6 research outputs found
Sulfur-Based Ylides in Transition-Metal-Catalysed Processes
- Author
- A Padwa
- A Padwa
- A Padwa
- AC Jones
- ACB Burtoloso
- AIO Suarez
- AM Phelps
- B Cimetière
- B Plietker
- BM Trost
- BM Trost
- C Molinaro
- C-Y Zhou
- CJ Moody
- CK Prier
- DS Carter
- EM McGarrigle
- G Kim
- G Kim
- G Li
- G Mlostoń
- H Koezuka
- H Nakano
- H Zhang
- I Aviv
- I Kawafune
- I Klose
- IK Mangion
- IK Mangion
- IK Mangion
- J Diekmann
- J Li
- J Sabbatani
- J Srogl
- J Vaitla
- J-P Qu
- J-R Chen
- JF Hooper
- JM Hatcher
- JR Fulton
- JV Matlock
- K Miki
- KJ Hock
- KJ Hock
- KK Ellis-Holder
- KL Greenman
- L Peng
- L Wang
- L Weber
- L-Q Lu
- M Barday
- M Clagett
- M Gandelman
- M Gandelman
- M Liao
- M Ma
- M Peña-López
- M Yar
- MD Santos
- MG Unthank
- MG Unthank
- MH Shaw
- MP Doyle
- MP Doyle
- MS Holzwarth
- N Tokitoh
- ND Shapiro
- P Bravo
- P Lu
- P Müller
- PW Davies
- PW Davies
- Q Wang
- Q Wang
- Q Xiao
- R Lin
- R Oost
- R Prabharasuth
- RH Crabtree
- S Kitagaki
- S Klimczyk
- S Klimczyk
- S Kramer
- S-F Zhu
- SJ Sabounchei
- SJ Sabounchei
- SJ Sabounchei
- SJ Sabounchei
- SJ Sabounchei
- SJ Sabounchei
- SJ Sabounchei
- T Cohen
- T Fukuda
- T Miura
- T-R Li
- V Nair
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- VK Aggarwal
- W Ando
- W Ando
- W Kirmse
- W-W Chan
- X Huang
- X Huang
- X Huang
- X Xu
- X Xu
- X Xu
- X Zhang
- X-D Xia
- Y Deng
- Y Deng
- Y Duan
- Y Duan
- Y Kato
- Y Li
- Y Li
- Y Nishibayashi
- Y Xu
- Y Xu
- Y Zhang
- Y-Y Liu
- Z Sheng
- Z Song
- Z Zhang
- Z Zhang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Recent developments in biocatalysis beyond the laboratory
- Author
- A Gog
- A Illanes
- AM Rouhi
- AP Green
- B Smerdel
- BM Brena
- BM Nestl
- BM Nestl
- BY Hwang
- C Kuraishi
- CE Olivier
- CK Savile
- CVL Giosafatto
- D Adachi
- D Zhang
- DA Clare
- DP Erickson
- GAH Jong De
- GW Huisman
- H Kohls
- IK Mangion
- IM Martins
- J Huang
- J James
- J Rudat
- J Stangierski
- J Yan
- JA Gerrard
- Jasmina Nikodinovic-Runic
- JH Seo
- JM Woodley
- K Buettner
- K Yokoyama
- Kevin E. O’ Connor
- KR Jegannathan
- KS Midelfort
- L Frodsham
- LH Han
- LP Christopher
- M Girardin
- M Kieliszek
- M Lee
- M Svedendahl
- Markets and Markets
- MD Truppo
- MD Truppo
- NG Heredia-Sandoval
- NM Rachel
- OS Ramos
- P Pierro Di
- P Tufvesson
- PJ Dunn
- R Dach
- R Schoenlechner
- RC Simon
- RE Meadows
- Reeta Davis
- S Chattopadhyay
- S Goes-Favoni de
- S Hama
- S Mathew
- S Renzetti
- SE Yew
- T Kanaji
- Tanja Narancic
- TJ Lim
- TP Korman
- TPN Ngo
- W Kroutil
- X Peng
- XW Yu
- XW Yu
- Y Lv
- Y Xie
- YT Hwang
- Z Jin
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Antibiotics in the clinical pipeline in 2013
- Author
- A Al-Lahham
- A Bonnefoy
- A Borghi
- A Dalhoff
- A Dalhoff
- A Gin
- A Koul
- A Malabarba
- A Malabarba
- A Rodríguez-Rojas
- A Sharma
- A Toda
- A Tupin
- A Wookey
- A Zumla
- AC Haagsma
- AC Rodloff
- AD So
- AG Brown
- AI Smolentsev
- Anonymous.
- B Cavalleri
- B Hofer
- B Spellberg
- B-Y Kim
- BJ Morrow
- BJ Morrow
- C Coronelli
- C Francavilla
- C Reading
- C van Delden
- CK Stover
- CRH Raetz
- CS Osborne
- CTM Mascio
- D Bertrand
- D Golparian
- D Grushkin
- D Landman
- D Vandamme
- DE Ehmann
- DI Andersson
- DJ Farrell
- DJ Farrell
- DJ Farrell
- DJ Payne
- DJ Payne
- DK Mercer
- DM Citron
- DM Citron
- DM Livermore
- DM Richards
- DM Shlaes
- DM Shlaes
- DR Ashtekar
- DR Snydman
- DT Moir
- DZ Chen
- E Azoulay-Dupuis
- E Bouza
- E Grunberg
- E Skripkin
- EA Nordahl
- EB Hirsch
- EMH Wellington
- F Parenti
- F-Y Lin
- FC Tenover
- FME Wagenlehner
- FP Gonzales
- G Zhanel
- G Zhanel
- GG Zhanel
- GJ Noel
- GN Tew
- GS Crowther
- H Lu
- H Patel
- H Reimann
- H Sasaki
- H-S Park
- HA Kirst
- HA Kirst
- HB Yu
- HH Fox
- HP Schweizer
- HS Park
- HS Park
- HS Sader
- HS Sader
- HS Sader
- HW Boucher
- HW Boucher
- HW Boucher
- I Galani
- I Rodríguez-Avial
- IK Mangion
- J Berdy
- J Isaksson
- J Kuti
- J Turner
- J Zhang
- J Zhou
- J Zhou
- J-W Jeong
- JA Karlowsky
- JA Karlowsky
- JA Leeds
- JA Leeds
- JA Sutcliffe
- JB Aggen
- JB Locke
- JB Parsons
- JE Hochlowski
- JH Yum
- JJ Gordon
- JL Crandon
- JM Hughes
- JM Rolain
- JW Larrick
- JWC Alffenaar
- K Andries
- K Bush
- K Coleman
- K Drlica
- K Michalska
- K O’Dwyer
- K Tahlan
- KB Waites
- KJ Shaw
- KN Williams
- L Lawrence
- L Wang
- LD Saravolatz
- LL Silver
- LL Silver
- LSL Ting
- M Castanheira
- M Gurumurthy
- M Matsumoto
- M Ronn
- M-S Hsu
- M-U Rashid
- MA Cooper
- MB Gravestock
- MG Scott
- MGP Page
- MJ Dawson
- MJ LaMarche
- MJ Weinstein
- MR Barbachyn
- MR Islam
- MR Jacobs
- MS Butler
- MS Butler
- MS Butler
- MT Gler
- MT Guskey
- MV Ranall
- MW Garrison
- N Kaplan
- N Ooi
- N Ooi
- N Srinivas
- N-C Emrich
- NJ de Souza
- P Prokocimer
- PG Higgins
- PG Higgins
- R Laxminarayan
- R Novak
- R Novak
- R O'Shea
- R Singh
- RB Clark
- RDG Cooper
- RE Lee
- REW Hancock
- RG Micetich
- RJ Theriault
- RN Jones
- RS Wallis
- RS Wallis
- S Boakes
- S Choi
- S Hawser
- S Higuchi
- S Kanthawong
- S Lemaire
- S Lemaire
- S Lemaire
- S Mushtaq
- S Omura
- S Sergio
- S Takeda
- S Takeda
- S Webb
- SD Putnam
- SM Bhavnani
- SS Bhagwat
- T Bogdanovich
- T Maisch
- T Mima
- T Stachyra
- T Yamakawa
- T-L Lauderdale
- TH Grossman
- TJ Falla
- TP Shiau
- TS Ryge
- U Manjunatha
- V Gerusz
- VN Kokryakov
- W Gottardi
- W Rodgers
- W Stubbings
- WB Im
- WT Prince
- X-Y Xiao
- Y Wang
- Z Oren
- ZA Kanafani
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 04/09/2013
- Field of study
The continued emergence of multi-drug-resistant bacteria is a major public health concern. The identification and development of new antibiotics, especially those with new modes of action, is imperative to help treat these infections. This review lists the 22 new antibiotics launched since 2000 and details the two first-in-class antibiotics, fidaxomicin (1) and bedaquiline (2), launched in 2011 and 2012, respectively. The development status, mode of action, spectra of activity, historical discovery and origin of the drug pharmacophore (natural product, natural product derived, synthetic or protein/mammalian peptide) of the 49 compounds and 6 β-lactamase/β-lactam combinations in active clinical development are discussed, as well as compounds that have been discontinued from clinical development since 2011. New antibacterial pharmacophore templates are also reviewed and analyzed
Investigational Antimicrobial Agents of 2013
- Author
- Abbanat D
- Aktas Z
- Allen NE
- Armstrong ES
- Balasubramanian V
- Barbachyn MR
- Barrett JF
- Biedenbach DJ
- Blondeau JM
- Bogatcheva E
- Boucher HW
- Bouchillon S
- Bozdogan B
- Bush K
- Bush K
- Bush K
- Bush K
- Candiani G
- Chen DZ
- Chen HY
- Chiba M
- Chu DT
- Collin F
- Craft JC
- Crowther GS
- Das D
- Day IP
- De Vriese AS
- Deane J
- Deane J
- Diacon AH
- Dunkle JA
- Echols RM
- Eckburg PB
- Ehmann DE
- Emrich NC
- Endimiani Choudhary A Y
- Fisher J
- Flamm RK
- Flamm RK
- Ford CW
- Gerding DN
- Gler MT
- Goh S
- Gomi K
- Gould IM
- Gould JK
- Gregory WA
- Gregory WA
- Griffith DC
- Grosset JH
- Grossman TH
- Guilloteau JP
- Hecker SJ
- Heine HS
- Hogenauer G
- Horn P
- Howden Grayson BP ML
- Hu C
- Hutchinson DK
- Jain R
- Johnson AP
- Kamboj M
- Kanafani ZA
- Katopodis GD
- Kavanagh F
- Ke Sampson W
- Kelley PG
- Kim EJ
- Kitagawa H
- Kitagawa H
- Kollef MH
- Koripella RK
- Kreusch A
- Kronvall G
- Kuramoto Y
- Kurosaka Y
- LaMarche MJ
- Landman D
- Lawrence L
- Lee M
- Lessa FC
- Li CR
- Li GQ
- Li GQ
- Livermore DM
- Livermore DM
- Livermore DM
- Livermore DM
- Livermore DM
- Livermore DM
- Lomovskaya O
- Louie A
- Macone A
- Macone AB
- Mangion IK
- Mansour H
- Mazel D
- Mega W
- Migliori GB
- Miida H
- Mitscher LA
- Moazed D
- Moir DT
- Morrisey I
- Morrissey I
- Mushtaq S
- Mushtaq S
- Mushtaq S
- Naderer OJ
- Nelson ML
- Novak R
- O'Brien W
- Page MGP
- Park CH
- Piddock LJ
- Powers RA
- Prince WT
- Protopopova M
- Putnam SD
- Rafie S
- Ramnauth J
- Reele S
- Remy JM
- Riddle V
- Rodríguez JC
- Russo TA
- Rustomjee R
- Ruzin A
- Ruzin A
- Sabet M
- Sacksteder KA
- Sader HS
- Sader HS
- Sader HS
- Sampson PB
- Seo MD
- Serero A
- Soulama C
- Stachyra T
- Starosta AL
- Steiert M
- Sum PE
- Sun H
- Sutcliffe JA
- Tan Q
- Tang YZ
- Tenover FC
- Titelman E
- Traczewski MM
- Tremolieres F
- Villemagne B
- Waksman SA
- Washington JA
- Weir S
- Werneburg M
- Wilbraham S
- Wiles JA
- Yang Y
- Young K
- Yount NY
- Zasloff M
- Zervosen A
- Zhanel GG
- Zhanel GG
- Zhang J
- Zhang J
- Zhong P
- Zhu DM
- Publication venue
- 'American Society for Microbiology'
- Publication date
- Field of study
Imino Transfer Hydrogenation Reductions
- Author
- A Bartoszewicz
- A Buchard
- A Landwehr
- A McSkimming
- A McSkimming
- A Nova
- A Quintard
- A Robertson
- A Ros
- AM Gulamhussen
- B Vilhanová
- B Zhao
- C Schüttler
- C Sui-Seng
- C Wang
- C Wang
- C Wang
- C Wang
- C Zheng
- CP Casey
- CR Graves
- D Blackmond
- D Gnanamgari
- D Guijarro
- D Guijarro
- D Guijarro
- D Gülcemal
- D Talwar
- D Talwar
- D Wang
- E Menéndez-Pedregal
- E Mizushima
- E Peris
- E Streckham
- E Vedejs
- ES Nogueira
- F Schwizer
- FE Fernández
- FE Fernández
- FW Monnard
- G Chelucci
- G Zhang
- GD Williams
- GJ Sherborne
- GKM Verzijl
- H Guan
- H Sugie
- H Xu
- H Šillová
- I Chatterjee
- I Kaldor
- IK Mangion
- J Blacker
- J Canivet
- J Han
- J Li
- J Long
- J Mao
- J Pecháčcek
- J Přech
- J Szawkalo
- J Szawkalo
- J Szawkalo
- J Tan
- J Václavik
- J Václavik
- J Václavik
- J Václavik
- J Václavik
- J Václavik
- J Václavik
- J Wu
- J Wu
- J-A Kim
- J-J Cheng
- JED Martins
- JF Collados
- JG Vries de
- JJ Soldevila-Barreda
- JM Zimbron
- JR Miecznikowski
- JSM Samec
- JSM Samec
- JSM Samec
- K Nishide
- K-I Fujita
- KA Nolin
- KH Ahn
- L Evanno
- L Li
- L Rubio-Pérez
- L Wang
- LF Tietze
- LS Santos
- M Duerrenberger
- M Dürrenberger
- M Genz
- M Kitamura
- M Kuzma
- M Ringenberg
- M Wills
- M Wu
- M Zhang
- MP Magee
- MR Ringenberg
- MV Jiménez
- N Haraguchi
- N Haraguchi
- N Uematsu
- NA Strotman
- O Pablo
- O Pablo
- O Pablo
- O Pamies
- O Saidi
- P Roszkowski
- P Roszkowski
- P Šot
- P Šot
- PE Sues
- QA Chen
- R Corberán
- R Kadyrov
- R Liu
- R Soni
- RM Bullock
- S Betanzos-Lara
- S Burling
- S Diez-Gonzalez
- S Gladiali
- S Guizzetti
- S Guizzetti
- S Gülcemal
- S Kang
- S Kuhl
- S Ogo
- S Ogo
- S Richards
- S Zhou
- SA Lee
- SD Boggs
- SE Clapham
- SJ Lucas
- SN Sluijter
- T Heinisch
- T Heinisch
- T Ikariya
- T Itoh
- T Koike
- T Quinto
- T Quinto
- TC Nugent
- TD Nixon
- TR Ward
- V Dragutan
- V Galmari
- V Köhler
- V Köhler
- V Parekh
- V Samano
- VS Shende
- W Tang
- W Tang
- W Zuo
- W Zuo
- X Dai
- X Yang
- X-H Zhu
- Y Fu
- Y Kondo
- Y Mirabal-Gallardo
- Y Watanabe
- Y Wei
- Y Wei
- Y Zhang
- Y-C Chen
- YC Chen
- YJ Seo
- YM Wilson
- Z Liu
- Z Wu
- Z-Q Rong
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Antibiotics in the clinical pipeline at the end of 2015
- Author
- A Al-Lahham
- A Belley
- A Bonnefoy
- A Dalhoff
- A Gin
- A Ito
- A Jekle
- A Morinaka
- A Sattar
- A Toda
- A Walkty
- AB Macone
- AC Nilsson
- AC Rodloff
- AG Brown
- AI Smolentsev
- AJ Sucher
- AM Upton
- AP Johnson
- B Hafkin
- B Hofer
- BD Brooks
- BE Erickson
- BT Tsuji
- C Francavilla
- C Lok
- C Lucasti
- C Reading
- C van Delden
- C-H Huang
- CA Michael
- CK Stover
- CL Ventola
- CL Ventola
- CR Li
- CT Walsh
- D Brown
- D Dominey-Howes
- D Golparian
- D Landman
- DE Ehmann
- DJ Farrell
- DJ Farrell
- DJ Farrell
- DJ Payne
- DJ Payne
- DM Citron
- DM Citron
- DM Livermore
- DM Richards
- DM Shlaes
- DR Ashtekar
- DR Snydman
- E Bettiola
- E Bouza
- E Grunberg
- E Skripkin
- F Pea
- F Van Bambeke
- FM Aarestrup
- FM Wagenlehner
- FP Gonzales
- G Kern
- G Piccinelli
- G Sinha
- G Zhanel
- G Zhanel
- GG Zhanel
- GG Zhanel
- GJ Patti
- GM Rossolini
- GN Tew
- H Lu
- H Reimann
- H Sasaki
- HA Blair
- HH Fox
- HH Locher
- HH Locher
- HL Haver
- HS Sader
- HS Sader
- I Galani
- I Karaiskos
- I Rodríguez-Avial
- IA Critchley
- IK Mangion
- J Blais
- J Isaksson
- J Zhou
- J Zhou
- J-W Jeong
- JA Karlowsky
- JA Karlowsky
- JA Sutcliffe
- JB Aggen
- JB Locke
- JB Parsons
- JE Ross
- JG Owen
- JL Crandon
- JL Crandon
- JL Crandon
- JL Fox
- JL Fox
- JS Jensen
- JW Lee
- K Chotikanatis
- K Coleman
- K Drlica
- K Li
- K McKeage
- K Pethe
- K Servick
- KMG O'Connell
- KN Rao
- L Bouillaut
- L Czaplewski
- L Honeyman
- L Jarvis
- L Lawrence
- L Wang
- LD Saravolatz
- LJ Shallcross
- LL Ling
- M Cheng
- M Gurumurthy
- M Matsumoto
- M Ronn
- M Woolhouse
- M-S Hsu
- M-U Rashid
- MA Banevicius
- MA Cooper
- MA Cooper
- MAT Blaskovich
- ME Stryjewski
- MEJ Woolhouse
- MF Gordeev
- MGP Page
- MJ Weinstein
- MJB Melchers
- MP Draper
- MR Jacobs
- MS Butler
- MS Butler
- MS Butler
- MT Guskey
- MZ Alam
- N Kaplan
- N Kaplan
- N Kohira
- N Ooi
- N Ooi
- N Srinivas
- N Yin
- N-C Emrich
- NE Allen
- NG Anthony
- NJ de Souza
- P Fernandes
- P Gopal
- P Nunn
- P Prokocimer
- P Veiga-Santos
- PG Higgins
- R Almaghrabi
- R CK
- R Gupta
- R Novak
- R Novak
- R Singh
- R Tasneen
- R Tommasi
- RB Clark
- RE Lee
- RG Micetich
- RK Flamm
- RM Anderson
- RM Poole
- RW Meek
- S Choi
- S Jacobsson
- S Kang
- S Lemaire
- S Mushtaq
- S Reardon
- S Shapiro
- S Takeda
- SB Singh
- SC Olsen
- SD Burdette
- SD Putnam
- SJ Kim
- SJ Kim
- SS Bhagwat
- T Maisch
- T Mima
- T Stachyra
- T Yamakawa
- T-L Lauderdale
- TH Grossman
- TH Grossman
- TP Shiau
- TS Ryge
- U Manjunatha
- V Gerusz
- V Knight-Connoni
- V Ong
- VN Kokryakov
- VR Anderson
- W Gottardi
- W Li
- W Qin
- W Rodgers
- W So
- W Stubbings
- WB Im
- WT Prince
- X-Y Xiao
- Y Kobayashi
- Y López
- YQ Huang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study