188 research outputs found
Metformin inhibits melanoma development through autophagy and apoptosis mechanisms
- Author
- A Decensi
- A Kalender
- AJ Meijer
- B Liu
- B Zheng
- CJ Bailey
- D Alonso-Curbelo
- D Tormo
- DJ Klionsky
- DM Smith
- E Morselli
- F Scarlatti
- F Scarlatti
- G Robert
- G Sarrabayrouse
- G Zhou
- HS Hundal
- I Ben Sahra
- I Ben Sahra
- I Ben Sahra
- J Woodard
- JD Lalau
- JT Zilfou
- K Hosono
- K Janjetovic
- L Larribere
- LW Wang
- M Buzzai
- M Pollak
- M Stumvoll
- MC Maiuri
- MC Maiuri
- MF Demierre
- P Colosetti
- P Gao
- R Rattan
- RG Jones
- S Conus
- T Botton
- T Botton
- Publication venue
- Nature Publishing Group
- Publication date
- Field of study
Metformin is the most widely used antidiabetic drug because of its proven efficacy and limited secondary effects. Interestingly, recent studies have reported that metformin can block the growth of different tumor types. Here, we show that metformin exerts antiproliferative effects on melanoma cells, whereas normal human melanocytes are resistant to these metformin-induced effects. To better understand the basis of this antiproliferative effect of metformin in melanoma, we characterized the sequence of events underlying metformin action. We showed that 24 h metformin treatment induced a cell cycle arrest in G0/G1 phases, while after 72 h, melanoma cells underwent autophagy as demonstrated by electron microscopy, immunochemistry, and by quantification of the autolysosome-associated LC3 and Beclin1 proteins. In addition, 96 h post metformin treatment we observed robust apoptosis of melanoma cells. Interestingly, inhibition of autophagy by knocking down LC3 or ATG5 decreased the extent of apoptosis, and suppressed the antiproliferative effect of metformin on melanoma cells, suggesting that apoptosis is a consequence of autophagy. The relevance of these observations were confirmed in vivo, as we showed that metformin treatment impaired the melanoma tumor growth in mice, and induced autophagy and apoptosis markers. Taken together, our data suggest that metformin has an important impact on melanoma growth, and may therefore be beneficial in patients with melanoma
A chemical biology screen reveals a role for Rab21-mediated control of actomyosin contractility in fibroblast-driven cancer invasion
- Author
- A Yuge
- AD Dubash
- AS Meshel
- C Gaggioli
- C Gaggioli
- C Laezza
- E Sahai
- EC Brockbank
- F Grinnell
- J Riedl
- JP Burke
- K Walker
- M Egeblad
- M Honjo
- MC Jones
- MF Demierre
- MF Olson
- N Werner
- P Friedl
- P Ngo
- R Ghittoni
- S Hooper
- S Huveneers
- S Pinner
- SA Holstein
- SA Holstein
- T Kusama
- T Meyer-Ter-Vehn
- T Pellinen
- T Pellinen
- T Pellinen
- TJ Murtola
- XD Ren
- Y Liu
- Publication venue
- Nature Publishing Group
- Publication date
- Field of study
Virtual pathway explorer (viPEr) and pathway enrichment analysis tool (PEANuT): creating and analyzing focus networks to identify cross-talk between molecules and pathways
- Author
- A Corsini
- A Kamburov
- A Leszczynska
- A Schröder
- AL Mammen
- B Paulweber
- Benjamin A. Kandel
- Bianca Hermine Habermann
- C Rodríguez-Antona
- CF Schaefer
- DS King
- DW Huang
- E Cerami
- EG Cerami
- EW Dijkstra
- Falko Hofmann
- G Bebek
- G Joshi-Tope
- G Vemana
- H Ceelie
- H Tatewaki
- H-Y Lee
- J Shimada
- J Supper
- JR Friedman
- JW Clendening
- JW Jukema
- K Howe
- KM Swanson
- L Ekström
- L Song
- LD Stein
- LJ Jensen
- LN Griner
- M Ashburner
- M Hafner
- M Kanehisa
- M Kuhn
- M Merli
- M Moya
- M-F Demierre
- Maria Thomas
- Marius Garmhausen
- MB Eisen
- MP Iersel van
- MS Katz
- MW Medina
- NCBI Resource Coordinators
- OJ Dunn
- P Convertini
- R Rodrigues Díez
- SE Moody
- TJ Antes
- TJ Murtola
- V Bombail
- VI Zannis
- Viktor Senderov
- WG Wood
- WikiPathways
- WWL Wong
- Y Benjamini
- Y Ohoka
- Y-H Cheng
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/2015
- Field of study
BACKGROUND: Interpreting large-scale studies from microarrays or next-generation sequencing for further experimental testing remains one of the major challenges in quantitative biology. Combining expression with physical or genetic interaction data has already been successfully applied to enhance knowledge from all types of high-throughput studies. Yet, toolboxes for navigating and understanding even small gene or protein networks are poorly developed. RESULTS: We introduce two Cytoscape plug-ins, which support the generation and interpretation of experiment-based interaction networks. The virtual pathway explorer viPEr creates so-called focus networks by joining a list of experimentally determined genes with the interactome of a specific organism. viPEr calculates all paths between two or more user-selected nodes, or explores the neighborhood of a single selected node. Numerical values from expression studies assigned to the nodes serve to score identified paths. The pathway enrichment analysis tool PEANuT annotates networks with pathway information from various sources and calculates enriched pathways between a focus and a background network. Using time series expression data of atorvastatin treated primary hepatocytes from six patients, we demonstrate the handling and applicability of viPEr and PEANuT. Based on our investigations using viPEr and PEANuT, we suggest a role of the FoxA1/A2/A3 transcriptional network in the cellular response to atorvastatin treatment. Moreover, we find an enrichment of metabolic and cancer pathways in the Fox transcriptional network and demonstrate a patient-specific reaction to the drug. CONCLUSIONS: The Cytoscape plug-in viPEr integrates –omics data with interactome data. It supports the interpretation and navigation of large-scale datasets by creating focus networks, facilitating mechanistic predictions from –omics studies. PEANuT provides an up-front method to identify underlying biological principles by calculating enriched pathways in focus networks. ELECTRONIC SUPPLEMENTARY MATERIAL: The online version of this article (doi:10.1186/s12864-015-2017-z) contains supplementary material, which is available to authorized users
The pp elastic scattering analyzing power measured with the polarized beam and the unpolarized target between 1.98 and 2.80 GeV
- Author
- Allgower C E.
- Ball J.
- Beddo M.
- Bedfer Y.
- Boutefnouchet A.
- Bystricky J.
- Chamouard P A.
- de Lesquen A.
- Demierre P.
- Fontaine J M.
- Ghazikhanian V.
- Grosnick D.
- Hess R.
- Janout Z.
- Kalinnikov V A.
- Kasprzyk T E.
- Khachaturov B A.
- Kunne R.
- Lehar F.
- Lopiano D.
- Matafonov V N.
- Pisarev I L.
- Popov a A.
- Prokofiev a N.
- Rapin D.
- Sans J L.
- Spinka H M.
- Teglia A.
- Usov Yu A.
- Vikhrov V V.
- Vuaridel B.
- Whitten C A.
- Zhdanov a A.
- Publication venue
- 'Elsevier BV'
- Publication date
- 01/01/1998
- Field of study
Iron Behaving Badly: Inappropriate Iron Chelation as a Major Contributor to the Aetiology of Vascular and Other Progressive Inflammatory and Degenerative Diseases
- Author
- A Abbott
- A Abou-Raya
- A Aljandali
- A Ambesi-Impiombato
- A Aydin
- A Balcerczyk
- A Besarab
- A Brzezinski
- A Campbell
- A Carrillo-Vico
- A Cavalli
- A Chattopadhyay
- A Chattopadhyay
- A Cherubini
- A Dey
- A Doms
- A Donovan
- A Donovan
- A Dávalos
- A Gaeta
- A Garny
- A Gnjec
- A Gomes
- A Gopalakrishnan
- A Hald
- A Henney
- A Hirayama
- A Hoffmann
- A Huber
- A Hugman
- A Iannetti
- A Ide-Ektessabi
- A Jacobs
- A Jeyabalan
- A Kahvejian
- A Karrar
- A Kasztler
- A Kibel
- A Kocyigit
- A Kotha
- A Kumral
- A Lass
- A Lecube
- A Lewén
- A Lotery
- A Maggio
- A Malek
- A Malik
- A Mantovani
- A Matsuzawa
- A Mitra
- A Monge
- A Murakami
- A Murakami
- A Murakami
- A Murakami
- A Mutti
- A Nijnik
- A Nunomura
- A Nunomura
- A Patt
- A Persson
- A Pietrangelo
- A Piga
- A Pirat
- A Post
- A Pradhan
- A Protti
- A Rattner
- A Ravati
- A Rehman
- A Reynolds
- A Richmond
- A Roetto
- A Roetto
- A Rostom
- A Rumbold
- A Russo
- A Rötig
- A Saltelli
- A Saltelli
- A Sandek
- A Sassano
- A Scalbert
- A Scalbert
- A Scalbert
- A Sica
- A Smahi
- A Sola
- A Stintzi
- A Szewczyk
- A Taguchi
- A Tedgui
- A Terman
- A Terman
- A Terman
- A Undas
- A Virdis
- A Wagner
- A Wagner
- A Wagner
- A Wagner
- A Wojas-Pelc
- A Wong
- A Xu
- A Yoritaka
- A Yoshimura
- A-L Barabási
- AA Andreadis
- AA Borisy
- AA Farooqui
- AA Qutub
- AA Qutub
- AA Vlessis
- AB Nathens
- AB Parsons
- AB Parsons
- AB Thompson
- AB Thomson
- AC Bayne
- AC Bharti
- AC Cave
- AC Mello Filho
- AD d'Hardemare
- AD de Silva
- Ad hoc committee on systemic lupus erythematosus response criteria for fatigue
- ADL van der
- AE Aust
- AE Baue
- AE Finefrock
- AE Heazell
- AE Heazell
- AE Kartikasari
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- AF Tramontano
- AH Berg
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- AH Tong
- AI Bush
- AI Bush
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- AJ Ghio
- AJ Ghio
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- AJ Hulbert
- AJ Kowaltowski
- AJ Lusis
- AJ Matthews
- AJ Reyes
- AJ van Oostrom
- AJ Watson
- AJ White
- AJ Williams
- AK Junk
- AL Beal
- AL Hemdahl
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- AL Sirén
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- AT McKie
- AV Lebedev
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- AY Andreyev
- AY Sun
- B Chakravarti
- B Chance
- B Cronin
- B de Valk
- B De Vries
- B Desoize
- B Drayer
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- B Goodell
- B Halliwell
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- B Shipley
- B Skibska
- B Sturm
- B Thorand
- B Wang
- B Wolff
- B Wolozin
- B Wolozin
- B Xu
- B Zhang
- B Zhou
- BA Maddux
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- BB Aggarwal
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- C Arnaud
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- C Finch
- C Fleury
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- C Gasche
- C Gasche
- C Gerhäuser
- C Goble
- C Henry
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- C Herder
- C Hershko
- C Hershko
- C Hershko
- C Hershko
- C Jacob
- C Kenyon
- C Knox
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- C Li
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- SY Qian
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- SZ Xu
- T Amit
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- T Finkel
- T Finkel
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- T Ganz
- T Ganz
- T Ganz
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- TG Kazi
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- The Long-Term Intervention with Pravastatin in Ischaemic Disease (LIPID) Study Group
- TJ Gibson
- TJ Shah
- TK Kvien
- TL Duarte
- TL Nickolas
- TM Dawson
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- TO Scholl
- TO Scholl
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- U Eckstein-Ludwig
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- UN Das
- V Adam-Vizi
- V Adam-Vizi
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- V Braun
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- V Campuzano
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- V Irazusta
- V Irazusta
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- X Chen
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- X Huang
- X Huang
- X Li
- X Zhang
- X Zhu
- X Zhu
- XD Huang
- XJ Li
- XM Yuan
- XM Yuan
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- Y Almog
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- Y Bao
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- Y Takada
- Y Wang
- Y Wang
- Y Wei
- Y Wei
- Y Wu
- Y Wu
- Y Zhang
- Y Zhang
- Y Zhang
- Y Zhao
- Y Zheng
- YE Henrotin
- YF Chu
- YH Lee
- YH Suh
- YH Wei
- YJ Surh
- YJ Surh
- YJ Surh
- YK Wu
- YM Kim
- YS Keum
- YS Sohn
- YX Ma
- YZ Fang
- Z Cai
- Z Cai
- Z Cheng
- Z Pei
- Z Serdar
- Z Tong
- Z Tong
- Z Yu
- Z Zhang
- ZD Liu
- ZD Liu
- ZE Karanjawala
- ZE Suntres
- ZI Cabantchik
- ZZ Chong
- ZZ Chong
- Publication venue
- Publication date
- 09/08/2008
- Field of study
The production of peroxide and superoxide is an inevitable consequence of
aerobic metabolism, and while these particular "reactive oxygen species" (ROSs)
can exhibit a number of biological effects, they are not of themselves
excessively reactive and thus they are not especially damaging at physiological
concentrations. However, their reactions with poorly liganded iron species can
lead to the catalytic production of the very reactive and dangerous hydroxyl
radical, which is exceptionally damaging, and a major cause of chronic
inflammation. We review the considerable and wide-ranging evidence for the
involvement of this combination of (su)peroxide and poorly liganded iron in a
large number of physiological and indeed pathological processes and
inflammatory disorders, especially those involving the progressive degradation
of cellular and organismal performance. These diseases share a great many
similarities and thus might be considered to have a common cause (i.e.
iron-catalysed free radical and especially hydroxyl radical generation). The
studies reviewed include those focused on a series of cardiovascular, metabolic
and neurological diseases, where iron can be found at the sites of plaques and
lesions, as well as studies showing the significance of iron to aging and
longevity. The effective chelation of iron by natural or synthetic ligands is
thus of major physiological (and potentially therapeutic) importance. As
systems properties, we need to recognise that physiological observables have
multiple molecular causes, and studying them in isolation leads to inconsistent
patterns of apparent causality when it is the simultaneous combination of
multiple factors that is responsible. This explains, for instance, the
decidedly mixed effects of antioxidants that have been observed, etc...Comment: 159 pages, including 9 Figs and 2184 reference
Off-chip passivated-electrode, insulator-based dielectrophoresis (OπDEP)
- Author
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Statin-induced anti-proliferative effects via cyclin D1 and p27 in a window-of-opportunity breast cancer trial
- Author
- A Arnold
- A Mohammed
- A Wachtershauser
- B Glimelius
- B Lebe
- B Relja
- C Gomez-Fernandez
- DO Morgan
- Dorthe Grabau
- E Luporsi
- EA Musgrove
- ER Garwood
- ER Nelson
- ER Nelson
- F Lopez
- FL Zhang
- FY Wu
- HB El-Serag
- IM Chu
- Ingrid Hedenfalk
- J Kuoppala
- J Massague
- JB Park
- JF Robertson
- JK Liao
- JL Goldstein
- JN Lavoie
- JW Clendening
- K Keyomarsi
- Karin Jirström
- KM Dale
- LM McShane
- M Cimino
- M Malumbres
- Maria Feldt
- MF Buckley
- MF Demierre
- MJ Campbell
- ML Coleman
- N Ishida
- NL Barbosa-Morais
- O Bjarnadottir
- Olöf Bjarnadottir
- P Desai
- Pär-Ola Bendahl
- Q Zhou
- RA Irizarry
- S Bellosta
- SF Nielsen
- Signe Borgquist
- Siker Kimbung
- Srinivas Veerla
- SW Blain
- TJ Murtola
- TP Ahern
- TP Ahern
- V Baldin
- WB Zhong
- X Chen
- X Guan
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
ATLAS detector and physics performance: Technical Design Report, 1
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- van der Graaf H.
- van Eijk B.
- Van Hille H.
- Vanickova M.
- Vanini S.
- Vanko J.
- Vanyashin A.
- Varanda M.
- Vartapetian A.
- Vassilieva L.
- Vassiliou M.
- Vazeille F.
- Vegni G.
- Veillet J-J.
- Velikzhanin Y.
- Veneziano S.
- Vercesi V.
- Vermeulen J.C.
- Vernay E.
- Vertogradov L.
- Vichou I.
- Vigeolas E.
- Vincke H.
- Vinogradov V.
- Virchaux M.
- Volpini G.
- von Boehn-Bucholz R.
- Vorobiev A.P.
- Vorozhtsov S.
- Voss R.
- Vovenko A.S.
- Vrba V.
- Vreeswijk M.
- Vuandel B.
- Vuillemin V.
- Wadsworth B.F.
- Wagner R.G.
- Wahlen H.
- Waldner F.
- Walkowiak W.
- Wampler L.
- Wang C.
- Wang C.H.
- Wappler F.
- Wastie R.L.
- Watase Y.
- Watkins P.M.
- Watson A.T.
- Watson N.K.
- Weaverdyck C.
- Webel M.
- Weber C.
- Webster A.
- Weerts H.
- Weichert J.
- Weidberg A.R.
- Weilhammer P.
- Wellenstein H.
- Wells D.
- Wermes N.
- Werneke P.
- Werner P.
- Wheeler S.
- Whitaker J.S.
- White A.
- White D.J.
- Wickens F.J.
- Wicklund A.B.
- Wielers M.
- Wijnen Th.A.M.
- Wilhelm I.
- Williams H.H.
- Willis S.E.
- Willis W.
- Wilson J.A.
- Wingerter-Seez I.
- Witzeling W.
- Wolter M.
- Wolters H.
- Wotschack J.
- Woudstra M.
- Wu H.
- Wu S.L.
- Wu X.
- Wuestenfeld J.
- Wunsch M.
- Wunstorf R.
- Wyllie K.H.
- Xie Y.G.
- Xu G.F.
- Xue L.
- Yakimenko M.
- Yamamoto A.
- Yamartino J.M.
- Yamdagni N.
- Yanagisawa C.
- Yang B.
- Yang T.
- Yarygin G.
- Yasu Y.
- Ye B.
- Ye J.
- Yoshida H.
- Yoshida R.
- Yu B.
- Yu X.Q.
- Zaets V.G.
- Zaitsev A.M.
- Zaitsev V.
- Zalite A.
- Zamani M.
- Zamora Y.
- Zanello L.
- Zdrazil M.
- Zeitnitz C.
- Zeldovich S.
- Zerwas D.
- Zhang B.
- Zhang L.
- Zhang N.
- Zhang Q.J.
- Zhao J.
- Zhao T.
- Zhichao L.
- Zhou B.
- Zhou B.
- Zhuravlev V.
- Zimin S.
- Ziolkowski M.
- Zitek K.
- Zitoun R.
- Zmouchhko V.
- Zobernig G.
- Zolnierowski Y.
- Zontar D.
- Zuffranieri F.
- Zuk G.
- Zverev E.G.
- Fasssouliotis D.
- Publication venue
- Union of Concerned Scientists
- Publication date
- 01/01/1999
- Field of study
Repurposing of approved cardiovascular drugs
- Author
- A González-Pérez
- A Izadpanah
- AE Buhl
- AE Durazzo
- AF Lever
- AH Otake
- AH Wagner
- AK Sood
- AK Sood
- AM Algra
- ARB Trialists Collaboration
- B Bernard
- B Pasternak
- B Stenkvist
- B Stenkvist
- B Stenkvist
- B Vandewalle
- BL Devine
- BS Brooke
- BS Rao
- C Bosetti
- C Denoyelle
- C Espineda
- C Leaute-Labreze
- C Leaute-Labreze
- C Léauté-Labrèze
- C Pees
- C Quintavalle
- CH Choi
- CR Meier
- D Bansal
- D Herr
- D Jacobs
- D Sardana
- D Spiegel
- D Spiegel
- D Westaby
- DA Goldfarb
- DG Powe
- DL Weddle
- E Flossmann
- EA Olsen
- EA Platz
- EK Sloan
- ES Diaz
- EV Yang
- F Elefteriou
- F Gueler
- G Garcia-Tsao
- G Ronquist
- G Zang
- GA Kune
- GJ Gasic
- H Desai
- H Graf
- HC Diener
- HC Dietz
- HC Dietz
- HH Grytli
- HJ Song
- HM Wang
- I Sipahi
- J Avila
- J Bertrand
- J Bosch
- J Bukberg
- J Gribbin
- J Haux
- J Shao
- J Springer
- J Tumlin
- J-Q Chen
- JH Neo
- JJ Kolenich
- JL Roberts
- Jochen Springer
- JP Fryzek
- JP Habashi
- JR Emberson
- Junichi Ishida
- K Bielawski
- K Hindler
- K Masur
- K Okamoto
- KA Toulis
- L Blais
- LA Fleisher
- LA Lipsitz
- LH Lindholm
- LL Gluud
- M Groenink
- M Hogeling
- M Leoncini
- M Nesher
- M Tan
- M Thiele
- M-F Demierre
- Masaaki Konishi
- ME Lindsay
- MJ Thun
- MR Graaf
- MT Ruffin
- N Kawazoe
- Nicole Ebner
- O Shiratori
- OO Ogunwobi
- P Ducy
- P Hillon
- PA Ganz
- PB Raghavendra
- PC Elwood
- PH Thaker
- PK Lindenauer
- PM Ridker
- PM Rothwell
- PM Rothwell
- PM Rothwell
- Q Zhou
- R Anandanadesan
- R Franchis de
- R Yasumatsu
- RC Wester
- RE Moore
- RJ Biggar
- RJ Biggar
- RJ Groszmann
- RV Lacro
- S Friis
- S John
- S Kang
- S Lachgar
- S Lemeshow
- S Marsigliante
- S Pugh
- S Singh
- S Takeda
- S Yang
- SA Rajasekaran
- SD Silberstein
- SK Manna
- SM Kornblau
- T Poynard
- T Serste
- T Sjoberg
- T Suganuma
- TG Kreindler
- TI Barron
- TL Assimes
- TP Ahern
- V Sans
- VH Price
- W Schoner
- WC Lau
- WK Wu
- WL Smith
- X Li
- X-D Wu
- Y Chida
- Y Fujimoto
- Y Li
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Primary cutaneous marginal zone B-cell lymphoma in a patient with chronic lymphocytic leukaemia
- Author
- Publication venue
- 'Wiley'
- Publication date
- Field of study
- …