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9 research outputs found
Structural determinant for inducing RORgamma specific inverse agonism triggered by a synthetic benzoxazinone ligand
Author
A Vagin
AK Shiau
+32Â more
BP Fauber
C Lock
CM Koth
Craig P. Wildes
Douglas J. Marcotte
GN Murshudov
H Xie
I Muegge
II Ivanov
J Chao
JA Kallen
Jayanth V. Chodaparambil
John H. Jones
Kevin Little
KK Singarapu
L Jin
Laura F. Silvian
M Chabaud
Noel A. Powell
O René
P Emsley
PS Danielian
S Fujino
S Fujita-Sato
S Kurebayashi
T Wang
TGG Battye
V Nahoum
Y Wang
Y Zhang
Y Zhang
YuTing Liu
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
Full text link
Crossref
Identification of an allosteric binding site for RORγt inhibition
Author
A Chaikuad
AJ McCoy
+42Â more
AM Brzozowski
BP Fauber
BP Fauber
BP Fauber
BP Fauber
C Stehlin
DM Heery
F Isono
FW Studier
H Gronemeyer
II Ivanov
IJ Bruno
JM Harris
JP Overington
K Ichiyama
L Jin
L Nagy
LA Solt
LA Solt
M Nichols
M Scheepstra
MD Winn
N Kumar
P Emsley
PD Adams
PR Evans
PV Afonine
RA Laskowski
S Fujita-Sato
SD Weeks
T Kanai
T Xu
T Yang
TGG Battye
TS Hughes
TW Moore
VB Chen
XO Yang
Y Wang
Y Yang
YW He
Z Huang
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Discovery and structural optimization of 4-(4-(benzyloxy)phenyl)-3,4-dihydropyrimidin-2(1H)-ones as RORc inverse agonists
Author
AM Jetten
BP Fauber
+40Â more
BP Fauber
BP Fauber
C Gege
Chun Wu
FH Niesen
H Toyama
HS Ranhotra
J Chao
Jian-qin Jiang
JR Huh
JR Huh
K Suino-Powell
L Jin
LA Solt
LA Solt
LA Solt
M Dubernet
MB van Niel
MW Pantoliano
N Kumar
PM Khan
RA Friesner
Rui Wang
S Fujita-Sato
T Xu
T Yang
TM Kamenecka
W Ouyang
Xi-shan Wu
Xiao-qian Xue
Xiao-yu Luo
Y Wang
Y Zhang
Yan Zhang
Yan-li Xing
Yong Xu
Yong-zhi Lu
Yu Song
Yu-lai Zhou
Z Li
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Metabolic plasticity underpins innate and acquired resistance to LDHA inhibition
Author
A Le
A Viale
+72Â more
AA Borisy
Aaron Boudreau
Aihe Zhou
Alex Vanderbilt
Anna Hitz
Anneleen Daemen
B Magnuson
Binqing Wei
BP Fauber
BP Fauber
C Granchi
Charles Eigenbrot
Christopher Del Nagro
David Peterson
DC Gray
Deepak Sampath
DG Hardie
DM Gwinn
E Vanderporten
G Qing
Georgia Hatzivassiliou
GL Semenza
H Busch
H Girgis
H Shim
H Xie
Hans E Purkey
HN Aithal
Ivana Yen
J Billiard
Jodie Pang
K Birsoy
K Inoki
KA Brand
Kirk Robarge
L Copeland
Laura Corson
Laurent Salphati
LR Pearce
Mandy Kwong
Marcia Belvin
Marie Evangelista
Mark McCleland
MI Koukourakis
MI Koukourakis
MI Koukourakis
Min Gao
MR Owen
NA Shirwany
P Seth
Peter K Jackson
PS Dragovich
PS Dragovich
RA Ward
Raju Pusapati
Rebecca Hong
Ron Firestein
Sharada Labadie
Shiva Malek
Shuguang Ma
Simon Williams
Steve Sideris
Thomas O'Brien
Tommy Lai
VR Fantin
WB Novoa
XM Ma
Y Shitara
Yingjie Li
Z Feng
Zhongguo Chen
ZJ Reitman
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Human Lactate Dehydrogenase A Inhibitors: A Molecular Dynamics Investigation
Author
A Kohlmann
A Le
+54Â more
B Hess
B Hess
B. Mario Pinto
BK Mai
BP Fauber
C Granchi
C Granchi
C Jarzynski
CI Bayly
Claudio M. Soares
CM Eszes
CR Dunn
D Hanahan
DA Case
E Vanquelef
F Colizzi
FB Straub
FY Dupradeau
G Bussi
GM Torrie
H Xie
HJC Berendsen
I Banga
J Gore
J Wang
JA Read
K Swiderek
K Swiderek
KS Rebecca
L Zhuang
LM Deck
M Parrinello
MI Koukourakis
MI Koukourakis
O Trott
O Warburg
P Cieplak
P Nicolini
PS Dragovich
PS Ward
RA Gatenby
RA Ward
RD Goldman
S McClendon
S Park
S Park
T Darden
T Kanno
U Essmann
V Hornak
VB Chen
WG Hoover
Y Kolev
Yun Shi
Publication venue
'Public Library of Science (PLoS)'
Publication date
Field of study
No full text
Crossref
Development of a Topical Treatment for Psoriasis Targeting RORγ: From Bench to Skin
Author
AM Bowcock
AM Jetten
+52Â more
AM Lin
Andrzej T Slominski
Anton M. Jetten
AT Slominski
AT Slominski
BP Fauber
C Leonardi
Carlos E. Peredo
David Rickard
DJ Cua
DJ Kojetin
E Witte
Edwige Nicodeme
EL Berg
Elizabeth Millerman
Fabrice Viviani
G Bergamini
Hans Hofland
II Ivanov
J Skepner
Javier Cote-Sierra
Jean-Marie Brusq
Jean-Philippe Therrien
Jessica Neil
JG Krueger
JM Reynolds
JR Huh
JR Huh
KA Papp
KE Nograles
L van der Fits
LA Solt
N Kumar
N Kumar
N Manel
O Rene
P Di Meglio
RA Clark
S Kurebayashi
S Xiao
Susan H. Smith
T Xu
Thi Bui
Veronique Birault
W Zhang
XA Qu
XO Yang
Y Cai
Y Takeda
Y Wang
Y Zheng
Yukimasa Takeda
Publication venue
'Public Library of Science (PLoS)'
Publication date
Field of study
No full text
Crossref
RORγt and RORα signature genes in human Th17 cells
Author
A Kramer
Aimee De Leon-Tabaldo
+54Â more
AM Jetten
Anne Fourie
BP Fauber
C Carlberg
C Leonardi
C Luci
EV Acosta-Rodriguez
FR Santori
G Eberl
G Eberl
Glenda Castro
I Dzhagalov
I Dzhagalov
I Villey
II Ivanov
II Ivanov
J Du
J Kallen
J Skepner
J Yang
JA Kallen
JC Clemente
Jingxue Yu
Jonathan Blevitt
KA Papp
Karen Ngo
KJ Livak
Krystal Herman
M Becker-Andre
M Ciofani
MA Ortiz
Marina I. Nelen
MJ McGeachy
N Manel
P Miossec
P Soroosh
Patrick Wilkinson
Q Ruan
Robert Kuhn
Rosa Luna-Roman
S Xiao
S Zhao
Shanrong Zhao
T Hirose
Tinghua Cao
U Matysiak-Scholze
V Giguere
W Hueber
Wai-Ping Fung-Leung
Xiaohua Xue
XO Yang
Xuejun Liu
Yeonseok Chung
YW He
Publication venue
'Public Library of Science (PLoS)'
Publication date
Field of study
No full text
Crossref
Preclinical and clinical characterization of the RORγt inhibitor JNJ-61803534
Author
A Deodhar
AL Gomes
+59Â more
AM Jetten
AT Slominski
AT Slominski
AT Slominski
BP Fauber
BS McKenzie
C Dong
C Gege
C Leonardi
C Liu
C Luci
C Nunez
C Ritchlin
CE Sutton
CL Leonardi
DA Kummer
E Safrany
F Ramirez-Valle
FR Santori
GS LluÃs Puig
H Spits
HA Blair
HR Yen
IB McInnes
IB McInnes
II Ivanov
J Bowes
JC-C Wei
JK Barbay
K Ichiyama
K Venken
KA Papp
KA Papp
KA Papp
L van der Fits
L Zhou
M Gazouli
M Gilliet
M Leppkes
MR Chang
N Sun
NE Martinez
P Mease
P Nash
P Rahman
P Soroosh
PJ Mease
R Du
RL Thurmond
S Kurebayashi
S Nakae
SL Gaffen
T Kuwabara
VM Tanis
X Hu
X Xue
Y Kochi
YJ Lee
Z Sun
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref
Pharmacologic modulation of RORγt translates to efficacy in preclinical and translational models of psoriasis and inflammatory arthritis
Author
AM Jetten
AV Rachitskaya
+65Â more
BP Fauber
BS McKenzie
C Dong
C Leonardi
C Nunez
C Ritchlin
CE Sutton
CE Sutton
CL Leonardi
CL Roark
DA Martin
DR Withers
E Safrany
FR Santori
H Sofen
H Spits
HL Rizzo
HR Yen
IB McInnes
IB McInnes
II Ivanov
J Bowes
J Skepner
JK Kolls
JP Sherlock
JR Chan
JR Huh
K Ichiyama
K Pavelka
KA Papp
KA Papp
KA Papp
KE Webster
KS Voo
L Moreira-Teixeira
L Zhou
LA Solt
LK Stamp
M Chabaud
M Ciofani
M Ferran
M Gazouli
M Leppkes
M Suarez-Farinas
MC Genovese
MC Genovese
MR Chang
N Caccamo
P Rahman
P Soroosh
PJ Mease
PJ Mease
S Kotake
S Peternel
S Xiao
SL Gaffen
SP Singh
T Xu
TN Canavan
TN Collingwood
TP Burris
X Hu
Y Cai
Y Kochi
Z Sun
Publication venue
'Springer Science and Business Media LLC'
Publication date
Field of study
No full text
Crossref