Declamatio de pueris ad virtutem ad literas liberaliter instituendis idque protinus a nativitate [499. C7-504. A13.] Desiderius Erasmus

原著 : エラスムス　翻訳 : 中城

Desiderius Erasmus, Concio de puero Jesu (599.C 1.-604.A 9)

原著 : エラスムス　翻訳 : 中城

Cancio de puero Jesu (604.A 10.-610.A 9) Desiderius Erasmus

原著 : エラスムス　翻訳 : 中城

[Translation] Declamatio de pueris ad virtutem ac literas liberaliter instituendis idque protinus a nativitate [504. A14. -509. F2.] Desiderius Erasmus

原著 : エラスムス　翻訳 : 中城

Nucleophilic substitution reaction of 1-methoxyindole-3-carbaldehyde

1-Methoxyindole-3-carbaldehyde is proved to be a versatile electrophile and reacts regioselectively at the 2-position with various types of nucleophiles providing 2-substituted indole-3-carbaldehydes. © 2012 The Japan Institute of Heterocyclic Chemistry

A novel synthetic method of pyrrolo[2,3-b]indoles and its application to the synthesis of (±)-debromoflustramine B1

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学部1-Methoxy-3-(2-nitrovinyl)indole (4) functions as an electrophile and reacted with various nucleophiles regioselectively at the 2-position. Employing allyl alkoxides as nucleophiles, a novel synthetic method of pyrrolo[2,3-b]indoles has been elaborated. Utilizing the method, the synthesis of (±)-debromofIustramine B (10b) was achieved

Nucleophilic substitution reaction of 3-acetyl-1-methoxyindole and its application for the synthesis of novel 2-substituted methyl 2,3-dihydro-1- methyl-3-oxo-5H-pyrido-[4,3-b]indole-4-carboxylates

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学部A simple synthetic route was established for 3-acetyl-1-methoxyindole, which was found to undergo nucleophilic substitution reactions selectively at the 2-position. Applying the reaction, novel 2-substituted methyl 2,3- dihydro-1-methyl-3-oxo-5H-pyrido[4,3-b]indole-4-carboxylates were prepared