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5 research outputs found
Novel 2′,6′-Dimethyl-l-Tyrosine-Containing Pyrazinone Opioid Mimetic μ-Agonists with Potent Antinociceptive Activity in Mice
Author
Akihiro Ambo
Kimitaka Shiotani
+6Â more
Lawrence H. Lazarus
Sharon D. Bryant
Yoshio Okada
Yuko Tsuda
Yunden Jinsmaa
Yusuke Sasaki
Publication venue
'American Society for Pharmacology & Experimental Therapeutics (ASPET)'
Publication date
Field of study
No full text
Crossref
Bifunctional [2,6-Dimethyl-l-tyrosine1]endomorphin-2 Analogues Substituted at Position 3 with Alkylated Phenylalanine Derivatives Yield Potent Mixed m-Agonist/d-Antagonist and Dual m-Agonist/d-Agonist Opioid Ligands
Author
Akihiro Ambo
Anna Miyazaki
+9Â more
Ewa Marczak
Kimitaka Shiotani
Lawrence H. Lazarus
Sharon D. Bryant
Tingyou Li
Yoshio Okada
Yuko Tsuda
Yunden Jinsmaa
Yusuke Sasaki
Publication venue
'American Chemical Society (ACS)'
Publication date
Field of study
No full text
Crossref
Application of liquid chromatography–tandem mass spectrometry for the determination of opioidmimetics in the brain dialysates from rats treated with opioidmimetics intraperitoneally
Author
Almquist
Anna Miyazaki
+24Â more
Desiderio
Desiderio
Dygos
Fumiyo Kasuya
Hermanson
Kazuo Igarashi
Kimata
Kimitaka Shiotani
Koichiro Hotta
Li Tingyou
Lundin
Nakahara
Nimura
Oda
Okada
Samii
Shoji Fukushima
Smith
Yang
Yokohama
Yoshio Okada
Youji Kitamura
Yuki Murabayashi
Yuko Tsuda
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Design and synthesis of opioidmimetics containing 2′,6′-dimethyl-l-tyrosine and a pyrazinone-ring platform
Author
Akihiro Ambo
Anna Miyazaki
+37Â more
Broccardo
Cox
Dygos
Erspamer
Erspamer
Fujita
Goldstein
Hruby
Hughes
Igarashi
Jinsmaa
Jinsmaa
Kimitaka Shiotani
Koda
Kreil
Lawrence H. Lazarus
Lazarus
Lazarus
Li
Ling
Melchiorri
Meunier
Montecucchi
Montecucchi
Okada
Okada
Okada
Salvadori
Sasaki
Sharon D. Bryant
Stromberg
Tingyou Li
Toshio Yokoi
Yoshio Okada
Yuko Tsuda
Yusuke Sasaki
Zadina
Publication venue
'Elsevier BV'
Publication date
Field of study
No full text
Crossref
Studies on the Mechanism of 1,2-Dihydropyrazin-2-one Ring Formation from Dipeptidyl Chloromethyl Ketone and Its Chemical Properties: Immediate Deamination during Catalytic Hydrogenation
Author
Almquist G. R. Kadambi R. S., Yasu
Anna Miyazaki
+23Â more
Colm ó
Dahn H. Garbarino J. A., O'Mu
Haas H. J.
House H. O.
Jinsmaa Y. Okada Y., Tsuda Y., Shi
Kimitaka Shiotani
Lawrence H. Lazarus
Mitui S. Sugi Y.
Okada Y. Tsukatani M., Taguchi H.,
Powers J. C. Tuhy P. M.
Schnabel E.
Sharefkin J. G. Zaltzman H.
Sharon D. Bryant
TAGUCHI H
Tingyou Li
Toshio Yokoi
Velluz L. Amiard G., Heyness R.
Velluz L. Anatol J., Amiard G.
Yagupolskii L. M. Maletina I. I.,
Yoshio Fujita
Yoshio Okada
Yuko Tsuda
Yutaka Fujisawa
Publication venue
'Pharmaceutical Society of Japan'
Publication date
01/01/2005
Field of study
No full text
Crossref