11 research outputs found
Exploiting loss of heterozygosity for allele-selective colorectal cancer chemotherapy
- Author
- A Gschwind
- A Untergasser
- AK Iyer
- AL Hubbard
- AS Nikonova
- BR Paolella
- C Cunningham
- C Sawyers
- D Nijhawan
- DW Hein
- DW Hein
- E Lindhagen
- EA Chiocca
- F Innocenti
- F Mertens
- FL Muller
- GR Abecasis
- GV Kryukov
- H Maiato
- I Aliagas-Martin
- I Niculescu-Duvaz
- IA Kesisova
- JP Basilion
- KJ Martell
- KJ Mavrakis
- LR Howe
- M Uhlen
- MJ Ratain
- N Issaeva
- P Baranczewski
- P Dey
- S Boukouvala
- S Kilpinen
- S Sakaushi
- SR Viswanathan
- T O’Hare
- WS El-Deiry
- Y Liu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Selective Aurora Kinase Inhibitors Identified Using a Taxol-Induced Checkpoint Sensitivity Screen
- Author
- Abe Y.
- Aliagas-Martin I.
- Andrea Musacchio
- Bayliss R.
- Bird A. W.
- Bishop J. D.
- Bolton M. A.
- Cheeseman I. M.
- Chen J.
- Deng X.
- Deng X.
- Eyers P. A.
- Fabian M. A.
- Fabrizio Villa
- George J.
- Giet R.
- Girdler F.
- Glover D. M.
- Hannak E.
- Harrington E. A.
- Hirota T.
- Honda R.
- Hsiao-Chun Huang
- Huang H. C.
- Hutterer A.
- Jelluma N.
- Jeyaprakash A. A.
- Jinhua Wang
- Kelly A. E.
- Kimura M.
- Koffa M. D.
- Kufer T. A.
- Kwiatkowski N.
- Lampson M. A.
- Lenart P.
- Li Tan
- Manfredi M. G.
- Mori D.
- Mortlock A. A.
- Nathanael Gray
- Nicholas Kwiatkowski
- Patricelli M. P.
- Rieder C. L.
- Santaguida S.
- Santaguida S.
- Saurin A. T.
- Sessa F.
- Shi J.
- Stefano Santaguida
- Tan N.
- Tanaka T. U.
- Terada Y.
- Tim Mitchison
- Toji S.
- Tsai M. Y.
- Vader G.
- Wertz I. E.
- Xianming Deng
- Yasui Y.
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
Phthalazinone Pyrazole Enhances the Hepatic Functions of Human Embryonic Stem Cell-Derived Hepatocyte-Like Cells via Suppression of the Epithelial-Mesenchymal Transition
- Author
- A Treyer
- AB D’Assoro
- AK Reka
- AM Wobus
- AV Bakin
- B Li
- C Billottet
- C Cicchini
- Chang-Woo Song
- D Chen
- Dae-Sung Kim
- DR Xu
- F Garibaldi
- H Katayama
- Han-Jin Park
- HJ Park
- HM Kim
- Hyemin Kim
- I Aliagas-Martin
- J Chen
- J Corchero
- J Yang
- JC Davila
- JE Lee
- Ji-Woo Kim
- JP Li
- JP Li
- JP Thiery
- JP Thiery
- K Anderson
- M Baxter
- ME Prime
- MG Manfredi
- MI Yovchev
- MJ Zamek-Gliszczynski
- N Kaplowitz
- N Keen
- O Goldman
- P Godoy
- P Samavarchi-Tehrani
- RA Wilke
- S Grotegut
- S Hauf
- S Kawashima
- Seokjoo Yoon
- SJ Grille
- SS Choi
- T Shimomura
- U Cavallaro
- V Sehdev
- XB Wan
- Y Kamiyama
- Y Xi
- YH Ding
- Young-Jun Choi
- Z Li
- Z Lu
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
A MYC–aurora kinase A protein complex represents an actionable drug target in p53-altered liver cancer
- Author
- A Katsha
- A Khwaja
- A Klein
- A Tannapfel
- AD Tward
- Anja Hohmeyer
- Antti Poso
- B Amati
- C Welsch
- CJ Sherr
- CJ Sherr
- CM Carlson
- CM Schmidt
- CM Shachaf
- D Fancelli
- D Huesken
- Daniel Dauch
- DF Calvisi
- DJ Burgess
- DL White
- DW Felsher
- DW Meek
- EE Calle
- G Falchook
- Giacomo Cossa
- H Beltran
- H BraumĂĽller
- H Katayama
- H Yuan
- I Aliagas-Martin
- J Bruix
- J Liu
- J Zuber
- JD Watson
- JE Delmore
- Jean-Charles Nault
- Jessica Zucman-Rossi
- JM Mosquera
- JP Vert
- K Podsypanina
- KL Chan
- L Lu
- L Soucek
- L Zender
- L Zender
- Lars Zender
- Lisa Hoenicke
- LY Lu
- M Brockmann
- M Eilers
- M Eilers
- Martin Eilers
- ME Diefenbacher
- MT Kimura
- N Meyer
- Nisar P Malek
- P Carpinelli
- P White
- PA Farazi
- Przemyslaw Bozko
- R Crane
- R Lord
- R PĂ©rez Tamayo
- R Rudalska
- R Taub
- Ramona Rudalska
- Sandrine Imbeaud
- Stefan Laufer
- T Otto
- T Wuestefeld
- Tae-Won Kang
- Tatu Pantsar
- Tetyana Yevsa
- Thomas Longerich
- Torsten Wuestefeld
- TW Kang
- V Krizhanovsky
- WC Gustafson
- Y Ito
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Aurora Kinases as Druggable Targets in Pediatric Leukemia: Heterogeneity in Target Modulation Activities and Cytotoxicity by Diverse Novel Therapeutic Agents
- Author
- Aarthi Jayanthan
- Aru Narendran
- AS Moore
- C Ditchfield
- C Soncini
- C-H Pui
- C-H Pui
- Claude Prigent
- CS Nabzdyk
- D Akahane
- D Bhojwani
- D Fancelli
- EA Harrington
- F Broekman
- F Chan
- F Locatelli
- H Hochegger
- H Katayama
- I Aliagas-Martin
- J Curry
- J How
- J Khan
- J Yang
- JA Seamon
- JD Oslob
- JJ Tentler
- JP Arbitrario
- JR Pollard
- JR Sierra
- K Yoshida
- KR Kelly
- KR Molhoek
- M Carmena
- M Kimura
- M Li
- M Steegmaier
- M Tanudji
- ME Tanenbaum
- N HĂ©garat
- N Keen
- N Steeghs
- O Gautschi
- P Carpinelli
- P Kaestner
- P Meraldi
- R Hrabakova
- RK Tyler
- S Emanuel
- S Howard
- S Lapenna
- S Okabe
- S Okabe
- S Wang
- SA Doggrell
- SE Puumala
- SMA Lens
- T Ota
- T Yamauchi
- Tony H. Truong
- W Lok
- W Qi
- Y Yakushijin
- Yibing Ruan
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- Field of study
A Computational Model for Overcoming Drug Resistance Using Selective Dual-Inhibitors for Aurora Kinase A and Its T217D Variant
- Author
- Ali H. I.
- Aliagas-Martin I.
- Barakat K.
- Barakat K.
- Barakat K. H.
- Bavetsias V.
- Baxter C. A.
- Constantinos Evangelinos
- Davies D. L.
- Dodson C. A.
- Dolinsky T. J.
- Dunbrack R. L.
- Fancelli D.
- Fenner A.
- Friesen D. E.
- Fu T.
- Garcia A. E.
- Goodsell D. S.
- Grazioso G.
- Greenman C.
- He W.
- Hess B.
- Hornak V.
- Howard S.
- J. Torin Huzil
- Jack Tuszynski
- Jakalian A.
- Jordheim L. P.
- Kalé L.
- Karaman M. W.
- Khaled H. Barakat
- Kirk E. Jordan
- Kollareddy M.
- Kollman P. A.
- Kroemer R. T.
- Kuhn B.
- Leonis G.
- Lin J. H.
- Liu J.
- Liu Q.
- Michael Houghton
- Morris G. M.
- Morshed M. N.
- Nowakowski J.
- Pettersen E. F.
- Sali A.
- Sardon T.
- Schoffski P.
- Sen S.
- Shao J.
- Shi H.
- Sloane D. A.
- Tari L. W.
- Totrov M.
- Wishart D. S.
- Wissing M. D.
- Xie L.
- Yang Y.
- Zhao B.
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
Physicochemical and DMPK In Silico Models: Facilitating Their Use by Medicinal Chemists
- Author
- Bickerton G. R.
- Cruciani G.
- Cruciani G.
- Daniel F. Ortwine
- Desai P. V.
- Faller B.
- Forina M.
- Gao H.
- Ghose A. K.
- Gleeson M. P.
- Gleeson M. P.
- Gleeson M. P.
- Gleeson M. P.
- Gupta R.
- Hann M. M.
- Heffron T. P.
- Hewitt M.
- Hill A. P.
- Hopfinger A. J.
- Ignacio Aliagas
- Kozopas K. M.
- Lee P. H.
- Leeson P. D.
- Leeson P. D.
- Lipinski C. A.
- Liu L.
- Liu L.
- Lobell M.
- Martin Y. C.
- Milletti F.
- Muchmore S. W.
- Nicola G.
- Obrezanova O.
- Patterson D. E.
- Peng Z.
- Plewczynski D.
- Ritchie T. J.
- Rush T. S.
- Sastry G. M.
- Scannell J. W.
- Segall M.
- Segall M. D.
- Stewart K. D.
- Sushko I.
- Tarcsay A.
- Thai K.-M.
- Wager T. T.
- Wager T. T.
- Wenlock M. C.
- Willett P.
- Zientek M.
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
Aurora Isoform Selectivity: Design and Synthesis of Imidazo[4,5- b
- Author
- Adams P. D.
- Alan Henley
- Aliagas-Martin I.
- Amar Joshi
- Amir Faisal
- Araki K.
- Barr A. R.
- Bavetsias V.
- Bavetsias V.
- Bavetsias V.
- Bayliss R.
- Bischoff J. R.
- Blagg J.
- Bolanos-Garcia V. M.
- Bouloc N.
- Brockmann M.
- Butrus Atrash
- Carmena M.
- Chan F.
- Cheung C. H. A.
- Chieffi P.
- Chongbo Sun
- Coumar M. S.
- Dodson C. A.
- Dodson C. A.
- Ducat D.
- Finaru A.
- Florence I. Raynaud
- Girdler F.
- Graczyk P. P.
- Green M. R.
- Gritsko T. M.
- Jessica A. Schmitt
- Jones G.
- Julian Blagg
- Kalgutkar A. S.
- Katherine Bush
- Katherine J. Boxall
- Kelly K. R.
- Knapp S.
- Larock R. C.
- Magda Kosmopoulou
- Malumbres M.
- Manfredi M. G.
- Manfredi M. G.
- Marumoto T.
- Mortlock A. A.
- Nathan Brown
- Otto T.
- Paul Workman
- Pollard J. R.
- Prime M. E.
- Reichardt W.
- Richard Bayliss
- Rosemary Burke
- Shimomura T.
- Sian Avery
- Simon Crumpler
- Sorrentino R.
- Spiros Linardopoulos
- Tanaka T.
- Ujjainwalla F.
- Vassilios Bavetsias
- Workman P.
- Yang D.
- Yolanda PĂ©rez-Fuertes
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
Development of o
- Author
- Adams N. D.
- Aliagas-Martin I.
- Anandan S.-K.
- Anastassiadis T.
- Asteriti I. A.
- Bardelle C.
- Barlaam B.
- Bearss D. J.
- Beattie J. F.
- Bebbington D.
- Belanger D. B.
- Berndt N.
- Boss D. S.
- Breault G. A.
- Brunger A. T.
- Cee V. J.
- Chakravarty A.
- Charter N. W.
- Cheung C. H. A.
- Cheung C. H. A.
- Coumar M. S.
- Dar A. A.
- DeLano W. L.
- Dodson C. A.
- Emsley P.
- Ernst Schonbrunn
- Fancelli D.
- Fancelli D.
- Fancelli D.
- Garuti L.
- Girdler F.
- Gizatullin F.
- Gorgun G.
- Green M. R.
- Harrington E. A.
- Harshani R. Lawrence
- Harsukh Gevariya
- Herr R. J.
- Hua Yang
- Jester B. W.
- Jin Q. Cheng
- Jin-Yi Zhu
- Kabsch W.
- Kang N. S.
- Keen N.
- Keen N.
- Koresawa M.
- Libertini S.
- Lietha D.
- Liu M.
- Lok W.
- Manfredi M. G.
- Manfredi M. G.
- Martin M. P.
- Marumoto T.
- Mathew P. Martin
- Mercedes Rodriguez
- Moriarty K. J.
- Mortlock A. A.
- Nicholas J. Lawrence
- Ochi T.
- Pearce L. R.
- Perez Fidalgo J. A.
- Pollard J. R.
- Portella G.
- Robert Kendig
- Roberta Pireddu
- Roy Elias
- Saeki T.
- SaĂŻd M. Sebti
- Sevil Ozcan
- Shang X.
- Shimomura T.
- Sloane D. A.
- Soncini C.
- Tari L. W.
- Tomita M.
- Vader G.
- Wilkinson R. W.
- Yeung S.-C. J.
- Yu T.
- Yunting Luo
- Zhang J.
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
Issues in interpreting the in vivo
- Author
- Abe Y
- Agnese V
- Aliagas-Martin I
- Anand S
- Bai M
- Bai M
- Bai M
- Bayliss R
- Bibby RA
- Brockmann M
- Carol H
- Castro A
- Cervantes-Ruiperez A
- Chen SS
- Chowdhury A
- Clark MA
- Crane R
- Dadke D
- de Carcer G
- Do TV
- Dodson CA
- Dodson CA
- Dutertre S
- Elena Shagisultanova
- Erica A Golemis
- Eyers PA
- Eyers PA
- Giubettini M
- Gorgun G
- Han YG
- Haydon CE
- Hirota T
- Huang YH
- Hutterer A
- Ice RJ
- Infante J DE
- Jackman M
- Johnson EO
- Johnson EO
- Joukov V
- Kashatus DF
- Katayama H
- Kelly KR
- Kelly KR
- Krystyniak A
- Kufer TA
- Lawrence HR
- Lefkowitz GK
- Littlepage LE
- Littlepage LE
- Liu Q
- Manfredi MG
- Matallanas D
- Meraldi P
- Mori D
- Mori D
- Nam HJ
- Nikonova AS
- Nikonova AS
- Nurse P
- Otto T
- Ouchi M
- Pascreau G
- Pascreau G
- Patel AV
- Perez de Castro I
- Plotnikova OV
- Plotnikova OV
- Plotnikova OV
- Plotnikova OV
- Pugacheva EN
- Pugacheva EN
- Qi W
- Qi W
- Radu M
- Ratushny V
- Reboutier D
- Roland L Dunbrack
- Rowan FC
- Sabino D
- Sarkissian M
- Satinover DL
- Schneider L
- Seeger-Nukpezah T
- Sehdev V
- Seki A
- Shao S
- Shi Y
- Sloane DA
- Tatsuka M
- Tomita M
- Vader G
- Weinstein IB
- Xu X
- Zeng K
- Zhang D
- Zhang M HJ
- Zhao ZS
- Zheng M
- Zorba A
- Publication venue
- 'Informa Healthcare'
- Publication date
- Field of study