The first and simple synthesis of indole alkaloid, bipolaramide

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学部The first and simple total synthesis of bipolaramide was achieved in 31 % overall yield from (2S)-2,3-dihydroindole-2-carboxylic acid in three (or two) steps. Derivatives of bipolaramide having halogen, alkenyl, nitro, or azido substitueras were also prepared

Rhe first total syntheses of 9-methoxycarbazole-3-carboxaldehyde and methoxybrassinin1 (the chemistry of 1-methoxyindole)

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学

A new and simple synthesis of 1-hydroxyindole derivatives

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学

A simple synthesis of 7-substituted 1-acetyl-2,3-dihydroindoles

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学

A simple synthesis of a phytoalexin, methoxybrassinin

金沢大学大学院自然科学研究科生理活性物質科学金沢大学薬学