7 research outputs found
Synthetic lethal therapies for cancer: what's next after PARP inhibitors?
- Author
- A Ashworth
- A Dixit
- A Drean
- A Drean
- A Fujimoto
- A Goga
- A Prahallad
- A Tsherniak
- A Tutt
- AA Chakraborty
- AC Palmer
- AH Tong
- AH Tong
- AJ Aguirre
- AJ Gill
- Alan Ashworth
- B Li
- B Vogelstein
- BG Bitler
- BG Bitler
- BG Wilson
- BG Wilson
- BH Lok
- C Bertoli
- C Bridges
- C Frezza
- C Kadoch
- C Scholl
- Cancer Genome Atlas Research Network
- Christopher J. Lord
- CJ Lord
- CJ Lord
- CJ Lord
- CJ Ryan
- CM Koh
- CT Williamson
- CV Dang
- D Horiuchi
- D Nittner
- D Robinson
- D Zhao
- DA Barbie
- DA Chan
- DF DeLair
- E Grabocka
- E Gurpinar
- EM Stein
- EM Swisher
- EM Tacconi
- EP Samartzis
- ER McDonald III
- F Dietlein
- FL Muller
- FL Muller
- G Karpel-Massler
- G Poortinga
- G Rancati
- GM Gordon
- GR Hoffman
- GV Kryukov
- H Farmer
- H Liu
- H Rokutan
- H Xiao
- HC Reinhardt
- HE Bryant
- I Murfuni
- J Campbell
- J Downward
- J Luo
- J Mora
- J Shen
- J Tischler
- JA Ledermann
- JD Kessler
- JI Garaycoechea
- JM Ostrem
- JM Thompson
- JR Whitfield
- JS Brown
- K Buchkovich
- K Cramer-Morales
- K Marjon
- KC Helming
- KC Wiegand
- KH Kim
- KJ Mavrakis
- KJ McManus
- KN Mohni
- L Dang
- LH Hartwell
- M Kampmann
- M Kwok
- M Robson
- M Steckel
- M Toyoshima
- MR Mirza
- MS Kumar
- MT Pickering
- MW Audeh
- N McCabe
- N Takebe
- N Waddell
- O Gilad
- P Dey
- PA Mateos-Gomez
- PC Fong
- PL Chen
- PL Sulkowski
- R Camarda
- R Ceccaldi
- R Marcotte
- RE Miller
- RJ Molenaar
- RM Meyers
- S Campaner
- S Cardaci
- S Chantalat
- S Frohling
- S Turcotte
- SM Chan
- SR Hengel
- SX Pfister
- SX Pfister
- T Dobzhansky
- T Januario
- T Nobori
- T Oike
- T Orvis
- T Raedt De
- T Wang
- T Zhang
- TR Brummelkamp
- WG Kaelin Jr.
- X Lai
- X Wang
- Y Wang
- Z Feng
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/09/2018
- Field of study
The genetic concept of synthetic lethality has now been validated clinically through the demonstrated efficacy of poly(ADP-ribose) polymerase (PARP) inhibitors for the treatment of cancers in individuals with germline loss-of-function mutations in either BRCA1 or BRCA2. Three different PARP inhibitors have now been approved for the treatment of patients with BRCA-mutant ovarian cancer and one for those with BRCA-mutant breast cancer; these agents have also shown promising results in patients with BRCA-mutant prostate cancer. Here, we describe a number of other synthetic lethal interactions that have been discovered in cancer. We discuss some of the underlying principles that might increase the likelihood of clinical efficacy and how new computational and experimental approaches are now facilitating the discovery and validation of synthetic lethal interactions. Finally, we make suggestions on possible future directions and challenges facing researchers in this field
Kinetic Investigation and Anticoagulant Activity of Amide Analogues of Isoform 2 and 3 of Antistasin
- Author
- A Atanasov
- A Rupin
- AV Basanova
- AZ Fernandez
- CK Marlowe
- CT Dunwiddie
- D Danalev
- D Danalev
- D Danalev
- D Danalev
- D Danalev
- D Longrois
- Dancho Danalev
- Dessislava Marinkova
- E Clyne
- F Faria
- F Markwardt
- Galina Obretenova
- GP Tuszynski
- GW Stone
- HJ Lee
- HK Caldwell
- Iren Tsibranska
- J Nienaber
- JA Ostrem
- KH Strube
- Konstantin Savov
- Lyubov Yotova
- M Kurzyna
- M Moser
- M Nisio Di
- M Smythe
- Raya Raykova
- S Alban
- S Bajusz
- S Iwanaga
- SS Mao
- X Zang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Non-monotonic dynamics and crosstalk in signaling pathways and their implications for pharmacology
- Author
- A Ramezanpour
- AF Fliri
- AL Hopkins
- AR Mashaghi
- BL Roth
- C Hadley
- CH Hansen
- CJ Marshall
- CT Keith
- DG Margineanu
- DR Hyduke
- EJ Calabrese
- F Shima
- FS vom Saal
- I Lokody
- J Inglese
- J Spiegel
- JA Papin
- JM Ostrem
- L Li
- L Yan
- M Kollmann
- M Natarajan
- MA Schwartz
- ML Skoge
- N Malo
- N Yin
- OJ Miller
- P Csermely
- P Kuzmic
- RCR Wootton
- S Frantz
- S Ishihara
- S Kaplan
- SK Mencher
- T Hampton
- TDC Fraser
- U Alon
- W de Ronde
- W de Ronde
- WC Hwang
- Y Tu
- YB Wetherill
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Targeting LKB1 in cancer – exposing and exploiting vulnerabilities
- Author
- A Hemminki
- A Hemminki
- A Osoegawa
- A Suzuki
- A Suzuki
- A Woods
- A Woods
- A Ylikorkala
- AA Ahmed
- AK Rines
- AM Strohecker
- B Apsel
- B Gan
- B Xiao
- B Zheng
- BJ Druker
- BY Shorning
- C Algire
- C Emmanuel
- C Nardella
- C Wei
- C Xu
- CJ Currie
- CM Contreras
- CM Fillmore
- CT Pineda
- D B Shackelford
- D Nakada
- DB Shackelford
- DB Shackelford
- DB Shackelford
- DB Shackelford
- DB Shackelford
- DB Shackelford
- DF Egan
- DG Hardie
- DG Hardie
- DJ Rossi
- DM Gwinn
- DR Gandara
- ED Segal
- ER Kline
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- F Martin-Belmonte
- FL Fimognari
- FX McCormack
- G Kusakai
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- H Alachkar
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- H Chen
- H Cheng
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- H Wang
- HS Kim
- J Barretina
- J Carretero
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- JD Lalau
- JJ Bissler
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- M Sanchez-Cespedes
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- MB Schneider
- MC Liang
- MD Wilkerson
- ME Feldman
- MM Mihaylova
- MN Corradetti
- MR Owen
- MR Pickard
- N Bardeesy
- N Janus
- OB Crofford
- P Fernandez
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- RJ Shaw
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- S Gurumurthy
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- SA Hawley
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- V Gorboulev
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- W Damsky
- W Liu
- WC Zhang
- WX Qi
- X Fu
- X Li
- XY Fu
- Y Gao
- Y Liu
- Y Nakada
- Z Chen
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Synthetic lethal therapies for cancer: what’s next after PARP inhibitors?
- Author
- A Ashworth
- A Dixit
- A Drean
- A Drean
- A Fujimoto
- A Goga
- A Prahallad
- A Tsherniak
- A Tutt
- AA Chakraborty
- AC Palmer
- AH Tong
- AH Tong
- AJ Aguirre
- AJ Gill
- Alan Ashworth
- B Li
- B Vogelstein
- BG Bitler
- BG Bitler
- BG Wilson
- BG Wilson
- BH Lok
- C Bertoli
- C Bridges
- C Frezza
- C Kadoch
- C Scholl
- Cancer Genome Atlas Research Network
- Christopher J. Lord
- CJ Lord
- CJ Lord
- CJ Lord
- CJ Ryan
- CM Koh
- CT Williamson
- CV Dang
- D Horiuchi
- D Nittner
- D Robinson
- D Zhao
- DA Barbie
- DA Chan
- DF DeLair
- E Grabocka
- E Gurpinar
- EM Stein
- EM Swisher
- EM Tacconi
- EP Samartzis
- ER McDonald III
- F Dietlein
- FL Muller
- FL Muller
- G Karpel-Massler
- G Poortinga
- G Rancati
- GM Gordon
- GR Hoffman
- GV Kryukov
- H Farmer
- H Liu
- H Rokutan
- H Xiao
- HC Reinhardt
- HE Bryant
- I Murfuni
- J Campbell
- J Downward
- J Luo
- J Mora
- J Shen
- J Tischler
- JA Ledermann
- JD Kessler
- JI Garaycoechea
- JM Ostrem
- JM Thompson
- JR Whitfield
- JS Brown
- K Buchkovich
- K Cramer-Morales
- K Marjon
- KC Helming
- KC Wiegand
- KH Kim
- KJ Mavrakis
- KJ McManus
- KN Mohni
- L Dang
- LH Hartwell
- M Kampmann
- M Kwok
- M Robson
- M Steckel
- M Toyoshima
- MR Mirza
- MS Kumar
- MT Pickering
- MW Audeh
- N McCabe
- N Takebe
- N Waddell
- O Gilad
- P Dey
- PA Mateos-Gomez
- PC Fong
- PL Chen
- PL Sulkowski
- R Camarda
- R Ceccaldi
- R Marcotte
- RE Miller
- RJ Molenaar
- RM Meyers
- S Campaner
- S Cardaci
- S Chantalat
- S Frohling
- S Turcotte
- SM Chan
- SR Hengel
- SX Pfister
- SX Pfister
- T Dobzhansky
- T Januario
- T Nobori
- T Oike
- T Orvis
- T Raedt De
- T Wang
- T Zhang
- TR Brummelkamp
- WG Kaelin Jr.
- X Lai
- X Wang
- Y Wang
- Z Feng
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Occupational Hazards in Modern Dentistry
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- Adebola FA Owotade FJ.
- Akesson I Hansson GA, balogh I, Moritz U.
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- 'Jaypee Brothers Medical Publishing'
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Small molecules in targeted cancer therapy: advances, challenges, and future perspectives
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- A Akinleye
- A Alshangiti
- A Ashkenazi
- A Awada
- A Beck
- A Chaturvedi
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- A Dlugosz
- A Drilon
- A Drilon
- A Drilon
- A Drilon
- A Drilon
- A Elshoury
- A Galanis
- A Gu
- A Hauschild
- A Hochhaus
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- A Italiano
- A James
- A Khunger
- A Krzyzosiak
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- A Morabito
- A Nakagawara
- A Noy
- A Patnaik
- A Quintas-Cardama
- A Redaelli
- A Sekulic
- A Spencer
- A Stathis
- A Suraweera
- A Tarakhovsky
- A Thomas
- A Vitkeviciene
- A Yokota
- A Yver
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- AC Hsieh
- AD Cox
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- AE Tron
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- T Ma
- T O’Hare
- T O’Hare
- T O’Hare
- T O’Hare
- T Sasaki
- T Yamaura
- TB Miranda
- TH Marsilje
- TJ Lynch
- TK Choueiri
- TM Herndon
- TM Sielecki
- TPS Perera
- TT Batchelor
- U Asghar
- V Cepero
- V Chau
- V Gibaja
- V Kasireddy
- V Santini
- V Serra
- V Strand
- VA Guerra
- VA Miller
- W Qi
- W Risau
- W Waggott
- WH Lin
- WH Yang
- WN Khan
- WS Huang
- WS Kim
- WTA van der Graaf
- X Chen
- X Dong
- X Huang
- X Jiang
- X Kong
- X Lin
- X Liu
- X Liu
- X Lu
- X Sheng
- X Wang
- X Wu
- X Xu
- X Zheng
- Y Bai
- Y Cheng
- Y Guo
- Y He
- Y Jia
- Y Li
- Y Ma
- Y Piao
- Y Pylayeva-Gupta
- Y Shi
- Y Wang
- Y Wang
- Y Xu
- Y Zhang
- Y Zhang
- Y Zhang
- Y Zhang
- Y Zhu
- YB Khotskaya
- YJ Choi
- YL Wu
- YM Abaza
- YS Cho
- YT Lee
- YX Yang
- YY Syed
- YY Syed
- YY Syed
- Z Chen
- Z Chen
- Z Dai
- Z Li
- Z Ma
- Z Zhang
- Z Zhou
- ZW Cai
- ZX Cao
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study