6 research outputs found
First Evaluation of [11C]R116301 as an In Vivo Tracer of NK1 Receptors in Man
- Author
- AA Megens
- Adriaan A. Lammertsma
- Albert D. Windhorst
- Anu J. Airaksinen
- Bart N. M. van Berckel
- BE Francis
- C Felipe De
- C Griffante
- CJ Hoekstra
- CSJ Walpole
- Dick J. Veltman
- E Livni
- F Maes
- G Brix
- J Hietala
- J West
- JM Kent
- Josée E. Leysen
- Kaoru Maruyama
- KRR Krishnan
- L Quartara
- L Quartara
- M Bergstrom
- M Bergstrom
- M Defrise
- M Keller
- M Mey Van der
- M Otsuka
- Mark Lubberink
- MB First
- MJ Nyman
- MJG Farthing
- MS Kramer
- NM Rupniak
- O Solin
- PJ Hesketh
- R Boellaard
- R Hargreaves
- R Hosoki
- RB Delrosario
- Ronald Boellaard
- Saskia P. A. Wolfensberger
- TM Dando
- WAP Breeman
- Wieb Reddingius
- William D. H. Carey
- YY Zhang
- Publication venue
- Springer-Verlag
- Publication date
- 01/01/2009
- Field of study
PURPOSE: NK1 receptors have been implicated in various neuropsychiatric and other disorders. R116301 is a selective NK1 receptor antagonist. In this pilot study, [(11)C]R116301 was evaluated as a potential positron emission tomography (PET) ligand for the NK1 receptor. PROCEDURES: Two dynamic PET studies were performed in three normal volunteers before and after a blocking dose of aprepitant. Data were analyzed using striatum to cerebellum standardized uptake value (SUV) ratios. RESULTS: Baseline SUV ratios at 60-90 min after injection ranged from 1.22 to 1.70. Following aprepitant administration, this specific signal was completely blocked. Aprepitant administration did not significantly affect uptake in cerebellum, confirming the absence of NK1 receptors in cerebellum. CONCLUSION: These preliminary results indicate that [(11)C]R116301 has potential as a radioligand for in vivo assessment of NK1 receptors in the human brai
RPF151, a novel capsaicin-like analogue: in vitro studies and in vivo preclinical antitumor evaluation in a breast cancer model
- Author
- A Gavezzotti
- A Szallasi
- AD Becke
- Adilson Kleber Ferreira
- AK Joe
- AL Gartel
- AM Sánchez
- AP Gilmore
- Ariane Matiello Bertin
- BR Blank
- C Amantini
- C-C Wu
- C-H Lin
- Carlos Rogério Figueiredo
- CM Breneman
- CSJ Walpole
- CSJ Walpole
- CSJ Walpole
- D Doherty
- DG Stupack
- DL Vaux
- F FaiĂŁo-Flores
- FE Koehn
- G Zeng
- GA Patani
- GI Evan
- GM Almeida
- GP Dotto
- H Akl
- H-F Lu
- H-M Wang
- H-S Jun
- HN BrandĂŁo
- IB Roninson
- IR Bukholm
- J Chow
- J Lee
- J Singh
- J-A Kim
- JE Meredith
- José Alexandre Marzagão Barbuto
- JY Kim
- K Ito
- K-L Lin
- Kerly Fernanda Mesquita Pasqualoto
- KH Forsythe
- M Zimmermann
- M-J Lee
- M-J Ludy
- Mariana Celestina Frojuello Costa B DamiĂŁo
- MaurĂcio Temotheo Tavares
- MC Guadamillas
- MCFCB DamiĂŁo
- ME Saez
- MJ Caterina
- MJ Caterina
- MJ Frisch
- MJ Reginato
- MJS Dewar
- ML Matter
- MY Jung
- N Bodor
- N Carragher
- P Bouillet
- P Sanphui
- Paulo Luiz de-Sá-Junior
- PL De-Sá-Júnior
- R Maity
- R Michalides
- RA Woo
- Ricardo Alexandre de Azevedo
- Roberto Parise-Filho
- S Fulda
- S Kim
- S Oikawa
- Sarah Fernandes Teixeira
- SH Oh
- SM Frisch
- SM Frisch
- SV Ekholm
- T Gurung
- T Takahashi
- VN Viswanadhan
- W Pendergrass
- Wilson Alves Ferreira-Junior
- X Deng
- Y Chai
- Y-H Yu
- Y-J Surh
- Y-L Huang
- Yara Cury
- Z Zhang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Peripheral Mediators of Pain
- Author
- A Czlonkowski
- A Dray
- A Dray
- A Dray
- A Dray
- A Dray
- A Dray
- A Dray
- A Dray
- A Mitchell
- A Rueff
- A Rueff
- A Szallasi
- AH Dickenson
- AJ Davis
- AJ Fox
- AN Akopian
- AN Akopian
- B Safieh-Garabedian
- BJ Undem
- BP Richardson
- C Bradley
- C Lewis
- C Stein
- C-C Chen
- CA Maggi
- CG Heapy
- CJ Woolf
- CM Gammon
- CSJ Walpole
- CW Tiffany
- D Weinreich
- DA Simone
- DL Tanelian
- DS McGehee
- DS Ragsdale
- E Kostyuk
- EM McLachlan
- F Marceau
- FQ Cunha
- FQ Cunha
- GD Nicol
- GJ Birrell
- GJ Keil
- GM Burgess
- GM Burgess
- GM Jonakait
- GR Lewin
- GR Seabrook
- H Holthusen
- H-G Scheible
- H-G Scheible
- HA Wieland
- HP Rang
- I Nagy
- IF James
- J Donnerer
- J Olesen
- J Sato
- J Szolcsányi
- J Winter
- J Winter
- J-C Meunier
- JC Lee
- JD Levine
- JG Menke
- JJ Toledo-Aral
- JM Hall
- JM Zhang
- JR Schwarz
- K Schepelmann
- K Seibert
- K-F Shen
- KD Bhoola
- KD Davis
- KD Davis
- KH Steen
- LG Aguayo
- LL Brand
- M Devor
- M Devor
- M Devor
- M Kurosawa
- M Malcangio
- M Petersen
- M Schmelz
- M Schäfer
- MA Moskowitz
- MC Crain
- MG Buzzi
- MN Perkins
- MN Perkins
- MS Gold
- N Andreev
- NN Ninkina
- O Matzner
- P Crunkhorn
- P Marchettini
- P Santicioli
- P Wei
- PJ Birch
- PPA Humphrey
- PR Elford
- PW Beck
- PW Mantyh
- R Karlsten
- R-D Treede
- RA Coleman
- RK Reinscheid
- RM Burch
- RR Steranka
- S Bevan
- S Bevan
- S Bevan
- S Boyce
- S Markowitz
- S Mense
- S Todorovic
- SB McMahon
- SC Cruwys
- SG Khasar
- SG Waxman
- SH Ferreira
- SH Kim
- SJ Bevan
- SM Moussaoui
- ST Meller
- SWN Thompson
- T Bleehan
- VMK Verge
- W Janig
- W-H Xiao
- WF Colmers
- X Zhang
- Y-P Lou
- YO Taiwo
- YO Taiwo
- YO Taiwo
- YO Taiwo
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/1997
- Field of study
Immune aspects of the bi-directional neuroimmune facilitator TRPV1
- Author
- A Jara-Oseguera
- A Liapi
- A Parenti
- A Perálvarez-MarĂn
- A Ray
- A SolĂs-LĂłpez
- AA Chora
- AG Szöllősi
- AJ Schain
- AM Bode
- B Liu
- BI TĂłth
- BJ Wainger
- BM Assas
- BU Schraml
- C Amantini
- C Goswami
- C Nathan
- CI Saunders
- CKY Cheung
- CSJ Walpole
- D Zhang
- DJ Cavanaugh
- E Nevius
- EM Singer
- ES Fernandes
- F Cevikbas
- F Nicoletti
- F Tsuji
- F Yang
- FN McNamara
- G Santoni
- G Shimosato
- H Zhang
- HE Gibson
- HS Kim
- I Devesa
- I Heiner
- I Heiner
- I Nikolic
- IM Hdud
- IV Duzen
- J Zhao
- JC Roberts
- JH Nam
- JP Lai
- K Magierowska
- K Shibasaki
- K Shibasaki
- K Stock
- K Venkatachalam
- K Yamashiro
- KS Park
- KW Ho
- M Entin-Meer
- M Entin-Meer
- M LĂ©vĂŞque
- M Mohammed
- M Murai
- M Nagasawa
- M-F Tsou
- MJ Caterina
- MW Doyle
- N Mikami
- P Fagone
- P Fagone
- P Fagone
- P Járomi
- PB Yaffe
- Puneet Gupta
- R Amachi
- R Marsch
- R Rehman
- R Samivel
- R Simeoli
- RK Majhi
- RS Boyd
- S Basu
- S Bertin
- S Bertin
- S Bertin
- S Caprodossi
- S Earley
- S Hassan
- S Marinelli
- S Rochlitzer
- S Talbot
- S Voedisch
- SA Omari
- SB Mazzone
- SE Wang
- T Miyake
- T Rodrigues
- TM Link
- TTL Wu
- TW Bailey
- X Zhen
- Y Dai
- Y Ninomiya
- Y Takayama
- Yan-Ruide Li
- YV Medvedeva
- Z Helyes
- É Borbély
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
The vanilloid receptor TRPV1: 10 years from channel cloning to antagonist proof-of-concept
- Author
- A Apostolidis
- A Apostolidis
- A Avelino
- A Babes
- A Dhaka
- A Hinman
- A Khachatryan
- A Mizuno
- A Moqrich
- A Sculptoreanu
- A Szallasi
- A Szallasi
- A Szallasi
- A Szallasi
- A Szallasi
- A Weil
- AB Malmberg
- AD Guler
- AJ Culshaw
- AM Patwardhan
- AM Peier
- AM Peier
- Arpad Szallasi
- B Ahren
- B Issekutz
- B Smith
- B Veronesi
- C Gennari
- Charles A. Blum
- CL Chan
- CSJ Walpole
- Daniel N. Cortright
- DC Immke
- DD McKemy
- DM Bautista
- DM Bautista
- DM Johnson
- DM Swanson
- DM Wu
- DP Mohapatra
- E Cuypers
- E Guillot
- E Mezey
- EC Wick
- G Bhave
- G Kallner
- G Lauria
- G Lu
- G MĂłzsik
- G Reid
- G Shimosato
- G Wang
- GD Smith
- GM Story
- GP Ahern
- H Katsura
- H Lee
- H Todaka
- H Watanabe
- H Xu
- HH Chuang
- HK Rami
- HL Pan
- HW Steenland
- HZ Hu
- I Fristad
- I Gatti
- I Marquez-Rodas
- I Vetter
- J Jung
- J Shin
- J Siemens
- J Szolcsányi
- J Szolcsányi
- J Vriens
- JB Davis
- JD Pomonis
- JE Keeble
- JE Krause
- JE Mitchell
- JF Sanchez
- JG Collier
- JJ Van Buren
- JR Ghilardi
- K Dai
- K Kobayashi
- K Talavera
- K Tousova
- KF Chung
- KG Sutton
- KJ Velanzano
- KM Walker
- KY Kwan
- L Klionsky
- L Liu
- L Negri
- L Wang
- LA Birder
- LJ Hudson
- LJ Macpherson
- LS Premkumar
- M Bandell
- M Belvisi
- M Cui
- M Dux
- M Hautkappe
- M McLeod
- M Numazaki
- M Numazaki
- M Pettersson
- M Suzuki
- M Suzuki
- M Tominaga
- M Tominaga
- M Trevisani
- MA Schumacher
- MD Dogan
- MH Rashid
- MH Rashid
- MJ Carr
- MJ Caterina
- MJ Caterina
- MJ Caterina
- MJ Gunthorpe
- MK Chung
- MM Hutter
- MR Zahner
- N Alessandri-Haber
- N Alessandri-Haber
- N Gavva
- N Sekiguchi
- NJ Barton
- NJ Gavva
- P Cesare
- P Dinis
- P Geppetti
- P Geppetti
- P Geppetti
- P Gopinath
- P Holzer
- P Holzer
- P Honore
- P Pacher
- P Tympanidis
- PJ Goadsby
- PJ Matthews
- PM Zygmunt
- Q Xue
- QP Ma
- R Marsch
- R Planells-Cases
- R Razavi
- R Sharif Naeini
- RC Jones
- RE Kouhen
- RJ Docherty
- S Akerman
- S Amadesi
- S Brauchi
- S Horie
- S Marinelli
- Samer R. Eid
- SE Jordt
- SE Jordt
- SE Jordt
- SF van de Graaf
- SG Moesgaard
- SM Huang
- SR Kim
- SW Hwang
- T Iida
- T Moriyama
- T Sano
- T Togashi
- TD Wilson-Gerwing
- U Binzen
- UG Lalloo
- VI Ognyanov
- W Chai
- W Liedtke
- W Tian
- XZ Xu
- Y Akiba
- Y Wang
- Y Wang
- Y Yiangou
- Z Zhang
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study
Anti-inflammatory Activity
- Author
- A Ahluwalia
- A Akeson
- A Alfieri
- A Blackham
- A Boris
- A Cabrero
- A Castrillo
- A Colorado
- A Crummey
- A Daniel
- A Ferrante
- A Golebiowski
- A GraneĂź
- A Hedberg
- A Lee
- A Mortellaro
- A Nagahisa
- A Naya
- A Nencioni
- A Pouleau
- A Robert
- A Rubino
- A Sabatino Di
- A Saria
- A Tanaka
- A Tomlinson
- A Tubaro
- A Zlotnik
- AA Miles
- AB Dietz
- AC Castro
- AC Issekutz
- AC Lennard
- AD Fryer
- AD Medhurst
- AE McEachern
- AEI Proudfoot
- AJ Bennett
- AJ Lewis
- AJ Miller
- AK Roshak
- AKW Tse
- AL Akeson
- AL Willis
- AM Wolf
- Anonymous
- AP Alexenko
- AP Alexenko
- AP Roszkowski
- AR Renzetti
- AS Kalgutkar
- AT Evans
- AW Ford-Hutchinson
- AW Yem
- B Beutler
- B Dubinsky
- B Goffe
- B Jarvis
- B Kaltschmidt
- B Moser
- B Rudas
- B Samuelsson
- B Sander
- B Sander
- BA Jakschik
- BA Whittle
- BB Aggarwal
- BB Aggarwal
- BD Gitter
- BL Daugherty
- C Blanquart
- C Bombardier
- C Brideau
- C Emond
- C Gloxhuber
- C Jiang
- C Kemal
- C Kunsch
- C Laudanna
- C Liebmann
- C Liebmann
- C Liu
- C Liu
- C Mendoza-Milla
- C Pfeifer
- C Shen
- C Takeguchi
- CA Dinarello
- CA Dinarello
- CA Dinarello
- CA Maggi
- CA Maggi
- CA Smith
- CA Winter
- CA Winter
- CC Chan
- CD Anderson
- CD Funk
- CH Hannum
- CH Pontzer
- CJ Dunn
- CJ Hawkey
- CJ Mussap
- CM Lee
- CM Yang
- CN Hensby
- CSJ Walpole
- CV Winder
- D Bishop-Bailey
- D Branceni
- D D’Ambrosio
- D Eggerickx
- D Faust
- D Ignar
- D Kollias
- D Kontoyiannis
- D Lorenz
- D Mastrangelo
- D O’Gradaigh
- D Pruneau
- D Riendeau
- D Riendeau
- D Rossi
- DA Flick
- DA Kalbhen
- DB Carter
- DB Colagiovanni
- DC Manning
- DE Furst
- DE Griswold
- DE Griswold
- DE Moller
- DF Woodward
- DJ Grainger
- DJ McCarty
- DJ McCarty
- DK Gemmel
- DL Saussy Jr
- DM Butler
- DM Crothers
- DM Knight
- DM Siegel
- DT Beattie
- E Arrigoni-Martelli
- E Bosio
- E Fujihira
- E Fujii
- E Moore
- E Sarrubi
- E Schött
- E Whitehorn
- E Wong
- EA Graham
- EA Higgs
- EE Opas
- EF Webb
- EG Weirich
- EH Karran
- EJ Fernandez
- EK Ainscow
- EM Eugui
- EM Kudlacz
- EM Lasché
- ES Alnemri
- ES Tai
- F D’Acquisto
- F Erdö
- F Gbahou
- F Gobeil
- F Herrmann
- F Lembeck
- F Marceau
- F Marceau
- F Nantel
- F Sallusto
- F Yan
- F Zhang
- FJ Legat
- FJT Staal
- FR Cochran
- G Buell
- G Camussi
- G Cirino
- G D’Amato
- G Hofrichter
- G Jancso
- G Tonelli
- G Wagner
- G Wiemer
- G Wilhelmi
- G Woerly
- GA FitzGerald
- GA Higgs
- GB Penn
- GC Sen
- GC Viscomi
- GD Anderson
- GJ Hankey
- GN Prado
- GP Lewis
- GP O’Neill
- GR Bobalik
- GR Drummond
- GT Le
- GV Lucca De
- GW Moe
- H Abt
- H Akiyama
- H Cambridge
- H Fahmi
- H Heitsch
- H Kojo
- H Safayhi
- H Salari
- H Schmidt
- H Selye
- H Shionoya
- H Shirota
- H Umehara
- HA Schreuder
- HD Lim
- HD Lim
- HG Alpermann
- HG Schaible
- HG Vogel
- HG Vogel
- HG Vogel
- HG Vogel
- HG Vogel
- HG Vogel
- I Nicoletti
- IE Bush
- IJ Esch De
- IL Bonta
- IM Adcock
- IM McLay
- IS Figari
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- J Veenstra
- J Waugh
- JA Gracie
- JA Kim
- JA Mitchell
- JB Calixto
- JB Cheng
- JB Warren
- JC Beaujouan
- JC Souza Pinto
- JD Winkler
- JF Kachur
- JG Meingassner
- JG Menke
- JG Vallejo
- JH Lee
- JH Ruth
- JI Braga da Motta
- JI Shigeta
- JJ Chen
- JJ Haringman
- JJ Moreno
- JJ Young
- JK Gierse
- JKF Hess
- JL Bascands
- JL Field
- JL Field
- JL Henry
- JL Kang
- JL Kang
- JL Martal
- JM Young
- JM Young
- JM Young
- JP Fortin
- JP Galizzi
- JP Portanova
- JP Tarayre
- JR Bing
- JR Burke
- JR Vane
- JS Faires
- JS Warren
- JS Yuan
- JT Whicher
- JW Christman
- JW Christman
- JW Watson
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- K Bon
- K Heynink
- K Hirota
- K Iwasaki
- K Nagata
- K Natarajan
- K Paulini
- K Paulini
- K Pfizenmaier
- K Redlich
- K Ren
- K Seibert
- K Seibert
- K Sugio
- K Tanaka
- K Thiam
- K Tiku
- K Tsumuri
- K Vuoltteenaho
- K Watanabe
- K Watanabe
- K Wirth
- KA Schneck
- KB Gordon
- KC Appell
- KH Sensch
- KJ Wirth
- KM Mohler
- KP Meyers
- KR Aupperle
- KU Weithmann
- KU Weithmann
- L Acarin
- L Chen
- L Harvath
- L Quartara
- L Reber
- L Sancilio
- L Seguin
- L Seguin
- L Singh
- LA Davis
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- LJ Crofford
- LL Iversen
- LM Blatt
- LM Young De
- LM Young De
- LMF Leeb-Lundberg
- LO Randall
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- M Bradford
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- M Feldmann
- M Frimmer
- M Félétou
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- M Katin
- M Katsumata
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- M Liang
- M Liang
- M Matsubara
- M Murakawa
- M MĂĽhlbauer
- M Otsuka
- M Ouellet
- M Peterfalvi
- M Roch-Arveiller
- M Tramontana
- M Zhang
- MA Botrel
- MA Cascieri
- MA Hull
- MA Matuszek
- MB Lawrence
- MD Brand
- MD Brand
- ME Poynter
- ME Rosenthale
- ME Rosenthale
- MG Fried
- MG O’Sullivan
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- MJ Uddin
- MK Pugsley
- ML Richards
- MM Campos
- MM Chang
- MM Chaturvedi
- MM Krause
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- MN Perkins
- MNJ Rupniak
- MR Shalaby
- MS Kramer
- MS Nanes
- MSS Palanki
- MSS Palanki
- N Ackerman
- N Fujioka
- N McClure
- N Minami
- N Mukaida
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- N Scheinfeld
- N Selve
- NE Rhaleb
- NE Rhaleb
- NJ Brenner
- NMJ Rupniak
- NMJ Rupniak
- NV Chandrasekharan
- O RĂĄdmark
- OP Gupta
- P Borgeat
- P Clarke
- P Cole
- P Delerive
- P D’Orléans-Juste
- P Holm-Pedersen
- P Houshmand
- P Kuhl
- P Li
- P Phelps
- P Schiatti
- P Schönhöfer
- P Traxler
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- PR Devchand
- PV Halushka
- QN Diep
- R Boopathy
- R Cirillo
- R Dewes
- R Fleischmann
- R Hicks
- R Hill
- R Hill
- R Hosoki
- R Lewis
- R Meier
- R Miesel
- R Moqbel
- R Nikolov
- R Panaccione
- R Patacchini
- R Schrenk
- R Sharma
- R William
- RA Bakker
- RA Coleman
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- RB Innis
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- RD Nelson
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- RJ Boucek
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- RM Atkinson
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- RM Burch
- RM Burch
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- RM Burch
- RM Hagan
- RN Williams
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- RR Bowers
- RR Brooks
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- RS Cvetkovic
- RT Palframan
- S Bourgoin
- S Boyden
- S Chen
- S Cheng
- S Daoui
- S Dion
- S Easthope
- S Eltayeb
- S Gosh
- S Gupta
- S Gupta
- S Hallé
- S Kargman
- S Kirchner
- S Kumar
- S Kunz
- S Leyck
- S McLean
- S McLean
- S Meini
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- S Mong
- S Nakae
- S Nakanishi
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- S Rosi
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- SA Alla
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- SC Bailey
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- SH Lee
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- SK Butt
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- SM Vogel
- SP Khanapure
- SW Martin
- T Croci
- T Feres
- T Griesbacher
- T Hökfelt
- T Ichiyama
- T Izumi
- T Jung
- T Kalajdzic
- T Kilic
- T Klein
- T Mijatovic
- T Mikami
- T Murata
- T Murata
- T Nishi
- T Oda
- T Peng
- T Pouw-Kraan Van der
- T Sakurada
- T Shimizu
- T Syrovets
- T Tatsuda
- T Wagner-Jauregg
- T Zielinski
- TA Bird
- TA Pugsley
- TC Nichols
- TJ Evans
- TJ Schall
- TM Cunha
- TR Jones
- TS Fröde
- TS Fröde
- TT Chau
- TW Lovenberg
- U Wagner
- US Euler Von
- V Chapman
- VJ Stecher
- W Dichtl
- W Eberhardt
- W Eberhardt
- W Feldberg
- W Hu
- W Spencer
- W Xie
- WA Cromlish
- WG Kaelin Jr
- WP Arend
- WP Arend
- WP Fung-Leung
- WS Powell
- X Edmonds-Alt
- X Emonds-Alt
- Y Harada
- Y Macotela
- Y Matzner
- Y Oyanagui
- Y Pande
- Y Pande
- Y Saita
- Y Tian
- Y Ushida
- Y Zhang
- YF Liu
- YH Joo
- YH Kim
- Z Geng
- ZE Mielens
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- Field of study