6 research outputs found
From Pan-Reactive KV7 Channel Opener to Subtype Selective Opener/Inhibitor by Addition of a Methyl Group
- Author
- A Schenzer
- AR Mackie
- Bernard Attali
- BH Bentzen
- C Biervert
- C Charlier
- Christoffer Bundgaard
- DA Brown
- F Miceli
- F Sotty
- G Blackburn-Munro
- GE Duncan
- Henrik Sindal Jensen
- HH Hansen
- HH Hansen
- HH Hansen
- HS Wang
- IA Greenwood
- JA Lieberman
- Jan Kehler
- JP Redrobe
- K Padilla
- KT Mueser
- L Cook
- Mario Rottländer
- MPG Korsgaard
- NA Singh
- Nicole Schmitt
- P Seeman
- PS Chadha
- PS Chadha
- Q Xiong
- R Risgaard
- R Søgaard
- S Khanamiri
- Sigrid Marie Blom
- SM Blom
- SM Blom
- SP Aiken
- TJ Jentsch
- TV Wuttke
- VJ Nickolson
- VK Gribkoff
- W Lange
- YJ Wu
- YJ Wu
- YJ Wu
- Z Talebizadeh
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- Field of study
Ion channel pharmacology
- Author
- A Luca De
- A Peretz
- A Szewczyk
- AD Wei
- B Hille
- C Heatwole
- C Munoz-Caro
- CA Vedeler
- CH Wallace
- CJ Weisz
- CR Bezzina
- D Conte Camerino
- D Tricarico
- D Tricarico
- D Tricarico
- D Tricarico
- D Tricarico
- Diana Conte Camerino
- Domenico Tricarico
- E Legroux-Crespel
- E Michelakis
- F Lehmann-Horn
- F Lesage
- FM Ashcroft
- G Meola
- GA Gutman
- GK Wang
- GO Skeie
- H Eguchi
- HC Hemmings
- IW Glaaser
- J Cuppoletti
- J Lai
- J Trip
- J-F Desaphy
- J-F Desaphy
- Jean-François Desaphy
- JF Desaphy
- JF Desaphy
- JJ Clare
- JJ Ligtenberg
- K Weckbecker
- L Wu
- M Cascio
- M Pusch
- MA Nassar
- MA Rogawski
- MJ Coghlan
- MP Takahashi
- MPG Korsgaard
- N Lenkey
- NCL McNaughton
- NG Bowery
- PD Dodson
- PT Lucas
- R Mannhold
- S Ghatta
- SC Cannon
- SD Spacey
- SE Heron
- SG Waxman
- SG Waxman
- SK Tate
- T Leniger
- TJ Jentsch
- V Yarov-Yarovoy
- WA Catteral
- Y Kubo
- YA Ruetsch
- Publication venue
- 'Elsevier BV'
- Publication date
- 01/01/2007
- Field of study
Because ion channels are involved in many cellular
processes, drugs acting on ion channels have long been used for the treatment of many diseases, especially those affecting electrically
excitable tissues. The present review discusses the pharmacology of voltage-gated and neurotransmitter-gated ion
channels involved in neurologic diseases, with emphasis on neurologic channelopathies. With the discovery of ion channelopathies,
the therapeutic value of many basic drugs targeting
ion channels has been confirmed. The understanding of the genotype–phenotype relationship has highlighted possible action mechanisms of other empirically used drugs. Moreover, other ion channels have been pinpointed as potential new drug targets. With regards to therapy of channelopathies, experimental
investigations of the intimate drug– channel interactions have demonstrated that channel mutations can either increase
or decrease affinity for the drug, modifying its potential
therapeutic effect. Together with the discovery of channel gene polymorphisms that may affect drug pharmacodynamics, these findings highlight the need for pharmacogenetic research to allow identification of drugs with more specific effects on
channel isoforms or mutants, to increase efficacy and reduce side effects. With a greater understanding of channel genetics, structure, and function, together with the identification of novel
primary and secondary channelopathies, the number of ion channel drugs for neurologic channelopathies will increase substantially
Recent advances in neurokinin-3 receptor antagonists
- Author
- BROCCARDO M
- BUELL G
- CANNING BJ
- CELLIER E
- CHEN MH CHUNG F-Z
- COUDORE-CIVIALE M-A COURTEIX C
- COUTURE R
- DAOUI S
- DONALDSON LF
- EMONDS-ALT X
- GAO Z
- GIARDINA GAM ARTICO M, CAVAGNERA S et al.
- GIARDINA GAM GRUGNI M, RIGOLIO R, VASSALLO M, ERHARD K, FARINA C
- GIARDINA GAM RAVEGLIA LF
- GIARDINA GAM RAVEGLIA LF, GRUGNI M
- GIARDINA GAM SARAU HM, FARINA C
- GIARDINA GAM SARAU HM, FARINA C et al.
- Giuseppe AM Giardina
- GOLDHILL J
- GUEUDET C
- HARRISON T KORSGAARD MPG
- JULIA V
- LINDEN DR
- LINDEN DR JIA Y-P
- Luca F Raveglia
- MANN PT
- Mario Grugni
- MEDHURST AD
- MEDHURST AD
- MILEUSNIC D
- MILEUSNIC D
- MYERS AC
- NALIVAIKO E
- OYAMADA H
- PIRRUNG MC
- RAVEGLIA LF
- REGOLI D
- RIBEIRO SJ
- RIBEIRO SJ
- SCHMID G
- SEYBOLD VS
- SNIDER RM CONSTANTINE SJW
- VON SPRECHER A
- YOUNG RC
- YUAN Y-D COUTURE
- ZERARI F
- Publication venue
- 'Informa Healthcare'
- Publication date
- Field of study
Ion channel pharmacology
- Author
- A Luca De
- A Peretz
- A Szewczyk
- AD Wei
- B Hille
- C Heatwole
- C Munoz-Caro
- CA Vedeler
- CH Wallace
- CJ Weisz
- CR Bezzina
- D Conte Camerino
- D Tricarico
- D Tricarico
- D Tricarico
- D Tricarico
- D Tricarico
- Diana Conte Camerino
- Domenico Tricarico
- E Legroux-Crespel
- E Michelakis
- F Lehmann-Horn
- F Lesage
- FM Ashcroft
- G Meola
- GA Gutman
- GK Wang
- GO Skeie
- H Eguchi
- HC Hemmings
- IW Glaaser
- J Cuppoletti
- J Lai
- J Trip
- J-F Desaphy
- J-F Desaphy
- Jean-François Desaphy
- JF Desaphy
- JF Desaphy
- JJ Clare
- JJ Ligtenberg
- K Weckbecker
- L Wu
- M Cascio
- M Pusch
- MA Nassar
- MA Rogawski
- MJ Coghlan
- MP Takahashi
- MPG Korsgaard
- N Lenkey
- NCL McNaughton
- NG Bowery
- PD Dodson
- PT Lucas
- R Mannhold
- S Ghatta
- SC Cannon
- SD Spacey
- SE Heron
- SG Waxman
- SG Waxman
- SK Tate
- T Leniger
- TJ Jentsch
- V Yarov-Yarovoy
- WA Catteral
- Y Kubo
- YA Ruetsch
- Publication venue
- 'Elsevier BV'
- Publication date
- Field of study
Tests for Anxiolytic Activity
- Author
- A AgĂĽero
- A AgĂĽero
- A Bachy
- A Bane
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- A Bilkei-Gorzo
- A Bilkei-Gorzo
- A Bourson
- A Butler
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- A Chagraoui
- A Clarke
- A Contarino
- A Czyrak
- A Célérier
- A Dumuis
- A Fernandez-Guasti
- A Fischer
- A Fleischmann
- A Fletcher
- A Fletcher
- A Frazer
- A Guidotti
- A Hausmann
- A Heest van
- A Holmes
- A Korte
- A Lecci
- A Lecci
- A Lenègre
- A McGregor
- A Newman-Tancredi
- A Newman-Tancredi
- A Pazos
- A Scriabine
- A Shekar
- A Siegel
- A Siegel
- A Siegel
- A Siegel
- A Siegel
- A Wiersma
- A Woods
- AB Davidson
- AD Rudzik
- AH Lewin
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- BL Roth
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- Publication venue
- 'Springer Science and Business Media LLC'
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Tests for Anxiolytic Activity
- Author
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- Bormann J
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- Costall B Domeney AM, Gerrard PA, Kelley ME, Naylor RJ
- Costall B Domeney AM, Naylor RJ, Tyers MB
- Costall B Hendrie CA, Kelly ME, Naylor RJ
- Costall B Kelley ME, Naylor RJ, Onaivi ES
- Costall B Kelly ME, Onaivi ES, Naylor RJ
- Costall B Naylor RJ, Tyers MB
- Costall B Naylor RT, Tyers MB
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