5 research outputs found
Siramesine triggers cell death through destabilisation of mitochondria, but not lysosomes
- Author
- A Grau
- AM Sadowska
- B Turk
- BA Spruce
- BJ Vilner
- BJ Vilner
- C Abate
- C Heading
- C Zeng
- C Zeng
- DJ Klionsky
- EE Kooijman
- EK Moltzen
- G Cassano
- G Droga-Mazovec
- J Perregaard
- J Spirkoski
- JM Walker
- JR Hornick
- JR Hornick
- KK Soby
- KW Crawford
- L Monassier
- M Nakanishi-Matsui
- MG Mamolo
- MJ Parry
- MS Ostenfeld
- MS Ostenfeld
- NA Colabufo
- R Quirion
- S Ivanova
- S Jonhede
- SB Hellewell
- SB Yang
- SD Banister
- SP Muench
- T Cirman
- U Repnik
- U Repnik
- VE Kagan
- VE Kagan
- WR Martin
- WT Bem
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Sigma-1 Agonist Binding in the Aging Rat Brain: a MicroPET Study with [11C]SA4503
- Author
- AL Gundlach
- Anna A. Rybczynska
- Anniek K. D. Visser
- Aren van Waarde
- C Julien-Dolbec
- Chantal Kwizera
- Csaba J. Nyakas
- DA Meyer
- DJ McCann
- DR Wallace
- E Hoekzema
- G Alonso
- GA Gudelsky
- GA Paleos
- H Goldman
- J Logan
- Jurgen W. A. Sijbesma
- JW Keyes
- K Ishiwata
- K Kawamura
- K Kawamura
- K Matsuno
- K Matsuno
- K Sahlholm
- Kiichi Ishiwata
- KK Soby
- LY Dong
- M Parent
- M Sakata
- M Suzuki
- M Takebayashi
- MD Majewska
- ML Leitner
- MP Morin-Surun
- Nisha K. Ramakrishnan
- NK Ramakrishnan
- NK Ramakrishnan
- NK Ramakrishnan
- P Bouchard
- P Schweinhardt
- Paul G. M. Luiten
- Philip H. Elsinga
- RM Ring
- RR Matsumoto
- Rudi A. J. O. Dierckx
- SL Patrick
- T Hayashi
- T Hayashi
- T Kobayashi
- T Maurice
- TA Mavlyutov
- Y Dong
- Y Kimura
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/2016
- Field of study
Purpose: Sigma-1 receptor ligands modulate the release of several neurotransmitters and intracellular calcium signaling. We examined the binding of a radiolabeled sigma-1 agonist in the aging rat brain with positron emission tomography (PET). Procedures: Time-dependent uptake of [11C]SA4503 was measured in the brain of young (1.5 to 3 months) and aged (18 to 32 months) Wistar Hannover rats, and tracer-kinetic models were fitted to this data, using metabolite-corrected plasma radioactivity as input function. Results: In aged animals, the injected probe was less rapidly metabolized and cleared. Logan graphical analysis and a 2-tissue compartment model (2-TCM) fit indicated changes of total distribution volume (VT) and binding potential (BPND) of the tracer. BPND was reduced particularly in the (hypo)thalamus, pons, and medulla. Conclusions: Some areas showed reductions of ligand binding with aging whereas binding in other areas (cortex) was not significantly affected. © 2015 The Author(s
The Role of Sigma Receptors in Depression
- Author
- Abellan MT Adell A, Honrubia MA, M
- Altamura CA Mauri MC, Ferrara A, M
- Andrade R Nicoll RA
- Bel N Artigas F
- BERGERON R
- Bergeron R Debonnel G
- BERMACK J E
- Bermack JE Debonnel G
- Blier P de Montigny C
- Blier P de Montigny C, Tardif D
- BOYER P-A
- Campbell BG Scherz MW, Keana JF, W
- CELADA P
- Chao MV
- Chaput Y de Montigny C, Blier P
- Couture S Debonnel G
- Debonnel G Bergeron R, de Montigny
- DeHaven-Hudkins D Fleissner L, For
- Delgado PL Charney DS, Price LH, A
- Delgado PL Moreno FA
- Duman R Heninger G, Nestler E
- FINKEL M S
- Gundlach AL Largent BL, Snyder SH
- Harvey BH
- HAYASHI T
- HUBER M T
- Jesberger JA Richardson JS
- KAMEI HIROYUKI
- Kia H Miquel MC, Brisorgueil MJ, D
- Kinsora JJ Jr Corbin A, Snider B,
- Lapin IP Oxenkrug GF
- LAUTERBORN J C
- Maes M Meltzer HY
- Maes M Verkerk R, Vandoolaeghe E,
- MALBERG J E
- Martin WR Eades CG, Thompson JA, H
- Maurice T Phan V-L, Su T-P
- Maurice T Roman FJ, Privat A
- McCann DJ Weissman AD, Su TP
- Mei J Pan Y-X, Xiu J, King M, Chan
- Middlemiss DN et al
- NODA YUKIHIRO
- Nowak G Paul I, Popik P, Young A,
- Pande AC Geneve J, Scherrer B
- Paul AP Layer RT, Skolnick P, Nowa
- PEJCHAL T
- Pepe GJ Rothchild I
- Pfleiderer B Michael N, Erfruth A,
- Quirion R Chichportiche R, Contrer
- Robichaud M Beauchemin V, Lavoie N
- Sanacora G Rothman DL, Mason G, Kr
- Sanchez C Papp M
- Schwarz S Pohl P, Zhou GZ
- SHELINE Y I
- SHIRAYAMA Y
- Skuza G Rogoz Z
- Soby KK Meier F, Mikkelsen JD
- Soriani O Le Foll F, Galas L, Roma
- Steinfels GF Alberici GP, Tam SW,
- TADA K
- Takebayashi M Hayashi T, Su TP
- Tsao LI Su TP
- URANI A
- Vilner BJ John CS, Bowen WD
- Wilke R Brettel M, Prince HM, Wolf
- Yamada S Uwahodo Y, Tottori K, Kik
- Young LT Bakish D, Beaulieu S
- Publication venue
- 'Japanese Pharmacological Society'
- Publication date
- 01/01/2005
- Field of study
Pterocarpans: interesting natural products with antifungal activity and other biological properties
- Author
- A Aragao Craveiro
- A Arnone
- A Haznagy
- A Rosa
- A Schoening
- A Subarnas
- A Ueno
- A Vanangamudi
- A Yagi
- A Yenesew
- A Yenesew
- A Yenesew
- A Yenesew
- AA Ajees
- AE Nkengfack
- AE Nkengfack
- AE Nkengfack
- AE Nkengfack
- AE Nkengfack
- AF Barrero
- AF Barrero
- AF Magalhaes
- AJ Brink
- AJ Brink
- AJ Demuner
- AJM Da Silva
- AK Jain
- AK Machocho
- AL Piccinelli
- AO Latunde-Dada
- AW Lenssen
- BCB Bezuidenhoudt
- BM Bandara
- BMR Bandara
- BR Baggett
- C Costa dos Santos
- C DeMartinis
- C Edwards
- C Selvam
- C Song
- C Triangali
- CC Joseph
- CCW Wanjala
- Cvd Brink
- CY Chuang
- D Durango
- D Gao
- DBF Juck
- DJ Robeson
- DK Datta
- DL Dornbos Jr.
- DL Gustine
- DL Gustine
- DMX Donnelly
- DMX Donnelly
- DR Perrin
- E Dagne
- E Dagne
- E Maekawa
- EE Shulâts
- EK Seo
- EV Rao
- F Cottiglia
- F Ferrari
- F Kiuchi
- F Manjary
- F Tian
- FA Macias
- FA Macias
- FD Dakora
- FJ Abreu Matos
- FR Van Heerden
- G Alagona
- G Alagona
- G Alagona
- G Belofsky
- G Belofsky
- G Dannhardt
- G Li
- G Palazzino
- GB Russell
- GCG Militao
- GCG Militao
- GF Spencer
- GI Seneviratne
- GJH Rall
- GJH Rall
- GL Da Silva
- H Bai
- H Duddeck
- H Kessmann
- H Matsuda
- H Orth
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Tanaka
- H Telikepalli
- H Yamamoto
- HB Xiao
- HD Van Etten
- HD Van Etten
- HH Dietrichs
- HJ Jung
- HM Sirat
- HMG Al-Hazimi
- HMG Al-Hazimi
- HMTB Herath
- I Kitagawa
- I Kitagawa
- IAM Cruickshank
- IAM Cruickshank
- IAM Cruickshank
- Ignacio RodrĂguez-GarcĂa
- J Armero
- JA Bailey
- JA Hargreaves
- JA Park
- JB Bredenberg
- JB Harborne
- JC Breytenbach
- JF Zeng
- JF Zeng
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JL Ingham
- JM Kim
- JS Kim
- JS Yoon
- JT Cook
- K Kajiyama
- K Kurosawa
- K Kurosawa
- K Ma
- K Nakamura
- KGR Pachler
- KH Shaker
- KK Atindehou
- KK Dorr
- KK Purushothaman
- L Alvarez
- L Pistelli
- L Pistelli
- L Van Puyvelde
- LA Mitscher
- LA Mitscher
- LA Mitscher
- LA Rabelo
- LC Chang
- Leticia Jiménez-Gonzålez
- LJ Wu
- Lq Hai
- LZ Lin
- M Arisawa
- M Brink
- M Chacha
- M Daniel
- M Iinuma
- M Iinuma
- M Iinuma
- M Iinuma
- M Iinuma
- M Iinuma
- M Iinuma
- M Iinuma
- M Iinuma
- M Komatsu
- M Komatsu
- M Mizuno
- M Mizuno
- M Mizuno
- M Morimoto
- M Nakagawa
- M Ohyama
- M Sato
- Manuel Muñoz-Dorado
- MH Hwang
- Miriam Ălvarez-Corral
- MJ OâNeill
- MJ OâNeill
- MM Salem
- MR Parthasarathy
- MS Abdel-Kader
- MS Abdel-Kader
- MSR Murthy
- N Matsuura
- N Mukherjee
- NT Keen
- NT Keen
- NW Preston
- OR Omobuwajo
- P Baruah
- P Erasto
- P Khaomek
- P Lebreton
- P Maximo
- P Maximo
- P Maximo
- P Maximo
- PC Stevenson
- PC Stevenson
- PC Stevenson
- PD Fraishtat
- PD Fraishtat
- PK Tarus
- PL Sawhney
- PM Dewick
- R Alencar
- R Braz Filho
- R Braz Filho
- R Braz Filho
- R Chanphen
- R Cook
- R Reyes-Chilpa
- R Reyes-Chilpa
- R Reyes-Chilpa
- R Roy
- R Sanduja
- R Vogelsang
- RM Letcher
- RW Miller
- S Awale
- S Koysomboon
- S Nagumo
- S Shibata
- S Soby
- S Tahara
- S Yahara
- SA Adesanya
- SA Fedoreyev
- SC Bhrara
- SC Chan
- SF Wang
- SG Pueppke
- SG Pueppke
- SK Chaudhuri
- SS Gnanamanickam
- SW Banks
- SY Ryu
- T Fukai
- T Fukai
- T Fukai
- T Fukai
- T Furuya
- T Kinoshita
- T Kinoshita
- T Konoshima
- T Maurich
- T Miyase
- T Miyase
- T Tanaka
- T Tanaka
- T Uchiyama
- TA Engler
- TA Engler
- TBH McMurry
- TH Kang
- TL Meragelman
- U Khera
- UV Babu
- VH Deshpande
- VNT Silva
- VS Batyuk
- VS Kamat
- VU Ahmad
- W Friedrichsen
- W Li
- W Li
- W Lwande
- W Mahabusarakam
- W Schaefer
- WB Mors
- WL Lo
- WL Lo
- XA Dominguez
- Y Deng
- Y Fujise
- Y Goda
- Y Goda
- Y Hayashi
- Y Kan
- Y Liu
- Y Obara
- Y Peleg
- Y Sakurai
- Y Shirataki
- Y Shirataki
- Y Shirataki
- Y Shirataki
- Y Wang
- Y Zhao
- YL Lin
- YN Shukla
- YS Kwon
- YS Kwon
- Z Jia
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Sigma receptors [ Ï
- Author
- Aanonsen L
- Aas P
- Abate C
- Abate C
- Abe K
- Abe T
- Abel T
- Abram S
- Aghajanian G
- Aizenman E
- Ajmo C
- Akunne H
- Al-Saif A
- Allahtavakoli M
- Allen D
- Altar C
- Amer M
- Anderson T
- Andrade R
- Angulo J
- Antonini V
- Antonini V
- Arnold J
- Arriza J
- Artola A
- Asztely F
- Awapara J
- Aydar E
- Aydar E
- Bai L
- Banister S
- Barb C
- Barbour B
- Barbour B
- Barnard E
- Barrot M
- Basile A
- Battaglia F
- Baulieu E
- Baur R
- Beart P
- Beck S
- Bel N
- Belanoff J
- Bem W
- Bergeron R
- Bergeron R
- Bergeron R
- Bergeron R
- Bergeron R
- Bermack J
- Bermack J
- Bermack J
- Bermack J
- Bertrand G
- Bertrand G
- Bettler B
- Bettler B
- Betz H
- Bhangu P
- Bhardwaj A
- Bhuiyan M
- Bhuiyan M
- Bhutada P
- Bitran D
- Blaylock R
- Blaylock R
- Blier P
- Blier P
- Blier P
- Blier P
- Bode B
- Boehme K
- Boldyrev A
- Bonnet K
- Bonomo V
- Boos R
- Booth R
- Borden L
- Borison R
- Bormann J
- Borowicz K
- Bouchard P
- Boulter J
- Bouvier M
- Bowen W
- Bowen W
- Bowen W
- Brammer M
- Brandes L
- Brent P
- Brent P
- Brent P
- Brew H
- Brimson J
- Brosnan J
- Brot M
- Brugmann WB
- Bruni J
- Bujalska M
- Bukusoglu C
- Burns G
- Burt D
- Butcher S
- Calabrese E
- Calabrese E
- Calabrese E
- Calabrese E
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- Calabrese E
- Callachan H
- Campbell B
- Cantiello H
- Carayon P
- Carlton S
- Carpenter C
- Carr D
- Caruso C
- Cassano G
- Cassano G
- Castellano C
- Castelli M
- Caveliers V
- Ceci A
- Celada P
- Celik I
- Cervo L
- Chaput Y
- Chaput Y
- Chaudhari N
- Chavez A
- Chen G
- Cheney D
- Chenu C
- Chien C
- Childers S
- Chiueh C
- Cho E
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- Cobos E
- Coccini T
- Coggeshall R
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- Collier T
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- Coutinho V
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- Cummings J
- Cunningham M
- Danysz W
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- Darnaudery M
- de Costa B
- Debonnel G
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- Delaunois A
- Dememes D
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- Dingledine R
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- Patel KD
- Patrick SL
- Paul IA
- Paul SM
- Pawlak G
- Peck V
- Peet NM
- Peeters M
- Pellegrino T
- Peng YG
- Pepe GJ
- Perl TM
- Perregaard J
- Phan VL
- Phan VL
- Phan VL
- Picaud S
- Picaud SA
- Pontecorvo MJ
- Prasad PD
- Prezzavento O
- Price MT
- Pritchett DB
- Pritchett DB
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- Puatanachokchai R
- Purcell WM
- Pyun K
- Quirion R
- Raab M
- Racchi M
- Ramamoorthy JD
- Rattan SI
- Rattan SI
- Renaudo A
- Renaudo A
- Renner R
- Rennie MJ
- Rhoades DJ
- Rison RA
- Roberts E
- Roberts E
- Roberts E
- Robichaud M
- Robson MJ
- Rockhold RW
- Rodvelt KR
- Roman F
- Romieu P
- Romieu P
- Romieu P
- Romieu P
- Ronsisvalle G
- Rosenberg PA
- Rosenmund C
- Rosin C
- Rothman RB
- Rousseaux CG
- Rousseaux CG
- Rupprecht R
- Ruscher K
- Ryan-Moro J
- Rybczynska AA
- Rybczynska AA
- Sabbatini R
- Sabino V
- Sacaan AI
- Saeki T
- Sagi N
- Said SI
- Said SI
- Sanchez C
- Sanchez C
- Sasa M
- Sasaki T
- Schaefer M
- Schatzberg AF
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- Schepmann D
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- Schofield PR
- Schultz K
- Schulz H
- Schulz H
- Schumacher M
- Schumacher M
- Schwab A
- Schwartz EA
- Schwarz S
- Seagard JL
- Seeburg PH
- Senda T
- Senda T
- Senkowska A
- Sershen H
- Seth P
- Shannon HE
- Sharp CD
- Shaw PJ
- Sheline YI
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- Shen MR
- Shioda N
- Shirayama Y
- Shirayama Y
- Shiue C
- Shu HJ
- Simony-Lafontaine J
- Simpson GM
- Singh P
- Skuza G
- Skuza G
- Skuza G
- Skuza G
- Skuza G
- Skuza G
- Smith KJ
- Soby KK
- Sommer B
- Soriani O
- Soriani O
- Soriani O
- Spillson AB
- Spirkoski J
- Stahl SM
- Starr MS
- Stefanski R
- Steinfels GF
- Stephanie F. Greene
- Stoffel-Wagner B
- Stone JM
- Stuhmer T
- Su TP
- Su TP
- Su TP
- Su TP
- Su TP
- Su TP
- Su TP
- Su TP
- Sugai N
- Sugimoto Y
- Supplisson S
- Sureda F
- Swegle JM
- Tabb JS
- Tachibana M
- Takahashi KA
- Takebayashi M
- Takebayashi M
- Takebayashi M
- Takebayashi M
- Tam SW
- Tan F
- Teichberg VI
- Terashvili M
- Thakur M
- Tokuyama S
- Tong Q
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- Toyohara J
- Truelove J
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- Truong DD
- Tryphonas L
- Tsai LH
- Tsai LH
- Tsai SY
- Tsai SY
- Tsao LI
- Tsumoto T
- Tucci M
- Tuerxun T
- Tung AS
- Uchida N
- Ujike H
- Ukai M
- Underhill SM
- Urani A
- Urani A
- Urani A
- Urani A
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- Vagnerova K
- Vallee M
- van Waarde A
- van Waarde A
- van Waarde A
- Varga EV
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- Vaupel DB
- Vignes M
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- Vilner BJ
- Vilner BJ
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- Vollrath JT
- Vu TH
- Vythilingam M
- Wakerley JB
- Walker JM
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- Walker R
- Wallace DR
- Walters RJ
- Wang B
- Wang H
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- Weaver CD
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- Whitlock BB
- Whittemore ER
- Widran J
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- Xu QX
- Xu W
- Yamada KA
- Yamada M
- Yamada S
- Yamaguchi I
- Yamamoto H
- Yamamoto H
- Yang JH
- Yang R
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- Yao X
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- Young GA
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- Yu W
- Yuzaki M
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- Zanardi R
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