6 research outputs found
The NCOR-HDAC3 co-repressive complex modulates the leukemogenic potential of the transcription factor ERG
- Author
- Aqaqe Nasma
- Birger Yehudit
- Bourquin Jean-Pierre
- Chen Chun-Wei
- Drakul Aneta
- Fishman Hila
- Geron Ifat
- Izraeli Shai
- Kugler Eitan
- Liedke Elisabeth
- Liu Qiao
- Madiwale Shreyas
- Milyavsky Michael
- Ogana Heather
- Pimanda John
- Priebe Valdemar
- Privé Gilbert G
- Raught Brian
- Rein Avigail
- Schmoellerl Johannes
- Sykes David B
- Thoms Julie A I
- Yassin Muhammad
- Yong Darren
- Zuber Johannes
- Publication venue
- Nature Publishing Group
- Publication date
- 21/09/2023
- Field of study
The ERG (ETS-related gene) transcription factor is linked to various types of cancer, including leukemia. However, the specific ERG domains and co-factors contributing to leukemogenesis are poorly understood. Drug targeting a transcription factor such as ERG is challenging. Our study reveals the critical role of a conserved amino acid, proline, at position 199, located at the 3' end of the PNT (pointed) domain, in ERG's ability to induce leukemia. P199 is necessary for ERG to promote self-renewal, prevent myeloid differentiation in hematopoietic progenitor cells, and initiate leukemia in mouse models. Here we show that P199 facilitates ERG's interaction with the NCoR-HDAC3 co-repressor complex. Inhibiting HDAC3 reduces the growth of ERG-dependent leukemic and prostate cancer cells, indicating that the interaction between ERG and the NCoR-HDAC3 co-repressor complex is crucial for its oncogenic activity. Thus, targeting this interaction may offer a potential therapeutic intervention
The NCOR-HDAC3 co-repressive complex modulates the leukemogenic potential of the transcription factor ERG
- Author
- Aneta Drakul
- Avigail Rein
- Brian Raught
- Chun-Wei Chen
- Darren Yong
- David B. Sykes
- Eitan Kugler
- Elisabeth Liedke
- Gilbert G. Privé
- Heather Ogana
- Hila Fishman
- Ifat Geron
- Jean-Pierre Bourquin
- Johannes Schmoellerl
- Johannes Zuber
- John Pimanda
- Julie A. I. Thoms
- Michael Milyavsky
- Muhammad Yassin
- Nasma Aqaqe
- Qiao Liu
- Shai Izraeli
- Shreyas Madiwale
- Valdemar Priebe
- Yehudit Birger
- Publication venue
- Nature Portfolio
- Publication date
- 01/09/2023
- Field of study
Abstract The ERG (ETS-related gene) transcription factor is linked to various types of cancer, including leukemia. However, the specific ERG domains and co-factors contributing to leukemogenesis are poorly understood. Drug targeting a transcription factor such as ERG is challenging. Our study reveals the critical role of a conserved amino acid, proline, at position 199, located at the 3’ end of the PNT (pointed) domain, in ERG’s ability to induce leukemia. P199 is necessary for ERG to promote self-renewal, prevent myeloid differentiation in hematopoietic progenitor cells, and initiate leukemia in mouse models. Here we show that P199 facilitates ERG’s interaction with the NCoR-HDAC3 co-repressor complex. Inhibiting HDAC3 reduces the growth of ERG-dependent leukemic and prostate cancer cells, indicating that the interaction between ERG and the NCoR-HDAC3 co-repressor complex is crucial for its oncogenic activity. Thus, targeting this interaction may offer a potential therapeutic intervention
Modernism and the Obscene
- Author
- Adrien Muriel
- Ali Saandia
- Arnold Wayne E.
- Birgy Philippe
- Bouzonviller Elisabeth
- Bozhkova Yasna
- Camus Cyril
- Châtel Laurent
- Cuisinier-Delorme Samuel
- Doumerc Eric
- Ferraty Franck
- Fitzgerald Annelie
- Friant-Kessler Brigitte
- Georges Emilie
- Gillespie Margaret
- Gould Sarah
- Guillain Aurélie
- Hercend Olivier
- Jouve Emeline
- Keller-Privat Isabelle
- Kennedy Kevin
- Liedke Heidi Lucja
- Marie Florence
- Michiels Laura
- Montefalcone Barbara
- Sabatier Armelle
- Savatier-Lahondès Céline
- Scarpa Sébastien
- Sippel Alexandra
- Tchamitchian Raphaëlle
- Vincent-Arnaud Nathalie
- Publication venue
- 'OpenEdition'
- Publication date
- 16/10/2020
- Field of study
REESTRUTURAÇÃO PRODUTIVA NO BRASIL: UM BALANÇO CRÍTICO INTRODUTÓRIO DA PRODUÇÃO BIBLIOGRÁFICA
- Author
- ABRANCHES Sérgio
- ANTUNES Jr. José Antonio Valle
- ANTUNES Ricardo
- BALTAR Paulo E. de A.
- BALTAR Paulo E. de A.
- BRAVERMAN Harry
- BRESCIANI Luis P.
- BRESCIANI Luis P.
- BURAWOY Michael
- CACCIAMALI Maria C.
- CANO Wilson
- CARLEIAL Liana
- CARVALHO Ruy de Quadros
- CARVALHO Ruy de Quadros
- CARVALHO Ruy de Quadros
- CASTRO Maria Silvia Portella de
- CASTRO Nadya
- CASTRO Nadya Araujo
- CATANI Antonio David
- CATANI Antonio David
- CORIAT Benjamin.
- DEDECCA Claudio Salvadori
- DELGADO Maria B. Godinho
- FERNANDES Florestan
- FERRETTI Celso J.
- Ferretti Celso J.
- FERRETTI Celso. J.
- FIDALGO Fernando Selmar
- FIDALGO Fernando Selmar
- FISCHER Rosa Maria
- FLEURY Afonso
- FLEURY Afonso
- FLEURY Maria Tereza Leme
- FLEURY Paulo Fernando
- FRANZOI Naira Lisboa
- FREEMAN Richard B
- GITAHY Leda
- GITAHY Leda
- GITAHY Leda
- Gitahy Leda
- GOLDENSTEIN Gisela T
- GOUNET Thomas
- HARVEY David
- HIRATA Helena
- HIRATA Helena
- HUMPHREY John
- JOFFILY Bernardo
- KON Anita
- KONIG Helmut
- KREIN José Dari
- LARANGEIRA Sonia M.G.
- LEITE Elenice M.
- LEITE Elenice M.
- LEITE Marcia de Paula
- LEONE Eugênia Troncoso
- LIEDKE Elida R.
- LOBO Elisabeth Souza
- LOPES Juarez R. Brandão
- MACHADO Lucília R. de Souza
- MACHADO Lucília R. de Souza
- MANDEL Ernest
- MANZANO Marcelo
- MANZANO Marcelo
- MARTINS Heloisa de S
- MARX Karl
- MARX Karl
- MATTOSO Jorge.
- MATTOSO Jorge.
- MEIKSINS Peter
- MORAES NETO Benedito Rodrigues de
- MÉSZAROS István
- NEDER R.T.
- NEDER Ricardo Toledo
- NEVES Magda de Almeida
- NEVES Magda de Almeida
- OLIVEIRA Carlos A.B.
- OLIVEIRA Marco Antonio de
- Paulo Sergio Tumolo
- PELIANO José Carlos
- PINHEIRO Ivan A .
- PIRES Elson L. Silva
- POCHMANN Marcio
- PORTUGAL Marcelo
- POSTHUMA Anne
- QUADROS Waldir José
- RAMALHO José Ricardo
- RATTNER Henrique
- REIS H. L.
- RIZEK Cibele S.
- RODRIGUES Iram Jácome
- ROSA Cláudio Porto da
- RUAS Roberto
- RUBIN Isaak Illich
- SALERNO Mário Sérgio
- SALERNO Mário Sérgio
- SALERNO Mário Sérgio
- SALM Claudio
- SALM Claudio
- SALM Claudio
- SANTOS Anselmo L. dos
- SANTOS Anselmo L. dos
- SILVA Elizabeth Bortolaia
- TUMOLO Paulo Sérgio
- TUMOLO Paulo Sérgio
- TUMOLO Paulo Sérgio
- VIDAL Manuel Cereceda
- WACHENDORFER Achim
- Publication venue
- 'FapUNIFESP (SciELO)'
- Publication date
- Field of study
Literatur
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- Pöhlmann Markus
- Rauchensteiner Manfried
- Rauchensteiner Manfried
- Reemtsma Jan Philipp
- Regele Oskar
- Rehbein Saalmann
- Reicher Dieter
- Remarque Erich Maria
- Riedl Joachim
- Rieks Rudolf
- Rosenstiel
- Rosenwein Barbara
- Rosenwein Barbara
- Roth Joseph
- Rothenberg Gunther E
- Rothenberg Gunther E
- Saar
- Safranski Rüdiger
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- Simmel Georg
- Simmel Georg
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- Sked Alan
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- Smith Anthony D
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- Uhl Heidemarie
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- Voranc Kuhar
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- ür Landesverteidigung
- Publication venue
- 'Vandenhoeck & Ruprecht GmbH & Co, KG'
- Publication date
- Field of study
Literatur
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- Proust Marcel
- Pçrksen Uwe
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