20 research outputs found
Studies in macrolide synthesis: A stereocontrolled synthesis of a (9S)-macrolide intermediate for oleandomycin using chiral boron reagents.
Full text linkSelective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): Discovery of EPPTB (RO5212773)
Full text linkOptimisation of imidazole compounds as selective TAAR1 agonists: Discovery of RO5073012
Full text linkSynthesis of Cytotoxic Marine Macrolides: An Aldol-Based Approach to Spongistatin 1 (Altohyrtin A)
Full text linkEnantio- and diastereoselective aldol reactions of achiral ethyl and methyl ketones with aldehydes: the use of enol diisopinocampheylborinates
Full text linkA UGT2B10 Splicing Polymorphism Common in African Populations May Greatly Increase Drug Exposure
Full text linkBis(oxazoline) and Bis(oxazolinyl)pyridine Copper Complexes as Enantioselective Diels−Alder Catalysts: Reaction Scope and Synthetic Applications
Full text link4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: Drug-like and non-xanthine based A2B adenosine receptor antagonists
Full text linkDiscovery of benzoylisoindolines as a novel class of potent, selective and orally active GlyT1 inhibitors
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