanzi S.
Dale N.
Das A.
Das A.
Deflorian F.
Deflorian F.
Doré A. S.
Fernández-Dueñas V.
Ferré S.
Fishman P.
Flögel U.
Fozard J. R.
Fredholm B. B.
Gallego D.
Gallo-Rodriguez C.
Gao Z. G.
Gao Z. G.
Gao Z. G.
Gao Z. G.
Gessi S.
Gessi S.
Ginsburg-Shmuel T.
Han Y.
Hechler B.
Hodgson R. A.
Horckmans M.
Hruba L.
IJzerman A. P.
Ivanov A .A.
Ivanov A. A.
Ivanov A. A.
Jaakola V. P.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jacobson K. A.
Jeong L. S.
Jeong L. S.
Katritch V.
Kecskés A.
Kecskés M.
Kenneth A. Jacobson
Kim J.
Kim J.
Koizumi S.
Kolb P.
Kozma E.
Kozma E.
Lane S. D.
Langmead C. J.
Lebon G.
Liu W.
Longhi M. S.
Mantell S.
Maruoka H.
Maruoka H.
Moro S.
Niiya K.
Oh Y. E.
Orru M.
Parandeh F.
Press N. J.
Rasmussen S. G. F.
Ravn J.
Reiter E.
Riksen N. P.
Scheerer P.
Sesma J. I.
Shearer J.
Siddiqi S. M.
Sirci F.
Sitkovsky M.
Stemmer S. M.
Tan C.
Tilley S. L.
Topiol S.
Tosh D. K.
Tosh D. K.
Tosh D. K.
Vaidya A.
Valant C.
van der Horst E.
Van Poecke S.
van Tilburg E. W.
van Westen G. J.
Venkatakrishnan A. J.
Volpini R.
von Kügelgen I.
Wan T. C.
Wang T. C.
Wu B.
Wu H.
Xu F.
Xu J.
Yang H.
Yelovitch S.
Zhang C.
Zhukov A.
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref