8 research outputs found
Tyrosine Phosphorylation of Rac1: A Role in Regulation of Cell Spreading
- Author
- A Briancon-Marjollet
- A Dovas
- AB Jaffe
- AJ Ridley
- BZ Katz
- C DerMardirossian
- C DerMardirossian
- Christopher Lemmon
- D Lietha
- Daniel Lietha
- E Nikolova
- E Tzima
- EE Bosco
- Erik H. J. Danen
- F Chang
- Fumin Chang
- H Abramovici
- H Fuss
- HH Grunicke
- JE Chrencik
- JH Choi
- JL Kissil
- JV Olsen
- K Moissoglu
- K Roepstorff
- KR Myers
- Lewis Romer
- LH Romer
- M Oyama
- MA Del Pozo
- MA Forget
- MD Schaller
- MD Schaller
- Michael Eck
- MJ Hart
- MP Playford
- MR Jezyk
- MV Milburn
- NO Carragher
- NS Bryce
- P Lang
- PL Hordijk
- S Li
- S Tu
- SA Moodie
- T Hunter
- T Kwon
- UK Laemmli
- V Benard
- X Wu
- XR Bustelo
- Y Gao
- Publication venue
- Public Library of Science
- Publication date
- 01/01/2011
- Field of study
Rac1 influences a multiplicity of vital cellular- and tissue-level control functions, making it an important candidate for targeted therapeutics. The activity of the Rho family member Cdc42 has been shown to be modulated by tyrosine phosphorylation at position 64. We therefore investigated consequences of the point mutations Y64F and Y64D in Rac1. Both mutations altered cell spreading from baseline in the settings of wild type, constitutively active, or dominant negative Rac1 expression, and were accompanied by differences in Rac1 targeting to focal adhesions. Rac1-Y64F displayed increased GTP-binding, increased association with βPIX, and reduced binding with RhoGDI as compared with wild type Rac1. Rac1-Y64D had less binding to PAK than Rac1-WT or Rac1-64F. In vitro assays demonstrated that Y64 in Rac1 is a target for FAK and Src. Taken together, these data suggest a mechanism for the regulation of Rac1 activity by non-receptor tyrosine kinases, with consequences for membrane extension
Conjugated Linoleic Acid Decreases MCF-7 Human Breast Cancer Cell Growth and Insulin-Like Growth Factor-1 Receptor Levels
- Author
- A Miglietta
- AA Spector
- AF Keating
- AG Renehan
- AJ Hulbert
- AL Lock
- AM Turpeinen
- B Majumder
- BA Corl
- C Cruz-Hernandez
- C desBordes
- C Ip
- C Ip
- C Ip
- Catherine J. Field
- CD Stubbs
- CJ Field
- DA Brown
- Danielle L. Amarù
- DD Guo
- DL Kleinberg
- DW Ma
- E Przybytkowski
- EJ Kim
- ES Schernhammer
- H Chujo
- H Huo
- H Uehara
- HH Grunicke
- HJ Cho
- J Folch
- J Zhang
- JH Seo
- JJ Yin
- JK Kramer
- JL Sebedio
- JP Peyrat
- LS Wang
- M Remacle-Bonnet
- M Yorek
- MD Sternlicht
- MM Ip
- MN Pollak
- MQ Kemp
- NE Hubbard
- NS Kelley
- P Tanmahasamut
- PD Schley
- PD Schley
- RF Grimble
- S Banni
- S Hardy
- S Hardy
- S Visonneau
- TR Dhiman
- Y Choi
- Y Kaburagi
- Y Park
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
PAR-4 as a possible new target for pancreatic cancer therapy
- Author
- Ahmad A
- Ahmed MM
- Ali S
- Ali S
- Asfar S Azmi
- Azmi AS
- Azmi AS
- Barradas M
- Bartsch DK
- Baud V
- Bhuiyan MM
- Boghaert ER
- Boghaert ER
- Buchholz M
- Burikhanov R
- Castagnola P
- Cejas P
- Chakraborty M
- Cheema SK
- Cho YS
- DeNicola GM
- Dobrzycka B
- El-Guendy N
- El-Guendy N
- Evans JD
- Fazlul H Sarkar
- Furukawa T
- Gallick GE
- Garcia-Cao I
- Gerdes B
- Gilmore TD
- Gonzalez IH
- Goswami A
- Greten FR
- Grunicke HH
- Gurumurthy S
- Gurumurthy S
- Hamacher R
- Hingorani SR
- Hua C
- Jemal A
- Jonson T
- Jonson T
- Keleg S
- Kimura M
- Kindler HL
- Kong D
- Kranenburg O
- Lessene G
- Li Y
- Macdonald JS
- Mollinedo F
- Moreno-Bueno G
- Moscat J
- Moskaluk CA
- Nalca A
- Neumann TE
- Olsen CC
- Perez-Mancera PA
- Perren A
- Philip A Philip
- Popovic HM
- Prost P
- Pruitt K
- Qiu G
- Rahman KM
- Ramzi M Mohammad
- Ranganathan P
- Rangnekar VM
- Regula KM
- Riely GJ
- Sato Y
- Schneider G
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- Sells SF
- Stehelin D
- Summy JM
- Syed F Zafar
- Tian B
- Truty MJ
- Truty MJ
- Van Custem E
- Vasudevan KM
- Xie J
- Xiong HQ
- Youssef EM
- Publication venue
- 'Informa Healthcare'
- Publication date
- Field of study
Cell-signaling targets for antitumour drug development
- Author
- A Asworth
- A Balmain
- A Basu
- A Basu
- A Fanidi
- A Gazit
- A Gazit
- A Gescher
- A Hall
- A Noseda
- A Wellstein
- AS Kraft
- AT Oosterom Van
- AV Schally
- B Margolis
- C Dive
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- C Liebow
- C Unger
- CA Koch
- CA O'Brian
- CA Stein
- CC Geilen
- CD Ferris
- CF Bennett
- CJ Tabin
- CL Arteaga
- CR Divgi
- CW Mahoney
- D Alberts
- D Lane
- DA Frank
- DC Heimbrook
- DJ Slamon
- DK Morrison
- DL Vaux
- DM Helfman
- DR Spriggs
- E Aboud-Pirak
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- JM Collins
- JW Hans
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- M Imoto
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- MB Kastan
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- MB Meyers
- MC Hancock
- MD Sklar
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- N Itoh
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- P Workman
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- PL Crowell
- PM Chaudhary
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- R Danesi
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- SH Ryu
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- SM Sebti
- SR Coughlin
- T Akiyama
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- YS Cho-Chung
- YS Cho-Chung
- Z Jamal
- Z Spigelman
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/1993
- Field of study
Regulation of gene expression by prolactin
- Author
- A Gertler
- A Gertler
- A Kanai
- A Kurtz
- A Mode
- A Ullrich
- AC Larner
- AF Wilks
- AM Stevens
- AM Vos De
- AR Buckley
- B Gellerson
- B Happ
- B Jehn
- B Pérez-Villamil
- B Staindl
- BC Cunningham
- BI Posner
- BJ Arey
- BJ Peters
- BK Vonderhaar
- BS Chilton
- C Cahoreau
- C Clapp
- C Collet
- C Collet
- C Jolicoeur
- C Legraverend
- C Puissant
- C Schindler
- C Schmidhauser
- C Schmidhauser
- C-A Schoenenberger
- CA Jagoda
- CG Prosser
- CJ Ormandy
- CJ Ormandy
- CJ Ormandy
- CKL Too
- CS Barker
- CS Lee
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- CS Nicoll
- CS Nicoll
- CV Clevenger
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- CW Pittius
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- DB Ray
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- DL Kleinberg
- DN Luck
- DW Leung
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- F Vizoso
- G Elberg
- G Fuh
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- G Thordarson
- GA Fan
- GA Jahn
- GA Jahn
- GC-K Chan
- GE Mattia Di
- GS Campbell
- GS Prins
- GW Randall
- H Rui
- H Wakao
- HB Sadowski
- HH Grunicke
- HS Goodman
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- I Pellegrini
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- J Wolff
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- KG Danielson
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- PA Furth
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- PG Campbell
- PJ Fielder
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- S Ali
- S Ali
- S Chiu
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- S Harris
- S Kleis-SanFrancisco
- S Mink
- S Pierre
- S Placido De
- S Sakai
- SB Waters
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- UM Wegenka
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- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/1994
- Field of study
Emerging therapeutic targets in colon cancer research
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- AHMAD S
- Antisense RNA
- ATTISANO L
- BARNARD JA.
- BARON PL
- BENCHIMOL S
- BLOBE GC
- BORDIER CG
- BORLINGHAUS P
- BRATTAIN MG
- BRATTAIN MG WILLSON JKV
- BROWDER TM
- Cancer of the colon and rectum. The Cancer Information Services.
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHAKRABARTY S
- CHEN RH
- CIARDIELLO F
- CIARDIELLO F
- CLARK EA
- COFFEY RJ
- COUSSENS L
- CROSS M
- DATTA MB
- DEAN DC
- DIRIX LY
- DISATNIK M-H
- DONALDSON RW
- EBNER R CHEN R-H
- EIDELMAN FJ
- ELLIS EM
- FRISCH SM
- GENG Y
- GIANCOTTI FG
- GRAVITT KR
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- HALLGREN B
- HARTWELL LH
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- MASSAGUE J
- MCNAMEE HP
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- MOSES HL
- MOUSTAKAS A
- MURTHY US
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- O'BRIAN CA
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- 'Informa Healthcare'
- Publication date
- Field of study
Issues and progress with protein kinase inhibitors for cancer treatment
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- A Bhattacharjee
- A Chakravarti
- A Lennon
- A Levitzki
- A Levitzki
- A Levitzki
- A Monks
- AD Catling
- AW Tolcher
- B Coudert
- B Geoerger
- B Nagar
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- BJ Druker
- BP Monia
- BP Rubin
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- DH Lynch
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- DJ Slamon
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- E Kerkhoff
- E Kerkhoff
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- E Rubin
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- Edward A. Sausville
- EE Cohen
- F Ciardiello
- F Ciardiello
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- FA Scappaticci
- FM Sirotnak
- G Gallardo
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- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Die Cytologie der Hepatocarcinogenese
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- A Forget
- A Gellhorn
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- A Graffi
- A Jacob
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- AB Novikoff
- AB Novikoff
- AB Novikoff
- AB Novikoff
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- AF Weber
- AF Weber
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- AK Laird
- AL Jones
- AL Jones
- AM Ambrose
- AM Rappaport
- AM Recondo
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- AS Mulay
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- B Flaks
- B Flaks
- B Flaks
- B Flaks
- B Flaks
- B Korpássy
- B Schulze
- B Tandler
- B Terracini
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- BH Ruebner
- BJ Horton
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- D Hadjiolov
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- H Ungar
- H-A Müller
- H-W Altmann
- H-W Altmann
- H-W Altmann
- H-W Altmann
- H-W Altmann
- H-W Altmann
- H-W Altmann
- HA Hartmann
- HB Andervont
- HC Grice
- HC Pitot
- HC Pitot
- HC Pitot
- HE Holling
- HF Stich
- HH Mason
- HJ Firminger
- HJ Firminger
- HL Richardson
- HL Stewart
- HM Rabes
- HM Rabes
- HP Hobik
- HP Morris
- HP Morris
- HS Taper
- I Hesse
- J Ashmore
- J Brodehl
- J Carneiro
- J Creemers
- J Côté
- J Davidson
- J Driessens
- J Driessens
- J Hoffmann
- J Locker
- J Maisin
- J Meldolesi
- J Meyer-Bertenrath
- J Meyer-Bertenrath
- J Meyer-Bertenrath
- J Reddy
- J Spain
- JC Arcos
- JC Arcos
- JC Arcos
- JC Arcos
- JC Arcos
- JC Garancis
- JC Man de
- JC Salomon
- JC Salomon
- JC Salomon
- JC Salomon
- JC Smith
- JD Spain
- JE Edwards
- JF Fraumeni
- JG Lafontaine
- JG Lafontaine
- JI Goodmann
- JJ Theron
- JLE Ericsson
- JM Price
- JM Price
- JM Price
- JN Chernozemski
- JP Chang
- JP Greenstein
- JR Allen
- JR Rüttner
- JS Carruthers
- JT Nodes
- JV Klavins
- JW Grisham
- JW Grisham
- JW Grisham
- JW Harman
- JW Orr
- JW Orr
- JW Orr
- JW Orr
- JW Steiner
- JW Steiner
- JW Steiner
- JW Steiner
- JW Steiner
- JW Wilson
- K Arakawa
- K Bélár
- K Goerttler
- K Miyai
- K Miyai
- K Miyai
- K Tempel
- KR Porter
- KR Porter
- KR Porter
- KS Narayan
- L Deckers-Passau
- L Ernster
- L Herman
- L Wiest
- LA Sordahl
- LB Bull
- LB Liu
- LC Strong
- LJ Rather
- LP Merkow
- LP Merkow
- LP Merkow
- LP Merkow
- LP Merkow
- M Arcasoy
- M Eder
- M Gronow
- M Gronow
- M Gronow
- M Heidenhain
- M Hoshino
- M Lopez
- M Müller
- M Wachstein
- M-C Moulin
- MA Lea
- MA Spycher
- MB Schmidt
- MB Sporn
- MD Reuber
- MD Reuber
- MD Reuber
- MD Reuber
- MF Argus
- MF Stanton
- MG Irving
- MG Kelly
- MH Ma
- MJ Phillips
- MJ Phillips
- MJ Striebich
- ML Watson
- MM Maini
- MM Maini
- MT White
- MW Woods
- N Brock
- N Heine
- N Ito
- NL Trotter
- O Klinge
- O Stein
- O Warburg
- OG Fitzhugh
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Bannasch
- P Baudhuin
- P Drochmans
- P Emmelot
- P Emmelot
- P Emmelot
- P Emmelot
- P Heizer
- P Melnick
- P Schmitz-Moormann
- PB Herdson
- PB Herdson
- PE Steiner
- PE Steiner
- PL Pederson
- PM Newberne
- PN Magee
- PN Magee
- PS Quinn
- R Cortell
- R Daoust
- R Daoust
- R Daoust
- R Daoust
- R Daoust
- R Daoust
- R Daoust
- R Daoust
- R Kinosita
- R Kinosita
- R Kullmann
- R Laumonier
- R Lesch
- R Lesch
- R Love
- R Potter van
- R Rondez
- R Schoental
- R Schoental
- R Simad
- R Simard
- R Sugihara
- R Vendrely
- R Wood
- RA McDonald
- RB Arhelger
- RC Reynolds
- RC Reynolds
- RE Albert
- RE Stowell
- RG Gustafsson
- RG Kessel
- RG Kleinfeld
- RG Kleinfeld
- RG Kleinfeld
- RGF Parker
- RJ Stenger
- RJ Stenger
- RL Hamilton
- RM Frank
- RM Sharma
- RO Christianson
- RO Recknagel
- RV Moseley
- S Fiala
- S Goldfarb
- S Goldfarb
- S Hori
- S Karasaki
- S Karasaki
- S Karasaki
- S Koulish
- S Koulish
- S Mironescu
- S Mironescu
- S Orrenius
- S Weinhouse
- S Weinhouse
- SA Luse
- SC Skoryna
- SM Epstein
- SM Epstein
- SW Henson Jr.
- T Hultin
- T Iwasaki
- T Kitagawa
- T Kitagawa
- T Mukherjee
- T Onoé
- T Sasaki
- T Schramm
- T Takano
- T Yoshida
- T-Y Lin
- TK Shnitka
- U Pfeifer
- U Pfeiffer
- U Quensel
- U Stenram
- V Desmet
- VJ Nigam
- VM Craddok
- W Bernhard
- W Bernhard
- W Bernhard
- W Djaczenko
- W Dontenwill
- W Hunstein
- W Jacobj
- W Lauber
- W Oehlert
- W Romen
- W Romen
- W Romen
- W Stäubli
- W Thoenes
- W Thoenes
- W Thoenes
- W Wessel
- WA Butler
- WC MacCarty
- WC Schneider
- WE Criss
- WE Criss
- WH Carnes
- WL Dunn
- WP Doherty
- WS Hartroft
- Y Furuta
- Y Inoaka
- Y Mochizuki
- Z Albert
- Z Albert
- Z Hruban
- Z Hruban
- Z Hruban
- Z Hruban
- Z Hruban
- Z Hruban
- Z Hruban
- Z Schaff
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/1975
- Field of study