8 research outputs found
Subarachnoidal Neurocysticercosis non-responsive to cysticidal drugs: a case series
- Author
- Publication venue
- BioMed Central
- Publication date
- 01/01/2010
- Field of study
<p>Abstract</p> <p>Background</p> <p>Neurocysticercosis (NC) is one of the most frequent parasitic diseases of the central nervous system. Cysticidal drugs, albendazole and praziquantel, are generally effective when parasites localize in the parenchyma. In contrast, parasites lodged in the subarachnoid basal cisterns are less responsive to treatment.</p> <p>Case Presentation</p> <p>The clinical and radiological pictures of six Mexican patients non-respondent to cysticidal treatment are presented.</p> <p>Conclusions</p> <p>The possible factors involved in the cysticidal non-response are discussed and hints are provided of potentially useful changes to therapeutic protocols.</p
Combination Treatment of Patients with BRAF-Mutant Melanoma: A New Standard of Care
- Author
- A Ackerman
- A Daud
- A Hauschild
- A Ribas
- A Ribas
- A Snyder
- Antonio M. Grimaldi
- C Robert
- C Robert
- D Frederick
- D Massi
- D Schadendorf
- D Schadendorf
- DB Johnson
- DR Minor
- EM Allen Van
- Ester Simeone
- F Hodi
- F Su
- G Long
- G Long
- G Long
- G Long
- G Moriceau
- GV Long
- J Galon
- J Larkin
- J Larkin
- J Wargo
- J Wilmott
- JA Jakob
- JA Sosman
- JJ Grob
- K Flaherty
- K Kim
- L Festino
- LA Diaz Jr
- Lucia Festino
- M Thakur
- Marco Palla
- PA Ascierto
- PA Ascierto
- PA Ascierto
- PA Ascierto
- PA Ascierto
- Paolo A. Ascierto
- PK Lau
- R Dummer
- R Mittapalli
- S Ugurel
- Vito Vanella
- X Jiang
- Y Yan
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Transcriptome analysis of the threatened snail Ellobium chinense reveals candidate genes for adaptation and identifies SSRs for conservation genetics
- Author
- A Conesa
- A Heyland
- A Kourtidis
- A Vasemagi
- B Dayrat
- BB Patnaik
- BB Patnaik
- BJ Haas
- C Camacho
- C Sim
- CJ Ramnanan
- CT Zimmer
- D Blankenberg
- DA Taylor
- DA Voronin
- DC Queller
- DF Mello
- E Novaes
- FM You
- G Zheng
- H Ogata
- H Shen
- HJ Lim
- J Boucher
- J Ge
- J Lv
- J Zhou
- JA Jost
- JH Spring
- JR Plenkowska
- L Wang
- L Wang
- LL Moroz
- M Ashburner
- M Kanehisa
- M Uliano-Silva
- MG Grabherr
- MI Mohd-Shamsudin
- MR Coscia
- O Mittapalli
- P Bouchet
- P Franchini
- PK Tucker
- RC Lovering
- SM Huse
- SW Kang
- SY Park
- SY Rhee
- T Ravasi
- TJ Fiedler
- W Xu
- WD Ong
- XJ Zhu
- Y Deng
- Y Yang
- Z Zhang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Clinical Relevance of BRAF V600E Mutation Status in Brain Tumors with a Focus on a Novel Management Algorithm
- Author
- A Banerjee
- A Bernstein
- A Drobysheva
- A Lassaletta
- A Mansouri
- A Roque
- AJ Sievert
- AM Marks
- B Beland
- BT Himes
- C Larochelle
- CM Ida
- D Aguilera
- D Dias-Santagata
- D Planchard
- DA Mordes
- DR Hargrave
- E Puxeddu
- E Tiacci
- EH Raabe
- F Bautista
- F Behling
- F Behling
- F del Bufalo
- G Schindler
- GA McArthur
- GV Long
- GV Long
- H Cin
- H Davies
- I Arozarena
- J Fangusaro
- J Larkin
- J-H Ahn
- JP Robinson
- JS Ross
- KC Schreck
- KC Schreck
- L Garnier
- L Sang
- L Sollfrank
- LL Ritterhouse
- M Dankner
- M Smith-Cohn
- M Stupp
- M Touat
- MA Karajannis
- MC Chamberlain
- MH Nissan
- MR Gilbert
- MW Kieran
- P Lito
- P Wen
- PI Poulikakos
- PK Brastianos
- PT Wan
- Q Breton
- R Dummer
- R Nazarian
- R Stupp
- R Stupp
- RK Mittapalli
- S Dahiya
- S Maraka
- S Rush
- S Vaidhyanathan
- SA Toll
- SK Meletath
- SY Lim
- T Kaley
- TM Johanns
- TW Yao
- WM Pardridge
- X Liu
- Y Lyustikman
- Y Piña
- Y Sun
- Y Tian
- YH Tan
- Z Tosuner
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Deciphering mechanisms of brain metastasis in melanoma - the gist of the matter
- Author
- A Hauschild
- A Kauffmann
- A Klein
- A Klein
- A Lehraiki
- A Mahajan
- A Muller
- A Roesch
- A Sandru
- AA Al-haidari
- AC Luissint
- AC Obenauf
- AD Boiko
- AD Boiko
- AD Bucheit
- AM Hong
- AM Mohammadi
- AW Silk
- B Ou
- BJ Wilson
- BP Murry
- C Crone
- C Fazakas
- C Nieder
- C Robert
- C Sun
- C Zhang
- CD McFarland
- CM Bailey
- D Capper
- D Dankort
- D Marchetti
- D Marchetti
- D Mathieu
- D Westphal
- DA Kircher
- DB Johnson
- DG Menter
- DS Vinay
- E McTyre
- E Monzani
- ES Anderson
- ES Park
- F Spagnolo
- FJ Huang
- FS Hodi
- G Chen
- G Cohn-Cedermark
- G Gampa
- G Rappa
- GA McArthur
- GB Deutsch
- GJ Freeman
- GJ Kaunitz
- GV Long
- GV Long
- GV Long
- H Davies
- H Easwaran
- H Lu
- H Niessner
- H Schwartz
- H Seifert
- H Soliman
- HA-H Tawbi
- HF Li
- I Arozarena
- I Bozic
- I Lee
- I Zubrilov
- IJ Fidler
- IJ Fidler
- J Chang
- J Gadiot
- J Gottschalk
- J Radke
- J Zhou
- JA Jakob
- JA Sosman
- JE Davies
- JF Jacobs
- JH Cho
- JJ Raizer
- JK Patel
- JN Poynter
- JV Cohen
- K Imafuku
- K Margolin
- K Yamada
- KT Flaherty
- L Cheng
- L Zhang
- LB Jilaveanu
- LJ Gardner
- LJ Schouten
- M Colombino
- M Kim
- M Labelle
- M Ngo
- M Qian
- M Saxena
- M Sensi
- M Yamamoto
- MA Davies
- MA Davies
- MA Davies
- MF Avril
- MR Middleton
- NJ Abbott
- NJ Bentley
- O Shakhova
- O Shonukan
- O Vornicova
- P Mu
- PB Chapman
- PB Chapman
- PE Valk
- PK Brastianos
- PW Sperduto
- Q Lin
- QF Wu
- R Dummer
- R Guo
- R Nazarian
- R Santarelli
- RB Corcoran
- RC Janzer
- RK Mittapalli
- S Bao
- S Gingis-Velitski
- S Hopkins
- S Spranger
- SA Haueis
- SB Goldberg
- SC Eisele
- SG Wu
- SL Topalian
- SS Choi
- T Carter
- T Pukrop
- T Redmer
- T Redmer
- T Sauka-Spengler
- T Schatton
- TC Gangadhar
- TG Simonsen
- TG Simonsen
- Torben Redmer
- TX Xie
- U Chukwueke
- V Chiarion-Sileni
- V Chiarion-Sileni
- V Gopalakrishnan
- V Lessmann
- V Nygaard
- V Stambolic
- W Cruz-Munoz
- W Stummer
- WO Greaves
- Y Cheli
- Y Denkins
- Y Kienast
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Role of Breast Cancer Resistance Protein (BCRP, ABCG2) in Cancer Outcomes and Drug Resistance
- Author
- A Au
- A Basseville
- A Brozik
- A Custodio
- A Dahlin
- A Pick
- A Porro
- A Sostelly
- A Telbisz
- AC Dankers
- AM Hamdan
- AM Wu
- B Fischer
- B Mohelnikova-Duchonova
- B Prasad
- B Shen
- B Vizio
- BC DiNatale
- C Scharenberg
- C Tian
- C Yang
- CG Dietrich
- CP Wu
- CP Wu
- D Campa
- D Hang
- DD Ross
- E Glodkowska-Mrowka
- E Herpel
- E Latorre
- E Mattia De
- E Turrini
- E Winter
- F Li
- F Lin
- F Lin
- F Wang
- F Wang
- FF Huang
- FF Huang
- FT Huang
- G Liu
- G Valdameri
- G Valdameri
- G Xiao
- H Boussac de
- H Kobuchi
- H Saranko
- H Tomiyasu
- H Yano
- H Zeng
- H Zhang
- HC Cooray
- HM Aliabadi
- HM Sim
- HR Kim
- J Bhullar
- J Hofman
- J Hofman
- J Lemmen
- J Merk
- J Selever
- J Xu
- J Zhao
- JD Allen
- JQ Feng
- JR Shaffer
- JW Xu
- K Juvale
- K Kage
- K Natarajan
- K Natarajan
- K Natarajan
- K Oda
- K Skoglund
- K Sodani
- K Yasuda
- KI Sereti
- KK To
- KK To
- KK To
- KK To
- KM Britton
- KM Giacomini
- KP Tan
- KW Tan
- L Xiang
- L Xiang
- LA Doyle
- LM Eldasher
- LM Tompkins
- LN Eadie
- LT Lima de
- M Delord
- M Fukudo
- M Grundy
- M Mogi
- M Rijavec
- M Suzuki
- M Tamura
- M Tiribelli
- M Vee Le
- M Zhang
- ML Cuestas
- ML Cuestas
- MM Zhu
- MT Hoque
- MT Ma
- MT Rosenfeldt
- N Baldini
- N Larbcharoensub
- N Memon
- NA Vries de
- NK Diop
- NV Litviakov
- OM Woodward
- P Bhatia
- P Chen
- P Goncalves
- P Lu
- P Zhang
- PA Koshkin
- PC Lin
- PK Campbell
- PL Ee
- PS Oh
- Q Chen
- Q Niu
- R Sane
- R Sane
- R Yamazaki
- RA Gilani
- RK Mittapalli
- RK Oberoi
- RR Singh
- S Agarwal
- S Agarwal
- S Benoki
- S Chuan Tang
- S Durmus
- S Gottschling
- S Hamada
- S Lheureux
- S Samanta
- S Shukla
- S Velamakanni
- S Zhao
- SA Zander
- SC Tang
- SC Tang
- SH Lee
- SJ Seong
- SJ Weroha
- SR Martins-Neves
- SS Vaidya
- SZ Ke
- T Ishikawa
- T Janvilisri
- T Minami
- T Mizuno
- T Nakanishi
- T Nakanishi
- T Nakanishi
- T Takada
- V Boso
- V Feinshtein
- V Goler-Baron
- V Goler-Baron
- V Martin
- VB Patel
- W Cheng
- W Huang
- W Li
- W Liu
- W Sun
- W Zhang
- WJ Yang
- WK Chau
- WL Furman
- WW Shen
- WY Liao
- X Jiao
- X Qian
- X Qian
- X Wu
- XQ Zhao
- XT Xu
- XX Li
- Y Adar
- Y An
- Y Honjo
- Y Imai
- Y Jiang
- Y Ma
- Y Ma
- Y Shinohara
- Y Shishido
- Y Wei
- Y Xie
- Y Xie
- Y Zong
- YH Lin
- YP Hu
- YP Liu
- YT Li
- YZ Pan
- Z Awada
- Z Ni
- Z Qin
- ZY Xu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Renal Drug Transporters and Drug Interactions.
- Author
- A Allen
- A Amphoux
- A Aslamkhan
- A Azzariti
- A Brandoni
- A Collett
- A Courtois
- A Crowe
- A Dahan
- A Dahan
- A Dahan
- A Dahlin
- A D’Emanuele
- A Enomoto
- A Enomoto
- A Futatsugi
- A Gaowa
- A Geick
- A Gupta
- A Hamada
- A Horie
- A Kamizono
- A Kawase
- A Koenen
- A Komatsuda
- A Kunze
- A Lazar
- A Lespine
- A Maeda
- A Maeda
- A McCormick
- A Milane
- A Mulgaonkar
- A Nakayama
- A Nies
- A Oka
- A Ose
- A Owen
- A Pawarode
- A Poirier
- A Rizwan
- A Servais
- A Soldner
- A Somogyi
- A Somogyi
- A Somogyi
- A Somogyi
- A Vildhede
- A Yamada
- A Yamada
- A Yonezawa
- A Yonezawa
- AA El-Sheikh
- AA Ela El
- AA Somogyi
- AA Somogyi
- AAK El-Sheikh
- AAK El-Sheikh
- AAK El-Sheikh
- AAK El-Sheikh
- AB Shapiro
- AE Busch
- AE Herwaarden van
- AE Kim
- AG Hotchkiss
- AH Schinkel
- AH Schinkel
- AH Schinkel
- AJ Dudley
- AJ Dudley
- AJ Scheen
- AL Dzierlenga
- AL VanWert
- AL VanWert
- AL Walker
- AM Al-Mohizea
- AM Bergman
- AM Hecken van
- AN Shaik
- Anton Ivanyuk
- AR Asif
- AS Mulato
- AS Ray
- AS Windass
- AS Windass
- AT Nies
- AT Wolman
- B Astorga
- B Feng
- B Feng
- B Fleisher
- B Greiner
- B Grover
- B Grover
- B Haenisch
- B Poller
- B Wenge
- BAC Acker van
- BC Burckhardt
- BC Ferslew
- BG Hardy
- BG Hardy
- BH Long
- BJ Gurley
- BL Lum
- BL Mason
- BM Schmitt
- BP Kearney
- BR Green
- C Chen
- C Chen
- C Chu
- C Fahrmayr
- C Fellner
- C Grammen
- C Hilgendorf
- C Jacobs
- C Jagannath
- C Kasserra
- C Kyrklund
- C Li
- C Luna-Tortós
- C Marzolini
- C Min-Koo
- C Pauli-Magnus
- C Pauli-Magnus
- C Pauli-Magnus
- C Pontier
- C Schmitt
- C Srimaroeng
- C Srimaroeng
- C Wandel
- C Wandel
- C Wang
- C Woodland
- C Xu
- C Zhang
- C Zhang
- C-H Ho
- CA Flynn
- CA Quezada
- CA Stanley
- CB Landersdorfer
- CB Landersdorfer
- CC Bridges
- CC Kuo
- CC Wong
- CC Wong
- CC Wong
- CE Frost
- CF Higgins
- CG Patel
- CGL Lee
- CH Rammelkamp
- CH Storch
- CL Noble
- CL Ronchera
- CO Kim
- Consortium IT
- CR Hill
- CR Yates
- CS Karyekar
- CS Lancaster
- CS Temple
- CV Fletcher
- D Capone
- D Cihalova
- D Devineni
- D Durr
- D Gründemann
- D Gründemann
- D Gründemann
- D Gründemann
- D Iusuf
- D Jung
- D Keppler
- D Lawlor
- D Li
- D Miura
- D Overbosch
- D Schrenk
- D Schwab
- D Siccardi
- D Taubert
- D Vishnuvardhan
- D Wang
- D Werner
- D Zhang
- Dai Cl
- DB Kell
- DE Burgio
- DE Martin
- DG Bailey
- DH Sweet
- DH Sweet
- DH Sweet
- DH Sweet
- DJ Tompson
- DL Bourdet
- DM Moss
- DM Truong
- DN Fish
- DS Miller
- DS Miller
- DW Boulton
- E Babu
- E Babu
- E Bakos
- E Cormet-Boyaka
- E Gozalpour
- E Kamiyama
- E Kimoto
- E Pasquier
- E Rytting
- E Rytting
- E Schwob
- E Stormer
- E Waller
- E-I Lepist
- E-S Jeong
- EE Robertson
- EF Choo
- EF Foote
- EG Schuetz
- EI Lepist
- EJ Guest
- EJ Wang
- EJ Wang
- EJ Wang
- EL Mariño
- EL Reyner
- EM Choi
- ES Oh
- F Faassen
- F Gimenez
- F Gutierrez
- F Leonessa
- F Müller
- F Müller
- F Pietruck
- F Shen
- F Tang
- F Tang
- F Trejtnar
- F Yamashita
- F Zhou
- FA Bainbridge
- FA Jong de
- FE O’Brien
- FE O’Brien
- FGM Russel
- FGM Russel
- Françoise Livio
- G Adamis
- G An
- G Ciarimboli
- G Ciarimboli
- G Ciarimboli
- G Ciarimboli
- G DiDiodato
- G He
- G Hill
- G Jayasagar
- G Kaler
- G Koren
- G Liu
- G Merino
- G Minuesa
- G Pan
- G Peytavin
- G Pottier
- G Reid
- G Reid
- GA Kullak-Ublick
- GC Williams
- GG Belz
- GJR Zaman
- GK Dresser
- GW Aherne
- H Chanteux
- H Duan
- H Endou
- H Fujimoto
- H Fujino
- H Gutmann
- H Hasannejad
- H Hasannejad
- H Honjo
- H Honjo
- H Honjo
- H Ishizuka
- H Izzedine
- H Jeong
- H Jones
- H Kidron
- H Ko
- H Kodaira
- H Koepsell
- H Koepsell
- H Komazawa
- H Kusuhara
- H Kusuhara
- H Kusuhara
- H Li
- H Liu
- H Matsuo
- H Matsuo
- H Motohashi
- H Motohashi
- H Nagy
- H Omote
- H Saitoh
- H Saitoh
- H Sasabe
- H Sato
- H Shen
- H Shen
- H Sun
- H Tahara
- H Tahara
- H Ueo
- H Yabuuchi
- H Yamaguchi
- H Yoon
- H Yuan
- H-K Lee
- HC Liu
- HE Jin
- HE Mellin
- HE Meyer zu Schwabedissen
- HH Kalsi
- HH Lee
- HJ Shin
- HM Faessel
- HM Kauffmann
- I Bachmakov
- I Badagnani
- I Ieiri
- I Ieiri
- I Ifergan
- I Leier
- I Massimi
- I Robieux
- I Tamai
- I Tamai
- I Tamai
- I Yano
- I-S Song
- IA Hauser
- IS Haslam
- IS Haslam
- IS Haslam
- IS Song
- IS Song
- IY Gong
- J Bai
- J Bentz
- J Biermann
- J Brillault
- J Crugten van
- J Cusato
- J Enokizono
- J Gao
- J He
- J Hunter
- J Knop
- J Knop
- J Koteff
- J Lee
- J Li
- J Li
- J Li
- J Lu
- J Mandikova
- J Mandíková
- J Müller
- J Naud
- J Oh
- J Rengelshausen
- J Rengelshausen
- J Shen
- J Shimada
- J Souza de
- J Stangier
- J Taipalensuu
- J Thomas
- J Weiss
- J Weiss
- J Weiss
- J Weiss
- J Weiss
- J Ye
- J Ye
- J Yin
- J Zhang
- J Zheng
- J Zong
- J-L Ghim
- J-Y Chung
- J-Y Han
- JB Pritchard
- JD Allen
- JD Schuetz
- JD Young
- JE Hibma
- JE Keskitalo
- JE Keskitalo
- JE Montfoort van
- JE Montfoort van
- JE Race
- JF Pouliot
- JH Choi
- JH Dalle
- JH Hochman
- JH Hooijberg
- JH Lee
- JJ Kiser
- JJ Kiser
- JJ Kohler
- JJ Kohler
- JL Morelle
- JM Burnell
- JM Davenport
- JM Kovarik
- JM Kovarik
- JM Kremer
- JN Santos Pereira Dos
- JP Sabo
- JP Wang
- JR Slizgi
- JS Hulot
- JS Lagas
- JS Wang
- JW Kim
- JW Massarella
- JW Polli
- JW Polli
- JW Smit
- JY Chatton
- Jérôme Biollaz
- K Bleasby
- K Dilger
- K Engel
- K Engel
- K Erik Pedersen
- K Fujiwara
- K Hacker
- K Horie
- K Ichida
- K Iwata
- K Jones
- K Kato
- K Kato
- K Köck
- K Maeda
- K Maeda
- K Nakano
- K Naruhashi
- K Naruhashi
- K Ogasawara
- K Shiba
- K Shirakawa
- K Stoeckel
- K Suzuki
- K Tahara
- K Takara
- K Takara
- K Takara
- K Takara
- K Titier
- K Toyama
- K Ueda
- K Vishwanathan
- K Wang
- K Yano
- K Yasuda
- K Yusa
- K Zhong
- K-A Kim
- K-I Umehara
- K-M Jalava
- K-M Kaukonen
- K-Y Yam
- KA Lentz
- KA Youdim
- KB Goralski
- KC Cundy
- KE Parrish
- KE Pedersen
- KHP Moore
- KI Umehara
- KJ Ullrich
- KJ Ullrich
- KJ Ullrich
- KK Adkison
- KK Adkison
- KK Filipski
- KM Barnes
- KM Hillgren
- KM Mahar Doan
- KM Morrissey
- KM Stray
- KP Arun
- KS Lips
- KW Kolb
- KY Jung
- KY Jung
- KY Ohta
- KY Ohta
- KY Ohta
- L Ci
- L Di
- L Diao
- L Granero
- L Gschwind
- L Hong
- L Lecureux
- L Li
- L Liu
- L Ma
- L Ma
- L Payen
- L Payen
- L Profit
- L Tong
- L Wang
- L Wang
- L Wang
- L Ye
- LA Bauer
- LCJ Ellis
- LH Lash
- LHM Brake te
- LL Moltke von
- LL Yacovino
- LM Vermeer
- LS Yu
- LW Maines
- M Alebouyeh
- M Bebawy
- M Bexten
- M Cvetkovic
- M Garthy
- M Grube
- M Grube
- M Hasegawa
- M Hasegawa
- M Hasegawa
- M Hayer-Zillgen
- M Hiasa
- M Homeida
- M Horikawa
- M Hosoyamada
- M Huls
- M Kagedal
- M Kajiwara
- M Kajiwara
- M Kakumoto
- M Katoh
- M Katoh
- M Komuro
- M Li
- M Masuda
- M Minocha
- M Miyajima
- M Motojima
- M Muirhead
- M Mukherjee
- M Naesens
- M Nishimura
- M Nomura
- M Obermeier
- M Okabe
- M Okuda
- M Okuda
- M Opravil
- M Otsuka
- M Rius
- M Rodríguez-Ibáñez
- M Sala-Rabanal
- M Sasaki
- M Sato
- M Sato
- M Schmidt
- M Shimizu
- M Sugawara
- M Sugie
- M Takaai
- M Takano
- M Takeda
- M Takeda
- M Takeda
- M Takeda
- M Takeda
- M Takeda
- M Tsuda
- M Tsuda
- M Tsuda
- M Uhr
- M Uhr
- M Wadelius
- M Wang
- M Yamazaki
- M Yamazaki
- M Zheng
- MA Hedaya
- MA Nagle
- MA Welch
- MB Wittwer
- MD Donovan
- MD Donovan
- MD Perloff
- MD Perloff
- MD Troutman
- ME Ganapathy
- ME Ganapathy
- ME Ganapathy
- MF Fromm
- MF Fromm
- MJ Borgnia
- MJ Cutler
- MJ Dresser
- MJ Gnoth
- MJ Jin
- MJ Knauer
- MJ Reese
- MJ Reese
- MK Choi
- ML Becker
- ML Lucero
- ML Rizk
- ML Ruiz
- MM Cornwell
- MM Parvez
- MM Posada
- MR Muirhead
- MS Joy
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- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/08/2017
- Field of study
Transporters in proximal renal tubules contribute to the disposition of numerous drugs. Furthermore, the molecular mechanisms of tubular secretion have been progressively elucidated during the past decades. Organic anions tend to be secreted by the transport proteins OAT1, OAT3 and OATP4C1 on the basolateral side of tubular cells, and multidrug resistance protein (MRP) 2, MRP4, OATP1A2 and breast cancer resistance protein (BCRP) on the apical side. Organic cations are secreted by organic cation transporter (OCT) 2 on the basolateral side, and multidrug and toxic compound extrusion (MATE) proteins MATE1, MATE2/2-K, P-glycoprotein, organic cation and carnitine transporter (OCTN) 1 and OCTN2 on the apical side. Significant drug-drug interactions (DDIs) may affect any of these transporters, altering the clearance and, consequently, the efficacy and/or toxicity of substrate drugs. Interactions at the level of basolateral transporters typically decrease the clearance of the victim drug, causing higher systemic exposure. Interactions at the apical level can also lower drug clearance, but may be associated with higher renal toxicity, due to intracellular accumulation. Whereas the importance of glomerular filtration in drug disposition is largely appreciated among clinicians, DDIs involving renal transporters are less well recognized. This review summarizes current knowledge on the roles, quantitative importance and clinical relevance of these transporters in drug therapy. It proposes an approach based on substrate-inhibitor associations for predicting potential tubular-based DDIs and preventing their adverse consequences. We provide a comprehensive list of known drug interactions with renally-expressed transporters. While many of these interactions have limited clinical consequences, some involving high-risk drugs (e.g. methotrexate) definitely deserve the attention of prescribers
Renal Drug Transporters and Drug Interactions
- Author
- A Allen
- A Amphoux
- A Aslamkhan
- A Azzariti
- A Brandoni
- A Collett
- A Courtois
- A Crowe
- A Dahan
- A Dahan
- A Dahan
- A Dahlin
- A D’Emanuele
- A Enomoto
- A Enomoto
- A Futatsugi
- A Gaowa
- A Geick
- A Gupta
- A Hamada
- A Horie
- A Kamizono
- A Kawase
- A Koenen
- A Komatsuda
- A Kunze
- A Lazar
- A Lespine
- A Maeda
- A Maeda
- A McCormick
- A Milane
- A Mulgaonkar
- A Nakayama
- A Nies
- A Oka
- A Ose
- A Owen
- A Pawarode
- A Poirier
- A Rizwan
- A Servais
- A Soldner
- A Somogyi
- A Somogyi
- A Somogyi
- A Somogyi
- A Vildhede
- A Yamada
- A Yamada
- A Yonezawa
- A Yonezawa
- AA El-Sheikh
- AA Ela El
- AA Somogyi
- AA Somogyi
- AAK El-Sheikh
- AAK El-Sheikh
- AAK El-Sheikh
- AAK El-Sheikh
- AB Shapiro
- AE Busch
- AE Herwaarden van
- AE Kim
- AG Hotchkiss
- AH Schinkel
- AH Schinkel
- AH Schinkel
- AJ Dudley
- AJ Dudley
- AJ Scheen
- AL Dzierlenga
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- AM Hecken van
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- Anton Ivanyuk
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- N Glube
- N Inotsume
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- N Ishiguro
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- N Lloberas
- N Mizuno
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- N Shiraki
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- R Maitra
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- R Nakagomi-Hagihara
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